btm 1042 has been researched along with afdx 116 in 2 studies
Studies (btm 1042) | Trials (btm 1042) | Recent Studies (post-2010) (btm 1042) | Studies (afdx 116) | Trials (afdx 116) | Recent Studies (post-2010) (afdx 116) |
---|---|---|---|---|---|
11 | 0 | 0 | 367 | 1 | 24 |
Protein | Taxonomy | btm 1042 (IC50) | afdx 116 (IC50) |
---|---|---|---|
Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | 1.8 | |
Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | 2.927 | |
Muscarinic acetylcholine receptor M3 | Rattus norvegicus (Norway rat) | 3.4558 | |
Muscarinic acetylcholine receptor M4 | Rattus norvegicus (Norway rat) | 2.927 | |
Muscarinic acetylcholine receptor M5 | Rattus norvegicus (Norway rat) | 2.927 | |
Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | 2.5994 | |
Muscarinic acetylcholine receptor M2 | Mus musculus (house mouse) | 6.2 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Baron, E; Boer, R; Eltze, M; Kromer, W | 1 |
Jackson, KN; Kachur, JF; Lowe, VC; Noronha-Blob, L; Sturm, BL | 1 |
2 other study(ies) available for btm 1042 and afdx 116
Article | Year |
---|---|
Telenzepine inhibits electrically-stimulated, acetylcholine plus histamine-mediated acid secretion in the mouse isolated stomach by blockade of M1 muscarine receptors.
Topics: Acetylcholine; Alkaloids; Animals; Anti-Ulcer Agents; Electric Stimulation; Furans; Gastric Acid; Gastric Mucosa; Histamine; Mice; Muscarinic Antagonists; Naphthalenes; p-Methoxy-N-methylphenethylamine; Parasympatholytics; Piperidines; Pirenzepine; Stomach; Thiazepines; Vagus Nerve | 1991 |
In vitro and in vivo antimuscarinic effects of (-)cis 2,3-dihydro-3-(4-methylpiperazinylmethyl)-2-phenyl-1,5 benzothiazepin-4-(5H)one HCl (BTM-1086) in guinea pig peripheral tissues.
Topics: Animals; Atropine; Calcium; Female; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Neurons; Parasympatholytics; Piperidines; Pirenzepine; Structure-Activity Relationship; Thiazepines; Tumor Cells, Cultured; Urinary Bladder; Vas Deferens | 1990 |