Page last updated: 2024-08-05 15:44:31

tropomyosin-related kinase B receptor antagonist

An antagonist that binds to and deactivates the tropomyosin-related kinase B (TrkB) receptor, the main signaling receptor of the neurotrophin brain-derived neurotrophic factor (BDNF).

ChEBI ID: 78681

Members (2)

MemberDefinitionClass
ANA-12A secondary carboxamide that is anthranilic acid in which the carboxy group has undergone condensation with the primary amino group of alpha-amino-epsilon-caprolactam, while the aryl-amino group has undergone condensation with the carboxy group of 1-benzothiophene-2-carboxylic acid. It is a selective, non-competitive antagonist of tropomyosin receptor kinase B (TrkB, also known as tyrosine receptor kinase B).ANA-12
sf 2370A organic heterooctacyclic compound that is a potent inhibitor of protein kinase C and is isolated from Nocardiopsis sp K-252aK-252a

Research

Studies (24)

TimeframeStudies, Drugs with This Role(%)All Drugs %
pre-19902 (8.33)18.7374
1990's3 (12.50)18.2507
2000's7 (29.17)29.6817
2010's8 (33.33)24.3611
2020's4 (16.67)2.80

Study Types

Publication TypeStudies, Drugs with this Role (%)All Drugs (%)
Trials0 (0.00%)5.53%
Reviews1 (4.17%)6.00%
Case Studies0 (0.00%)4.05%
Observational0 (0.00%)0.25%
Other23 (95.83%)84.16%

Protein Targets (325)

Potency Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
cytochrome P450 2C9, partialHomo sapiens (human)Potency0.379111
cytochrome P450 family 3 subfamily A polypeptide 4Homo sapiens (human)Potency10.684011
GVesicular stomatitis virusPotency0.379111
HLA class I histocompatibility antigen, B alpha chain Homo sapiens (human)Potency0.379111
Inositol hexakisphosphate kinase 1Homo sapiens (human)Potency0.379112
Interferon betaHomo sapiens (human)Potency0.379111

Inhibition Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
cAMP-dependent protein kinase Oryctolagus cuniculus (rabbit)IC500.000011
cAMP-dependent protein kinase catalytic subunit alphaBos taurus (cattle)IC500.145012
Chain A, Serine/threonine-protein kinase pknBMycobacterium tuberculosisIC501.000011
Cyclin-dependent kinase 2Homo sapiens (human)IC500.145012
Cyclin-dependent kinase 4Homo sapiens (human)IC500.145012
G1/S-specific cyclin-D1Homo sapiens (human)IC500.145012
G1/S-specific cyclin-E1Homo sapiens (human)IC500.145012
High affinity nerve growth factor receptorHomo sapiens (human)IC500.009533
Mitogen-activated protein kinase kinase kinase 10Homo sapiens (human)IC500.026713
Mitogen-activated protein kinase kinase kinase 11Homo sapiens (human)IC500.026713
Mitogen-activated protein kinase kinase kinase 9Homo sapiens (human)IC500.026713
Myosin light chain kinase, smooth muscleGallus gallus (chicken)IC500.000011
Myosin light chain kinase, smooth muscleHomo sapiens (human)IC500.022011
Myosin light chain kinase, smooth muscleHomo sapiens (human)Ki0.020011
Phosphorylase b kinase gamma catalytic chain, liver/testis isoformHomo sapiens (human)IC500.001722
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoformHomo sapiens (human)IC500.001722
Phosphorylase b kinase regulatory subunit alpha, liver isoformHomo sapiens (human)IC500.001722
Phosphorylase b kinase regulatory subunit alpha, skeletal muscle isoformHomo sapiens (human)IC500.001722
Phosphorylase b kinase regulatory subunit betaHomo sapiens (human)IC500.001722
Protein kinase C alpha typeHomo sapiens (human)IC500.250011
Protein kinase C alpha typeRattus norvegicus (Norway rat)IC500.125022
Protein kinase C beta typeHomo sapiens (human)IC500.250011
Protein kinase C beta typeRattus norvegicus (Norway rat)IC500.125022
Protein kinase C delta typeHomo sapiens (human)IC500.250011
Protein kinase C delta typeRattus norvegicus (Norway rat)IC500.125022
Protein kinase C epsilon typeHomo sapiens (human)IC500.250011
Protein kinase C epsilon typeRattus norvegicus (Norway rat)IC500.125022
Protein kinase C eta typeHomo sapiens (human)IC500.250011
Protein kinase C eta typeRattus norvegicus (Norway rat)IC500.125022
Protein kinase C gamma typeHomo sapiens (human)IC500.250011
Protein kinase C gamma typeRattus norvegicus (Norway rat)IC500.240033
Protein kinase C iota typeHomo sapiens (human)IC500.250011
Protein kinase C theta typeHomo sapiens (human)IC500.390022
Protein kinase C theta typeRattus norvegicus (Norway rat)IC500.125022
Protein kinase C zeta typeHomo sapiens (human)IC500.250011
Protein kinase C zeta typeRattus norvegicus (Norway rat)IC500.125022
Serine/threonine-protein kinase D1Homo sapiens (human)IC500.250011
Serine/threonine-protein kinase D3Homo sapiens (human)IC500.250011
Serine/threonine-protein kinase LMTK3Homo sapiens (human)IC500.079411
Serine/threonine-protein kinase pim-1Homo sapiens (human)IC500.150011
Vascular endothelial growth factor receptor 2Homo sapiens (human)IC500.043022

