Page last updated: 2024-08-05 14:59:18

fibroblast growth factor receptor antagonist

An antagonist at the fibroblast growth factor receptor.

ChEBI ID: 63457

Members (8)

MemberDefinitionClass
3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-(4-(4-ethylpiperazin-1-yl)-phenylamino)pyrimidin-4-yl)-1-methylureaA member of the class of phenylureas that is urea in which a hydrogen attached to one of the nitrogens is replaced by a 2,6-dichloro-3,5-dimethoxyphenyl group, while the hydrogens attached to the other nitrogen are replaced by a methyl group and a 6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl group. It is a potent and selective fibroblast growth factor receptor inhibitor.BGJ-398
azd4547A member of the class of benzamides that is a carboxamide resulting from the formal condensation of the carboxy group of 4-(cis-3,5-dimethylpiperazin-1-yl)benzoic acid with the amino substituent of 5-[2-(3,5-dimethoxyphenyl)ethyl]-1H-pyrazol-3-amine. It is an inhibitor of the fibroblast growth factor receptor (FGFR).AZD4547
brivanibA secondary alcohol resulting from the hydrolysis of the carboxylic ester group of brivanib alaninate. It is a dual VEGFR-2/FGFR-1 kinase inhibitor whose alanine prodrug, brivanib alaninate is currently under development as an oral agent for the treatment of cancer.(2R)-1-[[4-[(4-fluoro-2-methyl-1H-indol-5-yl)oxy]-5-methyl-6-pyrrolo[2,1-f][1,2,4]triazinyl]oxy]-2-propanol; brivanib
lenvatinibA member of the class of quinolines that is the carboxamide of 4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxylic acid. A multi-kinase inhibitor and orphan drug used (as its mesylate salt) for the treatment of various types of thyroid cancer that do not respond to radioiodine.lenvatinib
lucitanibA naphthalenecarboxamide obtained from formal condensation of the carboxy group of aminocyclopropyl)methoxy]-6-methoxyquinolin-4-yl}oxy)-1-naphthoic acid with methylamine.E-3810 free base
pd 173074A member of the class of ureas that is 1-tert-butylurea in which one of the hydrogens attached to N(3) is substituted by a pyrido[2,3-d]pyrimidin-7-yl group, which is itself substituted at positions 2 and 6 by a 4-(diethylamino)butyl]amino group and a 3,5-dimethoxyphenyl group, respectively. It is a FGF/VEGF receptor tyrosine kinase inhibitor.PD173074
ssr128129eAn organic sodium salt having 2-amino-5-[(1-methoxy-2-methylindolizin-3-yl)carbonyl]benzoate as the counterion.sodium 2-amino-5-[(1-methoxy-2-methylindolizin-3-yl)carbonyl]benzoate
SU5402An oxindole that is 3-methyleneoxindole in which one of the hydrogens of the methylene group is substituted by a 3-(2-carboxyethyl)-4-methyl-1H-pyrrol-2-yl group. It is an ATP-competitive inhibitor of the tyrosine kinase activity of fibroblast growth factor receptor 1.SU5402

Research

Studies (1,397)

TimeframeStudies, Drugs with This Role(%)All Drugs %
pre-19900 (0.00)18.7374
1990's3 (0.21)18.2507
2000's52 (3.72)29.6817
2010's576 (41.23)24.3611
2020's766 (54.83)2.80

Study Types

Publication TypeStudies, Drugs with this Role (%)All Drugs (%)
Trials147 (9.77%)5.53%
Reviews196 (13.03%)6.00%
Case Studies149 (9.91%)4.05%
Observational18 (1.20%)0.25%
Other994 (66.09%)84.16%

Protein Targets (539)

Potency Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
67.9K proteinVaccinia virusPotency12.672822
alpha-galactosidaseHomo sapiens (human)Potency31.622811
ATAD5 protein, partialHomo sapiens (human)Potency29.081011
Chain A, Beta-lactamaseEscherichia coli K-12Potency19.952611
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASEHomo sapiens (human)Potency0.794311
cytochrome P450 2C9, partialHomo sapiens (human)Potency14.490013
cytochrome P450 2D6Homo sapiens (human)Potency23.918511
cytochrome P450 family 3 subfamily A polypeptide 4Homo sapiens (human)Potency9.564213
DNA polymerase kappa isoform 1Homo sapiens (human)Potency15.003011
EWS/FLI fusion proteinHomo sapiens (human)Potency17.2315421
Fumarate hydrataseHomo sapiens (human)Potency28.149614
GVesicular stomatitis virusPotency14.490013
gemininHomo sapiens (human)Potency8.083022
glp-1 receptor, partialHomo sapiens (human)Potency4.466811
glucocerebrosidaseHomo sapiens (human)Potency25.285512
histone-lysine N-methyltransferase 2A isoform 2 precursorHomo sapiens (human)Potency44.668411
HLA class I histocompatibility antigen, B alpha chain Homo sapiens (human)Potency14.490013
IDH1Homo sapiens (human)Potency16.360111
Inositol hexakisphosphate kinase 1Homo sapiens (human)Potency14.490016
Interferon betaHomo sapiens (human)Potency21.5266218
nuclear factor erythroid 2-related factor 2 isoform 2Homo sapiens (human)Potency23.109311
nuclear receptor ROR-gamma isoform 1Mus musculus (house mouse)Potency35.481311
plasminogen precursorMus musculus (house mouse)Potency7.079511
polyproteinZika virusPotency28.149614
PPM1D proteinHomo sapiens (human)Potency22.9339110
serine-protein kinase ATM isoform aHomo sapiens (human)Potency39.810711
Smad3Homo sapiens (human)Potency22.387211
Spike glycoproteinSevere acute respiratory syndrome-related coronavirusPotency4.477222
TDP1 proteinHomo sapiens (human)Potency29.092922
tyrosine-protein kinase YesHomo sapiens (human)Potency4.967413
urokinase plasminogen activator surface receptor precursorMus musculus (house mouse)Potency7.079511
urokinase-type plasminogen activator precursorMus musculus (house mouse)Potency7.079511

