isoxazoles and urea
isoxazoles has been researched along with urea in 24 studies
Research
Studies (24)
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 2 (8.33) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 9 (37.50) | 29.6817 |
| 2010's | 9 (37.50) | 24.3611 |
| 2020's | 4 (16.67) | 2.80 |
Authors
| Authors | Studies |
|---|---|
| Chapman, AG | 1 |
| Gerok, W; Häussinger, D; Holstege, A; Pausch, J; Rasenack, J | 1 |
| Kristensen, AS; Madsen, U; Mathiesen, C; Nielsen, EØ; Peters, D; Valgeirsson, J; Varming, T | 1 |
| Achebe, F; Bowling, ME; Bullock, WH; Campbell, AM; Clairmont, KB; Cook, J; Hong, Z; Keiper, C; Kluender, H; Lowe, DB; Magnuson, S; Qi, N; Rodriguez, M; Salhanick, AI; Wang, M; Witman-Jones, T; Wong, WC | 1 |
| Barrow, JC; Connolly, TM; Nantermet, PG; Selnick, HG | 1 |
| Desai, KG; Liu, C | 1 |
| Ryng, S; Zimecki, M | 1 |
| Gonçalves, RB; Katpally, U; Mendes, YS; Oliveira, AC; Silva, JL; Smith, TJ; Soares, MR | 1 |
| Nylander, O; Pihl, L; Wilander, E | 1 |
| Bialer, M; Shimshoni, JA; Yagen, B | 1 |
| Hatanaka, M; Onitsuka, K; Sasai, H; Shinohara, T; Takenaka, K; Takizawa, S; Tsujihara, T | 1 |
| Li, Y; Liu, Y; Sun, R; Wang, Q; Xiong, L | 1 |
| Brahma, MK; Deshmukh, NJ; Dixit, A; Doshi, L; Enose, AA; Gangopadhyay, AK; Guha, T; Gupte, A; Jadhav, RD; Kadam, KS; Kandre, S; Nemmani, KV; Potdar, N; Reddy, MM; Sharma, R; Sivaramakrishnan, H; Srinivasan, S; Vishwakarma, RA | 1 |
| Arvidsson, PI; Besidski, Y; Bueters, T; Bylund, J; Macsari, I; Olofsson, S; Petersson, C | 1 |
| Beller, A; Hoenke, C; Isambert, T; Lessel, U; Nosse, B; Wellenzohn, B | 1 |
| Gowda, DC; Shantharam, CS; Sridhara, MB; Suhas, R; Suyoga Vardhan, DM | 1 |
| Bryszewska, M; Denisov, AA; Gurinovich, TA; Kazbanov, VV; Kletskov, AV; Kulchitsky, VA; Lapotko, DO; Paschkevich, SG; Petkevich, SK; Potkin, VI; Shcharbin, D | 1 |
| Azam, MA; Jubie, S; Thathan, J | 1 |
| Chen, LJ; Cheng, C; Li, LL; Ma, S; Niu, T; Wei, YQ; Xiang, R; Xiong, Y; Yang, LL; Yang, SY; Zheng, MW; Zhong, L; Zhou, Q | 1 |
| Burmistrov, V; Butov, GM; Dalinger, I; Danilov, D; Hammock, BD; Harris, TR; Morisseau, C; Shkineva, T; Vatsadze, I | 1 |
| Channe Gowda, D; Kumara, HK; Pavan Kumar, H; Suhas, R | 1 |
| Abou-Seri, SM; Behery, MGM; Eissa, AAM; Omar, FA | 1 |
| Becker, S; Carell, T; Crisp, A; Dubini, RCA; Hübner, S; Rovó, P; Schelter, F; Schinkel, T; Xu, F | 1 |
| Ahmad, MN; Chopra, S; Dasgupta, A; Kaul, G; Maddipatla, S; Nanduri, S; Ommi, O; Sahoo, SK; Singh, P; Yaddanapudi, VM | 1 |
Reviews
3 review(s) available for isoxazoles and urea
| Article | Year |
|---|---|
Valproate and myoclonus.
Topics: 5-Hydroxytryptophan; Amino Acids; Animals; Aspartic Acid; Clonazepam; DDT; Disease Models, Animal; Flurazepam; gamma-Aminobutyric Acid; Glycine; Isoxazoles; Light; Morphine; Muscimol; Myoclonus; Serotonin; Urea; Valproic Acid | 1986 |
Non-peptidic small-molecule antagonists of the human platelet thrombin receptor PAR-1.