Activation Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
26S proteasome regulatory subunit 6BHomo sapiens (human)Kd30.000012
5'-AMP-activated protein kinase catalytic subunit alpha-1Homo sapiens (human)Kd0.461011
5'-AMP-activated protein kinase subunit gamma-1Homo sapiens (human)Kd0.352011
5'-AMP-activated protein kinase subunit gamma-2Homo sapiens (human)Kd0.868011
AarF domain-containing protein kinase 1Homo sapiens (human)Kd6.090011
Actin-related protein 2Homo sapiens (human)Kd30.000011
Actin-related protein 3Homo sapiens (human)Kd30.000011
Activated CDC42 kinase 1Homo sapiens (human)Kd1.717011
Activin receptor type-1Homo sapiens (human)Kd30.000011
Activin receptor type-1BHomo sapiens (human)Kd15.258011
Activin receptor type-2BHomo sapiens (human)Kd30.000011
Acyl-CoA dehydrogenase family member 10Homo sapiens (human)Kd30.000011
Acyl-CoA dehydrogenase family member 11Homo sapiens (human)Kd30.000011
Adenosine kinaseHomo sapiens (human)Kd30.000011
Adenylate kinase 2, mitochondrialHomo sapiens (human)Kd30.000011
ADP/ATP translocase 2Homo sapiens (human)Kd30.000011
ADP/ATP translocase 3Homo sapiens (human)Kd30.000011
ALK tyrosine kinase receptorHomo sapiens (human)Kd30.000011
AP2-associated protein kinase 1Homo sapiens (human)Kd0.005011
ATP-dependent 6-phosphofructokinase, platelet typeHomo sapiens (human)Kd30.000011
ATP-dependent RNA helicase DDX1Homo sapiens (human)Kd30.000011
ATP-dependent RNA helicase DDX3XHomo sapiens (human)Kd30.000011
ATP-dependent RNA helicase DDX42Homo sapiens (human)Kd30.000011
ATP-dependent RNA helicase DHX30Homo sapiens (human)Kd30.000011
Atypical kinase COQ8A, mitochondrialHomo sapiens (human)Kd30.000012
Aurora kinase AHomo sapiens (human)Kd0.020011
Aurora kinase BHomo sapiens (human)Kd0.353011
Beta-adrenergic receptor kinase 1Homo sapiens (human)Kd30.000011
BMP-2-inducible protein kinaseHomo sapiens (human)Kd0.090011
Bone morphogenetic protein receptor type-1AHomo sapiens (human)Kd30.000011
Bone morphogenetic protein receptor type-1BHomo sapiens (human)Kd30.000011
Bone morphogenetic protein receptor type-2Homo sapiens (human)Kd30.000011
Breakpoint cluster region proteinHomo sapiens (human)Kd30.000011
Calcium/calmodulin-dependent protein kinase kinase 2Homo sapiens (human)Kd2.277011
Calcium/calmodulin-dependent protein kinase type II subunit deltaHomo sapiens (human)Kd0.190011
Calcium/calmodulin-dependent protein kinase type II subunit gammaHomo sapiens (human)Kd0.173011
Calcium/calmodulin-dependent protein kinase type IVHomo sapiens (human)Kd30.000011
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)Kd30.000011
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)Kd30.000011
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)Kd30.000011
cAMP-dependent protein kinase type II-alpha regulatory subunitHomo sapiens (human)Kd30.000011
Casein kinase I isoform alphaHomo sapiens (human)Kd30.000011
Casein kinase I isoform deltaHomo sapiens (human)Kd30.000011
Casein kinase I isoform epsilonHomo sapiens (human)Kd30.000011
Casein kinase I isoform gamma-1Homo sapiens (human)Kd30.000011
Casein kinase I isoform gamma-2Homo sapiens (human)Kd30.000011
Casein kinase I isoform gamma-3Homo sapiens (human)Kd30.000011
Casein kinase II subunit alpha'Homo sapiens (human)Kd30.000011
cGMP-dependent protein kinase 1 Homo sapiens (human)Kd30.000011
Chain A, Hepatocyte growth factor receptorHomo sapiens (human)Kd0.010011
Chromodomain-helicase-DNA-binding protein 4Homo sapiens (human)Kd30.000011
Citron Rho-interacting kinaseHomo sapiens (human)Kd30.000011
Cyclin-dependent kinase 1Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 10Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 12Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 13Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 16Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 17Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 2Homo sapiens (human)Kd0.101011
