fentanyl has been researched along with f 7302 in 64 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 14 (21.88) | 18.7374 |
1990's | 36 (56.25) | 18.2507 |
2000's | 12 (18.75) | 29.6817 |
2010's | 2 (3.13) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Chi, ZQ; Masuo, Y; Pélaprat, D; Rostène, W; Wang, H | 1 |
Lin, FS; Wang, CQ; Zhu, GY | 2 |
Chi, ZQ; Gu, JJ; Zhao, GM | 1 |
Yang, HQ; Zhang, KM; Zhao, ZQ | 2 |
Brine, GA; Carroll, FI; Jacobson, AE; Rice, KC; Rothman, RB; Seggel, M; Xu, H | 1 |
Chi, ZQ; Pélaprat, D; Roques, BP; Rostène, W; Vanhove, A; Wang, H | 1 |
Hu, ST; Xu, T | 1 |
Chi, ZQ; Kopp, N; Pélaprat, D; Roques, BP; Rostène, W; Sarrieau, A; Vanhove, A; Wang, H | 1 |
Chi, ZQ; Jin, WQ; Zhao, GM; Zheng, WJ; Zhou, HY | 1 |
Chen, JQ; Chi, ZQ; Jin, WQ | 1 |
Nie, ZZ; Wang, CQ; Zhang, KG | 1 |
Chen, J; Chi, ZQ; Xu, H; Yao, YH; Zhu, YC | 1 |
Chi, ZQ; Yao, YH | 1 |
Chi, ZQ; Li, GF; Xu, H; Yao, YH | 1 |
Ge, BL; Wang, CH; Wu, CR; Zhu, YX | 1 |
Chi, ZQ; Zheng, WJ; Zhou, J | 2 |
Chen, J; Chi, ZQ; Xu, H | 1 |
Chi, ZQ; Li, GF; Ye, SZ | 1 |
Chen, XJ; Chi, ZQ; Jin, WQ | 1 |
Chen, WL; Chen, XJ; Chi, ZQ; Huang, ZM; Li, ZG; Zhang, HP; Zheng, WJ; Zhou, J | 1 |
Li, ZY; Liu, JZ; Ni, CH; Tang, GZ; Wu, YZ; Zhao, XL; Zhou, DH | 1 |
Chou, DP; Huang, ZM; Wu, RQ; Zhu, YC | 1 |
Dai, QY; Fang, SN; Ge, BJ; Huang, ZM; Li, QZ; Ni, CH; Wu, RQ; Zhou, DH | 1 |
Chen, J; Chen, XJ; Chi, ZQ; Ji, RY; Jin, WQ; Wang, ZX; Zhu, YC | 1 |
Li, XY; Xu, SF; Zhu, CB; Zhu, YH | 1 |
Cui, X; Han, JS; Xu, W | 1 |
Chen, SZ; Han, JS | 1 |
Brine, GA; Carroll, FI; Liu, Y; Rothman, RB; Singh, P; Stark, PA; Xu, H | 1 |
Chen, XJ; Chi, ZQ; Lin, SY; Lu, YF; Tong, CX; Wei, AL; Zhou, DH | 1 |
Shi, GG; Wei, DS; Xu, SF | 1 |
Chi, ZQ; Li, GF; Lu, YF | 1 |
Barth, A; Brandt, W; Höltje, HD | 1 |
Brine, GA; Carroll, FI; Ni, Q; Partilla, JS; Rothman, RB; Stark, PA; Xu, H | 1 |
Han, JS; Han, NL; Zhang, LJ | 1 |
Han, JS; Sun, YH; Zhou, Y | 1 |
Han, JS; Sun, YH; Zhang, ZW; Zhou, Y | 1 |
Han, JS; Kang, HG; Li, CQ; Liu, NJ; Xu, C; Xu, T; Yu, YX | 1 |
Brine, GA; Carroll, FI; Chen, C; Lai, J; Liu-Chen, LY; Lu, YF; Partilla, JS; Porreca, F; Rice, KC; Rothman, RB; Sadee, W; Xu, H | 1 |
Cheung, P; Li, JG; Liu-Chen, LY; Raffa, RB; Tzeng, TB | 1 |
Chen, KX; Chi, ZQ; Ji, RY; Jiang, HL; Tang, Y; Wang, ZX | 1 |
Chen, J; Chen, XJ; Chi, ZQ; Jin, WQ; Wang, ZX | 1 |
Chen, KX; Ji, RY; Jiang, HL; Rong, SB; Wang, QM; Zhao, SR; Zhu, YC | 1 |
Brine, GA; Carroll, FI; Chen, KX; Chi, ZQ; Lu, YF; Partilla, JS; Rice, KC; Rothman, RB; Wang, JB; Xu, H; Zheng, QX | 1 |