Topics: Blood Platelets; Humans; Inhibitory Concentration 50; Isoxazoles; Platelet Aggregation Inhibitors; Receptor, PAR-1; Structure-Activity Relationship; Urea | 2003 |
Dual targeting DNA gyrase B (GyrB) and topoisomerse IV (ParE) inhibitors: A review.
Topics: Amino Acid Sequence; Aminopyridines; Anti-Bacterial Agents; Barbiturates; Benzimidazoles; DNA Gyrase; DNA Topoisomerase IV; Fluoroquinolones; Indazoles; Isoxazoles; Morpholines; Organophosphates; Oxazolidinones; Prodrugs; Pyrazoles; Pyrroles; Pyrrolidines; Pyrrolidinones; Quinazolinones; Quinolines; Spiro Compounds; Topoisomerase II Inhibitors; Topoisomerase Inhibitors; Urea | 2015 |
Other Studies
21 other study(ies) available for isoxazoles and urea
| Article | Year |
|---|---|
The glutamine analog acivicin as antipyrimidine. Studies on the interrelationship between pyrimidine and urea synthesis in liver.
Topics: Animals; Antibiotics, Antineoplastic; Carbamyl Phosphate; Cytosol; Female; Isoxazoles; Liver; Mitochondria, Liver; Orotic Acid; Oxazoles; Pyrimidines; Rats; Rats, Inbred Strains; Urea | 1985 |
2-arylureidobenzoic acids: selective noncompetitive antagonists for the homomeric kainate receptor subtype GluR5.
Topics: Animals; Benzoates; Cell Line; Excitatory Amino Acid Agonists; Humans; Isoxazoles; Mice; Muscle Rigidity; Patch-Clamp Techniques; Propionates; Quantitative Structure-Activity Relationship; Radioligand Assay; Receptors, Kainic Acid; Urea | 2003 |
In vitro SAR of (5-(2H)-isoxazolonyl) ureas, potent inhibitors of hormone-sensitive lipase.
Topics: Enzyme Inhibitors; Hypoglycemic Agents; Isoxazoles; Sterol Esterase; Structure-Activity Relationship; Urea | 2004 |
Enhancement of dissolution rate of valdecoxib using solid dispersions with polyethylene glycol 4000.
Topics: Algorithms; Calorimetry, Differential Scanning; Chemistry, Pharmaceutical; Cyclooxygenase Inhibitors; Excipients; Isoxazoles; Kinetics; Mannitol; Microscopy, Electron, Scanning; Polyethylene Glycols; Povidone; Solubility; Spectroscopy, Fourier Transform Infrared; Sulfonamides; Urea; X-Ray Diffraction | 2005 |
Search for new lead structures for low-molecular-weight immune response modifiers.
Topics: Amides; Animals; Antibody Formation; Drug Design; Immunity, Cellular; Immunologic Factors; Indicators and Reagents; Isoxazoles; Mice; Mice, Inbred CBA; Molecular Weight; Urea | 2004 |
VP4 protein from human rhinovirus 14 is released by pressure and locked in the capsid by the antiviral compound WIN.
Topics: Antiviral Agents; Capsid; Capsid Proteins; Dose-Response Relationship, Drug; Drug Interactions; HeLa Cells; Humans; Hydrostatic Pressure; Isoxazoles; Rhinovirus; Temperature; Urea; Virus Assembly | 2007 |
Comparative study of the effect of luminal hypotonicity on mucosal permeability in rat upper gastrointestinal tract.
Topics: Animals; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Duodenum; Gastric Mucosa; Hydrogen-Ion Concentration; Hypotonic Solutions; Indomethacin; Intestinal Absorption; Intestinal Mucosa; Inulin; Isoxazoles; Jejunum; Male; Methylglucosides; Osmolar Concentration; Permeability; Rats; Rats, Inbred Strains; Sodium Chloride; Stomach; Upper Gastrointestinal Tract; Urea | 2008 |
Synthesis and anticonvulsant activity of aromatic tetramethylcyclopropanecarboxamide derivatives.
Topics: Administration, Oral; Amides; Animals; Anticonvulsants; Cyclopropanes; Electroshock; Isoxazoles; Mice; Motor Activity; Rats; Seizures; Sulfonamides; Urea; Valproic Acid; Zonisamide | 2008 |
Enantioselective intramolecular oxidative aminocarbonylation of alkenylureas catalyzed by palladium-spiro bis(isoxazoline) complexes.
Topics: Alkenes; Amination; Catalysis; Isoxazoles; Ligands; Models, Chemical; Organometallic Compounds; Oxidation-Reduction; Palladium; Pyrimidines; Pyrroles; Spiro Compounds; Stereoisomerism; Urea | 2009 |
Design, synthesis, and insecticidal evaluation of new benzoylureas containing isoxazoline and isoxazole group.
