Page last updated: 2024-08-05 15:48:14

c-Met tyrosine kinase inhibitor

An EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor that interferes with the action of c-Met tyrosine kinase.

ChEBI ID: 90199

Members (3)

MemberDefinitionClass
AMG-208A member of the class of quinolines that is 7-methoxyquinoline substituted at position 4 by a (6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methoxy group. AMG exhibits antitumour activity, particularly in prostate cancer.AMG-208
pha 665752A member of the class of indolones that is 1,3-dihydro-2H-indol-2-one which is substituted by a (2,6-dichlorobenzyl)sulfonyl group at position 5 and by a (1H-pyrrol-2-yl)methylidene group at position 2, the pyrrole ring of which is substituted by methyl groups at positions 3 and 5, and by a [2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]carbonyl group at position 4 (the Z,R isomer).PHA-665752
sgx 523A member of the class of triazolopyridazines that is 6-(1-methylpyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazine-3-thiol in which the thiol hydrogen is replaced by a quinolin-6-yl group.SGX-523

Research

Studies (33)

TimeframeStudies, Drugs with This Role(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's7 (21.21)29.6817
2010's18 (54.55)24.3611
2020's8 (24.24)2.80

Study Types

Publication TypeStudies, Drugs with this Role (%)All Drugs (%)
Trials1 (2.17%)5.53%
Reviews3 (6.52%)6.00%
Case Studies0 (0.00%)4.05%
Observational0 (0.00%)0.25%
Other42 (91.30%)84.16%

Protein Targets (499)

Potency Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
cytochrome P450 2C9, partialHomo sapiens (human)Potency0.756411
cytochrome P450 family 3 subfamily A polypeptide 4Homo sapiens (human)Potency0.756411
EWS/FLI fusion proteinHomo sapiens (human)Potency25.248422
GVesicular stomatitis virusPotency0.756411
HLA class I histocompatibility antigen, B alpha chain Homo sapiens (human)Potency0.756411
Inositol hexakisphosphate kinase 1Homo sapiens (human)Potency0.756412
Interferon betaHomo sapiens (human)Potency4.111624
PPM1D proteinHomo sapiens (human)Potency5.230012

Inhibition Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
ALK tyrosine kinase receptorHomo sapiens (human)IC500.076713
calcium-dependent protein kinase 4Plasmodium falciparum 3D7IC500.021011
Chain A, Hepatocyte growth factor receptorHomo sapiens (human)IC500.009012
Chain A, Hepatocyte growth factor receptorHomo sapiens (human)Ki5.001414
Cyclin-dependent kinase 2-associated protein 2Homo sapiens (human)IC5010.000011
Cytochrome P450 3A4Homo sapiens (human)IC5032.000011
Epidermal growth factor receptorHomo sapiens (human)IC501.007524
Fibroblast growth factor receptor 1Homo sapiens (human)IC503.000011
Glycogen synthase kinase-3 betaHomo sapiens (human)IC5010.000011
Hepatocyte growth factor receptorHomo sapiens (human)IC500.02401721
Homeodomain-interacting protein kinase 1Homo sapiens (human)IC500.100011
Homeodomain-interacting protein kinase 2Homo sapiens (human)IC500.100011
Homeodomain-interacting protein kinase 3Homo sapiens (human)IC500.100011
Homeodomain-interacting protein kinase 4Homo sapiens (human)IC500.100011
Insulin-like growth factor 1 receptorHomo sapiens (human)IC5010.000011
Macrophage-stimulating protein receptorHomo sapiens (human)IC500.068011
MAP kinase-activated protein kinase 2Homo sapiens (human)IC5010.000011
MAP kinase-activated protein kinase 3Homo sapiens (human)IC5010.000011
Mitogen-activated protein kinase 14Homo sapiens (human)IC5010.000011
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)IC500.076713
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)IC506.000011
Tyrosine-protein kinase ABL1Homo sapiens (human)IC501.400011
Vascular endothelial growth factor receptor 2Homo sapiens (human)IC500.531522

Activation Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
26S proteasome regulatory subunit 6BHomo sapiens (human)Kd30.000012
3-phosphoinositide-dependent protein kinase 1Homo sapiens (human)Kd10.000012
5'-AMP-activated protein kinase catalytic subunit alpha-1Homo sapiens (human)Kd17.577524
5'-AMP-activated protein kinase catalytic subunit alpha-2Homo sapiens (human)Kd5.385012
5'-AMP-activated protein kinase subunit gamma-1Homo sapiens (human)Kd30.000012
5'-AMP-activated protein kinase subunit gamma-2Homo sapiens (human)Kd30.000012
AarF domain-containing protein kinase 1Homo sapiens (human)Kd30.000012
Actin-related protein 2Homo sapiens (human)Kd30.000013
Actin-related protein 3Homo sapiens (human)Kd30.000012
Activated CDC42 kinase 1Homo sapiens (human)Kd20.000024
Activin receptor type-1Homo sapiens (human)Kd20.000024
Activin receptor type-1BHomo sapiens (human)Kd20.000024