Inhibition Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
Carbonic anhydrase 1Homo sapiens (human)Ki10.000011
Carbonic anhydrase 2Homo sapiens (human)Ki10.000011
Carbonic anhydrase 5A, mitochondrialHomo sapiens (human)Ki0.132711
Chain A, Protein (fibroblast Growth Factor (fgf) Receptor 1)Homo sapiens (human)Ki0.045211
Coiled-coil domain-containing protein 6Homo sapiens (human)IC500.010011
Cytochrome P450 1A2Homo sapiens (human)IC5040.000011
Cytochrome P450 2C19Homo sapiens (human)IC5040.000011
Cytochrome P450 2C9 Homo sapiens (human)IC5040.000011
Cytochrome P450 2D6Homo sapiens (human)IC5040.000011
Cytochrome P450 3A4Homo sapiens (human)IC5019.007044
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)IC5050.000011
Epidermal growth factor receptorHomo sapiens (human)IC5025.950022
Fibroblast growth factor receptor 1Homo sapiens (human)IC501.00814548
Fibroblast growth factor receptor 2Homo sapiens (human)IC500.46172729
Fibroblast growth factor receptor 3Homo sapiens (human)IC500.53032627
Fibroblast growth factor receptor 4Homo sapiens (human)IC500.72282328
Fibroblast growth factor receptor 4Mus musculus (house mouse)IC500.497224
Gastrin/cholecystokinin type B receptorRattus norvegicus (Norway rat)IC5050.000011
Insulin receptorHomo sapiens (human)IC5050.000022
Kinesin-1 heavy chainHomo sapiens (human)IC500.010011
Nuclear receptor coactivator 4Homo sapiens (human)IC500.010011
Platelet-derived growth factor receptor alphaHomo sapiens (human)IC500.051011
Platelet-derived growth factor receptor alphaRattus norvegicus (Norway rat)IC5017.000011
Platelet-derived growth factor receptor betaHomo sapiens (human)IC503.019522
Platelet-derived growth factor receptor betaMus musculus (house mouse)IC5012.007024
Platelet-derived growth factor receptor betaRattus norvegicus (Norway rat)IC5017.000011
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)IC5018.000011
Protein kinase C alpha typeHomo sapiens (human)IC5025.000011
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)IC500.016244
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)Ki0.001511
Proto-oncogene tyrosine-protein kinase SrcGallus gallus (chicken)IC5020.000011
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)IC5013.507024
Serine-protein kinase ATMHomo sapiens (human)IC5017.600011
Smoothened homologHomo sapiens (human)Ki0.046511
Tyrosine-protein kinase CSKHomo sapiens (human)IC5019.800011
Tyrosine-protein kinase JAK3Homo sapiens (human)IC5050.000011
Tyrosine-protein kinase LckHomo sapiens (human)IC502.500011
Vascular endothelial growth factor receptor 1 Homo sapiens (human)IC500.082178
Vascular endothelial growth factor receptor 1 Homo sapiens (human)Ki0.060011
Vascular endothelial growth factor receptor 2Homo sapiens (human)IC500.04012324
Vascular endothelial growth factor receptor 2Mus musculus (house mouse)IC500.089011
Vascular endothelial growth factor receptor 2Homo sapiens (human)Ki0.026011
Vascular endothelial growth factor receptor 2Mus musculus (house mouse)Ki0.028011
Vascular endothelial growth factor receptor 3Homo sapiens (human)IC500.033067

