Page last updated: 2024-09-03

btm 1042 and afdx 116

btm 1042 has been researched along with afdx 116 in 2 studies

Compound Research Comparison

Studies
(btm 1042)
Trials
(btm 1042)
Recent Studies (post-2010)
(btm 1042)
Studies
(afdx 116)
Trials
(afdx 116)
Recent Studies (post-2010) (afdx 116)
1100367124

Protein Interaction Comparison

ProteinTaxonomybtm 1042 (IC50)afdx 116 (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)1.8
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)2.927
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)3.4558
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.927
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.927
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.5994
Muscarinic acetylcholine receptor M2Mus musculus (house mouse)6.2

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baron, E; Boer, R; Eltze, M; Kromer, W1
Jackson, KN; Kachur, JF; Lowe, VC; Noronha-Blob, L; Sturm, BL1

Other Studies

2 other study(ies) available for btm 1042 and afdx 116

ArticleYear
Telenzepine inhibits electrically-stimulated, acetylcholine plus histamine-mediated acid secretion in the mouse isolated stomach by blockade of M1 muscarine receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:1

    Topics: Acetylcholine; Alkaloids; Animals; Anti-Ulcer Agents; Electric Stimulation; Furans; Gastric Acid; Gastric Mucosa; Histamine; Mice; Muscarinic Antagonists; Naphthalenes; p-Methoxy-N-methylphenethylamine; Parasympatholytics; Piperidines; Pirenzepine; Stomach; Thiazepines; Vagus Nerve

1991
In vitro and in vivo antimuscarinic effects of (-)cis 2,3-dihydro-3-(4-methylpiperazinylmethyl)-2-phenyl-1,5 benzothiazepin-4-(5H)one HCl (BTM-1086) in guinea pig peripheral tissues.
    Life sciences, 1990, Volume: 46, Issue:17

    Topics: Animals; Atropine; Calcium; Female; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neurons; Parasympatholytics; Piperidines; Pirenzepine; Structure-Activity Relationship; Thiazepines; Tumor Cells, Cultured; Urinary Bladder; Vas Deferens

1990