Chen, J; Chi, ZQ; Li, CL; Pei, G; Shen, QX; Wang, CH; Wei, Q; Zhou, DH | 1 |
Bi-Yi, C; Jie, C; Wen-Qiao, J; Xin-Jian, C; You-Cheng, Z; Zhi-Qiang, C | 1 |
Chi, ZQ; Guo, GW; He, Y; Jin, WQ; Zhu, YC; Zou, Y | 1 |
Chen, ZW; Han, JS; Wang, Y; Yang, K | 1 |
Li, XY; Wu, T | 1 |
Cao, Y; Chen, KX; Gu, JD; Huang, XQ; Ji, RY; Jiang, HL; Luo, XM; Rong, SB; Tan, XJ; Zhu, YC | 1 |
Chi, ZQ; Jin, WQ; Jin, XL; Li, GF; Zhou, DH | 1 |
Chen, XJ; Chi, ZQ; Guo, GW; Jin, WQ; Liu, ZH; Zhang, HP; Zhu, YC | 1 |
Han, JS; Wang, XM; Wang, Y | 1 |
Chen, BY; Chen, XJ; Chi, ZQ; Jin, WQ; Zhu, YC | 1 |
Chen, J; Chen, LW; Chi, ZQ; Feng, YP; Xu, XJ; Zhou, DH | 1 |
Can, G; De-He, Z; Jie, C; Li-Wei, C; Qiang, W; Xue-Jun, X; Zhi-Qiang, C | 1 |
Che, LW; Chen, J; Chi, ZQ; Gao, C; Xu, XJ | 1 |
Chen, J; Chen, LW; Chi, ZQ; Gao, C; Tao, YM; Xu, XJ | 1 |
Chen, XJ; Chi, ZQ; He, Y; Jin, WQ; Liu, ZH; Shen, QX | 1 |
Dong, H; Han, J; Wang, X; Xu, G; Yu, Y; Zhang, D; Zhang, M | 1 |
Chi, ZQ; Liu, JG; Sun, JF; Tao, YM; Wang, YH; Xu, XJ | 1 |
Bardel, C; Chatron, N; Huissoud, C; Massoud, M; Nouchy, M; Raymond, L; Sanlaville, D; Schluth-Bolard, C | 1 |
64 other study(ies) available for fentanyl and f 7302
Article | Year |
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Effect of brain lesions on [3H]ohmefentanyl binding site densities in the rat striatum and substantia nigra.
Topics: Animals; Brain Injuries; Corpus Striatum; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Fentanyl; Male; Rats; Rats, Wistar; Receptors, Opioid; Substantia Nigra | 1992 |
[Effects of microiontophoretically applied OMF and U-50488 on spontaneous discharges of respiration related units in the region of nucleus of solitary tract of rat].
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Depression, Chemical; Electrophysiology; Female; Fentanyl; Iontophoresis; Male; Medulla Oblongata; Naloxone; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid; Respiration | 1992 |
Effects of ohmefentanyl on CA1 field potentials in rat hippocampus slices.
Topics: Analgesics; Animals; Evoked Potentials; Fentanyl; Hippocampus; Male; Morphine; Naloxone; Rats; Rats, Wistar | 1992 |
[Inhibition of ohmefentanyl on articular afferent-induced responses of neurons in the spinal lamina X].
Topics: Analgesics; Animals; Cats; Electric Stimulation; Female; Fentanyl; Joints; Male; Neurons, Afferent; Nociceptors; Spinal Cord | 1992 |
RTI-4614-4: an analog of (+)-cis-3-methylfentanyl with a 27,000-fold binding selectivity for mu versus delta opioid binding sites.