Cyclin-dependent kinase 3Homo sapiens (human)Kd0.032011
Cyclin-dependent kinase 4Homo sapiens (human)Kd0.014011
Cyclin-dependent kinase 6Homo sapiens (human)Kd0.399011
Cyclin-dependent kinase 7Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 9Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase-like 5Homo sapiens (human)Kd30.000011
Cyclin-dependent-like kinase 5 Homo sapiens (human)Kd0.911011
Cyclin-G-associated kinaseHomo sapiens (human)Kd1.269011
Cytochrome c1, heme protein, mitochondrialHomo sapiens (human)Kd30.000011
dCTP pyrophosphatase 1Homo sapiens (human)Kd30.000011
Delta(24)-sterol reductaseHomo sapiens (human)Kd30.000011
Deoxycytidine kinaseHomo sapiens (human)Kd30.000011
Discoidin domain-containing receptor 2Homo sapiens (human)Kd30.000011
DNA replication licensing factor MCM4Homo sapiens (human)Kd30.000011
DNA topoisomerase 2-alphaHomo sapiens (human)Kd30.000011
DNA topoisomerase 2-betaHomo sapiens (human)Kd30.000011
DnaJ homolog subfamily A member 1Homo sapiens (human)Kd30.000011
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)Kd1.747011
Dual specificity mitogen-activated protein kinase kinase 2Homo sapiens (human)Kd0.474011
Dual specificity mitogen-activated protein kinase kinase 3Homo sapiens (human)Kd30.000011
Dual specificity mitogen-activated protein kinase kinase 4Homo sapiens (human)Kd30.000011
Dual specificity mitogen-activated protein kinase kinase 5Homo sapiens (human)Kd2.033011
Dual specificity mitogen-activated protein kinase kinase 6Homo sapiens (human)Kd0.088011
Dual specificity protein kinase CLK1Homo sapiens (human)Kd0.010011
Dual specificity protein kinase CLK2Homo sapiens (human)Kd3.809011
Dual specificity protein kinase CLK4Homo sapiens (human)Kd0.015011
Dual specificity protein kinase TTKHomo sapiens (human)Kd0.030011
Dual specificity testis-specific protein kinase 1Homo sapiens (human)Kd30.000011
Dual specificity testis-specific protein kinase 2Homo sapiens (human)Kd30.000011
Dual specificity tyrosine-phosphorylation-regulated kinase 1AHomo sapiens (human)Kd4.852011
Dual specificity tyrosine-phosphorylation-regulated kinase 1BHomo sapiens (human)Kd30.000011
Dynamin-like 120 kDa protein, mitochondrialHomo sapiens (human)Kd30.000011
EKC/KEOPS complex subunit TP53RKHomo sapiens (human)Kd3.840011
Electron transfer flavoprotein subunit betaHomo sapiens (human)Kd30.000011
Elongation factor Tu, mitochondrialHomo sapiens (human)Kd30.000012
Ephrin type-A receptor 1Homo sapiens (human)Kd30.000011
Ephrin type-A receptor 2Homo sapiens (human)Kd30.000011
Ephrin type-A receptor 4Homo sapiens (human)Kd30.000011
Ephrin type-A receptor 5Homo sapiens (human)Kd30.000011
Ephrin type-A receptor 7Homo sapiens (human)Kd30.000011
Ephrin type-B receptor 2Homo sapiens (human)Kd30.000011
Ephrin type-B receptor 3Homo sapiens (human)Kd30.000011
Ephrin type-B receptor 4Homo sapiens (human)Kd30.000011
Ephrin type-B receptor 6Homo sapiens (human)Kd30.000011
Epidermal growth factor receptorHomo sapiens (human)Kd30.000011
Epithelial discoidin domain-containing receptor 1Homo sapiens (human)Kd30.000011
Eukaryotic translation initiation factor 2-alpha kinase 1Homo sapiens (human)Kd30.000011
Eukaryotic translation initiation factor 5BHomo sapiens (human)Kd30.000011
Exosome RNA helicase MTR4Homo sapiens (human)Kd30.000011
Ferrochelatase, mitochondrialHomo sapiens (human)Kd30.000011
Fibroblast growth factor receptor 1Homo sapiens (human)Kd30.000011
Focal adhesion kinase 1Homo sapiens (human)Kd30.000011
General transcription and DNA repair factor IIH helicase subunit XPDHomo sapiens (human)Kd30.000011
Glycine--tRNA ligaseHomo sapiens (human)Kd30.000011
Glycogen phosphorylase, brain formHomo sapiens (human)Kd30.000011
Glycogen phosphorylase, liver formHomo sapiens (human)Kd30.000011
Glycogen synthase kinase-3 alphaHomo sapiens (human)Kd30.000011
