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Cannabinoid receptor 2
A cannabinoid receptor 2 that is encoded in the genome of rat. [OMA:Q9QZN9, PRO:DNx]
Synonyms
CB-2;
CB2;
rCB2
Research
Bioassay Publications (13)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 4 (30.77) | 18.2507 |
| 2000's | 4 (30.77) | 29.6817 |
| 2010's | 5 (38.46) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (20)
Drugs with Inhibition Measurements
Drugs with Activation Measurements
A novel probe for the cannabinoid receptor.Journal of medicinal chemistry, , May-29, Volume: 35, Issue:11, 1992
Synthesis and pharmacological evaluation of ether and related analogues of delta 8-, delta 9-, and delta 9,11-tetrahydrocannabinol.Journal of medicinal chemistry, , Volume: 34, Issue:11, 1991
Imine derivatives as new potent and selective CB2 cannabinoid receptor agonists with an analgesic action.Bioorganic & medicinal chemistry, , Feb-01, Volume: 16, Issue:3, 2008
Discovery and optimization of a novel series of N-arylamide oxadiazoles as potent, highly selective and orally bioavailable cannabinoid receptor 2 (CB2) agonists.Journal of medicinal chemistry, , Aug-28, Volume: 51, Issue:16, 2008
The importance of hydrogen bonding and aromatic stacking to the affinity and efficacy of cannabinoid receptor CB2 antagonist, 5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)methyl]-N-[(1S,2S,4R)-1,3,3-trimethylbicyclo[2.2.1]hept-2-yl]-1H-pyrazole-3-carboxJournal of medicinal chemistry, , Sep-12, Volume: 56, Issue:17, 2013
Oxygenated metabolites of anandamide and 2-arachidonoylglycerol: conformational analysis and interaction with cannabinoid receptors, membrane transporter, and fatty acid amide hydrolase.Journal of medicinal chemistry, , Aug-15, Volume: 45, Issue:17, 2002
(R)-methanandamide: a chiral novel anandamide possessing higher potency and metabolic stability.Journal of medicinal chemistry, , Jun-10, Volume: 37, Issue:12, 1994