Topics: Animals; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Fentanyl; In Vitro Techniques; Kinetics; Radioligand Assay; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu | 1991 |
[3H]ohmefentanyl preferentially binds to mu-opioid receptors but also labels sigma-sites in rat brain sections.
Topics: Amino Acid Sequence; Analgesics; Animals; Autoradiography; Binding Sites; Brain; Corpus Striatum; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Fentanyl; Male; Molecular Sequence Data; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Substrate Specificity; Tritium | 1991 |
[Relationship between central beta-endorphins and serotonin systems in mechanism of hypoxic ventilatory regulation].
Topics: Animals; beta-Endorphin; Fentanyl; Hypoxia; Injections, Intraventricular; Male; Naloxone; Rabbits; Respiration; Serotonin | 1991 |
Characterization and distribution of [3H]ohmefentanyl binding sites in the human brain.
Topics: Adult; Aged; Autoradiography; Basal Ganglia; Binding Sites; Binding, Competitive; Brain Chemistry; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Female; Fentanyl; Humans; In Vitro Techniques; Kinetics | 1991 |
[Pharmacokinetics of [3H]ohmefentanyl in rats].
Topics: Animals; Blood Proteins; Fentanyl; Male; Protein Binding; Rats; Rats, Inbred Strains; Tissue Distribution | 1990 |
[Opioid dependence and tolerance in the guinea-pig ileum in vitro].
Topics: Analgesics; Animals; Drug Tolerance; Fentanyl; Guinea Pigs; Ileum; Male; Morphine Derivatives; Muscle Contraction; Muscle, Smooth; Opioid-Related Disorders | 1990 |
Inhibition of nociceptive responses of dorsal horn neurones in the cat spinal cord by ohmefentanyl, a preferring mu opioid receptor agonist [corrected].
Topics: Action Potentials; Animals; Cats; Fentanyl; Narcotic Antagonists; Nociceptors; Receptors, Opioid; Receptors, Opioid, mu; Spinal Cord | 1990 |
[Effects of microiontophoretically applied OMF on spontaneous discharges of respiration related units (RRUs) in the region of nucleus ambigus of rat].
Topics: Animals; Electrophysiology; Female; Fentanyl; Iontophoresis; Male; Medulla Oblongata; Rats; Rats, Inbred Strains; Receptors, Opioid; Respiration | 1990 |
[Effects of ohmefentanyl on rat respiration].
Topics: Analgesics; Animals; Dose-Response Relationship, Drug; Female; Fentanyl; Male; Medulla Oblongata; Pons; Rats; Rats, Inbred Strains; Respiration | 1989 |
Potent 3-methylfentanyl analogs: morphine-like catalepsy and receptor binding characteristics.
Topics: Analgesics; Animals; Catalepsy; Female; Fentanyl; Male; Mice; Radioligand Assay; Rats; Receptors, Opioid; Receptors, Opioid, mu | 1987 |
Inhibitory regulations of ohmefentanyl and morphine on postsynaptic dopamine receptors.
Topics: Animals; Corpus Striatum; Fentanyl; Male; Morphine; Neurons; Rats; Receptors, Dopamine; Receptors, Neurotransmitter; Rotation; Substantia Nigra | 1988 |
[Autoradiographic distribution of [3H]ohmefentanyl binding sites in rat corpus striatum].
Topics: Analgesics; Animals; Autoradiography; Binding Sites; Corpus Striatum; Fentanyl; Hydroxydopamines; Kainic Acid; Male; Oxidopamine; Rats; Receptors, Opioid; Receptors, Opioid, mu | 1988 |
[Effects of ohmefentanyl on the content of endorphin in pituitary and brain areas of rats].
Topics: Analgesia; Animals; beta-Endorphin; Brain; Catalepsy; Dynorphins; Endorphins; Enkephalin, Methionine; Fentanyl; Male; Peptide Fragments; Pituitary Gland; Radioimmunoassay; Rats; Tissue Distribution | 1986 |
[Effects of potent analgesics, ohmefentanyl and mefentanyl, on respiration and electroencephalogram in rabbits].