Activin receptor type-2AHomo sapiens (human)Kd10.000012
Activin receptor type-2BHomo sapiens (human)Kd20.000024
Acyl-CoA dehydrogenase family member 10Homo sapiens (human)Kd30.000012
Acyl-CoA dehydrogenase family member 11Homo sapiens (human)Kd30.000012
Adenine phosphoribosyltransferaseHomo sapiens (human)Kd30.000012
Adenosine kinaseHomo sapiens (human)Kd30.000012
Adenylate kinase 2, mitochondrialHomo sapiens (human)Kd30.000012
ADP/ATP translocase 2Homo sapiens (human)Kd30.000012
ADP/ATP translocase 3Homo sapiens (human)Kd30.000012
ALK tyrosine kinase receptorHomo sapiens (human)Kd6.350012
Angiopoietin-1 receptorHomo sapiens (human)Kd8.350012
Ankyrin repeat and protein kinase domain-containing protein 1Homo sapiens (human)Kd10.000012
AP2-associated protein kinase 1Homo sapiens (human)Kd17.580024
ATP-dependent 6-phosphofructokinase, platelet typeHomo sapiens (human)Kd30.000011
ATP-dependent RNA helicase DDX1Homo sapiens (human)Kd30.000012
ATP-dependent RNA helicase DDX3XHomo sapiens (human)Kd30.000012
ATP-dependent RNA helicase DDX42Homo sapiens (human)Kd30.000012
Atypical kinase COQ8A, mitochondrialHomo sapiens (human)Kd20.000024
Atypical kinase COQ8B, mitochondrialHomo sapiens (human)Kd10.000012
Aurora kinase AHomo sapiens (human)Kd20.000024
Aurora kinase BHomo sapiens (human)Kd20.400025
Aurora kinase CHomo sapiens (human)Kd5.150012
BDNF/NT-3 growth factors receptorHomo sapiens (human)Kd5.400012
Beta-adrenergic receptor kinase 1Homo sapiens (human)Kd30.000012
BMP-2-inducible protein kinaseHomo sapiens (human)Kd20.009425
Bone morphogenetic protein receptor type-1AHomo sapiens (human)Kd20.000024
Bone morphogenetic protein receptor type-1BHomo sapiens (human)Kd20.000024
Bone morphogenetic protein receptor type-2Homo sapiens (human)Kd19.050024
Breakpoint cluster region proteinHomo sapiens (human)Kd30.000012
Calcium-dependent protein kinase 1Plasmodium falciparum 3D7Kd10.000012
Calcium/calmodulin-dependent protein kinase kinase 1Homo sapiens (human)Kd5.032012
Calcium/calmodulin-dependent protein kinase kinase 2Homo sapiens (human)Kd17.518324
Calcium/calmodulin-dependent protein kinase type 1Homo sapiens (human)Kd6.050012
Calcium/calmodulin-dependent protein kinase type 1DHomo sapiens (human)Kd5.750012
Calcium/calmodulin-dependent protein kinase type 1GHomo sapiens (human)Kd10.000012
Calcium/calmodulin-dependent protein kinase type II subunit alphaHomo sapiens (human)Kd6.700012
Calcium/calmodulin-dependent protein kinase type II subunit betaHomo sapiens (human)Kd10.000012
Calcium/calmodulin-dependent protein kinase type II subunit deltaHomo sapiens (human)Kd18.225024
Calcium/calmodulin-dependent protein kinase type II subunit gammaHomo sapiens (human)Kd18.000024
Calcium/calmodulin-dependent protein kinase type IVHomo sapiens (human)Kd20.000024
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)Kd20.000024
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)Kd20.000024
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)Kd15.001012
cAMP-dependent protein kinase catalytic subunit PRKXHomo sapiens (human)Kd10.000012
cAMP-dependent protein kinase type II-alpha regulatory subunitHomo sapiens (human)Kd30.000012
Casein kinase I isoform alphaHomo sapiens (human)Kd20.000024
Casein kinase I isoform alpha-likeHomo sapiens (human)Kd10.000012
Casein kinase I isoform deltaHomo sapiens (human)Kd18.550024
Casein kinase I isoform epsilonHomo sapiens (human)Kd17.715024
Casein kinase I isoform gamma-1Homo sapiens (human)Kd20.000024
Casein kinase I isoform gamma-2Homo sapiens (human)Kd16.666723
Casein kinase I isoform gamma-3Homo sapiens (human)Kd22.000025
Casein kinase II subunit alphaHomo sapiens (human)Kd10.000012
Casein kinase II subunit alpha'Homo sapiens (human)Kd18.900024
Cell division control protein 2 homologPlasmodium falciparum 3D7Kd10.000012
Cell division cycle 7-related protein kinaseHomo sapiens (human)Kd30.000011
cGMP-dependent protein kinase 1 Homo sapiens (human)Kd20.000024
cGMP-dependent protein kinase 2Homo sapiens (human)Kd10.000012
Choline-phosphate cytidylyltransferase AHomo sapiens (human)Kd30.000012
Chromodomain-helicase-DNA-binding protein 4Homo sapiens (human)Kd30.000012
Citron Rho-interacting kinaseHomo sapiens (human)Kd20.000024
Cyclin-dependent kinase 1Homo sapiens (human)Kd30.000012
Cyclin-dependent kinase 11AHomo sapiens (human)Kd10.000012
Cyclin-dependent kinase 11BHomo sapiens (human)Kd10.000012
Cyclin-dependent kinase 12Homo sapiens (human)Kd30.000012
Cyclin-dependent kinase 13Homo sapiens (human)Kd20.000024
Cyclin-dependent kinase 14Homo sapiens (human)Kd5.650012
Cyclin-dependent kinase 15Homo sapiens (human)Kd5.255012
