Proteins > Gamma-aminobutyric acid type B receptor subunit 2
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Gamma-aminobutyric acid type B receptor subunit 2
A gamma-aminobutyric acid type B receptor subunit 2 that is encoded in the genome of rat. [OMA:O88871, PRO:DNx]
Synonyms
GABA-B receptor 2;
GABA-B-R2;
GABA-BR2;
GABABR2;
Gb2;
G-protein coupled receptor 51
Research
Bioassay Publications (8)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 1 (12.50) | 18.7374 |
| 1990's | 6 (75.00) | 18.2507 |
| 2000's | 1 (12.50) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (14)
Drugs with Inhibition Measurements
Partial GABAA receptor agonists. Synthesis and in vitro pharmacology of a series of nonannulated analogs of 4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
3-Thienyl- and 3-furylaminobutyric acids. Synthesis and binding GABAB receptor studies.Journal of medicinal chemistry, , Volume: 34, Issue:8, 1991
Synthesis and pharmacological evaluation of gamma-aminobutyric acid analogues. New ligand for GABAB sites.Journal of medicinal chemistry, , Volume: 30, Issue:4, 1987
Synthesis and pharmacological evaluation of novel gamma-aminobutyric acid type B (GABAB) receptor agonists as gastroesophageal reflux inhibitors.Journal of medicinal chemistry, , Jul-24, Volume: 51, Issue:14, 2008
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
Synthesis and biochemical evaluation of baclofen analogues locked in the baclofen solid-state conformation.Journal of medicinal chemistry, , Volume: 34, Issue:4, 1991
3-Thienyl- and 3-furylaminobutyric acids. Synthesis and binding GABAB receptor studies.Journal of medicinal chemistry, , Volume: 34, Issue:8, 1991
Synthesis and pharmacological evaluation of gamma-aminobutyric acid analogues. New ligand for GABAB sites.Journal of medicinal chemistry, , Volume: 30, Issue:4, 1987
Synthesis and pharmacological evaluation of novel gamma-aminobutyric acid type B (GABAB) receptor agonists as gastroesophageal reflux inhibitors.Journal of medicinal chemistry, , Jul-24, Volume: 51, Issue:14, 2008
Phosphinic acid analogues of GABA. 2. Selective, orally active GABAB antagonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
Synthesis and pharmacology of the baclofen homologues 5-amino-4-(4-chlorophenyl)pentanoic acid and the R- and S-enantiomers of 5-amino-3-(4-chlorophenyl)pentanoic acid.Journal of medicinal chemistry, , Jun-03, Volume: 42, Issue:11, 1999
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
Synthesis and pharmacological evaluation of novel gamma-aminobutyric acid type B (GABAB) receptor agonists as gastroesophageal reflux inhibitors.Journal of medicinal chemistry, , Jul-24, Volume: 51, Issue:14, 2008
Phosphinic acid analogues of GABA. 2. Selective, orally active GABAB antagonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.Journal of medicinal chemistry, , Aug-18, Volume: 38, Issue:17, 1995