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colchicine and e 7010

colchicine has been researched along with e 7010 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (10.00)18.2507
2000's2 (20.00)29.6817
2010's6 (60.00)24.3611
2020's1 (10.00)2.80

Authors

AuthorsStudies
Bukhtiyarova, M; Chao, W; Dorsey, BD; Flubacher, D; Flynn, GA; Fujimoto, T; Husain, A; Joseph, RW; Kelly, MJ; Lee, KJ; Lee, Y; Liu, B; Lu, Y; Mihelcic, J; Moffett, KK; Moore, WR; Nelson, D; Ochman, AR; Saporito, MS; Schumacher, A; Shetty, RS; Springman, EB; Stojanovic, A; Williams, K1
Lama, R; Li, B; Sandhu, R; Su, B; Zhong, B1
Chang, CY; Chang, JY; Chang, YT; Kuo, CC; Lai, MJ; Lee, HY; Liou, JP; Liu, YM; Mehndiratta, S; Nien, CY; Pan, SL; Su, MC; Wu, JS; Wu, SY1
Chang, LH; Chen, MC; Chuang, HY; Huang, HL; Lai, MJ; Lee, HY; Liou, JP; Liu, YM; Mehndiratta, S; Pan, SL; Teng, CM; Tsai, AC; Wu, YW1
Guo, XL; Ji, YT; Liu, YN; Liu, ZP; Tang, LQ; Wang, JJ; Zhang, CM; Zhao, GD1
Chang, CY; Chang, JY; Chen, MC; Hsu, KC; Lai, MJ; Lee, HY; Lin, MH; Lin, TE; Liou, JP; Liu, YM; Nepali, K; Ojha, R1
Ahmed, SA; Althagafi, II; Ansari, MA; Kamal, A; Malik, MS1
Kitoh, K; Koyanagi, N; Yamaguchi, A; Yoshimatsu, K; Yoshino, H1
Kovar, P; Ng, SC; Rosenberg, SH; Tahir, SK1
Burnett, JC; Day, BW; Gussio, R; Hamel, E; Hermone, AR; McGrath, C; Nguyen, TL; Wipf, P; Zaharevitz, DW1

Reviews

1 review(s) available for colchicine and e 7010

ArticleYear
Application of triazoles as bioisosteres and linkers in the development of microtubule targeting agents.
    RSC medicinal chemistry, 2020, Mar-01, Volume: 11, Issue:3

    Topics:

2020

Other Studies

9 other study(ies) available for colchicine and e 7010

ArticleYear
Synthesis and pharmacological evaluation of N-(3-(1H-indol-4-yl)-5-(2-methoxyisonicotinoyl)phenyl)methanesulfonamide (LP-261), a potent antimitotic agent.
    Journal of medicinal chemistry, 2011, Jan-13, Volume: 54, Issue:1

    Topics: Animals; Biological Availability; Cell Line, Tumor; Cell Proliferation; Cell Survival; Colchicine; Drug Screening Assays, Antitumor; G2 Phase; Humans; Indoles; Isonicotinic Acids; Mice; Mice, Nude; Models, Molecular; Neoplasm Transplantation; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Sulfonamides; Transplantation, Heterologous; Tubulin; Tubulin Modulators

2011
Identification of selective tubulin inhibitors as potential anti-trypanosomal agents.
    Bioorganic & medicinal chemistry letters, 2012, Sep-01, Volume: 22, Issue:17

    Topics: Amino Acid Sequence; Animals; Cattle; Cell Proliferation; Cells, Cultured; Fibroblasts; Humans; Models, Molecular; Molecular Sequence Data; Structural Homology, Protein; Sulfonamides; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African; Tubulin; Tubulin Modulators

2012
Furanylazaindoles: potent anticancer agents in vitro and in vivo.
    Journal of medicinal chemistry, 2013, Oct-24, Volume: 56, Issue:20