Activation Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
26S proteasome regulatory subunit 6BHomo sapiens (human)Kd30.000013
3-phosphoinositide-dependent protein kinase 1Homo sapiens (human)Kd10.000011
5'-AMP-activated protein kinase catalytic subunit alpha-1Homo sapiens (human)Kd25.000024
5'-AMP-activated protein kinase catalytic subunit alpha-2Homo sapiens (human)Kd10.000011
5'-AMP-activated protein kinase subunit gamma-1Homo sapiens (human)Kd30.000013
5'-AMP-activated protein kinase subunit gamma-2Homo sapiens (human)Kd30.000013
AarF domain-containing protein kinase 1Homo sapiens (human)Kd30.000013
Actin-related protein 2Homo sapiens (human)Kd30.000013
Actin-related protein 3Homo sapiens (human)Kd30.000013
Activated CDC42 kinase 1Homo sapiens (human)Kd25.000024
Activin receptor type-1Homo sapiens (human)Kd25.000024
Activin receptor type-1BHomo sapiens (human)Kd25.000024
Activin receptor type-2AHomo sapiens (human)Kd10.000011
Activin receptor type-2BHomo sapiens (human)Kd25.000024
Acyl-CoA dehydrogenase family member 10Homo sapiens (human)Kd30.000013
Acyl-CoA dehydrogenase family member 11Homo sapiens (human)Kd30.000013
Adenine phosphoribosyltransferaseHomo sapiens (human)Kd30.000014
Adenosine kinaseHomo sapiens (human)Kd30.000013
Adenylate kinase 2, mitochondrialHomo sapiens (human)Kd30.000013
ADP/ATP translocase 2Homo sapiens (human)Kd30.000013
ADP/ATP translocase 3Homo sapiens (human)Kd30.000013
ALK tyrosine kinase receptorHomo sapiens (human)Kd10.000011
Angiopoietin-1 receptorHomo sapiens (human)Kd0.440011
Ankyrin repeat and protein kinase domain-containing protein 1Homo sapiens (human)Kd10.000011
AP2-associated protein kinase 1Homo sapiens (human)Kd25.000024
ATP-dependent 6-phosphofructokinase, platelet typeHomo sapiens (human)Kd30.000012
ATP-dependent RNA helicase DDX1Homo sapiens (human)Kd30.000013
ATP-dependent RNA helicase DDX3XHomo sapiens (human)Kd30.000014
ATP-dependent RNA helicase DDX42Homo sapiens (human)Kd30.000013
ATP-dependent RNA helicase DHX30Homo sapiens (human)Kd30.000012
Atypical kinase COQ8A, mitochondrialHomo sapiens (human)Kd25.000024
Atypical kinase COQ8B, mitochondrialHomo sapiens (human)Kd10.000011
Aurora kinase AHomo sapiens (human)Kd20.076235
Aurora kinase BHomo sapiens (human)Kd16.158224
Aurora kinase CHomo sapiens (human)Kd10.000011
BDNF/NT-3 growth factors receptorHomo sapiens (human)Kd10.000011
Beta-adrenergic receptor kinase 1Homo sapiens (human)Kd30.000013
BMP-2-inducible protein kinaseHomo sapiens (human)Kd25.000024
Bone morphogenetic protein receptor type-1AHomo sapiens (human)Kd25.000024
Bone morphogenetic protein receptor type-1BHomo sapiens (human)Kd25.000024
Bone morphogenetic protein receptor type-2Homo sapiens (human)Kd25.000024
Breakpoint cluster region proteinHomo sapiens (human)Kd23.528214
Calcium-dependent protein kinase 1Plasmodium falciparum 3D7Kd10.000011
Calcium/calmodulin-dependent protein kinase kinase 1Homo sapiens (human)Kd10.000011
Calcium/calmodulin-dependent protein kinase kinase 2Homo sapiens (human)Kd25.000024
Calcium/calmodulin-dependent protein kinase type 1Homo sapiens (human)Kd10.000011
Calcium/calmodulin-dependent protein kinase type 1DHomo sapiens (human)Kd10.000011
Calcium/calmodulin-dependent protein kinase type 1GHomo sapiens (human)Kd10.000011
Calcium/calmodulin-dependent protein kinase type II subunit alphaHomo sapiens (human)Kd10.000011
Calcium/calmodulin-dependent protein kinase type II subunit betaHomo sapiens (human)Kd10.000011
Calcium/calmodulin-dependent protein kinase type II subunit deltaHomo sapiens (human)Kd25.000024
Calcium/calmodulin-dependent protein kinase type II subunit gammaHomo sapiens (human)Kd25.000024
Calcium/calmodulin-dependent protein kinase type IVHomo sapiens (human)Kd25.000024
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)Kd25.000024
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)Kd25.000024
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)Kd30.000013
cAMP-dependent protein kinase catalytic subunit PRKXHomo sapiens (human)Kd10.000011
cAMP-dependent protein kinase type II-alpha regulatory subunitHomo sapiens (human)Kd30.000013
Casein kinase I isoform alphaHomo sapiens (human)Kd25.000024
Casein kinase I isoform alpha-likeHomo sapiens (human)Kd10.000011
Casein kinase I isoform deltaHomo sapiens (human)Kd25.000024
Casein kinase I isoform epsilonHomo sapiens (human)Kd25.000024
Casein kinase I isoform gamma-1Homo sapiens (human)Kd25.000024
Casein kinase I isoform gamma-2Homo sapiens (human)Kd23.333323
Casein kinase I isoform gamma-3Homo sapiens (human)Kd25.000024
Casein kinase II subunit alphaHomo sapiens (human)Kd10.000011
Casein kinase II subunit alpha'Homo sapiens (human)Kd25.000024
Cell division control protein 2 homologPlasmodium falciparum 3D7Kd10.000011
Cell division cycle 7-related protein kinaseHomo sapiens (human)Kd30.000011
cGMP-dependent protein kinase 1 Homo sapiens (human)Kd25.000024
cGMP-dependent protein kinase 2Homo sapiens (human)Kd10.000011
Choline-phosphate cytidylyltransferase AHomo sapiens (human)Kd30.000011
Chromodomain-helicase-DNA-binding protein 4Homo sapiens (human)Kd30.000013
Citron Rho-interacting kinaseHomo sapiens (human)Kd25.000024
Cyclin-dependent kinase 1Homo sapiens (human)Kd30.000013
Cyclin-dependent kinase 11AHomo sapiens (human)Kd10.000011
Cyclin-dependent kinase 11BHomo sapiens (human)Kd10.000011
Cyclin-dependent kinase 12Homo sapiens (human)Kd30.000013
Cyclin-dependent kinase 13Homo sapiens (human)Kd25.000024
Cyclin-dependent kinase 14Homo sapiens (human)Kd10.000011
Cyclin-dependent kinase 15Homo sapiens (human)Kd10.000011
Cyclin-dependent kinase 16Homo sapiens (human)Kd25.000024
