Page last updated: 2024-08-07 12:42:14
Growth hormone secretagogue receptor type 1
A growth hormone secretagogue receptor that is encoded in the genome of rat. [OMA:O08725, PRO:DNx]
Synonyms
GHS-R;
GH-releasing peptide receptor;
GHRP;
Ghrelin receptor
Research
Bioassay Publications (5)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 2 (40.00) | 18.2507 |
| 2000's | 1 (20.00) | 29.6817 |
| 2010's | 1 (20.00) | 24.3611 |
| 2020's | 1 (20.00) | 2.80 |
Compounds (7)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| l 692429 | Rattus norvegicus (Norway rat) | IC50 | 0.0600 | 1 | 1 |
| substance p, phe(5)-trp(7,9)-leu(11)- | Rattus norvegicus (Norway rat) | IC50 | 0.1337 | 3 | 3 |
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| l 692429 | Rattus norvegicus (Norway rat) | EC50 | 0.0600 | 1 | 1 |
| l 163191 | Rattus norvegicus (Norway rat) | EC50 | 0.0013 | 1 | 1 |
| cp 424391 | Rattus norvegicus (Norway rat) | EC50 | 0.0030 | 1 | 1 |
| tabimorelin | Rattus norvegicus (Norway rat) | EC50 | 0.0180 | 1 | 1 |
| l 162752 | Rattus norvegicus (Norway rat) | EC50 | 0.0140 | 1 | 1 |
| sk&f 110679 | Rattus norvegicus (Norway rat) | EC50 | 0.0058 | 2 | 2 |