Page last updated: 2024-09-05

darunavir and bms 806

darunavir has been researched along with bms 806 in 3 studies

Compound Research Comparison

Studies
(darunavir)
Trials
(darunavir)
Recent Studies (post-2010)
(darunavir)
Studies
(bms 806)
Trials
(bms 806)
Recent Studies (post-2010) (bms 806)
1,14822478045018

Protein Interaction Comparison

ProteinTaxonomydarunavir (IC50)bms 806 (IC50)
Cytochrome P450 2D6Homo sapiens (human)9.7
Envelope glycoprotein gp160 [Cleaved into: Surface protein gp120 Human immunodeficiency virus 18.7

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (66.67)24.3611
2020's1 (33.33)2.80

Authors

AuthorsStudies
De Clercq, E; Liu, X; Pannecouque, C; Zhan, P1
De Clercq, E; Kang, D; Kongsted, J; Liu, X; Namasivayam, V; Pannecouque, C; Poongavanam, V; Song, Y; Wu, G; Zhan, P; Zhang, J; Zhao, T1
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1

Reviews

2 review(s) available for darunavir and bms 806

ArticleYear
Anti-HIV Drug Discovery and Development: Current Innovations and Future Trends.
    Journal of medicinal chemistry, 2016, Apr-14, Volume: 59, Issue:7

    Topics: Anti-HIV Agents; Chemistry, Pharmaceutical; Chemoprevention; Drug Design; Drug Discovery; Drug Resistance, Viral; HIV Protease Inhibitors; Humans; Molecular Targeted Therapy; Mutation; Prodrugs; Solubility; Structure-Activity Relationship

2016
Overview of Recent Strategic Advances in Medicinal Chemistry.
    Journal of medicinal chemistry, 2019, 11-14, Volume: 62, Issue:21

    Topics: Chemistry, Pharmaceutical; Drug Discovery

2019

Other Studies

1 other study(ies) available for darunavir and bms 806

ArticleYear
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023