Cyclin-dependent kinase 17Homo sapiens (human)Kd25.000024
Cyclin-dependent kinase 18Homo sapiens (human)Kd10.000011
Cyclin-dependent kinase 19Homo sapiens (human)Kd10.000011
Cyclin-dependent kinase 2Homo sapiens (human)Kd25.000024
Cyclin-dependent kinase 3Homo sapiens (human)Kd23.333323
Cyclin-dependent kinase 4Homo sapiens (human)Kd22.000035
Cyclin-dependent kinase 6Homo sapiens (human)Kd30.000013
Cyclin-dependent kinase 7Homo sapiens (human)Kd25.000024
Cyclin-dependent kinase 8Homo sapiens (human)Kd10.000011
Cyclin-dependent kinase 9Homo sapiens (human)Kd25.000024
Cyclin-dependent kinase-like 1Homo sapiens (human)Kd10.000011
Cyclin-dependent kinase-like 2Homo sapiens (human)Kd10.000011
Cyclin-dependent kinase-like 3Homo sapiens (human)Kd10.000011
Cyclin-dependent kinase-like 5Homo sapiens (human)Kd23.333323
Cyclin-dependent-like kinase 5 Homo sapiens (human)Kd25.000024
Cyclin-G-associated kinaseHomo sapiens (human)Kd25.000024
Cysteine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000013
Cytochrome c1, heme protein, mitochondrialHomo sapiens (human)Kd30.000015
Cytoplasmic tyrosine-protein kinase BMXHomo sapiens (human)Kd10.000011
dCTP pyrophosphatase 1Homo sapiens (human)Kd30.000013
Death-associated protein kinase 1Homo sapiens (human)Kd10.000011
Death-associated protein kinase 2Homo sapiens (human)Kd10.000011
Death-associated protein kinase 3Homo sapiens (human)Kd10.000011
Delta(24)-sterol reductaseHomo sapiens (human)Kd30.000013
Deoxycytidine kinaseHomo sapiens (human)Kd30.000013
Discoidin domain-containing receptor 2Homo sapiens (human)Kd10.078024
DNA replication licensing factor MCM4Homo sapiens (human)Kd30.000013
DNA topoisomerase 2-alphaHomo sapiens (human)Kd30.000012
DNA topoisomerase 2-betaHomo sapiens (human)Kd30.000013
DnaJ homolog subfamily A member 1Homo sapiens (human)Kd30.000013
Dual serine/threonine and tyrosine protein kinaseHomo sapiens (human)Kd10.000011
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)Kd25.000024
Dual specificity mitogen-activated protein kinase kinase 2Homo sapiens (human)Kd26.000025
Dual specificity mitogen-activated protein kinase kinase 3Homo sapiens (human)Kd25.000024
Dual specificity mitogen-activated protein kinase kinase 4Homo sapiens (human)Kd10.000011
Dual specificity mitogen-activated protein kinase kinase 5Homo sapiens (human)Kd16.502524
Dual specificity mitogen-activated protein kinase kinase 6Homo sapiens (human)Kd25.000024
Dual specificity mitogen-activated protein kinase kinase 7Homo sapiens (human)Kd10.000011
Dual specificity protein kinase CLK1Homo sapiens (human)Kd25.000024
Dual specificity protein kinase CLK2Homo sapiens (human)Kd26.000025
Dual specificity protein kinase CLK3Homo sapiens (human)Kd23.333323
Dual specificity protein kinase CLK4Homo sapiens (human)Kd23.333323
Dual specificity protein kinase TTKHomo sapiens (human)Kd23.333323
Dual specificity testis-specific protein kinase 1Homo sapiens (human)Kd25.000024
Dual specificity tyrosine-phosphorylation-regulated kinase 1AHomo sapiens (human)Kd25.000024
Dual specificity tyrosine-phosphorylation-regulated kinase 1BHomo sapiens (human)Kd20.000022
Dual specificity tyrosine-phosphorylation-regulated kinase 2Homo sapiens (human)Kd10.000011
Dynamin-like 120 kDa protein, mitochondrialHomo sapiens (human)Kd30.000013
eIF-2-alpha kinase GCN2Homo sapiens (human)Kd10.000011
EKC/KEOPS complex subunit TP53RKHomo sapiens (human)Kd30.000013
Electron transfer flavoprotein subunit betaHomo sapiens (human)Kd30.000014
Elongation factor Tu, mitochondrialHomo sapiens (human)Kd30.000013
Ephrin type-A receptor 1Homo sapiens (human)Kd23.333323
Ephrin type-A receptor 2Homo sapiens (human)Kd25.000024
Ephrin type-A receptor 3Homo sapiens (human)Kd10.000011
Ephrin type-A receptor 4Homo sapiens (human)Kd25.000024
Ephrin type-A receptor 5Homo sapiens (human)Kd25.000024
Ephrin type-A receptor 6Homo sapiens (human)Kd0.190011
Ephrin type-A receptor 7Homo sapiens (human)Kd20.566723
Ephrin type-A receptor 8Homo sapiens (human)Kd10.000011
Ephrin type-B receptor 1Homo sapiens (human)Kd10.000011
Ephrin type-B receptor 2Homo sapiens (human)Kd25.000024
Ephrin type-B receptor 3Homo sapiens (human)Kd25.000024
Ephrin type-B receptor 4Homo sapiens (human)Kd25.000024
Ephrin type-B receptor 6Homo sapiens (human)Kd22.850024
Epidermal growth factor receptorHomo sapiens (human)Kd12.40001315
Epithelial discoidin domain-containing receptor 1Homo sapiens (human)Kd0.309724
Eukaryotic translation initiation factor 2-alpha kinase 1Homo sapiens (human)Kd25.000024
Eukaryotic translation initiation factor 5BHomo sapiens (human)Kd30.000013
Exosome RNA helicase MTR4Homo sapiens (human)Kd30.000013
Ferrochelatase, mitochondrialHomo sapiens (human)Kd16.476524
Fibroblast growth factor receptor 1Homo sapiens (human)EC500.021011
Fibroblast growth factor receptor 1Homo sapiens (human)Kd22.524824
Fibroblast growth factor receptor 2Homo sapiens (human)Kd0.110011
Fibroblast growth factor receptor 3Homo sapiens (human)EC500.030011
Fibroblast growth factor receptor 3Homo sapiens (human)Kd0.155022
Fibroblast growth factor receptor 4Homo sapiens (human)Kd0.600011
Focal adhesion kinase 1Homo sapiens (human)Kd25.000024
G protein-coupled receptor kinase 4Homo sapiens (human)Kd10.000011
G protein-coupled receptor kinase 6Homo sapiens (human)Kd30.000013
General transcription and DNA repair factor IIH helicase subunit XPDHomo sapiens (human)Kd30.000013
Glycine--tRNA ligaseHomo sapiens (human)Kd30.000014
Glycogen phosphorylase, brain formHomo sapiens (human)Kd30.000014
Glycogen phosphorylase, liver formHomo sapiens (human)Kd30.000013
Glycogen synthase kinase-3 alphaHomo sapiens (human)Kd25.000024
