Page last updated: 2024-08-16

zolpidem and gaboxadol

zolpidem has been researched along with gaboxadol in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's13 (65.00)29.6817
2010's7 (35.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Alva, H; Blednov, YA; Harris, RA; Jung, S; Rosahl, T; Wallace, D; Whiting, PJ1
Cagetti, E; Liang, J; Olsen, RW; Spigelman, I1
Bjerrum, OJ; Blackburn-Munro, G; Jensen, DG; Rode, F1
Goldstein, PA; Harrison, NL; Jia, F; Pignataro, L; Schofield, CM; Yue, M1
Deacon, S; Dijk, DJ; Lundahl, J; Walsh, JK1
Deacon, S; Loft, H; Lundahl, J; Staner, C; Staner, L1
Hutson, PH; McDonald, LM; Sheppard, WF; Sohal, B; Staveley, SM; Tattersall, FD1
Adrien, J; Aixendri, R; Alexandre, C; Dordal, A; Guzman, A; Hamon, M1
Ahring, PK; Erichsen, HK; Larsen, JS; Lopez-Garcia, JA; Mirza, NR; Munro, G; Nielsen, EØ; Rivera-Arconada, I1
Agrawal, N; Alexander, R; Boyle, J; Calder, N; Danjou, P; Fu, I; Gargano, C; McCrea, JB; Murphy, MG1
Cook, JM; Groenink, L; Hopkins, SC; Klanker, M; Korte, SM; Olivier, B; Van Linn, ML; Vinkers, CH1
Eglin, M; Hajak, G; Hedner, J; Loft, H; Lundahl, J; Lütolf, S; Stórustovu, SI1
Deacon, S; Dijk, DJ; James, LM; Peters, S; Walsh, JK1
Leufkens, TR; Lund, JS; Vermeeren, A1
Deacon, S; Ebert, B; Ferri, R; Ma, J; Ray, S; Snyder, E; Svetnik, V; Walsh, JK1
Deacon, S; Lundahl, J; Maurice, D; Staner, L1
Barberis, A; Benfenati, F; Cancedda, L; Fiumelli, H; Succol, F1
Brazhe, A; Jensen, K; Jessen, SB; Lauritzen, M; Lind, BL; Mathiesen, C; Thomsen, K1
Lingford-Hughes, A; Muthukumaraswamy, S; Myers, J; Nutt, D; Papadopoulos, A; Wilson, S1
Herring, WJ; Lines, C; Ma, J; Roth, T; Snyder, E; Svetnik, V1

Trials

9 trial(s) available for zolpidem and gaboxadol

ArticleYear
The selective extrasynaptic GABAA agonist, gaboxadol, improves traditional hypnotic efficacy measures and enhances slow wave activity in a model of transient insomnia.
    Sleep, 2007, Volume: 30, Issue:5

    Topics: Adolescent; Adult; Cross-Over Studies; Delta Rhythm; Dose-Response Relationship, Drug; Double-Blind Method; Female; GABA Agonists; GABA-A Receptor Agonists; Humans; Hypnotics and Sedatives; Isoxazoles; Male; Middle Aged; Polysomnography; Pyridines; Sleep; Sleep, REM; Theta Rhythm; Wakefulness; Zolpidem

2007
Short-term treatment with gaboxadol improves sleep maintenance and enhances slow wave sleep in adult patients with primary insomnia.
    Psychopharmacology, 2007, Volume: 195, Issue:1

    Topics: Adolescent; Adult; Aged; Cross-Over Studies; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Electroencephalography; GABA Agonists; Headache; Humans; Isoxazoles; Middle Aged; Nausea; Polysomnography; Pyridines; Sex Factors; Sleep Initiation and Maintenance Disorders; Sleep Stages; Tachycardia; Time Factors; Treatment Outcome; Zolpidem

2007
Tolerability, pharmacokinetics and night-time effects on postural sway and critical flicker fusion of gaboxadol and zolpidem in elderly subjects.
    British journal of clinical pharmacology, 2009, Volume: 67, Issue:2

    Topics: Aged; Cross-Over Studies; Double-Blind Method; Female; Flicker Fusion; GABA Agonists; Humans; Isoxazoles; Male; Postural Balance; Pyridines; Reaction Time; Zolpidem

2009
A 2-week efficacy and safety study of gaboxadol and zolpidem using electronic diaries in primary insomnia outpatients.
    Sleep medicine, 2009, Volume: 10, Issue:7

    Topics: Adolescent; Adult; Aged; Ambulatory Care; Diagnostic and Statistical Manual of Mental Disorders; Double-Blind Method; Drug Administration Schedule; Electronic Data Processing; Female; GABA Agonists; Humans; Isoxazoles; Male; Middle Aged; Pyridines; Severity of Illness Index; Single-Blind Method; Sleep Initiation and Maintenance Disorders; Substance Withdrawal Syndrome; Surveys and Questionnaires; Time Factors; Treatment Outcome; Young Adult; Zolpidem

