Page last updated: 2024-08-05 15:48:20

ryanodine receptor modulator

null

ChEBI ID: 38809

Members (1)

MemberDefinitionClass
flubendiamideflubendiamide

Research

Studies (97)

TimeframeStudies, Drugs with This Role(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's10 (10.31)29.6817
2010's66 (68.04)24.3611
2020's21 (21.65)2.80

Study Types

Publication TypeStudies, Drugs with this Role (%)All Drugs (%)
Trials0 (0.00%)5.53%
Reviews2 (2.02%)6.00%
Case Studies0 (0.00%)4.05%
Observational0 (0.00%)0.25%
Other97 (97.98%)84.16%

Protein Targets (15)

Potency Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
AR proteinHomo sapiens (human)Potency13.133322
Cellular tumor antigen p53Homo sapiens (human)Potency48.849311
estrogen nuclear receptor alphaHomo sapiens (human)Potency19.160222
estrogen-related nuclear receptor alphaHomo sapiens (human)Potency34.481366
farnesoid X nuclear receptorHomo sapiens (human)Potency36.953511
GLI family zinc finger 3Homo sapiens (human)Potency6.106533
heat shock protein beta-1Homo sapiens (human)Potency43.919322
nuclear factor erythroid 2-related factor 2 isoform 1Homo sapiens (human)Potency38.802322
nuclear receptor subfamily 1, group I, member 3Homo sapiens (human)Potency10.936011
peroxisome proliferator-activated receptor deltaHomo sapiens (human)Potency40.674511
pregnane X nuclear receptorHomo sapiens (human)Potency13.767611
RAR-related orphan receptor gammaMus musculus (house mouse)Potency41.953822
thyroid hormone receptor beta isoform 2Rattus norvegicus (Norway rat)Potency16.575233
v-jun sarcoma virus 17 oncogene homolog (avian)Homo sapiens (human)Potency34.886311
vitamin D (1,25- dihydroxyvitamin D3) receptorHomo sapiens (human)Potency41.531222