Glycogen synthase kinase-3 betaHomo sapiens (human)Kd25.000024
GTP-binding nuclear protein RanHomo sapiens (human)Kd30.000013
Guanine nucleotide-binding protein G(i) subunit alpha-2Homo sapiens (human)Kd30.000013
Heme oxygenase 2Homo sapiens (human)Kd30.000013
Hepatocyte growth factor receptorHomo sapiens (human)Kd20.000046
High affinity nerve growth factor receptorHomo sapiens (human)Kd23.333323
Homeodomain-interacting protein kinase 1Homo sapiens (human)Kd10.000011
Homeodomain-interacting protein kinase 2Homo sapiens (human)Kd10.000011
Homeodomain-interacting protein kinase 3Homo sapiens (human)Kd10.000011
Homeodomain-interacting protein kinase 4Homo sapiens (human)Kd10.000011
Hormonally up-regulated neu tumor-associated kinaseHomo sapiens (human)Kd10.000011
Inhibitor of nuclear factor kappa-B kinase subunit alphaHomo sapiens (human)Kd10.000011
Inhibitor of nuclear factor kappa-B kinase subunit betaHomo sapiens (human)Kd10.000011
Inhibitor of nuclear factor kappa-B kinase subunit epsilonHomo sapiens (human)Kd25.000024
Inosine-5'-monophosphate dehydrogenase 2Homo sapiens (human)Kd30.000013
Insulin receptorHomo sapiens (human)Kd26.666726
Insulin receptor-related proteinHomo sapiens (human)Kd10.000011
Insulin-like growth factor 1 receptorHomo sapiens (human)Kd25.000024
Integrin-linked protein kinaseHomo sapiens (human)Kd30.000013
Interferon-induced, double-stranded RNA-activated protein kinaseHomo sapiens (human)Kd10.000011
Interleukin-1 receptor-associated kinase 1Homo sapiens (human)Kd26.000025
Interleukin-1 receptor-associated kinase 3Homo sapiens (human)Kd25.000024
Interleukin-1 receptor-associated kinase 4Homo sapiens (human)Kd25.000024
Isoleucine--tRNA ligase, mitochondrialHomo sapiens (human)Kd30.000013
Leucine-rich repeat serine/threonine-protein kinase 2Homo sapiens (human)Kd10.000022
Leukocyte tyrosine kinase receptorHomo sapiens (human)Kd10.000011
Leukotriene C4 synthaseCavia porcellus (domestic guinea pig)Kd10.000011
LIM domain kinase 1Homo sapiens (human)Kd25.000024
LIM domain kinase 2Homo sapiens (human)Kd25.000024
Long-chain-fatty-acid--CoA ligase 5Homo sapiens (human)Kd30.000012
Macrophage colony-stimulating factor 1 receptorHomo sapiens (human)Kd1.900011
Macrophage-stimulating protein receptorHomo sapiens (human)Kd25.000024
MAP kinase-activated protein kinase 2Homo sapiens (human)Kd17.515824
MAP kinase-activated protein kinase 3Homo sapiens (human)Kd30.000011
MAP kinase-activated protein kinase 5Homo sapiens (human)Kd25.000024
MAP kinase-interacting serine/threonine-protein kinase 1Homo sapiens (human)Kd10.000011
MAP kinase-interacting serine/threonine-protein kinase 2Homo sapiens (human)Kd10.000011
MAP/microtubule affinity-regulating kinase 3Homo sapiens (human)Kd25.000024
MAP/microtubule affinity-regulating kinase 4Homo sapiens (human)Kd25.000024
Mast/stem cell growth factor receptor KitHomo sapiens (human)Kd3.019288
Maternal embryonic leucine zipper kinaseHomo sapiens (human)Kd25.000024
Megakaryocyte-associated tyrosine-protein kinaseHomo sapiens (human)Kd10.000011
Membrane-associated progesterone receptor component 1Homo sapiens (human)Kd30.000012
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinaseHomo sapiens (human)Kd26.000025
Microtubule-associated serine/threonine-protein kinase 1Homo sapiens (human)Kd10.000011
MidasinHomo sapiens (human)Kd30.000013
Misshapen-like kinase 1Homo sapiens (human)Kd20.103323
Mitogen-activated protein kinase 1Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase 10Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase 11Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase 12Homo sapiens (human)Kd10.000011
Mitogen-activated protein kinase 13Homo sapiens (human)Kd10.000011
Mitogen-activated protein kinase 14Homo sapiens (human)Kd17.554224
Mitogen-activated protein kinase 15Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase 3 Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase 4Homo sapiens (human)Kd10.000011
Mitogen-activated protein kinase 6Homo sapiens (human)Kd10.000011
Mitogen-activated protein kinase 7Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase 8Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase 9Homo sapiens (human)Kd26.000025
Mitogen-activated protein kinase kinase kinase 1Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase kinase kinase 10Homo sapiens (human)Kd10.000011
Mitogen-activated protein kinase kinase kinase 11Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase kinase kinase 12Homo sapiens (human)Kd10.000011
Mitogen-activated protein kinase kinase kinase 13Homo sapiens (human)Kd10.000011
Mitogen-activated protein kinase kinase kinase 15Homo sapiens (human)Kd10.000011
Mitogen-activated protein kinase kinase kinase 19Homo sapiens (human)Kd0.500011
Mitogen-activated protein kinase kinase kinase 2Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase kinase kinase 20Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase kinase kinase 3Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase kinase kinase 4Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase kinase kinase 5Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase kinase kinase 6Homo sapiens (human)Kd17.893824
Mitogen-activated protein kinase kinase kinase 7Homo sapiens (human)Kd10.000011
Mitogen-activated protein kinase kinase kinase 9Homo sapiens (human)Kd10.000011
Mitogen-activated protein kinase kinase kinase kinase 1Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase kinase kinase kinase 2Homo sapiens (human)Kd20.115625
Mitogen-activated protein kinase kinase kinase kinase 3Homo sapiens (human)Kd25.000024