Topics: Analgesics; Animals; Electroencephalography; Female; Fentanyl; Male; Rabbits; Respiration | 1986 |
Ohmefentanyl--a new agonist for mu-opiate receptor.
Topics: Analgesics; Animals; Binding Sites; Brain; Fentanyl; Male; Mice; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu | 1985 |
[Autoradiography of [3H]ohmefentanyl binding with opiate receptors in the rat brain].
Topics: Analgesics; Animals; Autoradiography; Binding, Competitive; Brain; Fentanyl; Male; Rats; Receptors, Opioid; Receptors, Opioid, mu | 1986 |
The choice of opioid receptor subtype in isolated preparations by ohmefentanyl.
Topics: Analgesics; Animals; Fentanyl; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Rabbits; Rats; Receptors, Opioid; Receptors, Opioid, mu; Species Specificity; Vas Deferens | 1987 |
[Effect of ohmefentanyl injection to the region of nucleus tractus solitarius on discharge of phrenic nerve in rabbits].
Topics: Analgesics; Animals; Electrophysiology; Female; Fentanyl; Male; Medulla Oblongata; Microinjections; Phrenic Nerve; Rabbits | 1988 |
[Analgesic activity and toxicity of potent analgesics, ohmefentanyl and mefentanyl].
Topics: Analgesics; Animals; Blood Pressure; Electrocardiography; Electroencephalography; Fentanyl; Mice; Nalorphine; Rabbits; Rats | 1984 |
[Preparation of [3H]-labelled N-[1-(beta-hydroxy beta-phenylethyl)-3-methyl-4-piperidyl]-N-phenylpropionamide and studies of its binding with opiate receptors of mouse brain].
Topics: Analgesics; Animals; Brain; Fentanyl; Mice; Receptors, Opioid; Tritium | 1982 |
[Studies on potent analgesics. VII. Synthesis and analgesic activity of diastereoisomers of 1-beta-hydroxy-3-methylfentanyl (7302) and related compounds].
Topics: Analgesics; Animals; Fentanyl; Male; Mice; Stereoisomerism; Structure-Activity Relationship | 1983 |
[Studies on potent analgesics. V. Synthesis and analgesic activity of the ester derivatives of N-(1-(2-hydroxy-2-phenylethyl)-3-methyl-4-piperidyl)-N-phenylpropan amide (7302)].
Topics: Analgesics; Animals; Female; Fentanyl; Mice | 1983 |
Stereoisomers of N-[1-hydroxy-(2-phenylethyl)-3-methyl-4-piperidyl]- N-phenylpropanamide: synthesis, stereochemistry, analgesic activity, and opioid receptor binding characteristics.
Topics: Analgesics; Animals; Crystallography, X-Ray; Female; Fentanyl; Guinea Pigs; Ileum; Male; Mice; Morphine; Muscle, Smooth; Rabbits; Receptors, Opioid; Stereoisomerism; Structure-Activity Relationship; Vas Deferens | 1995 |
Binding sites of mu receptor increased when acupuncture analgesia was enhanced by droperidol: an autoradiographic study.
Topics: Acupuncture Analgesia; Analgesics; Animals; Autoradiography; Binding Sites; Brain; Droperidol; Fentanyl; Male; Pain Threshold; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu | 1995 |
Spinal serotonin IA and IC/2 receptors mediate supraspinal mu opioid-induced analgesia.
Topics: Analgesia; Animals; Brain; Fentanyl; Injections, Intraventricular; Injections, Spinal; Male; Pain Threshold; Rats; Rats, Wistar; Reaction Time; Receptors, Opioid, mu; Receptors, Serotonin; Serotonin Antagonists; Spinal Cord | 1994 |
Protein c-fos induction in rat brain and spinal dorsal horn by sincalide and opioids in vitro.
Topics: Animals; Brain; Dynorphins; Fentanyl; Peptide Fragments; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sincalide; Spinal Cord | 1994 |
Enantiomers of diastereomeric cis-N-[1-(2-hydroxy-2-phenylethyl)- 3-methyl-4-piperidyl]-N-phenylpropanamides: synthesis, X-ray analysis, and biological activities.