Glycogen synthase kinase-3 betaHomo sapiens (human)Kd30.000011
GTP-binding nuclear protein RanHomo sapiens (human)Kd30.000011
Heme oxygenase 2Homo sapiens (human)Kd30.000011
Hepatocyte growth factor receptorHomo sapiens (human)Kd30.000011
High affinity nerve growth factor receptorHomo sapiens (human)Kd1.739011
Inhibitor of nuclear factor kappa-B kinase subunit epsilonHomo sapiens (human)Kd0.494011
Inosine-5'-monophosphate dehydrogenase 2Homo sapiens (human)Kd30.000011
Insulin receptorHomo sapiens (human)Kd30.000011
Insulin-like growth factor 1 receptorHomo sapiens (human)Kd30.000011
Integrin-linked protein kinaseHomo sapiens (human)Kd30.000011
Interleukin-1 receptor-associated kinase 1Homo sapiens (human)Kd30.000011
Interleukin-1 receptor-associated kinase 3Homo sapiens (human)Kd0.254011
Interleukin-1 receptor-associated kinase 4Homo sapiens (human)Kd0.009011
LIM domain kinase 1Homo sapiens (human)Kd30.000011
LIM domain kinase 2Homo sapiens (human)Kd30.000011
Long-chain-fatty-acid--CoA ligase 5Homo sapiens (human)Kd30.000011
Macrophage-stimulating protein receptorHomo sapiens (human)Kd30.000011
MAP kinase-activated protein kinase 2Homo sapiens (human)Kd30.000011
MAP kinase-activated protein kinase 3Homo sapiens (human)Kd30.000011
MAP kinase-activated protein kinase 5Homo sapiens (human)Kd30.000011
MAP/microtubule affinity-regulating kinase 3Homo sapiens (human)Kd0.384011
MAP/microtubule affinity-regulating kinase 4Homo sapiens (human)Kd0.028011
Maternal embryonic leucine zipper kinaseHomo sapiens (human)Kd0.083011
Membrane-associated progesterone receptor component 1Homo sapiens (human)Kd30.000011
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinaseHomo sapiens (human)Kd30.000011
MidasinHomo sapiens (human)Kd30.000011
Misshapen-like kinase 1Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 1Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 10Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 11Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 14Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 15Homo sapiens (human)Kd0.167011
Mitogen-activated protein kinase 3 Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 7Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 8Homo sapiens (human)Kd0.551011
Mitogen-activated protein kinase 9Homo sapiens (human)Kd0.986011
Mitogen-activated protein kinase kinase kinase 1Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 11Homo sapiens (human)Kd0.572011
Mitogen-activated protein kinase kinase kinase 2Homo sapiens (human)Kd4.118011
Mitogen-activated protein kinase kinase kinase 20Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 3Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 4Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 5Homo sapiens (human)Kd0.182011
Mitogen-activated protein kinase kinase kinase 6Homo sapiens (human)Kd0.335011
Mitogen-activated protein kinase kinase kinase kinase 1Homo sapiens (human)Kd0.452011
Mitogen-activated protein kinase kinase kinase kinase 2Homo sapiens (human)Kd0.131011
Mitogen-activated protein kinase kinase kinase kinase 3Homo sapiens (human)Kd2.374011
Mitogen-activated protein kinase kinase kinase kinase 4Homo sapiens (human)Kd0.019011
Mitogen-activated protein kinase kinase kinase kinase 5Homo sapiens (human)Kd0.193011
Mitotic checkpoint serine/threonine-protein kinase BUB1Homo sapiens (human)Kd30.000011
Multifunctional protein ADE2Homo sapiens (human)Kd30.000011
Myosin light chain kinase 3Homo sapiens (human)Kd0.098011
Myosin light chain kinase, smooth muscleHomo sapiens (human)Kd30.000011
Myosin-14Homo sapiens (human)Kd30.000011
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13Homo sapiens (human)Kd30.000011
Non-receptor tyrosine-protein kinase TNK1Homo sapiens (human)Kd0.287011
Non-receptor tyrosine-protein kinase TYK2Homo sapiens (human)Kd30.000011
NUAK family SNF1-like kinase 2Homo sapiens (human)Kd30.000011