Mitogen-activated protein kinase kinase kinase kinase 4Homo sapiens (human)Kd20.836824
Mitogen-activated protein kinase kinase kinase kinase 5Homo sapiens (human)Kd18.903425
Mitotic checkpoint serine/threonine-protein kinase BUB1Homo sapiens (human)Kd30.000013
Multifunctional protein ADE2Homo sapiens (human)Kd30.000013
Muscle, skeletal receptor tyrosine-protein kinaseHomo sapiens (human)Kd10.000011
Myosin light chain kinase 2, skeletal/cardiac muscleHomo sapiens (human)Kd10.000011
Myosin light chain kinase 3Homo sapiens (human)Kd26.000025
Myosin light chain kinase family member 4Homo sapiens (human)Kd10.000011
Myosin light chain kinase, smooth muscleHomo sapiens (human)Kd23.333323
Myosin-10Homo sapiens (human)Kd30.000013
Myosin-14Homo sapiens (human)Kd30.000015
Myosin-IIIaHomo sapiens (human)Kd10.000011
Myosin-IIIbHomo sapiens (human)Kd10.000011
Myotonin-protein kinaseHomo sapiens (human)Kd10.000011
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13Homo sapiens (human)Kd30.000013
Non-receptor tyrosine-protein kinase TNK1Homo sapiens (human)Kd25.000024
Non-receptor tyrosine-protein kinase TYK2Homo sapiens (human)Kd22.000035
NT-3 growth factor receptorHomo sapiens (human)Kd10.000011
NUAK family SNF1-like kinase 1Homo sapiens (human)Kd10.000011
NUAK family SNF1-like kinase 2Homo sapiens (human)Kd25.000024
Nucleolar GTP-binding protein 1Homo sapiens (human)Kd30.000013
Obg-like ATPase 1Homo sapiens (human)Kd30.000013
PAS domain-containing serine/threonine-protein kinaseHomo sapiens (human)Kd30.000012
Peripheral plasma membrane protein CASKHomo sapiens (human)Kd10.000011
Peroxisomal acyl-coenzyme A oxidase 1Homo sapiens (human)Kd30.000013
Peroxisomal acyl-coenzyme A oxidase 3Homo sapiens (human)Kd30.000013
Phenylalanine--tRNA ligase beta subunitHomo sapiens (human)Kd30.000013
Phosphatidylethanolamine-binding protein 1Homo sapiens (human)Kd30.000013
Phosphatidylinositol 4-kinase betaHomo sapiens (human)Kd10.000011
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit betaHomo sapiens (human)Kd10.000011
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gammaHomo sapiens (human)Kd10.000011
Phosphatidylinositol 4-phosphate 5-kinase type-1 alphaHomo sapiens (human)Kd10.000011
Phosphatidylinositol 4-phosphate 5-kinase type-1 gammaHomo sapiens (human)Kd10.000011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformHomo sapiens (human)Kd10.00001010
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformHomo sapiens (human)Kd10.000011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformHomo sapiens (human)Kd10.000011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)Kd10.000011
Phosphatidylinositol 5-phosphate 4-kinase type-2 alphaHomo sapiens (human)Kd30.000013
Phosphatidylinositol 5-phosphate 4-kinase type-2 betaHomo sapiens (human)Kd10.000011
Phosphatidylinositol 5-phosphate 4-kinase type-2 gammaHomo sapiens (human)Kd25.000024
Phosphorylase b kinase gamma catalytic chain, liver/testis isoformHomo sapiens (human)Kd25.000024
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoformHomo sapiens (human)Kd10.000011
Platelet-derived growth factor receptor alphaHomo sapiens (human)Kd0.011011
Platelet-derived growth factor receptor betaHomo sapiens (human)Kd0.795224
Probable ATP-dependent RNA helicase DDX6Homo sapiens (human)Kd30.000013
Prostaglandin G/H synthase 2Homo sapiens (human)Kd10.000011
Protein kinase C alpha typeHomo sapiens (human)Kd30.000013
Protein kinase C beta typeHomo sapiens (human)Kd30.000013
Protein kinase C delta typeHomo sapiens (human)Kd26.000025
Protein kinase C epsilon typeHomo sapiens (human)Kd10.000011
Protein kinase C eta typeHomo sapiens (human)Kd10.000011
Protein kinase C iota typeHomo sapiens (human)Kd25.000024
Protein kinase C theta typeHomo sapiens (human)Kd25.000024
Protein kinase C zeta typeHomo sapiens (human)Kd30.000011
Protein-tyrosine kinase 2-betaHomo sapiens (human)Kd25.000024
Protein-tyrosine kinase 6Homo sapiens (human)Kd17.543224
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)Kd3.374957
Proto-oncogene tyrosine-protein kinase ROSHomo sapiens (human)Kd10.000011
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)Kd22.900024
Putative heat shock protein HSP 90-beta 2Homo sapiens (human)Kd30.000015
Pyridoxal kinaseHomo sapiens (human)Kd25.468013
Rab-like protein 3Homo sapiens (human)Kd30.000012
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)Kd25.000024
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)Kd25.000024
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)Kd25.000024
RAF proto-oncogene serine/threonine-protein kinaseHomo sapiens (human)Kd10.000011
Ras-related protein Rab-10Homo sapiens (human)Kd30.000013
Ras-related protein Rab-27AHomo sapiens (human)Kd30.000013
Ras-related protein Rab-6AHomo sapiens (human)Kd30.000013
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)Kd10.000011
Receptor tyrosine-protein kinase erbB-3Homo sapiens (human)Kd10.000011
Receptor tyrosine-protein kinase erbB-4Homo sapiens (human)Kd10.000011
Receptor-interacting serine/threonine-protein kinase 1Homo sapiens (human)Kd10.000011
Receptor-interacting serine/threonine-protein kinase 2Homo sapiens (human)Kd8.277524
Receptor-interacting serine/threonine-protein kinase 3Homo sapiens (human)Kd20.105313
Receptor-interacting serine/threonine-protein kinase 4Homo sapiens (human)Kd10.000011
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)Kd16.0000810
Rho-associated protein kinase 1Homo sapiens (human)Kd25.000024
Rho-associated protein kinase 2Homo sapiens (human)Kd25.000024
Rhodopsin kinase GRK1Homo sapiens (human)Kd10.000011
Rhodopsin kinase GRK7Homo sapiens (human)Kd10.000011
