Page last updated: 2024-09-03

zd 7114 and brl 37344

zd 7114 has been researched along with brl 37344 in 5 studies

Compound Research Comparison

Studies
(zd 7114)
Trials
(zd 7114)
Recent Studies (post-2010)
(zd 7114)
Studies
(brl 37344)
Trials
(brl 37344)
Recent Studies (post-2010) (brl 37344)
3523290046

Protein Interaction Comparison

ProteinTaxonomyzd 7114 (IC50)brl 37344 (IC50)
Beta-2 adrenergic receptorHomo sapiens (human)3
Beta-1 adrenergic receptorHomo sapiens (human)5
Beta-2 adrenergic receptorRattus norvegicus (Norway rat)0.8697

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (80.00)18.2507
2000's1 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Green, M; Growcott, JW; Holloway, B; Wilson, C1
Cannon, B; Dicker, A; Nedergaard, J1
Grant, TL; Holloway, BR; Mayers, RM; Quayle, SP; Thompson, AJ1
Feller, DR; Konkar, AA; Lezama, EJ; Miller, DD; Salazar-Bookaman, MM1
Badawi, JK; Bross, S; Honeck, P; Kwon, ST; Langbein, S; Seja, T; Uecelehan, H1

Other Studies

5 other study(ies) available for zd 7114 and brl 37344

ArticleYear
Zeneca ZD7114 acts as an antagonist at beta 3-adrenoceptors in rat isolated ileum.
    British journal of pharmacology, 1993, Volume: 110, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Ethanolamines; Female; Ileum; In Vitro Techniques; Male; Phenoxyacetates; Phenoxypropanolamines; Propranolol; Rats; Receptors, Adrenergic, beta

1993
Stimulation of nonshivering thermogenesis in the Syrian hamster by norepinephrine and beta-selective adrenergic agents: a phenomenon of refractoriness.
    Comparative biochemistry and physiology. Part C, Pharmacology, toxicology & endocrinology, 1996, Volume: 113, Issue:1

    Topics: Acclimatization; Adipose Tissue, Brown; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Body Temperature Regulation; Cold Temperature; Cricetinae; Drug Interactions; Ethanolamines; Female; Isoproterenol; Male; Mesocricetus; Norepinephrine; Oxygen Consumption; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Reproducibility of Results; Shivering

1996
The acid metabolite of ZD7114 is a partial agonist of lipolysis mediated by the rat beta 3-adrenoceptor.
    European journal of pharmacology, 1996, Jan-11, Volume: 295, Issue:2-3

    Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Dose-Response Relationship, Drug; Ethanolamines; Isoproterenol; Lipolysis; Male; Phenoxyacetates; Phenoxypropanolamines; Rats; Rats, Wistar

1996
Pharmacological study of atypical beta-adrenoceptors in rat esophageal smooth muscle.
    European journal of pharmacology, 1996, Jul-11, Volume: 308, Issue:1

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Carbachol; Clenbuterol; Cyclohexane Monoterpenes; Esophagus; Ethanolamines; Female; Heart Atria; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Phenethylamines; Phenoxyacetates; Phenoxypropanolamines; Pindolol; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Serotonin Antagonists; Trachea; Tretoquinol

1996
Relaxation of human detrusor muscle by selective beta-2 and beta-3 agonists and endogenous catecholamines.
    Urology, 2007, Volume: 69, Issue:4

    Topics: Adrenergic beta-Agonists; Aged; Catecholamines; Clenbuterol; Dose-Response Relationship, Drug; Ethanolamines; Female; Humans; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Phenoxyacetates; Phenoxypropanolamines; Propanolamines; Terbutaline; Urinary Bladder

2007
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