Nucleolar GTP-binding protein 1Homo sapiens (human)Kd30.000011
Peroxisomal acyl-coenzyme A oxidase 1Homo sapiens (human)Kd30.000011
Peroxisomal acyl-coenzyme A oxidase 3Homo sapiens (human)Kd30.000011
Phenylalanine--tRNA ligase beta subunitHomo sapiens (human)Kd30.000011
Phosphatidylinositol 5-phosphate 4-kinase type-2 alphaHomo sapiens (human)Kd30.000011
Phosphatidylinositol 5-phosphate 4-kinase type-2 gammaHomo sapiens (human)Kd30.000011
Phosphorylase b kinase gamma catalytic chain, liver/testis isoformHomo sapiens (human)Kd3.263011
Platelet-derived growth factor receptor betaHomo sapiens (human)Kd1.006011
Probable ATP-dependent RNA helicase DDX6Homo sapiens (human)Kd30.000011
Protein kinase C alpha typeHomo sapiens (human)Kd2.280011
Protein kinase C beta typeHomo sapiens (human)Kd30.000011
Protein kinase C delta typeHomo sapiens (human)Kd30.000012
Protein kinase C iota typeHomo sapiens (human)Kd30.000011
Protein kinase C theta typeHomo sapiens (human)Kd30.000011
Protein kinase C zeta typeHomo sapiens (human)Kd30.000011
Protein-tyrosine kinase 2-betaHomo sapiens (human)Kd1.360011
Protein-tyrosine kinase 6Homo sapiens (human)Kd30.000011
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)Kd0.669011
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)Kd30.000011
Putative heat shock protein HSP 90-beta 2Homo sapiens (human)Kd30.000012
Pyridoxal kinaseHomo sapiens (human)Kd30.000011
Rab-like protein 3Homo sapiens (human)Kd30.000011
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)Kd30.000011
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)Kd30.000011
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)Kd30.000011
Ras-related protein Rab-10Homo sapiens (human)Kd30.000011
Ras-related protein Rab-27AHomo sapiens (human)Kd30.000011
Ras-related protein Rab-6AHomo sapiens (human)Kd30.000012
Receptor-interacting serine/threonine-protein kinase 2Homo sapiens (human)Kd0.526011
Receptor-interacting serine/threonine-protein kinase 3Homo sapiens (human)Kd30.000011
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)Kd0.227011
Rho-associated protein kinase 1Homo sapiens (human)Kd30.000011
Rho-associated protein kinase 2Homo sapiens (human)Kd30.000011
Ribosomal protein S6 kinase alpha-1Homo sapiens (human)Kd2.994011
Ribosomal protein S6 kinase alpha-3Homo sapiens (human)Kd2.990011
Ribosomal protein S6 kinase alpha-4Homo sapiens (human)Kd0.432011
Ribosomal protein S6 kinase alpha-5Homo sapiens (human)Kd14.659011
Ribosomal protein S6 kinase alpha-6Homo sapiens (human)Kd2.181011
Ribosomal protein S6 kinase beta-1Homo sapiens (human)Kd30.000011
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiens (human)Kd4.031011
RNA cytidine acetyltransferaseHomo sapiens (human)Kd30.000011
S-adenosylmethionine synthase isoform type-2Homo sapiens (human)Kd30.000011
Septin-9Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 10Homo sapiens (human)Kd0.481011
Serine/threonine-protein kinase 16Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 24Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 26Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 3Homo sapiens (human)Kd0.043011
Serine/threonine-protein kinase 38Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 38-likeHomo sapiens (human)Kd2.137011
Serine/threonine-protein kinase 4Homo sapiens (human)Kd0.029011
Serine/threonine-protein kinase A-RafHomo sapiens (human)Kd30.000012
Serine/threonine-protein kinase B-rafHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Chk1Homo sapiens (human)Kd0.122011
Serine/threonine-protein kinase D2Homo sapiens (human)Kd0.030011
Serine/threonine-protein kinase D3Homo sapiens (human)Kd0.038011
Serine/threonine-protein kinase ICKHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase LATS1Homo sapiens (human)Kd0.067011
Serine/threonine-protein kinase MARK2Homo sapiens (human)Kd0.704011
