An antagonist at G-protein-coupled receptor.
ChEBI ID: 88295
| Member | Definition | Class |
|---|---|---|
| gallein | A xanthene dye that is fluoran carrying four hydroxy substituents at positions 3', 4', 5' and 6'. | gallein |
| Timeframe | Studies, Drugs with This Role(%) | All Drugs % |
|---|---|---|
| pre-1990 | 1 (2.27) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 8 (18.18) | 29.6817 |
| 2010's | 30 (68.18) | 24.3611 |
| 2020's | 5 (11.36) | 2.80 |
| Publication Type | Studies, Drugs with this Role (%) | All Drugs (%) |
|---|---|---|
| Trials | 0 (0.00%) | 5.53% |
| Reviews | 1 (2.27%) | 6.00% |
| Case Studies | 0 (0.00%) | 4.05% |
| Observational | 0 (0.00%) | 0.25% |
| Other | 43 (97.73%) | 84.16% |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|---|---|---|---|---|
| Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2 | Homo sapiens (human) | IC50 | 0.2000 | 1 | 1 |
| Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1 | Homo sapiens (human) | IC50 | 0.2000 | 1 | 1 |