    Topics: Animals; Antineoplastic Agents; Cell Cycle Checkpoints; Cell Line, Tumor; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Design; Female; Heterocyclic Compounds, 2-Ring; HT29 Cells; Humans; Indoles; Inhibitory Concentration 50; Mice, Nude; Molecular Structure; Neoplasms; Polymerization; Sulfonamides; Tubulin; Xenograft Model Antitumor Assays

2013
N-Sulfonyl-aminobiaryls as Antitubulin Agents and Inhibitors of Signal Transducers and Activators of Transcription 3 (STAT3) Signaling.
    Journal of medicinal chemistry, 2015, Aug-27, Volume: 58, Issue:16

    Topics: Antineoplastic Agents; Apoptosis; Binding, Competitive; Cell Line, Tumor; Colchicine; Humans; Phosphorylation; STAT3 Transcription Factor; Structure-Activity Relationship; Sulfonamides; Tubulin Modulators

2015
Design, Synthesis, and Biological Evaluation of 1-Methyl-1,4-dihydroindeno[1,2-c]pyrazole Analogues as Potential Anticancer Agents Targeting Tubulin Colchicine Binding Site.
    Journal of medicinal chemistry, 2016, 06-09, Volume: 59, Issue:11

    Topics: Animals; Antineoplastic Agents; Binding Sites; Cell Line, Tumor; Cell Proliferation; Colchicine; Dose-Response Relationship, Drug; Drug Design; Drug Screening Assays, Antitumor; Humans; Mice; Mice, Nude; Models, Molecular; Molecular Structure; Neoplasms, Experimental; Pyrazoles; Structure-Activity Relationship; Tubulin; Tubulin Modulators

2016
1-Arylsulfonyl indoline-benzamides as a new antitubulin agents, with inhibition of histone deacetylase.
    European journal of medicinal chemistry, 2019, Jan-15, Volume: 162

    Topics: A549 Cells; Animals; Antineoplastic Agents; Benzamides; Carcinoma, Non-Small-Cell Lung; Catalytic Domain; Cell Line, Tumor; Cell Proliferation; Heterografts; Histone Deacetylase Inhibitors; Humans; Indoles; Lymphoma, B-Cell; Mice; Models, Molecular; Protein Binding; Tubulin Modulators

2019
Mechanism of action of E7010, an orally active sulfonamide antitumor agent: inhibition of mitosis by binding to the colchicine site of tubulin.
    Cancer research, 1997, Aug-01, Volume: 57, Issue:15

    Topics: Aminophenols; Animals; Antineoplastic Agents; Binding, Competitive; Cell Cycle; Colchicine; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Humans; Leukemia; Lung Neoplasms; Mice; Microtubules; Mitosis; Sulfonamides; Tubulin; Tumor Cells, Cultured; Vincristine

1997
Rapid colchicine competition-binding scintillation proximity assay using biotin-labeled tubulin.
    BioTechniques, 2000, Volume: 29, Issue:1

    Topics: Aminophenols; Bibenzyls; Binding Sites; Binding, Competitive; Biotinylation; Colchicine; Demecolcine; Mebendazole; Microspheres; Podophyllotoxin; Scintillation Counting; Solvents; Stilbenes; Streptavidin; Sulfonamides; Tritium; Tubulin; Yttrium

2000
A common pharmacophore for a diverse set of colchicine site inhibitors using a structure-based approach.
    Journal of medicinal chemistry, 2005, Sep-22, Volume: 48, Issue:19

    Topics: 2-Methoxyestradiol; 4-Butyrolactone; Aminophenols; Binding Sites; Chalcone; Colchicine; Cyclopropanes; Estradiol; Indans; Lignans; Models, Molecular; Molecular Structure; Nocodazole; Podophyllotoxin; Protein Binding; Stilbenes; Structure-Activity Relationship; Sulfonamides; Thiazoles; Tubulin; Tubulin Modulators

2005
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