Page last updated: 2024-08-21

indazoles and rifampin

indazoles has been researched along with rifampin in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Garrett, M; Hee, B; Klamerus, KJ; Kuruganti, U; Ni, G; Pithavala, YK; Toh, M; Tortorici, M1
Adhikari, C; Krishna, VS; Reshma, RS; Sharada, DS; Sriram, D; Vidyacharan, S1
Chen, EC; Chen, Y; Choo, EF; Liu, L; Ma, F; Mao, J; Sahasranaman, S; Zhu, R1

Trials

1 trial(s) available for indazoles and rifampin

ArticleYear
Effect of rifampin on the pharmacokinetics of Axitinib (AG-013736) in Japanese and Caucasian healthy volunteers.
    Cancer chemotherapy and pharmacology, 2010, Volume: 65, Issue:3

    Topics: Adult; Area Under Curve; Asian People; Axitinib; Cross-Over Studies; Cytochrome P-450 CYP3A; Enzyme Inhibitors; Genotype; Glucuronosyltransferase; Humans; Imidazoles; Indazoles; Japan; Male; Metabolic Clearance Rate; Middle Aged; Rifampin; White People; Young Adult

2010

Other Studies

2 other study(ies) available for indazoles and rifampin

ArticleYear
A robust synthesis of functionalized 2H-indazoles via solid state melt reaction (SSMR) and their anti-tubercular activity.
    Bioorganic & medicinal chemistry letters, 2017, 04-01, Volume: 27, Issue:7

    Topics: Antitubercular Agents; Ciprofloxacin; Ethambutol; Indazoles; Isoniazid; Mycobacterium tuberculosis; Rifampin; Structure-Activity Relationship

2017
Assessment of OATP transporter-mediated drug-drug interaction using physiologically-based pharmacokinetic (PBPK) modeling - a case example.
    Biopharmaceutics & drug disposition, 2018, Volume: 39, Issue:9

    Topics: Area Under Curve; Cinnamates; Cyclosporine; Drug Interactions; Gemfibrozil; Humans; Indazoles; Liver-Specific Organic Anion Transporter 1; Models, Biological; Pravastatin; Rifampin; Solute Carrier Organic Anion Transporter Family Member 1B3

2018