Page last updated: 2024-09-04

canertinib and spc-839

canertinib has been researched along with spc-839 in 2 studies

Compound Research Comparison

Studies
(canertinib)
Trials
(canertinib)
Recent Studies (post-2010)
(canertinib)
Studies
(spc-839)
Trials
(spc-839)
Recent Studies (post-2010) (spc-839)
12496537018

Protein Interaction Comparison

ProteinTaxonomycanertinib (IC50)spc-839 (IC50)
Inhibitor of nuclear factor kappa-B kinase subunit betaHomo sapiens (human)0.0538
Inhibitor of nuclear factor kappa-B kinase subunit alphaHomo sapiens (human)1.3
Transcription factor AP-1Homo sapiens (human)0.008
Nuclear factor NF-kappa-B p105 subunitHomo sapiens (human)0.008
Cannabinoid receptor 1Rattus norvegicus (Norway rat)0.344
Mu-type opioid receptorRattus norvegicus (Norway rat)0.2527
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)0.618
Nuclear factor NF-kappa-B p100 subunit Homo sapiens (human)0.008
Transcription factor p65Homo sapiens (human)0.008
Cannabinoid receptor 2Rattus norvegicus (Norway rat)0.344

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Das, D; Hong, J1

Reviews

1 review(s) available for canertinib and spc-839

ArticleYear
Recent advancements of 4-aminoquinazoline derivatives as kinase inhibitors and their applications in medicinal chemistry.
    European journal of medicinal chemistry, 2019, May-15, Volume: 170

    Topics: Animals; Antineoplastic Agents; Chemistry Techniques, Synthetic; Humans; Neoplasms; Protein Kinase Inhibitors; Quinazolines

2019

Other Studies

1 other study(ies) available for canertinib and spc-839

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013
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