Page last updated: 2024-09-03

gr 73632 and senktide

gr 73632 has been researched along with senktide in 17 studies

Compound Research Comparison

Studies
(gr 73632)
Trials
(gr 73632)
Recent Studies (post-2010)
(gr 73632)
Studies
(senktide)
Trials
(senktide)
Recent Studies (post-2010) (senktide)
7719292150

Protein Interaction Comparison

ProteinTaxonomygr 73632 (IC50)senktide (IC50)
Neuromedin-K receptorRattus norvegicus (Norway rat)0.011
Neuromedin-K receptorHomo sapiens (human)0.0263
Neuromedin-K receptorCavia porcellus (domestic guinea pig)0.012

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's11 (64.71)18.2507
2000's5 (29.41)29.6817
2010's1 (5.88)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Clark, D; Elliott, PJ; Hagan, RM; Overton, P1
Hall, JM; Mitchell, D; Morton, IK1
Elliott, PJ; Hagan, RM; Mason, GS; Stephens-Smith, M1
Beresford, IJ; Deal, MJ; Hagan, RM; Ireland, SJ; Jordan, CC; Ward, P1
Hall, JM; Morton, IK1
Arkinstall, S; Beresford, IJ; Hagan, RM; Ireland, SJ; Seale, PW; Stables, JM; Walsh, DM; Ward, P1
Bentley, GN; Gent, JP1
Chizh, BA; Cumberbatch, MJ; Headley, PM1
Dalforno, G; Gaviraghi, G; Hagan, RM; Palea, S; Pietra, C; Trist, DG1
Altier, N; Stewart, J1
Cody, C; Jones, RS; Maubach, KA1
Holzer, P; Shahbazian, A1
Greenwood-Van Meerveld, B; Sutkowski-Markmann, DM; Venkova, K1
Greenwood-Van Meerveld, B; Venkova, K1
Adolfsson, R; Ahlstedt, I; de Verdier, J; Drmota, T; Engberg, S; Johansson, A; Jussila, R; Kristensson, E; Leffler, A; Lindström, E; Novén, A; Påhlman, I; Sigfridsson, K; Sundqvist, M; von Mentzer, B1
Bongianni, F; Cinelli, E; Mutolo, D; Pantaleo, T1
Navarro, VM; Ohkura, S; Okamura, H; Wakabayashi, Y; Yamamura, T1

Other Studies

17 other study(ies) available for gr 73632 and senktide

ArticleYear
Neurokinin agonists differentially affect A9 and A10 dopamine cells in the rat.
    European journal of pharmacology, 1992, Mar-17, Volume: 213, Issue:1

    Topics: Animals; Dopamine; Neurokinin A; Neurons; Peptide Fragments; Rats; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Substantia Nigra; Tegmentum Mesencephali

1992
Neurokinin receptors in the rabbit iris sphincter characterised by novel agonist ligands.
    European journal of pharmacology, 1991, Jun-18, Volume: 199, Issue:1

    Topics: Animals; In Vitro Techniques; Iris; Kinetics; Ligands; Male; Neurokinin A; Peptide Fragments; Rabbits; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P

1991
Behavioural and biochemical responses following activation of midbrain dopamine pathways by receptor selective neurokinin agonists.
    Neuropeptides, 1991, Volume: 19, Issue:2

    Topics: Amino Acid Sequence; Animals; Chromatography, High Pressure Liquid; Dopamine; Haloperidol; Limbic System; Male; Mesencephalon; Molecular Sequence Data; Motor Activity; Neural Pathways; Neurokinin A; Peptide Fragments; Rats; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Substantia Nigra; Tegmentum Mesencephali

1991
Receptor-selective, peptidase-resistant agonists at neurokinin NK-1 and NK-2 receptors: new tools for investigating neurokinin function.
    Neuropeptides, 1991, Volume: 19, Issue:2

    Topics: Administration, Cutaneous; Amino Acid Sequence; Animals; Bronchoconstriction; Capillary Permeability; Chromatography, High Pressure Liquid; Guinea Pigs; Male; Molecular Sequence Data; Neurokinin A; Neurokinin B; Peptide Fragments; Rats; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Trachea

1991
Novel ligands confirm NK-1 receptor-mediated modulation of neurotransmission in the guinea pig vas deferens preparation.
    Annals of the New York Academy of Sciences, 1991, Volume: 632

    Topics: Animals; Electric Stimulation; Evoked Potentials; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Neurokinin A; Neurokinin B; Peptide Fragments; Receptors, Neurotransmitter; Receptors, Tachykinin; Substance P; Synaptic Transmission; Vas Deferens

1991
GR138676, a novel peptidic tachykinin antagonist which is potent at NK3 receptors.
    Neuropeptides, 1994, Volume: 27, Issue:6

    Topics: Amino Acid Sequence; Animals; Arachidonic Acid; Astrocytoma; Binding, Competitive; Calcium; CHO Cells; Cricetinae; Humans; Male; Molecular Sequence Data; Neurokinin B; Oligopeptides; Peptide Fragments; Portal Vein; Rats; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Transfection; Tumor Cells, Cultured