2009
Sex differences and the effect of gaboxadol and zolpidem on EEG power spectra in NREM and REM sleep.
    Journal of psychopharmacology (Oxford, England), 2010, Volume: 24, Issue:11

    Topics: Adolescent; Adult; Cross-Over Studies; Electroencephalography; Female; Humans; Hypnotics and Sedatives; Isoxazoles; Male; Middle Aged; Pyridines; Receptors, GABA-A; Sex Factors; Sleep; Sleep Stages; Sleep, REM; Young Adult; Zolpidem

2010
Alterations in cyclic alternating pattern associated with phase advanced sleep are differentially modulated by gaboxadol and zolpidem.
    Sleep, 2010, Volume: 33, Issue:11

    Topics: Adolescent; Adult; Cross-Over Studies; Double-Blind Method; Female; GABA Agonists; GABA-A Receptor Agonists; Humans; Isoxazoles; Male; Middle Aged; Polysomnography; Pyridines; Self Report; Sleep Initiation and Maintenance Disorders; Sleep Stages; Young Adult; Zolpidem

2010
EEG spectral power density profiles during NREM sleep for gaboxadol and zolpidem in patients with primary insomnia.
    Journal of psychopharmacology (Oxford, England), 2012, Volume: 26, Issue:8

    Topics: Adolescent; Adult; Aged; Brain Waves; Cross-Over Studies; Dose-Response Relationship, Drug; Double-Blind Method; Electroencephalography; Humans; Hypnotics and Sedatives; Isoxazoles; Middle Aged; Pyridines; Sleep; Sleep Initiation and Maintenance Disorders; Zolpidem

2012
Differences between magnetoencephalographic (MEG) spectral profiles of drugs acting on GABA at synaptic and extrasynaptic sites: a study in healthy volunteers.
    Neuropharmacology, 2015, Volume: 88

    Topics: Adult; Brain; Brain Waves; Cross-Over Studies; Female; GABA Agonists; gamma-Aminobutyric Acid; Humans; Isoxazoles; Magnetoencephalography; Male; Nipecotic Acids; Pyridines; Rest; Single-Blind Method; Synapses; Tiagabine; Young Adult; Zolpidem

2015
Electroencephalographic power spectral density profile of the orexin receptor antagonist suvorexant in patients with primary insomnia and healthy subjects.
    Sleep, 2014, Oct-01, Volume: 37, Issue:10

    Topics: Adult; Aged; Azepines; Cross-Over Studies; Double-Blind Method; Electroencephalography; Female; Healthy Volunteers; Humans; Isoxazoles; Male; Middle Aged; Orexin Receptor Antagonists; Polysomnography; Pyridines; Sleep; Sleep Initiation and Maintenance Disorders; Triazoles; Young Adult; Zolpidem

2014

Other Studies

11 other study(ies) available for zolpidem and gaboxadol

ArticleYear
Deletion of the alpha1 or beta2 subunit of GABAA receptors reduces actions of alcohol and other drugs.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 304, Issue:1

    Topics: Animals; Behavior, Animal; Brain; Central Nervous System Depressants; Chlorides; Ethanol; Etomidate; Female; Flurazepam; GABA Agonists; GABA Modulators; Gene Deletion; Hypnotics and Sedatives; Isoxazoles; Male; Mice; Mice, Knockout; Pentobarbital; Postural Balance; Pyridines; Receptors, GABA; Receptors, GABA-A; Sex Characteristics; Sleep; Time Factors; Zolpidem

2003
Altered pharmacology of synaptic and extrasynaptic GABAA receptors on CA1 hippocampal neurons is consistent with subunit changes in a model of alcohol withdrawal and dependence.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 310, Issue:3

    Topics: Alcoholism; Animals; Azides; Benzodiazepines; Diazepam; Drug Interactions; Ethanol; GABA Agonists; Hippocampus; Isoxazoles; Neurons; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Substance Withdrawal Syndrome; Zolpidem

2004
Centrally-mediated antinociceptive actions of GABA(A) receptor agonists in the rat spared nerve injury model of neuropathic pain.
    European journal of pharmacology, 2005, Jun-01, Volume: 516, Issue:2

    Topics: Analgesics; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; GABA Agonists; GABA-A Receptor Agonists; Isonicotinic Acids; Isoxazoles; Male; Muscimol; Neuralgia; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Stress, Mechanical; Time Factors; Trauma, Nervous System; Zolpidem

2005
An extrasynaptic GABAA receptor mediates tonic inhibition in thalamic VB neurons.
    Journal of neurophysiology, 2005, Volume: 94, Issue:6