Cyclin-dependent kinase 16Homo sapiens (human)Kd17.775024
Cyclin-dependent kinase 17Homo sapiens (human)Kd17.720024
Cyclin-dependent kinase 18Homo sapiens (human)Kd5.750012
Cyclin-dependent kinase 19Homo sapiens (human)Kd10.000012
Cyclin-dependent kinase 2Homo sapiens (human)Kd20.000024
Cyclin-dependent kinase 3Homo sapiens (human)Kd22.000025
Cyclin-dependent kinase 4Homo sapiens (human)Kd13.813336
Cyclin-dependent kinase 6Homo sapiens (human)Kd30.000012
Cyclin-dependent kinase 7Homo sapiens (human)Kd17.532524
Cyclin-dependent kinase 8Homo sapiens (human)Kd10.000012
Cyclin-dependent kinase 9Homo sapiens (human)Kd17.950024
Cyclin-dependent kinase-like 1Homo sapiens (human)Kd10.000012
Cyclin-dependent kinase-like 2Homo sapiens (human)Kd6.200012
Cyclin-dependent kinase-like 3Homo sapiens (human)Kd10.000012
Cyclin-dependent kinase-like 5Homo sapiens (human)Kd20.000024
Cyclin-dependent-like kinase 5 Homo sapiens (human)Kd20.000024
Cyclin-G-associated kinaseHomo sapiens (human)Kd17.825024
Cysteine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000013
Cytochrome c1, heme protein, mitochondrialHomo sapiens (human)Kd30.000012
Cytoplasmic tyrosine-protein kinase BMXHomo sapiens (human)Kd10.000012
dCTP pyrophosphatase 1Homo sapiens (human)Kd30.000012
Death-associated protein kinase 1Homo sapiens (human)Kd10.000012
Death-associated protein kinase 2Homo sapiens (human)Kd10.000012
Death-associated protein kinase 3Homo sapiens (human)Kd10.000012
Delta(24)-sterol reductaseHomo sapiens (human)Kd30.000012
Deoxycytidine kinaseHomo sapiens (human)Kd30.000012
Discoidin domain-containing receptor 2Homo sapiens (human)Kd19.400024
DNA replication licensing factor MCM4Homo sapiens (human)Kd30.000012
DNA topoisomerase 2-alphaHomo sapiens (human)Kd30.000012
DNA topoisomerase 2-betaHomo sapiens (human)Kd30.000012
DnaJ homolog subfamily A member 1Homo sapiens (human)Kd30.000012
Dual serine/threonine and tyrosine protein kinaseHomo sapiens (human)Kd10.000012
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)Kd17.775024
Dual specificity mitogen-activated protein kinase kinase 2Homo sapiens (human)Kd17.745024
Dual specificity mitogen-activated protein kinase kinase 3Homo sapiens (human)Kd20.000024
Dual specificity mitogen-activated protein kinase kinase 4Homo sapiens (human)Kd16.666723
Dual specificity mitogen-activated protein kinase kinase 5Homo sapiens (human)Kd17.850024
Dual specificity mitogen-activated protein kinase kinase 6Homo sapiens (human)Kd20.000024
Dual specificity mitogen-activated protein kinase kinase 7Homo sapiens (human)Kd10.000012
Dual specificity protein kinase CLK1Homo sapiens (human)Kd17.682524
Dual specificity protein kinase CLK2Homo sapiens (human)Kd17.602524
Dual specificity protein kinase CLK3Homo sapiens (human)Kd14.533323
Dual specificity protein kinase CLK4Homo sapiens (human)Kd20.000024
Dual specificity protein kinase TTKHomo sapiens (human)Kd10.000012
Dual specificity testis-specific protein kinase 1Homo sapiens (human)Kd20.000024
Dual specificity testis-specific protein kinase 2Homo sapiens (human)Kd30.000012
Dual specificity tyrosine-phosphorylation-regulated kinase 1AHomo sapiens (human)Kd17.695024
Dual specificity tyrosine-phosphorylation-regulated kinase 1BHomo sapiens (human)Kd20.360025
Dual specificity tyrosine-phosphorylation-regulated kinase 2Homo sapiens (human)Kd10.000012
Dynamin-like 120 kDa protein, mitochondrialHomo sapiens (human)Kd30.000012
eIF-2-alpha kinase GCN2Homo sapiens (human)Kd6.700012
EKC/KEOPS complex subunit TP53RKHomo sapiens (human)Kd30.000012
Electron transfer flavoprotein subunit betaHomo sapiens (human)Kd30.000012
Elongation factor Tu, mitochondrialHomo sapiens (human)Kd30.000013
Ephrin type-A receptor 1Homo sapiens (human)Kd20.000024
Ephrin type-A receptor 2Homo sapiens (human)Kd20.000024
Ephrin type-A receptor 3Homo sapiens (human)Kd10.000012
Ephrin type-A receptor 4Homo sapiens (human)Kd22.000025
Ephrin type-A receptor 5Homo sapiens (human)Kd20.000024
Ephrin type-A receptor 6Homo sapiens (human)Kd10.000012
Ephrin type-A receptor 7Homo sapiens (human)Kd20.000024
Ephrin type-A receptor 8Homo sapiens (human)Kd6.950012
Ephrin type-B receptor 1Homo sapiens (human)Kd10.000012
Ephrin type-B receptor 2Homo sapiens (human)Kd20.000024
Ephrin type-B receptor 3Homo sapiens (human)Kd20.000024
Ephrin type-B receptor 4Homo sapiens (human)Kd20.000024
Ephrin type-B receptor 6Homo sapiens (human)Kd18.225024
Epidermal growth factor receptorHomo sapiens (human)Kd11.53851326
Epithelial discoidin domain-containing receptor 1Homo sapiens (human)Kd17.517524
Eukaryotic peptide chain release factor GTP-binding subunit ERF3BHomo sapiens (human)Kd30.000011