Ribosomal protein S6 kinase alpha-1Homo sapiens (human)Kd22.000035
Ribosomal protein S6 kinase alpha-2Homo sapiens (human)Kd10.000022
Ribosomal protein S6 kinase alpha-3Homo sapiens (human)Kd25.000024
Ribosomal protein S6 kinase alpha-4Homo sapiens (human)Kd22.000035
Ribosomal protein S6 kinase alpha-5Homo sapiens (human)Kd22.000035
Ribosomal protein S6 kinase alpha-6Homo sapiens (human)Kd22.000035
Ribosomal protein S6 kinase beta-1Homo sapiens (human)Kd23.333323
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiens (human)Kd20.507713
RNA cytidine acetyltransferaseHomo sapiens (human)Kd30.000013
S-adenosylmethionine synthase isoform type-2Homo sapiens (human)Kd30.000013
Septin-9Homo sapiens (human)Kd30.000013
Serine/threonine-protein kinase 10Homo sapiens (human)Kd10.293224
Serine/threonine-protein kinase 16Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase 17AHomo sapiens (human)Kd10.000011
Serine/threonine-protein kinase 17BHomo sapiens (human)Kd10.000011
Serine/threonine-protein kinase 24Homo sapiens (human)Kd26.000025
Serine/threonine-protein kinase 25Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase 26Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase 3Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase 32AHomo sapiens (human)Kd10.000011
Serine/threonine-protein kinase 32BHomo sapiens (human)Kd3.900011
Serine/threonine-protein kinase 32CHomo sapiens (human)Kd10.000011
Serine/threonine-protein kinase 33Homo sapiens (human)Kd3.200011
Serine/threonine-protein kinase 35Homo sapiens (human)Kd0.026011
Serine/threonine-protein kinase 36Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase 38Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase 38-likeHomo sapiens (human)Kd23.333323
Serine/threonine-protein kinase 4Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase A-RafHomo sapiens (human)Kd30.000013
Serine/threonine-protein kinase ATRHomo sapiens (human)Kd30.000012
Serine/threonine-protein kinase B-rafHomo sapiens (human)Kd23.333336
Serine/threonine-protein kinase BRSK1Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase BRSK2Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase Chk1Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase Chk2Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase D1Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase D2Homo sapiens (human)Kd26.000025
Serine/threonine-protein kinase D3Homo sapiens (human)Kd26.000025
Serine/threonine-protein kinase DCLK1Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase DCLK2Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase DCLK3Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase ICKHomo sapiens (human)Kd26.000025
Serine/threonine-protein kinase LATS1Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase LATS2Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase MAKHomo sapiens (human)Kd10.000011
Serine/threonine-protein kinase MARK1Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase MARK2Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase MRCK alphaHomo sapiens (human)Kd25.000024
Serine/threonine-protein kinase MRCK betaHomo sapiens (human)Kd26.000025
Serine/threonine-protein kinase MRCK gammaHomo sapiens (human)Kd25.000024
Serine/threonine-protein kinase mTORHomo sapiens (human)Kd10.000011
Serine/threonine-protein kinase N1Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase N2Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase N3Homo sapiens (human)Kd30.000013
Serine/threonine-protein kinase Nek1Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase Nek11Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase Nek2Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase Nek3Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase Nek4Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase Nek5Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase Nek6Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase Nek7Homo sapiens (human)Kd26.000025
Serine/threonine-protein kinase Nek9Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase NIM1Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase NLKHomo sapiens (human)Kd25.000024
Serine/threonine-protein kinase OSR1Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase PAK 1Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase PAK 2Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase PAK 3Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase PAK 4Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase PAK 5Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase PAK 6Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase pim-1Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase pim-2Homo sapiens (human)Kd23.333323
Serine/threonine-protein kinase pim-3Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase PknBMycobacterium tuberculosis H37RvKd10.000011
Serine/threonine-protein kinase PLK1Homo sapiens (human)Kd20.000022
Serine/threonine-protein kinase PLK2Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase PLK3Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase PLK4Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase PRP4 homologHomo sapiens (human)Kd10.000011
Serine/threonine-protein kinase receptor R3Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase RIO1Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase RIO2Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase RIO3Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase SBK1Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase Sgk3Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase SIK1Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase SIK2Homo sapiens (human)Kd26.000025