Topics: Analgesics; Animals; Crystallography, X-Ray; Fentanyl; Macaca mulatta; Magnetic Resonance Spectroscopy; Mice; Rats; Stereoisomerism | 1995 |
Monoclonal antibodies specific for ohmefentanyl.
Topics: Animals; Antibodies, Monoclonal; Female; Fentanyl; Guinea Pigs; Hybridomas; Ileum; Male; Mice; Mice, Inbred BALB C; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Opioid | 1994 |
[Effect of agonists of opioid receptor on coronary arterial strips in porcine].
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Coronary Vessels; Fentanyl; Haloperidol; In Vitro Techniques; Morphine; Muscle Contraction; Muscle, Smooth, Vascular; Naloxone; Pyrrolidines; Receptors, Opioid; Swine | 1994 |
Characterization and distribution of mu opioid receptors in rabbit cerebellum.
Topics: Animals; Autoradiography; Binding Sites; Cerebellum; Etorphine; Female; Fentanyl; Male; Rabbits; Radioligand Assay; Receptors, Opioid, mu | 1993 |
A new consistent model explaining structure (conformation)-activity relationships of opiates with mu-selectivity.
Topics: Analgesics; Crystallography, X-Ray; Fentanyl; Models, Molecular; Molecular Conformation; Narcotics; Phenazocine; Receptors, Opioid, mu; Stereoisomerism; Structure-Activity Relationship; Tomography, Emission-Computed | 1993 |
Stereochemical requirements for pseudoirreversible inhibition of opioid mu receptor binding by the 3-methylfentanyl congeners, RTI-46144 and its enantiomers: evidence for different binding domains.
Topics: Animals; Binding Sites; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Fentanyl; Ligands; Molecular Conformation; Rats; Receptors, Opioid, mu; Stereoisomerism | 1993 |
Regulation by lithium of the antagonistic effect of cholecystokinin octapeptide on ohmefentanyl-induced antinociception.
Topics: Analgesics; Animals; Fentanyl; Injections, Spinal; Lithium; Male; Nociceptors; Pain Measurement; Phosphatidylinositols; Rats; Rats, Wistar; Receptors, Opioid, mu; Sincalide | 1994 |
[Potentiation of morphine- and ohmefentanyl-induced analgesia by cholecystokinin receptor antagonists in rat].
Topics: Analgesics; Animals; Benzodiazepinones; Devazepide; Fentanyl; Morphine; Pain Threshold; Phenylurea Compounds; Rats; Rats, Wistar; Receptors, Cholecystokinin; Spinal Cord | 1993 |
Increased release of immunoreactive cholecystokinin octapeptide by morphine and potentiation of mu-opioid analgesia by CCKB receptor antagonist L-365,260 in rat spinal cord.
Topics: Analgesia; Analgesics; Animals; Benzodiazepinones; Devazepide; Dose-Response Relationship, Drug; Fentanyl; Injections, Spinal; Male; Morphine; Naloxone; Nociceptors; Pain Threshold; Phenylurea Compounds; Radioimmunoassay; Rats; Rats, Wistar; Receptors, Cholecystokinin; Receptors, Opioid, mu; Sincalide; Spinal Cord; Subarachnoid Space | 1993 |
Cholecystokinin octapeptide reverses mu-opioid-receptor-mediated inhibition of calcium current in rat dorsal root ganglion neurons.
Topics: Animals; Calcium Channel Blockers; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Fentanyl; Ganglia, Spinal; Ion Channel Gating; Male; Neurons; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, mu; Sincalide | 1995 |
Opioid peptide receptor studies. 7. The methylfentanyl congener RTI-4614-4 and its four enantiomers bind to different domains of the rat mu opioid receptor.
Topics: Affinity Labels; Analgesics; Analgesics, Opioid; Animals; Binding Sites; Binding, Competitive; COS Cells; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Etorphine; Fentanyl; Melphalan; Membrane Proteins; Protein Structure, Tertiary; Radioligand Assay; Rats; Receptors, Opioid, mu; Recombinant Fusion Proteins; Stereoisomerism | 1998 |
Apparent thermodynamic parameters of ligand binding to the cloned rat mu-opioid receptor.