Eukaryotic translation initiation factor 2-alpha kinase 1Homo sapiens (human)Kd20.000024
Eukaryotic translation initiation factor 5BHomo sapiens (human)Kd30.000012
Exosome RNA helicase MTR4Homo sapiens (human)Kd30.000012
Ferrochelatase, mitochondrialHomo sapiens (human)Kd30.000013
Fibroblast growth factor receptor 1Homo sapiens (human)Kd20.000024
Fibroblast growth factor receptor 2Homo sapiens (human)Kd7.600012
Fibroblast growth factor receptor 3Homo sapiens (human)Kd8.800024
Fibroblast growth factor receptor 4Homo sapiens (human)Kd10.000012
Focal adhesion kinase 1Homo sapiens (human)Kd17.975024
G protein-coupled receptor kinase 4Homo sapiens (human)Kd5.210012
G protein-coupled receptor kinase 6Homo sapiens (human)Kd30.000011
General transcription and DNA repair factor IIH helicase subunit XPDHomo sapiens (human)Kd30.000012
Glycine--tRNA ligaseHomo sapiens (human)Kd30.000012
Glycogen phosphorylase, brain formHomo sapiens (human)Kd30.000012
Glycogen phosphorylase, liver formHomo sapiens (human)Kd30.000012
Glycogen synthase kinase-3 alphaHomo sapiens (human)Kd20.000024
Glycogen synthase kinase-3 betaHomo sapiens (human)Kd20.000024
GTP-binding nuclear protein RanHomo sapiens (human)Kd30.000012
Guanine nucleotide-binding protein G(i) subunit alpha-2Homo sapiens (human)Kd30.000011
Heme oxygenase 2Homo sapiens (human)Kd30.000012
Hepatocyte growth factor receptorHomo sapiens (human)EC500.042011
Hepatocyte growth factor receptorHomo sapiens (human)Kd3.754348
High affinity nerve growth factor receptorHomo sapiens (human)Kd13.440023
Homeodomain-interacting protein kinase 1Homo sapiens (human)Kd5.046512
Homeodomain-interacting protein kinase 2Homo sapiens (human)Kd5.060012
Homeodomain-interacting protein kinase 3Homo sapiens (human)Kd5.031512
Homeodomain-interacting protein kinase 4Homo sapiens (human)Kd5.650012
Hormonally up-regulated neu tumor-associated kinaseHomo sapiens (human)Kd5.700012
Inhibitor of nuclear factor kappa-B kinase subunit alphaHomo sapiens (human)Kd10.000012
Inhibitor of nuclear factor kappa-B kinase subunit betaHomo sapiens (human)Kd10.000012
Inhibitor of nuclear factor kappa-B kinase subunit epsilonHomo sapiens (human)Kd17.675024
Inosine-5'-monophosphate dehydrogenase 2Homo sapiens (human)Kd30.000012
Insulin receptorHomo sapiens (human)Kd18.075024
Insulin receptor-related proteinHomo sapiens (human)Kd6.750012
Insulin-like growth factor 1 receptorHomo sapiens (human)Kd20.000024
Integrin-linked protein kinaseHomo sapiens (human)Kd30.000012
Interferon-induced, double-stranded RNA-activated protein kinaseHomo sapiens (human)Kd10.000012
Interleukin-1 receptor-associated kinase 1Homo sapiens (human)Kd17.900024
Interleukin-1 receptor-associated kinase 3Homo sapiens (human)Kd17.652524
Interleukin-1 receptor-associated kinase 4Homo sapiens (human)Kd18.125024
Isoleucine--tRNA ligase, mitochondrialHomo sapiens (human)Kd30.000013
Leucine-rich repeat serine/threonine-protein kinase 2Homo sapiens (human)Kd10.000024
Leukocyte tyrosine kinase receptorHomo sapiens (human)Kd10.000012
Leukotriene C4 synthaseCavia porcellus (domestic guinea pig)Kd10.000012
LIM domain kinase 1Homo sapiens (human)Kd20.000024
LIM domain kinase 2Homo sapiens (human)Kd20.000024
Long-chain-fatty-acid--CoA ligase 5Homo sapiens (human)Kd30.000013
Macrophage colony-stimulating factor 1 receptorHomo sapiens (human)Kd5.350012
Macrophage-stimulating protein receptorHomo sapiens (human)EC500.900011
Macrophage-stimulating protein receptorHomo sapiens (human)Kd18.000024
MAP kinase-activated protein kinase 2Homo sapiens (human)Kd20.000024
MAP kinase-activated protein kinase 3Homo sapiens (human)Kd30.000011
MAP kinase-activated protein kinase 5Homo sapiens (human)Kd20.000024
MAP kinase-interacting serine/threonine-protein kinase 1Homo sapiens (human)Kd10.000012
MAP kinase-interacting serine/threonine-protein kinase 2Homo sapiens (human)Kd10.000012
MAP/microtubule affinity-regulating kinase 3Homo sapiens (human)Kd20.000024
MAP/microtubule affinity-regulating kinase 4Homo sapiens (human)Kd20.000024
Mast/stem cell growth factor receptor KitHomo sapiens (human)Kd7.0681816
Maternal embryonic leucine zipper kinaseHomo sapiens (human)Kd20.000024
Megakaryocyte-associated tyrosine-protein kinaseHomo sapiens (human)Kd10.000012
Membrane-associated progesterone receptor component 1Homo sapiens (human)Kd30.000012
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinaseHomo sapiens (human)Kd20.000024
Microtubule-associated serine/threonine-protein kinase 1Homo sapiens (human)Kd10.000012
MidasinHomo sapiens (human)Kd30.000012
Misshapen-like kinase 1Homo sapiens (human)Kd5.125012