Topics: Animals; Culicidae; Drug Design; Insecticides; Isoxazoles; Moths; Structure-Activity Relationship; Urea | 2011 |
Synthesis and biological evaluation of isoxazole, oxazole, and oxadiazole containing heteroaryl analogs of biaryl ureas as DGAT1 inhibitors.
Topics: Animals; Chemistry Techniques, Synthetic; Diacylglycerol O-Acyltransferase; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Isoxazoles; Mice; Oxadiazoles; Solubility; Structure-Activity Relationship; Urea; Water | 2012 |
Novel bioactivation mechanism of reactive metabolite formation from phenyl methyl-isoxazoles.
Topics: Carbamates; Carbon; Cysteine; Glutathione; Humans; Isoxazoles; Liver; Magnetic Resonance Spectroscopy; Mass Spectrometry; Microsomes, Liver; NADP; NAV1.1 Voltage-Gated Sodium Channel; Nitrogen; Oxidation-Reduction; Urea; Voltage-Gated Sodium Channel Blockers | 2012 |
Identification of new potent GPR119 agonists by combining virtual screening and combinatorial chemistry.
Topics: Cell Line; Combinatorial Chemistry Techniques; Databases, Factual; High-Throughput Screening Assays; Humans; Isoxazoles; Models, Molecular; Oxadiazoles; Receptors, G-Protein-Coupled; Spiro Compounds; Structure-Activity Relationship; Urea | 2012 |
Inhibition of protein glycation by urea and thiourea derivatives of glycine/proline conjugated benzisoxazole analogue - synthesis and structure-activity studies.
Topics: Animals; Cattle; Dose-Response Relationship, Drug; Glycine; Isoxazoles; Molecular Structure; Proline; Serum Albumin, Bovine; Structure-Activity Relationship; Urea | 2013 |
The influence of heterocyclic compound-PAMAM dendrimer complexes on evoked electrical responses in slices of hypoxic brain tissue.
Topics: Animals; Brain; Carboxylic Acids; Dendrimers; Electrophysiological Phenomena; Excitatory Postsynaptic Potentials; Hippocampus; Hypoxia; In Vitro Techniques; Isoxazoles; Male; Oxygen; Rats; Urea | 2014 |
SKLB-677, an FLT3 and Wnt/β-catenin signaling inhibitor, displays potent activity in models of FLT3-driven AML.
Topics: Animals; Animals, Genetically Modified; Antineoplastic Agents; Apoptosis; beta Catenin; Cell Line, Tumor; Cell Proliferation; Cell Survival; Drug Resistance, Neoplasm; Female; fms-Like Tyrosine Kinase 3; G1 Phase Cell Cycle Checkpoints; Humans; Isoxazoles; Leukemia, Myeloid, Acute; Mice; Mice, Inbred NOD; Mice, SCID; Phenylurea Compounds; Pyrazoles; Pyrimidines; Urea; Wnt Proteins; Wnt Signaling Pathway; Zebrafish | 2015 |
1,3-Disubstituted and 1,3,3-trisubstituted adamantyl-ureas with isoxazole as soluble epoxide hydrolase inhibitors.
Topics: Adamantane; Drug Stability; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Inhibitory Concentration 50; Isoxazoles; Microsomes; Solubility; Structure-Activity Relationship; Urea | 2015 |
Multitarget-directed therapeutics: (Urea/thiourea)
Topics: Anti-Infective Agents; Anti-Inflammatory Agents; Antioxidants; Heterocyclic Compounds; Humans; Isoxazoles; Lysine; Molecular Docking Simulation; Piperazines; Piperidines; Structure-Activity Relationship; Thiourea; Urea | 2021 |
Synthesis, in vitro anticancer activity and in silico studies of certain isoxazole-based carboxamides, ureates, and hydrazones as potential inhibitors of VEGFR2.
Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Hydrazones; Isoxazoles; Molecular Structure; Protein Kinase Inhibitors; Structure-Activity Relationship; Urea; Vascular Endothelial Growth Factor Receptor-2 | 2021 |
Isoxazole Nucleosides as Building Blocks for a Plausible Proto-RNA.
Topics: Cytidine; Isoxazoles; Nucleosides; RNA; Urea | 2022 |
Isoxazole carboxylic acid methyl ester-based urea and thiourea derivatives as promising antitubercular agents.
Topics: Animals; Antitubercular Agents; Carboxylic Acids; Chlorocebus aethiops; Esters; Isoxazoles; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Structure-Activity Relationship; Thiourea; Urea; Vero Cells | 2023 |