Page last updated: 2024-08-18

pyrroles and Malaria

pyrroles has been researched along with Malaria in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19904 (20.00)18.7374
1990's1 (5.00)18.2507
2000's6 (30.00)29.6817
2010's9 (45.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrew, AK; Cooper, CA; Moore, JM; Morffy Smith, CD; Russ, BN1
Arang, N; Bello, T; Dudgeon, DR; Glennon, EK; Gujral, TS; Kain, HS; Kaushansky, A; Walter, ENF1
Çavdar, H; Ekinci, D; Kocaoğlu, E; Şentürk, M; Supuran, CT; Talaz, O1
Douglass, AN; Kain, HS; Kappe, SH; Kaushansky, A; Lakshmanan, V; Metzger, PG; Mikolajczak, SA1
Hempel, C; Hoyer, N; Kurtzhals, JA; Staalsø, T1
Abdullahi, M; Arang, N; Austin, LS; Billman, ZP; Douglass, AN; Hume, JCC; Kain, HS; Kappe, SHI; Kaushansky, A; Mikolajczak, SA; Murphy, SC1
Kancharla, P; Kelly, JX; Reynolds, KA1
Basilico, N; Brun, R; Casagrande, M; Parapini, S; Sparatore, A; Sparatore, F; Taramelli, D; Wittlin, S1
Bhanot, P; Panchal, D1
Cortopassi, WA; França, TC; Krettli, AU; Oliveira, AA; Penna-Coutinho, J1
Schramm, VL1
Ager, A; Gerena, L; Guan, J; Lin, AJ; O'Neil, M; Obaldia, N; Zhang, Q1
Li, Q; Lin, AJ; Skillman, DS; Smith, K; Xie, LH; Zhang, J1
Gendler, PL; Rapoport, H1
Hayashi, M; Hirata, H; Horii, T; Kawauchi, K; Kim, HS; Mitamura, T; Moriyama, Y; Shibata, Y; Tsuboi, S; Wataya, Y1
Ang, KK; Hamann, MT; Higa, T; Holmes, MJ; Kara, UA1
Ang, KK; Holmes, MJ; Kara, UA1
Blanton, CD; Sowell, JW1
Bailey, DM; Johnson, RE; Salvador, UJ1
Aviado, DM1

Reviews

2 review(s) available for pyrroles and Malaria

ArticleYear
Immucillins as antibiotics for T-cell proliferation and malaria.
    Nucleosides, nucleotides & nucleic acids, 2004, Volume: 23, Issue:8-9

    Topics: Animals; Anti-Bacterial Agents; Cell Proliferation; Deoxyguanosine; Erythrocytes; Humans; Hypoxanthine; Kinetics; Lymphocyte Activation; Malaria; Models, Chemical; Phenotype; Plasmodium falciparum; Purine Nucleosides; Purines; Pyrimidinones; Pyrroles; T-Lymphocytes

2004
Chemotherapy of Plasmodium berghei.
    Experimental parasitology, 1969, Volume: 25, Issue:1

    Topics: Animals; Anthracenes; Anti-Bacterial Agents; Anti-Infective Agents; Antimalarials; Benzene Derivatives; Cardiovascular System; Central Nervous System; Coloring Agents; Enzyme Inhibitors; Erythropoiesis; Histamine; Hormones; Malaria; Malaria, Avian; Mice; Naphthyridines; Organometallic Compounds; Plasmodium; Pteridines; Pyrimidines; Pyrroles; Quinolines; Rats; Sulfonamides; Sulfones; Thiazoles; Vitamins

1969

Other Studies

18 other study(ies) available for pyrroles and Malaria

ArticleYear
A novel murine model for assessing fetal and birth outcomes following transgestational maternal malaria infection.
    Scientific reports, 2019, 12-20, Volume: 9, Issue:1