Mitogen-activated protein kinase 1Homo sapiens (human)Kd20.000024
Mitogen-activated protein kinase 10Homo sapiens (human)Kd17.975024
Mitogen-activated protein kinase 11Homo sapiens (human)Kd20.000024
Mitogen-activated protein kinase 12Homo sapiens (human)Kd10.000012
Mitogen-activated protein kinase 13Homo sapiens (human)Kd10.000012
Mitogen-activated protein kinase 14Homo sapiens (human)Kd20.000024
Mitogen-activated protein kinase 15Homo sapiens (human)Kd20.000024
Mitogen-activated protein kinase 3 Homo sapiens (human)Kd20.000024
Mitogen-activated protein kinase 4Homo sapiens (human)Kd10.000012
Mitogen-activated protein kinase 6Homo sapiens (human)Kd10.000012
Mitogen-activated protein kinase 7Homo sapiens (human)Kd17.925024
Mitogen-activated protein kinase 8Homo sapiens (human)Kd18.550024
Mitogen-activated protein kinase 9Homo sapiens (human)Kd20.000024
Mitogen-activated protein kinase kinase kinase 1Homo sapiens (human)Kd20.000024
Mitogen-activated protein kinase kinase kinase 10Homo sapiens (human)Kd10.000012
Mitogen-activated protein kinase kinase kinase 11Homo sapiens (human)Kd20.000024
Mitogen-activated protein kinase kinase kinase 12Homo sapiens (human)Kd5.335012
Mitogen-activated protein kinase kinase kinase 13Homo sapiens (human)Kd6.600012
Mitogen-activated protein kinase kinase kinase 15Homo sapiens (human)Kd10.000012
Mitogen-activated protein kinase kinase kinase 19Homo sapiens (human)Kd3.239012
Mitogen-activated protein kinase kinase kinase 2Homo sapiens (human)Kd18.800024
Mitogen-activated protein kinase kinase kinase 20Homo sapiens (human)Kd20.000024
Mitogen-activated protein kinase kinase kinase 3Homo sapiens (human)Kd18.975024
Mitogen-activated protein kinase kinase kinase 4Homo sapiens (human)Kd17.950024
Mitogen-activated protein kinase kinase kinase 5Homo sapiens (human)Kd20.000024
Mitogen-activated protein kinase kinase kinase 6Homo sapiens (human)Kd20.000024
Mitogen-activated protein kinase kinase kinase 7Homo sapiens (human)Kd7.650012
Mitogen-activated protein kinase kinase kinase 9Homo sapiens (human)Kd10.000012
Mitogen-activated protein kinase kinase kinase kinase 1Homo sapiens (human)Kd17.537524
Mitogen-activated protein kinase kinase kinase kinase 2Homo sapiens (human)Kd18.400024
Mitogen-activated protein kinase kinase kinase kinase 3Homo sapiens (human)Kd20.098025
Mitogen-activated protein kinase kinase kinase kinase 4Homo sapiens (human)Kd17.570024
Mitogen-activated protein kinase kinase kinase kinase 5Homo sapiens (human)Kd17.519824
Mitotic checkpoint serine/threonine-protein kinase BUB1Homo sapiens (human)Kd30.000012
Multifunctional protein ADE2Homo sapiens (human)Kd30.000012
Muscle, skeletal receptor tyrosine-protein kinaseHomo sapiens (human)Kd10.000012
Myosin light chain kinase 2, skeletal/cardiac muscleHomo sapiens (human)Kd5.480012
Myosin light chain kinase 3Homo sapiens (human)Kd20.000024
Myosin light chain kinase family member 4Homo sapiens (human)Kd10.000012
Myosin light chain kinase, smooth muscleHomo sapiens (human)Kd19.475024
Myosin-10Homo sapiens (human)Kd30.000013
Myosin-14Homo sapiens (human)Kd30.000012
Myosin-IIIaHomo sapiens (human)Kd10.000012
Myosin-IIIbHomo sapiens (human)Kd10.000012
Myotonin-protein kinaseHomo sapiens (human)Kd10.000012
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13Homo sapiens (human)Kd30.000012
Non-receptor tyrosine-protein kinase TNK1Homo sapiens (human)Kd20.000024
Non-receptor tyrosine-protein kinase TYK2Homo sapiens (human)Kd16.100036
NT-3 growth factor receptorHomo sapiens (human)Kd5.465012
NUAK family SNF1-like kinase 1Homo sapiens (human)Kd5.310012
NUAK family SNF1-like kinase 2Homo sapiens (human)Kd13.636723
Nucleolar GTP-binding protein 1Homo sapiens (human)Kd30.000012
Obg-like ATPase 1Homo sapiens (human)Kd30.000012
PAS domain-containing serine/threonine-protein kinaseHomo sapiens (human)Kd30.000011
Peripheral plasma membrane protein CASKHomo sapiens (human)Kd5.850012
Peroxisomal acyl-coenzyme A oxidase 1Homo sapiens (human)Kd30.000012
Peroxisomal acyl-coenzyme A oxidase 3Homo sapiens (human)Kd30.000012
Phenylalanine--tRNA ligase beta subunitHomo sapiens (human)Kd30.000012
Phosphatidylethanolamine-binding protein 1Homo sapiens (human)Kd30.000012
Phosphatidylinositol 4-kinase betaHomo sapiens (human)Kd10.000012
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit betaHomo sapiens (human)Kd10.000012
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gammaHomo sapiens (human)Kd10.000012
Phosphatidylinositol 4-phosphate 5-kinase type-1 alphaHomo sapiens (human)Kd5.140012
Phosphatidylinositol 4-phosphate 5-kinase type-1 gammaHomo sapiens (human)Kd10.000012