Serine/threonine-protein kinase MRCK alphaHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase MRCK betaHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase MRCK gammaHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase N1Homo sapiens (human)Kd0.264011
Serine/threonine-protein kinase N2Homo sapiens (human)Kd0.361011
Serine/threonine-protein kinase N3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Nek1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Nek2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Nek3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Nek7Homo sapiens (human)Kd0.003011
Serine/threonine-protein kinase Nek9Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase NLKHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase PAK 2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase PAK 4Homo sapiens (human)Kd0.344011
Serine/threonine-protein kinase PAK 6Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase pim-1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase pim-2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase PLK4Homo sapiens (human)Kd0.073011
Serine/threonine-protein kinase SIK2Homo sapiens (human)Kd0.058011
Serine/threonine-protein kinase SIK3Homo sapiens (human)Kd4.027011
Serine/threonine-protein kinase STK11Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase TAO1Homo sapiens (human)Kd18.757011
Serine/threonine-protein kinase TAO2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase TAO3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase TBK1Homo sapiens (human)Kd1.157011
Serine/threonine-protein kinase ULK1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase ULK3Homo sapiens (human)Kd0.107011
Serine/threonine-protein kinase/endoribonuclease IRE1Homo sapiens (human)Kd0.019011
Serine/threonine-protein kinase/endoribonuclease IRE2Homo sapiens (human)Kd0.908011
STE20-like serine/threonine-protein kinase Homo sapiens (human)Kd3.305011
STE20-related kinase adapter protein alphaHomo sapiens (human)Kd30.000011
Structural maintenance of chromosomes protein 1AHomo sapiens (human)Kd30.000011
Structural maintenance of chromosomes protein 2Homo sapiens (human)Kd30.000011
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrialHomo sapiens (human)Kd30.000011
TGF-beta receptor type-1Homo sapiens (human)Kd2.179011
TGF-beta receptor type-2Homo sapiens (human)Kd30.000011
Thyroid hormone receptor-associated protein 3Homo sapiens (human)Kd30.000011
TRAF2 and NCK-interacting protein kinaseHomo sapiens (human)Kd0.010011
Tyrosine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase ABL1Homo sapiens (human)Kd30.000011
Tyrosine-protein kinase ABL2Homo sapiens (human)Kd30.000011
Tyrosine-protein kinase BTKHomo sapiens (human)Kd1.567011
Tyrosine-protein kinase CSKHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase FerHomo sapiens (human)Kd0.455011
Tyrosine-protein kinase Fes/FpsHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase FRKHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase FynHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase HCKHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase JAK1Homo sapiens (human)Kd30.000011
Tyrosine-protein kinase LckHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase LynHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase MerHomo sapiens (human)Kd0.041011
Tyrosine-protein kinase SYKHomo sapiens (human)Kd0.545011
Tyrosine-protein kinase TecHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase YesHomo sapiens (human)Kd30.000011
U5 small nuclear ribonucleoprotein 200 kDa helicaseHomo sapiens (human)Kd30.000011
Uncharacterized aarF domain-containing protein kinase 5Homo sapiens (human)Kd30.000011
Uncharacterized protein FLJ45252Homo sapiens (human)Kd0.021011
Very long-chain specific acyl-CoA dehydrogenase, mitochondrialHomo sapiens (human)Kd30.000011
Wee1-like protein kinaseHomo sapiens (human)Kd30.000011