    Topics: Animals; Cell Survival; Chromosome Pairing; Disease Models, Animal; Female; Finite Element Analysis; Malaria; Malaria, Falciparum; Mice; Nerve Regeneration; Polymers; Pregnancy; Pregnancy Complications, Parasitic; Pyrroles; Tissue Scaffolds

2019
Identifying host regulators and inhibitors of liver stage malaria infection using kinase activity profiles.
    Nature communications, 2017, 11-01, Volume: 8, Issue:1

    Topics: Animals; Cell Line, Tumor; HEK293 Cells; Hepatocytes; Host-Parasite Interactions; Humans; Indoles; Liver; Malaria; Mice; Piperazines; Plasmodium yoelii; Protein Kinase Inhibitors; Protein Kinases; Purines; Pyrroles; RNA Interference; Roscovitine; Sporozoites; Sunitinib

2017
Determination of the inhibitory effects of N-methylpyrrole derivatives on glutathione reductase enzyme.
    Journal of enzyme inhibition and medicinal chemistry, 2019, Volume: 34, Issue:1

    Topics: Antimalarials; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glutathione Reductase; Malaria; Molecular Structure; Pyrroles; Structure-Activity Relationship

2019
Malaria parasite liver stages render host hepatocytes susceptible to mitochondria-initiated apoptosis.
    Cell death & disease, 2013, Aug-08, Volume: 4

    Topics: Animals; Apoptosis; Hepatocytes; Indoles; Malaria; Mice; Mice, Inbred BALB C; Mitochondria; Parasite Load; Pyrroles; Signal Transduction

2013
Effects of the vascular endothelial growth factor receptor-2 (VEGFR-2) inhibitor SU5416 on in vitro cultures of Plasmodium falciparum.
    Malaria journal, 2014, May-28, Volume: 13

    Topics: Animals; Antimalarials; Cytosol; Disease Models, Animal; Erythrocytes; Female; Flow Cytometry; Humans; Immunohistochemistry; Indoles; Malaria; Mice, Inbred C57BL; Plasmodium berghei; Plasmodium falciparum; Pyrroles; Tyrosine; Vascular Endothelial Growth Factor Receptor-2

2014
Host-based Prophylaxis Successfully Targets Liver Stage Malaria Parasites.
    Molecular therapy : the journal of the American Society of Gene Therapy, 2015, Volume: 23, Issue:5

    Topics: Animals; Antimalarials; Cell Line; Disease Models, Animal; Female; Imidazoles; Indoles; Life Cycle Stages; Liver; Malaria; Malaria, Falciparum; Mice; Mice, Transgenic; Parasite Load; Piperazines; Plasmodium; Plasmodium falciparum; Post-Exposure Prophylaxis; Proto-Oncogene Proteins c-bcl-2; Pyrroles; Tumor Suppressor Protein p53

2015
Synthesis and Structure-Activity Relationships of Tambjamines and B-Ring Functionalized Prodiginines as Potent Antimalarials.
    Journal of medicinal chemistry, 2015, Sep-24, Volume: 58, Issue:18

    Topics: Animals; Antimalarials; Drug Resistance, Multiple; Female; Hep G2 Cells; Humans; Malaria; Mice; Plasmodium falciparum; Plasmodium yoelii; Pyrroles; Structure-Activity Relationship

2015
Antimalarial activity of novel pyrrolizidinyl derivatives of 4-aminoquinoline.
    Bioorganic & medicinal chemistry letters, 2008, Jul-01, Volume: 18, Issue:13

    Topics: Aminoquinolines; Animals; Antimalarials; Body Weight; Cell Line; Chloroquine; Humans; Malaria; Mice; Microsomes; Models, Chemical; Plasmodium berghei; Plasmodium falciparum; Pyrroles

2008
Activity of a trisubstituted pyrrole in inhibiting sporozoite invasion and blocking malaria infection.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:10

    Topics: Animals; Antimalarials; Female; Hep G2 Cells; Humans; Malaria; Mice; Plasmodium berghei; Plasmodium yoelii; Polymerase Chain Reaction; Pyrroles; Sporozoites