    Topics: Action Potentials; Animals; Animals, Newborn; Azides; Benzodiazepines; Bicuculline; Blotting, Western; Cells, Cultured; Chlorides; Dose-Response Relationship, Drug; Electric Stimulation; GABA Agonists; GABA Antagonists; Humans; Immunohistochemistry; Immunoprecipitation; In Vitro Techniques; Indoles; Isoxazoles; Membrane Potentials; Mice; Mice, Inbred C57BL; Neural Inhibition; Neurons; Patch-Clamp Techniques; Prokaryotic Initiation Factors; Protein Subunits; Pyridines; Receptors, GABA-A; Synapses; Synaptophysin; Transfection; Ventral Thalamic Nuclei; Zinc Compounds; Zolpidem

2005
Discriminative stimulus effects of tiagabine and related GABAergic drugs in rats.
    Psychopharmacology, 2008, Volume: 197, Issue:4

    Topics: Administration, Oral; Amines; Animals; Anticonvulsants; Azabicyclo Compounds; Baclofen; Benzodiazepines; Bicuculline; Brain; Cyclohexanecarboxylic Acids; Discrimination Learning; Dose-Response Relationship, Drug; GABA Agents; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; Gabapentin; gamma-Aminobutyric Acid; Generalization, Stimulus; Hypnotics and Sedatives; Injections, Intraperitoneal; Isoxazoles; Male; Nipecotic Acids; Piperazines; Pyridines; Rats; Thiophenes; Tiagabine; Zolpidem

2008
Sleep-stabilizing effects of E-6199, compared to zopiclone, zolpidem and THIP in mice.
    Sleep, 2008, Volume: 31, Issue:2

    Topics: Animals; Azabicyclo Compounds; Electroencephalography; Hypnotics and Sedatives; Isoxazoles; Mice; Piperazines; Polysomnography; Pyridines; Sleep; Sleep Stages; Sleep Wake Disorders; Zolpidem

2008
Comparison of the novel subtype-selective GABAA receptor-positive allosteric modulator NS11394 [3'-[5-(1-hydroxy-1-methyl-ethyl)-benzoimidazol-1-yl]-biphenyl-2-carbonitrile] with diazepam, zolpidem, bretazenil, and gaboxadol in rat models of inflammatory
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 327, Issue:3

    Topics: Allosteric Regulation; Animals; Benzimidazoles; Benzodiazepinones; Diazepam; GABA Modulators; Humans; Inflammation; Isoxazoles; Neuralgia; Pyridines; Rats; Receptors, GABA-A; Zolpidem

2008
Dissociating anxiolytic and sedative effects of GABAAergic drugs using temperature and locomotor responses to acute stress.
    Psychopharmacology, 2009, Volume: 204, Issue:2

    Topics: Acute Disease; Anesthetics; Animals; Anti-Anxiety Agents; Body Temperature; Carbolines; Central Nervous System Depressants; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; GABA Agents; GABA Agonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Hypnotics and Sedatives; Isoxazoles; Male; Motor Activity; Pyridines; Rats; Rats, Wistar; Receptors, GABA-A; Stress, Psychological; Telemetry; Zolpidem

2009
Highway driving performance and cognitive functioning the morning after bedtime and middle-of-the-night use of gaboxadol, zopiclone and zolpidem.
    Journal of sleep research, 2009, Volume: 18, Issue:4

    Topics: Adult; Affect; Arousal; Attention; Automobile Driving; Azabicyclo Compounds; Cognition; Cross-Over Studies; Double-Blind Method; Drug Administration Schedule; Female; GABA Agonists; Humans; Isoxazoles; Male; Memory, Short-Term; Neuropsychological Tests; Orientation; Piperazines; Postural Balance; Psychomotor Performance; Pyridines; Reaction Time; Retention, Psychology; Sleep Initiation and Maintenance Disorders; Young Adult; Zolpidem

2009
Intracellular chloride concentration influences the GABAA receptor subunit composition.
    Nature communications, 2012, Mar-13, Volume: 3

    Topics: Animals; Bumetanide; Carboxylic Acids; Cells, Cultured; Cerebellum; Chlorides; gamma-Aminobutyric Acid; Indenes; Isoxazoles; K Cl- Cotransporters; Mice; Neurons; Patch-Clamp Techniques; Protein Subunits; Pyridines; Receptors, GABA-A; RNA Interference; RNA, Small Interfering; Symporters; Zolpidem

2012
GABAA Receptor-Mediated Bidirectional Control of Synaptic Activity, Intracellular Ca2+, Cerebral Blood Flow, and Oxygen Consumption in Mouse Somatosensory Cortex In Vivo.
    Cerebral cortex (New York, N.Y. : 1991), 2015, Volume: 25, Issue:9

    Topics: Action Potentials; Animals; Biophysics; Calcium; Cerebrovascular Circulation; Dose-Response Relationship, Drug; Egtazic Acid; Electric Stimulation; Functional Laterality; GABA Agonists; gamma-Aminobutyric Acid; Isoxazoles; Mice; Oxygen Consumption; Partial Pressure; Pyridines; Receptors, GABA-A; Somatosensory Cortex; Sulfonamides; Thiazoles; Vibrissae; Zolpidem

2015
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