Topics: Analgesics; Animals; Binding, Competitive; CHO Cells; Cricetinae; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Fentanyl; Ligands; Methadone; Morphine; Naltrexone; Narcotic Antagonists; Pentazocine; Peptide Fragments; Peptides; Radioligand Assay; Rats; Receptors, Opioid, mu; Somatostatin; Sufentanil; Thermodynamics; Time Factors | 1998 |
Molecular modeling of mu opioid receptor and its interaction with ohmefentanyl.
Topics: Amino Acid Sequence; Analgesics; Binding Sites; Fentanyl; Models, Molecular; Molecular Sequence Data; Receptors, Opioid, mu; Sequence Alignment | 1996 |
Analgesic activity and selectivity for opioid receptors of enantiomers of ohmefentanyl.
Topics: Analgesics; Animals; Female; Fentanyl; Guinea Pigs; Ileum; Male; Mice; Muscle Contraction; Rabbits; Receptors, Opioid, mu; Stereoisomerism; Structure-Activity Relationship; Vas Deferens | 1996 |
Interaction models of 3-methylfentanyl derivatives with mu opioid receptors.
Topics: Analgesics; Drug Interactions; Fentanyl; Models, Molecular; Receptors, Opioid, mu; Structure-Activity Relationship | 1997 |
Opioid peptide receptor studies, 11: involvement of Tyr148, Trp318 and His319 of the rat mu-opioid receptor in binding of mu-selective ligands.
Topics: Animals; Cloning, Molecular; COS Cells; Fentanyl; Histidine; Ligands; Models, Molecular; Molecular Structure; Mutagenesis, Site-Directed; Rats; Receptors, Opioid, mu; Stereoisomerism; Tryptophan; Tyrosine | 1999 |
Human mu-opioid receptor overexpressed in baculovirus system and its pharmacological characterizations.
Topics: Animals; Baculoviridae; Cells, Cultured; Cyclic AMP; Diprenorphine; Etorphine; Fentanyl; Gene Expression; Insecta; Radioligand Assay; Receptors, Opioid, mu; Transfection | 1998 |
Analgesic activity and selectivity of isothiocyanate derivatives of fentanyl analogs for opioid receptors.
Topics: Amides; Analgesics, Opioid; Animals; Fentanyl; Isothiocyanates; Male; Mice; Muscle Contraction; Nociceptors; Pain Measurement; Receptors, Opioid; Receptors, Opioid, delta; Stereoisomerism; Structure-Activity Relationship; Substrate Specificity; Vas Deferens | 1999 |
Comparison of physical dependence of ohmefentanyl stereoisomers in mice.
Topics: Analgesics; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Fentanyl; Male; Mice; Morphine Dependence; Stereoisomerism; Substance Withdrawal Syndrome; Substance-Related Disorders | 2000 |
The metabolic evidence of synergistic effect between ohmefentanyl and [D-Pen2, D-Pen5] enkephalin on differentiated SH-SY5Y cells in humans.
Topics: Acids; Analgesics; Analgesics, Opioid; Animals; Cell Differentiation; CHO Cells; Cricetinae; Drug Synergism; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Extracellular Space; Fentanyl; Humans; Naloxone; Narcotic Antagonists; Neuroblastoma; Neurons; Tumor Cells, Cultured | 2001 |
Evidence for mu opioid receptor on mouse spleen lymphocytes.
Topics: Animals; Cell Division; Female; Fentanyl; Mice; Mice, Inbred ICR; Naloxone; Receptors, Opioid, mu; Spleen; T-Lymphocytes | 1999 |
Molecular modeling on solvent effect and interaction mechanism of fentanyl analogs to mu-opioid receptor.
Topics: Analgesics; Binding Sites; Drug Interactions; Fentanyl; Models, Molecular; Receptors, Opioid, mu; Solvents; Structure-Activity Relationship | 2000 |
[Effects of ohmefentanyl at anesthetic dose on plasma levels of corticosterone, cortisol and antidiuretic hormone in rats].
Topics: Analgesics; Animals; Corticosterone; Fentanyl; Male; Rats; Stress Disorders, Post-Traumatic; Vasopressins | 1997 |
Quantitative comparison of ohmefentanyl isomers induced conditioning place preference in mice.