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformHomo sapiens (human)Kd10.00001020
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformHomo sapiens (human)Kd10.000012
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformHomo sapiens (human)Kd10.000012
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)Kd10.000012
Phosphatidylinositol 5-phosphate 4-kinase type-2 alphaHomo sapiens (human)Kd30.000012
Phosphatidylinositol 5-phosphate 4-kinase type-2 betaHomo sapiens (human)Kd5.800012
Phosphatidylinositol 5-phosphate 4-kinase type-2 gammaHomo sapiens (human)Kd18.325024
Phosphorylase b kinase gamma catalytic chain, liver/testis isoformHomo sapiens (human)Kd20.480025
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoformHomo sapiens (human)Kd5.950012
Platelet-derived growth factor receptor alphaHomo sapiens (human)Kd6.000012
Platelet-derived growth factor receptor betaHomo sapiens (human)Kd17.975024
Probable ATP-dependent RNA helicase DDX6Homo sapiens (human)Kd30.000012
Prostaglandin G/H synthase 2Homo sapiens (human)Kd5.235012
Protein kinase C alpha typeHomo sapiens (human)Kd30.000012
Protein kinase C beta typeHomo sapiens (human)Kd30.000012
Protein kinase C delta typeHomo sapiens (human)Kd22.000025
Protein kinase C epsilon typeHomo sapiens (human)Kd10.000012
Protein kinase C eta typeHomo sapiens (human)Kd10.000012
Protein kinase C iota typeHomo sapiens (human)Kd20.000024
Protein kinase C theta typeHomo sapiens (human)Kd20.000024
Protein-tyrosine kinase 2-betaHomo sapiens (human)Kd17.727524
Protein-tyrosine kinase 6Homo sapiens (human)Kd20.000024
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)Kd10.2240510
Proto-oncogene tyrosine-protein kinase ROSHomo sapiens (human)Kd6.500012
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)Kd20.000024
Putative heat shock protein HSP 90-beta 2Homo sapiens (human)Kd30.000012
Pyridoxal kinaseHomo sapiens (human)Kd30.000012
Rab-like protein 3Homo sapiens (human)Kd30.000012
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)Kd20.000024
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)Kd20.000024
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)Kd20.000024
RAF proto-oncogene serine/threonine-protein kinaseHomo sapiens (human)Kd10.000012
Ras-related protein Rab-10Homo sapiens (human)Kd30.000012
Ras-related protein Rab-27AHomo sapiens (human)Kd30.000013
Ras-related protein Rab-6AHomo sapiens (human)Kd30.000012
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)Kd10.000012
Receptor tyrosine-protein kinase erbB-3Homo sapiens (human)Kd10.000012
Receptor tyrosine-protein kinase erbB-4Homo sapiens (human)Kd10.000012
Receptor-interacting serine/threonine-protein kinase 1Homo sapiens (human)Kd5.750012
Receptor-interacting serine/threonine-protein kinase 2Homo sapiens (human)Kd20.000024
Receptor-interacting serine/threonine-protein kinase 3Homo sapiens (human)Kd30.000012
Receptor-interacting serine/threonine-protein kinase 4Homo sapiens (human)Kd10.000012
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)Kd8.4928816
Rho-associated protein kinase 1Homo sapiens (human)Kd20.000024
Rho-associated protein kinase 2Homo sapiens (human)Kd19.675024
Rhodopsin kinase GRK1Homo sapiens (human)Kd5.550012
Rhodopsin kinase GRK7Homo sapiens (human)Kd5.030512
Ribosomal protein S6 kinase alpha-1Homo sapiens (human)Kd18.571437
Ribosomal protein S6 kinase alpha-2Homo sapiens (human)Kd10.000024
Ribosomal protein S6 kinase alpha-3Homo sapiens (human)Kd19.975024
Ribosomal protein S6 kinase alpha-4Homo sapiens (human)Kd16.666736
Ribosomal protein S6 kinase alpha-5Homo sapiens (human)Kd15.183336
Ribosomal protein S6 kinase alpha-6Homo sapiens (human)Kd16.133336
Ribosomal protein S6 kinase beta-1Homo sapiens (human)Kd18.525024
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiens (human)Kd15.062012
RNA cytidine acetyltransferaseHomo sapiens (human)Kd30.000012
S-adenosylmethionine synthase isoform type-2Homo sapiens (human)Kd30.000012
Septin-9Homo sapiens (human)Kd30.000012
Serine/threonine-protein kinase 10Homo sapiens (human)Kd17.572524
Serine/threonine-protein kinase 16Homo sapiens (human)Kd18.700024
Serine/threonine-protein kinase 17AHomo sapiens (human)Kd7.000012
Serine/threonine-protein kinase 17BHomo sapiens (human)Kd6.750012
Serine/threonine-protein kinase 24Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase 25Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase 26Homo sapiens (human)Kd18.450024
Serine/threonine-protein kinase 3Homo sapiens (human)Kd17.975024
Serine/threonine-protein kinase 32AHomo sapiens (human)Kd10.000012
Serine/threonine-protein kinase 32BHomo sapiens (human)Kd10.000012
