Page last updated: 2024-08-07 17:29:24
Cannabinoid receptor 2
A cannabinoid receptor 2 that is encoded in the genome of rat. [OMA:Q9QZN9, PRO:DNx]
Synonyms
CB-2;
CB2;
rCB2
Research
Bioassay Publications (13)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 4 (30.77) | 18.2507 |
| 2000's | 4 (30.77) | 29.6817 |
| 2010's | 5 (38.46) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (20)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| dronabinol | Rattus norvegicus (Norway rat) | IC50 | 0.2180 | 1 | 1 |
| dronabinol | Rattus norvegicus (Norway rat) | Ki | 0.0460 | 1 | 1 |
| cp-55,940 | Rattus norvegicus (Norway rat) | IC50 | 0.0021 | 1 | 1 |
| 1,1-dimethylheptyl-11-hydroxytetrahydrocannabinol | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| delta(9-11)-tetrahydrocannabinol | Rattus norvegicus (Norway rat) | IC50 | 0.3340 | 1 | 1 |
| n,n-di-n-propylserotonin | Rattus norvegicus (Norway rat) | IC50 | 0.8200 | 1 | 1 |
| delta-8-tetrahydrocannabinol | Rattus norvegicus (Norway rat) | IC50 | 0.1790 | 1 | 1 |
| tandutinib | Rattus norvegicus (Norway rat) | IC50 | 0.2000 | 1 | 2 |
| anandamide | Rattus norvegicus (Norway rat) | Ki | 0.5393 | 3 | 3 |
| glyceryl 2-arachidonate | Rattus norvegicus (Norway rat) | Ki | 0.1000 | 1 | 1 |
| virodhamine | Rattus norvegicus (Norway rat) | Ki | 0.9120 | 1 | 1 |
| am-356 | Rattus norvegicus (Norway rat) | Ki | 0.0240 | 2 | 2 |
| spc-839 | Rattus norvegicus (Norway rat) | IC50 | 0.3440 | 2 | 6 |
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| cp-55,940 | Rattus norvegicus (Norway rat) | EC50 | 0.0003 | 1 | 1 |
| 2-chloro-n(6)cyclopentyladenosine | Rattus norvegicus (Norway rat) | EC50 | 0.0046 | 1 | 1 |
| n(6)-cyclopentyladenosine | Rattus norvegicus (Norway rat) | EC50 | 0.0063 | 1 | 1 |
| sr 144528 | Rattus norvegicus (Norway rat) | EC50 | 0.0233 | 1 | 1 |
| (3r)-((2,3-dihydro-5-methyl-3-((4-morpholinyl)methyl)pyrrolo-(1,2,3-de)-1,4-benzoxazin-6-yl)(1-naphthalenyl))methanone | Rattus norvegicus (Norway rat) | EC50 | 0.0015 | 1 | 1 |
| n-((1s,trans)-2-hydroxycyclopentyl)adenosine | Rattus norvegicus (Norway rat) | EC50 | 0.0059 | 1 | 1 |
| am 1241 | Rattus norvegicus (Norway rat) | EC50 | 0.2655 | 1 | 2 |
| gw 842166x | Rattus norvegicus (Norway rat) | EC50 | 0.0910 | 1 | 1 |
| a-796260 | Rattus norvegicus (Norway rat) | EC50 | 0.0016 | 1 | 1 |