Topics: Analgesics, Opioid; Animals; Behavior, Addictive; Conditioning, Operant; Dose-Response Relationship, Drug; Fentanyl; Injections, Subcutaneous; Isomerism; Male; Mice; Mice, Inbred Strains; Morphine; Reinforcement, Psychology | 2001 |
Discrimination between peptide and non-peptide opioid agonists on the transcription of opioid receptors in two cell lines.
Topics: Benzamides; Cell Line; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Fentanyl; Piperazines; Polymerase Chain Reaction; Receptors, Opioid, delta; Receptors, Opioid, mu; RNA, Messenger; Transcription, Genetic | 2001 |
Analgesic activity and opioid receptor selectivity of stereoisomers of ohmefentanyl isothiocyanate.
Topics: Analgesics, Opioid; Animals; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Female; Fentanyl; Guinea Pigs; Ileum; In Vitro Techniques; Isothiocyanates; Male; Mice; Muscle Contraction; Nociceptors; Pain; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Stereoisomerism; Vas Deferens | 2001 |
Analysis of binding domain and function of chimeric mu/kappa opioid receptors to ohmefentanyl stereoisomers.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Binding Sites; Chlorocebus aethiops; COS Cells; Cyclic AMP; Dynorphins; Fentanyl; Peptide Fragments; Protein Structure, Tertiary; Receptors, Opioid, kappa; Receptors, Opioid, mu; Recombinant Fusion Proteins; Stereoisomerism | 2001 |
Homodimerization of human mu-opioid receptor overexpressed in Sf9 insect cells.
Topics: Animals; Baculoviridae; Blotting, Western; Cell Line; Dimerization; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Fentanyl; GTP-Binding Proteins; Humans; Insecta; Ligands; Narcotics; Peptides; Receptors, Opioid, mu; Sodium Dodecyl Sulfate; Time Factors | 2002 |
Ohmefentanyl stereoisomers induce changes of CREB phosphorylation in hippocampus of mice in conditioned place preference paradigm.
Topics: Analgesics; Animals; Behavior, Animal; Conditioning, Psychological; Cyclic AMP Response Element-Binding Protein; Dose-Response Relationship, Drug; Fentanyl; Hippocampus; Ketamine; Male; Mice; Morphine; Morphine Dependence; Phosphorylation; Reward; Stereoisomerism; Substance Withdrawal Syndrome; Substance-Related Disorders | 2003 |
Effects of ohmefentanyl stereoisomers on phosphorylation of cAMP- response element binding protein in cultured rat hippocampal neurons.
Topics: Analgesics; Animals; Cells, Cultured; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Fentanyl; Hippocampus; Morphine; Naloxone; Neurons; Phosphorylation; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Signal Transduction; Stereoisomerism | 2003 |
Effect of chronic treatment of ohmefentanyl stereoisomers on cyclic AMP formation in Sf9 insect cells expressing human mu-opioid receptors.
Topics: Analgesics; Animals; Binding, Competitive; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Drug Combinations; Fentanyl; Humans; Mice; Morphine Dependence; Naloxone; Receptors, Opioid, mu; Spodoptera; Stereoisomerism; Transfection | 2004 |
Orphanin FQ antagonizes the inhibition of Ca(2+) currents induced by mu-opioid receptors.
Topics: Analgesics; Animals; Calcium; Calcium Channels; Fentanyl; Ganglia, Spinal; Male; Neurons; Nociceptin; Nociceptin Receptor; Opioid Peptides; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, Opioid; Receptors, Opioid, mu; Reverse Transcriptase Polymerase Chain Reaction | 2005 |
Paradoxical relationship between RAVE (relative activity versus endocytosis) values of several opioid receptor agonists and their liability to cause dependence.
Topics: Analgesics, Opioid; Animals; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Endocytosis; Etorphine; Fentanyl; Guanosine 5'-O-(3-Thiotriphosphate); Morphine; Opioid-Related Disorders; Receptors, Opioid, mu | 2010 |
Comment on "Trisomy 21 noninvasive prenatal testing for twin pregnancies".
Topics: Down Syndrome; Female; Fentanyl; Humans; Pregnancy; Pregnancy, Twin; Prenatal Diagnosis; Trisomy | 2019 |