Page last updated: 2024-09-05

vx-745 and tak-715

vx-745 has been researched along with tak-715 in 2 studies

Compound Research Comparison

Studies
(vx-745)
Trials
(vx-745)
Recent Studies (post-2010)
(vx-745)
Studies
(tak-715)
Trials
(tak-715)
Recent Studies (post-2010) (tak-715)
5813516013

Protein Interaction Comparison

ProteinTaxonomyvx-745 (IC50)tak-715 (IC50)
Mitogen-activated protein kinase 13Homo sapiens (human)0.24
Mitogen-activated protein kinase 12Homo sapiens (human)0.24
Mitogen-activated protein kinase 11Homo sapiens (human)0.22
Mitogen-activated protein kinase 14Homo sapiens (human)0.1235

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hajduk, PJ; Johnson, EF; Kifle, L; Merta, PJ; Metz, JT; Soni, NB1
Azevedo, R; de Vlieg, J; Kazemier, B; Oubrie, A; Raaijmakers, H; van Zeeland, M1

Other Studies

2 other study(ies) available for vx-745 and tak-715

ArticleYear
Navigating the kinome.
    Nature chemical biology, 2011, Volume: 7, Issue:4

    Topics: Drug Design; Pharmacogenetics; Protein Kinases; Proteome; Systems Biology

2011
X-ray structure of p38α bound to TAK-715: comparison with three classic inhibitors.
    Acta crystallographica. Section D, Biological crystallography, 2012, Volume: 68, Issue:Pt 8

    Topics: Adenosine Triphosphate; Benzamides; Catalytic Domain; Cloning, Molecular; Crystallization; Crystallography, X-Ray; Humans; Imidazoles; Indoles; Ligands; p38 Mitogen-Activated Protein Kinases; Protein Binding; Protein Conformation; Protein Kinase Inhibitors; Pyridazines; Pyridines; Pyrimidines; Structure-Activity Relationship; Thiazoles

2012