Serine/threonine-protein kinase SIK3Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase STK11Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase TAO1Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase TAO2Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase TAO3Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase TBK1Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase TNNI3KHomo sapiens (human)Kd10.000011
Serine/threonine-protein kinase tousled-like 1Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase tousled-like 2Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase ULK1Homo sapiens (human)Kd26.000025
Serine/threonine-protein kinase ULK2Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase ULK3Homo sapiens (human)Kd25.000024
Serine/threonine-protein kinase VRK2Homo sapiens (human)Kd10.000011
Serine/threonine-protein kinase/endoribonuclease IRE1Homo sapiens (human)Kd18.060524
Serine/threonine-protein kinase/endoribonuclease IRE2Homo sapiens (human)Kd30.000013
Signal recognition particle receptor subunit alphaHomo sapiens (human)Kd30.000013
SNF-related serine/threonine-protein kinaseHomo sapiens (human)Kd10.000011
SRSF protein kinase 1Homo sapiens (human)Kd10.000011
SRSF protein kinase 2Homo sapiens (human)Kd10.000011
SRSF protein kinase 3Homo sapiens (human)Kd10.000011
STE20-like serine/threonine-protein kinase Homo sapiens (human)Kd9.190524
STE20-related kinase adapter protein alphaHomo sapiens (human)Kd20.379013
STE20/SPS1-related proline-alanine-rich protein kinaseHomo sapiens (human)Kd10.000011
Structural maintenance of chromosomes protein 1AHomo sapiens (human)Kd30.000014
Structural maintenance of chromosomes protein 2Homo sapiens (human)Kd30.000013
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrialHomo sapiens (human)Kd30.000013
Testis-specific serine/threonine-protein kinase 1Homo sapiens (human)Kd10.000011
TGF-beta receptor type-1Homo sapiens (human)Kd25.000024
TGF-beta receptor type-2Homo sapiens (human)Kd25.000024
Thyroid hormone receptor-associated protein 3Homo sapiens (human)Kd30.000012
TRAF2 and NCK-interacting protein kinaseHomo sapiens (human)Kd15.181224
Transient receptor potential cation channel subfamily M member 6Homo sapiens (human)Kd10.000011
Tyrosine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000013
Tyrosine-protein kinase ABL1Homo sapiens (human)Kd5.55121618
Tyrosine-protein kinase ABL2Homo sapiens (human)Kd24.360025
Tyrosine-protein kinase BlkHomo sapiens (human)Kd2.000011
Tyrosine-protein kinase BTKHomo sapiens (human)Kd25.000024
Tyrosine-protein kinase CSKHomo sapiens (human)Kd25.000024
Tyrosine-protein kinase FerHomo sapiens (human)Kd25.000024
Tyrosine-protein kinase Fes/FpsHomo sapiens (human)Kd25.000024
Tyrosine-protein kinase FgrHomo sapiens (human)Kd20.000022
Tyrosine-protein kinase FRKHomo sapiens (human)Kd25.000024
Tyrosine-protein kinase FynHomo sapiens (human)Kd26.000025
Tyrosine-protein kinase HCKHomo sapiens (human)Kd23.175024
Tyrosine-protein kinase ITK/TSKHomo sapiens (human)Kd10.000011
Tyrosine-protein kinase JAK1Homo sapiens (human)Kd22.000035
Tyrosine-protein kinase JAK2Homo sapiens (human)Kd23.333323
Tyrosine-protein kinase JAK3Homo sapiens (human)Kd10.000011
Tyrosine-protein kinase LckHomo sapiens (human)Kd22.775024
Tyrosine-protein kinase LynHomo sapiens (human)Kd20.552825
Tyrosine-protein kinase MerHomo sapiens (human)Kd20.000022
Tyrosine-protein kinase receptor Tie-1Homo sapiens (human)Kd1.100011
Tyrosine-protein kinase receptor TYRO3Homo sapiens (human)Kd10.000011
Tyrosine-protein kinase receptor UFOHomo sapiens (human)Kd10.000011
Tyrosine-protein kinase SrmsHomo sapiens (human)Kd10.000011
Tyrosine-protein kinase SYKHomo sapiens (human)Kd26.000025
Tyrosine-protein kinase TecHomo sapiens (human)Kd25.000024
Tyrosine-protein kinase TXKHomo sapiens (human)Kd10.000011
Tyrosine-protein kinase YesHomo sapiens (human)Kd25.000024
Tyrosine-protein kinase ZAP-70Homo sapiens (human)Kd10.000011
U5 small nuclear ribonucleoprotein 200 kDa helicaseHomo sapiens (human)Kd30.000013
UMP-CMP kinase Homo sapiens (human)Kd30.000014
Uncharacterized aarF domain-containing protein kinase 5Homo sapiens (human)Kd30.000012
Uncharacterized protein FLJ45252Homo sapiens (human)Kd30.000013
Uncharacterized serine/threonine-protein kinase SBK3Homo sapiens (human)Kd10.000011
Vascular endothelial growth factor receptor 1 Homo sapiens (human)Kd0.010011
Vascular endothelial growth factor receptor 2Homo sapiens (human)EC500.250011
Vascular endothelial growth factor receptor 2Homo sapiens (human)Kd0.003622
Vascular endothelial growth factor receptor 3Homo sapiens (human)Kd0.056011
Very long-chain specific acyl-CoA dehydrogenase, mitochondrialHomo sapiens (human)Kd30.000013
Wee1-like protein kinaseHomo sapiens (human)Kd25.000024
Wee1-like protein kinase 2Homo sapiens (human)Kd10.000011

Other Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
CholinesteraseHomo sapiens (human)Activity0.040011
Cytochrome P450 1A2Homo sapiens (human)Km45.000011
Cytochrome P450 3A4Homo sapiens (human)Km32.700011
Fibroblast growth factor receptor 1Homo sapiens (human)Activity0.276011
Fibroblast growth factor receptor 2Homo sapiens (human)Activity0.276011
Fibroblast growth factor receptor 3Homo sapiens (human)Activity0.276011
Fibroblast growth factor receptor 4Homo sapiens (human)Activity0.276011
Vascular endothelial growth factor receptor 1 Homo sapiens (human)Activity0.040011
Vascular endothelial growth factor receptor 2Homo sapiens (human)Activity0.040011
Vascular endothelial growth factor receptor 3Homo sapiens (human)Activity0.040011