Serine/threonine-protein kinase 32CHomo sapiens (human)Kd10.000012
Serine/threonine-protein kinase 33Homo sapiens (human)Kd5.420012
Serine/threonine-protein kinase 35Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase 36Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase 38Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase 38-likeHomo sapiens (human)Kd16.666723
Serine/threonine-protein kinase 4Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase A-RafHomo sapiens (human)Kd30.000012
Serine/threonine-protein kinase ATRHomo sapiens (human)Kd30.000012
Serine/threonine-protein kinase B-rafHomo sapiens (human)Kd16.666736
Serine/threonine-protein kinase BRSK1Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase BRSK2Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase Chk1Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase Chk2Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase D1Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase D2Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase D3Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase DCLK1Homo sapiens (human)Kd5.700012
Serine/threonine-protein kinase DCLK2Homo sapiens (human)Kd5.495012
Serine/threonine-protein kinase DCLK3Homo sapiens (human)Kd7.250012
Serine/threonine-protein kinase ICKHomo sapiens (human)Kd17.600024
Serine/threonine-protein kinase LATS1Homo sapiens (human)Kd22.000025
Serine/threonine-protein kinase LATS2Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase MAKHomo sapiens (human)Kd5.445012
Serine/threonine-protein kinase MARK1Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase MARK2Homo sapiens (human)Kd18.400024
Serine/threonine-protein kinase MRCK alphaHomo sapiens (human)Kd20.000024
Serine/threonine-protein kinase MRCK betaHomo sapiens (human)Kd20.000024
Serine/threonine-protein kinase MRCK gammaHomo sapiens (human)Kd20.000024
Serine/threonine-protein kinase mTORHomo sapiens (human)Kd10.000012
Serine/threonine-protein kinase N1Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase N2Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase N3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Nek1Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase Nek11Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase Nek2Homo sapiens (human)Kd17.650024
Serine/threonine-protein kinase Nek3Homo sapiens (human)Kd23.333326
Serine/threonine-protein kinase Nek4Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase Nek5Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase Nek6Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase Nek7Homo sapiens (human)Kd16.666723
Serine/threonine-protein kinase Nek9Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase NIM1Homo sapiens (human)Kd9.350012
Serine/threonine-protein kinase NLKHomo sapiens (human)Kd20.000024
Serine/threonine-protein kinase OSR1Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase PAK 1Homo sapiens (human)Kd6.450012
Serine/threonine-protein kinase PAK 2Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase PAK 3Homo sapiens (human)Kd5.550012
Serine/threonine-protein kinase PAK 4Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase PAK 5Homo sapiens (human)Kd6.300012
Serine/threonine-protein kinase PAK 6Homo sapiens (human)Kd16.666723
Serine/threonine-protein kinase pim-1Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase pim-2Homo sapiens (human)Kd16.666723
Serine/threonine-protein kinase pim-3Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase PknBMycobacterium tuberculosis H37RvKd10.000012
Serine/threonine-protein kinase PLK1Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase PLK2Homo sapiens (human)Kd9.150012
Serine/threonine-protein kinase PLK3Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase PLK4Homo sapiens (human)Kd17.602524
Serine/threonine-protein kinase PRP4 homologHomo sapiens (human)Kd6.300012
Serine/threonine-protein kinase receptor R3Homo sapiens (human)Kd16.666723
Serine/threonine-protein kinase RIO1Homo sapiens (human)Kd5.235012
Serine/threonine-protein kinase RIO2Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase RIO3Homo sapiens (human)Kd2.794524
Serine/threonine-protein kinase SBK1Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase Sgk3Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase SIK1Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase SIK2Homo sapiens (human)Kd18.125024
Serine/threonine-protein kinase SIK3Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase STK11Homo sapiens (human)Kd18.150024
Serine/threonine-protein kinase TAO1Homo sapiens (human)Kd17.615024