1994
Neurokinin actions on substantia gelatinosa neurones in an adult longitudinal spinal cord preparation.
    Brain research, 1995, Feb-27, Volume: 673, Issue:1

    Topics: Afferent Pathways; Animals; Electric Stimulation; Male; Peptide Fragments; Physalaemin; Rats; Rats, Wistar; Spinal Cord; Spinal Nerve Roots; Substance P; Substantia Gelatinosa; Time Factors

1995
Modulation of excitatory amino acid responses by tachykinins and selective tachykinin receptor agonists in the rat spinal cord.
    British journal of pharmacology, 1995, Volume: 115, Issue:6

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Electrophysiology; Excitatory Amino Acids; Male; N-Methylaspartate; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Tachykinin; Spinal Cord; Substance P; Tachykinins

1995
Further studies on the effects of selective neurokinin agonists upon the activation of micturition reflex in rats. Evidence for a dual NK-1 receptor mediated excitatory and inhibitory activity.
    Neuropeptides, 1993, Volume: 24, Issue:5

    Topics: Animals; Dose-Response Relationship, Drug; Injections, Intra-Arterial; Injections, Intraventricular; Male; Neurokinin A; Peptide Fragments; Physalaemin; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Reflex; Substance P; Urinary Bladder; Urination

1993
Tachykinin NK-1 and NK-3 selective agonists induce analgesia in the formalin test for tonic pain following intra-VTA or intra-accumbens microinfusions.
    Behavioural brain research, 1997, Volume: 89, Issue:1-2

    Topics: Amphetamine; Analgesics, Non-Narcotic; Animals; Central Nervous System Stimulants; Formaldehyde; Male; Microinjections; Nucleus Accumbens; Pain Measurement; Peptide Fragments; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Ventral Tegmental Area

1997
Tachykinins may modify spontaneous epileptiform activity in the rat entorhinal cortex in vitro by activating GABAergic inhibition.
    Neuroscience, 1998, Volume: 83, Issue:4

    Topics: Animals; Baclofen; Bicuculline; Entorhinal Cortex; Epilepsy; Evoked Potentials; In Vitro Techniques; Male; Membrane Potentials; Neurokinin A; Neurokinin B; Neurons; Peptide Fragments; Phosphinic Acids; Propanolamines; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Reaction Time; Receptors, GABA-A; Receptors, GABA-B; Substance P; Synapses; Tachykinins

1998
Differences in circular muscle contraction and peristaltic motor inhibition caused by tachykinin NK1 receptor agonists in the guinea-pig small intestine.
    Neurogastroenterology and motility, 2000, Volume: 12, Issue:2

    Topics: Adenosine Triphosphate; Animals; Enzyme Inhibitors; Female; Guinea Pigs; Intestine, Small; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Neurokinin A; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Peptide Fragments; Peristalsis; Piperidines; Purinergic P2 Receptor Antagonists; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Sincalide; Spasm; Substance P; Suramin; Tetrodotoxin

2000
Peripheral activity of a new NK1 receptor antagonist TAK-637 in the gastrointestinal tract.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 300, Issue:3

    Topics: Animals; Capsaicin; Digestive System; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Isometric Contraction; Male; Muscle, Smooth; Naphthyridines; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Substance P

2002
Effects of TAK-637 on NK(1) receptor-mediated mechanisms regulating colonic secretion.
    Toxicology and applied pharmacology, 2004, Apr-15, Volume: 196, Issue:2

    Topics: Animals; Capsaicin; Colforsin; Colon; Electric Stimulation; Electrophysiology; Guinea Pigs; In Vitro Techniques; Intestinal Absorption; Intestinal Mucosa; Male; Naphthyridines; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Receptors, Neurokinin-1; Statistics, Nonparametric; Substance P; Tetrodotoxin

2004
Senktide-induced gerbil foot tapping behaviour is blocked by selective tachykinin NK1 and NK3 receptor antagonists.
    European journal of pharmacology, 2007, Dec-22, Volume: 577, Issue:1-3

    Topics: Animals; Autoradiography; Behavior, Animal; Brain; Calcium; CHO Cells; Cloning, Molecular; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Foot; Gerbillinae; Injections, Intraventricular; Male; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Quinolines; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P

2007
Neurokinin receptor modulation of respiratory activity in the rabbit.
    The European journal of neuroscience, 2008, Volume: 27, Issue:12

    Topics: Animals; Exhalation; Inhalation; Male; Medulla Oblongata; Microinjections; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Phrenic Nerve; Piperidines; Rabbits; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Substance P; Vagotomy

2008
Effects of intravenous administration of neurokinin receptor subtype-selective agonists on gonadotropin-releasing hormone pulse generator activity and luteinizing hormone secretion in goats.
    The Journal of reproduction and development, 2015, Volume: 61, Issue:1

    Topics: Animals; Estradiol; Female; Goats; Gonadotropin-Releasing Hormone; Infusions, Intravenous; Kisspeptins; Ligands; Luteinizing Hormone; Neurokinin A; Peptide Fragments; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Signal Transduction; Substance P; Time Factors

2015