2010
Antimalarial activity of potential inhibitors of Plasmodium falciparum lactate dehydrogenase enzyme selected by docking studies.
    PloS one, 2011, Volume: 6, Issue:7

    Topics: Animals; Antimalarials; Atorvastatin; Catalytic Domain; Cells, Cultured; Enzyme-Linked Immunosorbent Assay; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Itraconazole; L-Lactate Dehydrogenase; Malaria; Mice; Plasmodium falciparum; Pyrroles; Triazoles

2011
Antimalarial activities of new pyrrolo[3,2-f]quinazoline-1,3-diamine derivatives.
    Antimicrobial agents and chemotherapy, 2005, Volume: 49, Issue:12

    Topics: Animals; Antimalarials; Disease Models, Animal; Malaria; Mice; Plasmodium berghei; Plasmodium falciparum; Pyrroles; Quinazolines

2005
New potential antimalarial agents: therapeutic-index evaluation of pyrroloquinazolinediamine and its prodrugs in a rat model of severe malaria.
    Antimicrobial agents and chemotherapy, 2006, Volume: 50, Issue:5

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Malaria; Maximum Tolerated Dose; Parasitemia; Plasmodium berghei; Prodrugs; Pyrroles; Quinazolines; Random Allocation; Rats; Rats, Sprague-Dawley; Sesquiterpenes; Therapeutic Equivalency

2006
Permethyl analogue of the pyrrolic antibiotic distamycin A.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:1

    Topics: Animals; Antimalarials; Cells, Cultured; Distamycins; Malaria; Mice; Plasmodium berghei; Pyrroles

1981
Cycloprodigiosin hydrochloride obtained from Pseudoalteromonas denitrificans is a potent antimalarial agent.
    Biological & pharmaceutical bulletin, 1999, Volume: 22, Issue:5

    Topics: Animals; Antimalarials; Disease Models, Animal; Drug Evaluation, Preclinical; Gram-Negative Aerobic Bacteria; Humans; In Vitro Techniques; Indoles; Malaria; Male; Mice; Mice, Inbred ICR; Plasmodium falciparum; Pyrroles

1999
In vivo antimalarial activity of the beta-carboline alkaloid manzamine A.
    Antimicrobial agents and chemotherapy, 2000, Volume: 44, Issue:6

    Topics: Animals; Antimalarials; Carbazoles; Indoles; Malaria; Male; Mice; Microscopy, Electron; Plasmodium berghei; Pyrroles

2000
Immune-mediated parasite clearance in mice infected with Plasmodium berghei following treatment with manzamine A.
    Parasitology research, 2001, Volume: 87, Issue:9

    Topics: Animals; Antibodies, Protozoan; Antimalarials; Carbazoles; Cytokines; Erythrocytes; Immunoglobulin G; Indoles; Malaria; Male; Mice; Parasitemia; Plasmodium berghei; Pyrroles

2001
New synthesis of substituted pyrrolo[1,2-alpha][1,3]diazepine and its pharmacological activity.
    Journal of pharmaceutical sciences, 1976, Volume: 65, Issue:6

    Topics: Animals; Anti-Inflammatory Agents; Antineoplastic Agents; Antiviral Agents; Azepines; Blood Pressure; Central Nervous System; Cholesterol; Diuretics; Hypoglycemic Agents; Lipoproteins; Malaria; Mice; Plasmodium berghei; Pyrroles; Rats

1976
Pyrrole antibacterial agents. 1. Compounds related to pyoluteorin.
    Journal of medicinal chemistry, 1973, Volume: 16, Issue:11

    Topics: Animals; Anti-Bacterial Agents; Benzoates; Escherichia coli; Klebsiella Infections; Malaria; Mice; Microbial Sensitivity Tests; Plasmodium berghei; Proteus vulgaris; Pseudomonas aeruginosa; Pyrroles; Schistosoma mansoni; Schistosomiasis; Staphylococcal Infections; Staphylococcus; Structure-Activity Relationship

1973