Serine/threonine-protein kinase TAO2Homo sapiens (human)Kd17.800024
Serine/threonine-protein kinase TAO3Homo sapiens (human)Kd17.510824
Serine/threonine-protein kinase TBK1Homo sapiens (human)Kd17.742524
Serine/threonine-protein kinase TNNI3KHomo sapiens (human)Kd10.000012
Serine/threonine-protein kinase tousled-like 1Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase tousled-like 2Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase ULK1Homo sapiens (human)Kd18.000024
Serine/threonine-protein kinase ULK2Homo sapiens (human)Kd5.750012
Serine/threonine-protein kinase ULK3Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase VRK2Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase/endoribonuclease IRE1Homo sapiens (human)Kd20.000024
Serine/threonine-protein kinase/endoribonuclease IRE2Homo sapiens (human)Kd30.000012
Signal recognition particle receptor subunit alphaHomo sapiens (human)Kd30.000012
SNF-related serine/threonine-protein kinaseHomo sapiens (human)Kd10.000012
SRSF protein kinase 1Homo sapiens (human)Kd5.020512
SRSF protein kinase 2Homo sapiens (human)Kd5.250012
SRSF protein kinase 3Homo sapiens (human)Kd5.800012
STE20-like serine/threonine-protein kinase Homo sapiens (human)Kd17.587524
STE20-related kinase adapter protein alphaHomo sapiens (human)Kd30.000013
STE20/SPS1-related proline-alanine-rich protein kinaseHomo sapiens (human)Kd10.000012
Structural maintenance of chromosomes protein 1AHomo sapiens (human)Kd30.000012
Structural maintenance of chromosomes protein 2Homo sapiens (human)Kd30.000013
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrialHomo sapiens (human)Kd30.000013
Testis-specific serine/threonine-protein kinase 1Homo sapiens (human)Kd6.050012
TGF-beta receptor type-1Homo sapiens (human)Kd20.000024
TGF-beta receptor type-2Homo sapiens (human)Kd20.000024
Thyroid hormone receptor-associated protein 3Homo sapiens (human)Kd30.000012
TRAF2 and NCK-interacting protein kinaseHomo sapiens (human)Kd17.577524
Transient receptor potential cation channel subfamily M member 6Homo sapiens (human)Kd10.000012
Tyrosine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000012
Tyrosine-protein kinase ABL1Homo sapiens (human)Kd9.27411632
Tyrosine-protein kinase ABL2Homo sapiens (human)Kd19.225024
Tyrosine-protein kinase BlkHomo sapiens (human)Kd5.950012
Tyrosine-protein kinase BTKHomo sapiens (human)Kd20.000024
Tyrosine-protein kinase CSKHomo sapiens (human)Kd20.000024
Tyrosine-protein kinase FerHomo sapiens (human)Kd20.000024
Tyrosine-protein kinase Fes/FpsHomo sapiens (human)Kd20.000024
Tyrosine-protein kinase FgrHomo sapiens (human)Kd13.966723
Tyrosine-protein kinase FRKHomo sapiens (human)Kd20.000024
Tyrosine-protein kinase FynHomo sapiens (human)Kd20.000024
Tyrosine-protein kinase HCKHomo sapiens (human)Kd20.000024
Tyrosine-protein kinase ITK/TSKHomo sapiens (human)Kd10.000012
Tyrosine-protein kinase JAK1Homo sapiens (human)Kd15.450036
Tyrosine-protein kinase JAK2Homo sapiens (human)Kd13.476723
Tyrosine-protein kinase JAK3Homo sapiens (human)Kd5.235012
Tyrosine-protein kinase LckHomo sapiens (human)Kd17.580024
Tyrosine-protein kinase LynHomo sapiens (human)Kd20.000024
Tyrosine-protein kinase MerHomo sapiens (human)Kd17.825024
Tyrosine-protein kinase receptor Tie-1Homo sapiens (human)Kd5.600012
Tyrosine-protein kinase receptor TYRO3Homo sapiens (human)Kd6.000012
Tyrosine-protein kinase receptor UFOHomo sapiens (human)Kd5.055012
Tyrosine-protein kinase SrmsHomo sapiens (human)Kd10.000012
Tyrosine-protein kinase SYKHomo sapiens (human)Kd20.000024
Tyrosine-protein kinase TecHomo sapiens (human)Kd20.000024
Tyrosine-protein kinase TXKHomo sapiens (human)Kd10.000012
Tyrosine-protein kinase YesHomo sapiens (human)Kd17.850024
Tyrosine-protein kinase ZAP-70Homo sapiens (human)Kd10.000012
U5 small nuclear ribonucleoprotein 200 kDa helicaseHomo sapiens (human)Kd30.000012
UMP-CMP kinase Homo sapiens (human)Kd30.000012
Uncharacterized aarF domain-containing protein kinase 5Homo sapiens (human)Kd30.000012
Uncharacterized protein FLJ45252Homo sapiens (human)Kd30.000013
Uncharacterized serine/threonine-protein kinase SBK3Homo sapiens (human)Kd10.000012
Vascular endothelial growth factor receptor 1 Homo sapiens (human)Kd10.000012
Vascular endothelial growth factor receptor 2Homo sapiens (human)EC502.500011
Vascular endothelial growth factor receptor 2Homo sapiens (human)Kd10.000012
Vascular endothelial growth factor receptor 3Homo sapiens (human)Kd5.700012
Very long-chain specific acyl-CoA dehydrogenase, mitochondrialHomo sapiens (human)Kd30.000012
Wee1-like protein kinaseHomo sapiens (human)Kd20.000024
Wee1-like protein kinase 2Homo sapiens (human)Kd10.000012