Page last updated: 2024-09-03

cgp 52432 and glycine

cgp 52432 has been researched along with glycine in 5 studies

Compound Research Comparison

Studies
(cgp 52432)
Trials
(cgp 52432)
Recent Studies (post-2010)
(cgp 52432)
Studies
(glycine)
Trials
(glycine)
Recent Studies (post-2010) (glycine)
7202935,1637568,415

Protein Interaction Comparison

ProteinTaxonomycgp 52432 (IC50)glycine (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)1.4852
Sodium- and chloride-dependent glycine transporter 1Homo sapiens (human)106
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.3253
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.3253
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.3253
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.3253
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.3253
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.3253
Sodium- and chloride-dependent glycine transporter 2Homo sapiens (human)128

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (20.00)29.6817
2010's4 (80.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Luccini, E; Raiteri, L; Raiteri, M; Romei, C1
Brooks, PL; Peever, JH2
Di Prisco, S; Grilli, M; Marchi, M; Pittaluga, A; Summa, M; Usai, C1
Georgopoulos, P; Papatheodoropoulos, C; Petrides, T; Pofantis, H1

Other Studies

5 other study(ies) available for cgp 52432 and glycine

ArticleYear
GABA(B) presynaptic receptors modulate glycine exocytosis from mouse spinal cord and hippocampus glycinergic nerve endings.
    Pharmacological research, 2009, Volume: 59, Issue:3

    Topics: Animals; Baclofen; Benzylamines; Exocytosis; Glycine; Glycine Plasma Membrane Transport Proteins; Hippocampus; Mice; Nerve Endings; Organophosphorus Compounds; Phosphinic Acids; Receptors, GABA-B; Spinal Cord

2009
GABAergic and glycinergic control of upper airway motoneurons in rapid eye movement sleep.
    Advances in experimental medicine and biology, 2010, Volume: 669

    Topics: Animals; Benzylamines; Electroencephalography; Electromyography; gamma-Aminobutyric Acid; Glycine; Male; Masseter Muscle; Motor Neurons; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Respiratory System; Sleep, REM

2010
Presynaptic mGlu7 receptors control GABA release in mouse hippocampus.
    Neuropharmacology, 2013, Volume: 66

    Topics: Adenylyl Cyclase Inhibitors; Aminobutyrates; Animals; Baclofen; Benzhydryl Compounds; Benzoates; Benzylamines; Colforsin; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Exocytosis; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Hippocampus; Imines; Mice; Phosphinic Acids; Potassium Chloride; Pyridones; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Synaptosomes; Syntaxin 1; Vesicular Inhibitory Amino Acid Transport Proteins

2013
Identification of the transmitter and receptor mechanisms responsible for REM sleep paralysis.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Jul-18, Volume: 32, Issue:29

    Topics: Animals; Benzylamines; Bicuculline; Electromyography; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glycine; Glycine Agents; Male; Motor Neurons; Neural Inhibition; Paresis; Phosphinic Acids; Rats; Rats, Sprague-Dawley; Sleep, REM; Strychnine; Trigeminal Nuclei

2012
Differences in paired-pulse inhibition and facilitation in the dentate gyrus and CA3 field between dorsal and ventral rat hippocampus.
    Brain research, 2015, May-22, Volume: 1608

    Topics: Animals; Benzylamines; Biophysics; CA3 Region, Hippocampal; Cyclopropanes; Dentate Gyrus; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; Glycine; In Vitro Techniques; Male; Nerve Net; Organophosphorus Compounds; Phosphinic Acids; Piperazines; Rats; Rats, Wistar; Statistics, Nonparametric

2015
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