An EC 2.7.10.* (protein-tyrosine kinase) inhibitor that specifically blocks the action of non-specific protein-tyrosine kinase (EC 2.7.10.2).
| Member | Definition | Class |
|---|
| 1,2,3,4,5,6-hexabromocyclohexane | A bromohydrocarbon that is cyclohexane in which the hydrogen at positions 1,2,3,4,5 and 6 have been replaced by bromo groups. It is a potent inhibitor of JAK2 tyrosine kinase autophosphorylation. | 1,2,3,4,5,6-hexabromocyclohexane |
| 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz(h)imidazo(4,5-f)isoquinoline-7-one | An organic heterotetracyclic compound that is 1,6-dihydrobenzo[h]imidazo[4,5-f]isoquinolin-7-one bearing additional tert-butyl and fluoro substituents at positions 2 and 9 respectively. | 2-tert-butyl-9-fluoro-1,6-dihydrobenzo[h]imidazo[4,5-f]isoquinolin-7-one |
| acp-196 | A member of the class of imidazopyrazines that is imidazo[1,5-a]pyrazine substituted by 4-(pyridin-2-ylcarbamoyl)phenyl, (2S)-1-(but-2-ynoyl)pyrrolidin-2-yl, and amino groups at positions 1, 3 and 8, respectively. It is an irreversible second-generation Bruton's tyrosine kinase (BTK) inhibitor that is approved by the FDA for the treatment of adult patients with mantle cell lymphoma (MCL) who have received at least one prior therapy. | acalabrutinib |
| ag 1879 | A member of the class of pyrazolopyrimidine that is pyrazolo[3,4-d]pyrimidin-4-amine bearing additional tert-butyl and 4-chlorophenyl substituents at positions 1 and 3 respectively. It is a potent ATP-competitive inhibitor of the Src family of protein tyrosine kinases. | PP2 |
| ag-490 | A monocarboxylic acid amide obtained by formal condensation of the carboxy group of (2E)-2-cyano-3-(3,4-dihydroxyphenyl)prop-2-enoic acid with the amino group of benzylamine. | tyrphostin B42 |
| b 43 | A member of the class of pyrrolopyrimidines that is 7H-pyrrolo[2,3-d]pyrimidine substituted by amino, 4-phenoxyphenyl, and cyclopentyl groups at positions 4, 5 and 7, respectively. It is a potent inhibitor of Lck that inhibits Lck (64-509) and LckCD isoforms (IC50 of less than 1 and 2 nM, respectively). | RK-24466 |
| baricitinib | A pyrrolopyrimidine that is 7H-pyrrolo[2,3-d]pyrimidine substituted by a 1-[3-(cyanomethyl)-1-(ethanesulfonyl)azetidin-3-yl]-1H-pyrazol-4-yl group at position 5. It is an FDA approved selective Janus Kinase 1 and 2 (JAK1 and JAK2) inhibitor used for the treatment of rheumatoid arthritis. | baricitinib |
| curcumin | A beta-diketone that is methane in which two of the hydrogens are substituted by feruloyl groups. A natural dyestuff found in the root of Curcuma longa. | curcumin |
| delgocitinib | A pyrrolopyrimidine that is 7H-pyrrolo[2,3-d]pyrimidine substituted by a (3S,4R)-1-(cyanoacetyl)-3-methyl-1,6-diazaspiro[3.4]octan-6-yl group at position 4. It is a pan-Janus kinase (JAK) inhibitor and is approved for treatment of atopic dermatitis (AD) in Japan. | delgocitinib |
| incb-018424 | A pyrazole substituted at position 1 by a 2-cyano-1-cyclopentylethyl group and at position 3 by a pyrrolo[2,3-d]pyrimidin-4-yl group. Used as the phosphate salt for the treatment of patients with intermediate or high-risk myelofibrosis, including primary myelofibrosis, post-polycythemia vera myelofibrosis and post-essential thrombocythemia myelofibrosis. | ruxolitinib |
| lfm a13 | An enamide obtained by formal condensation of the carboxy group of (2Z)-2-cyano-3-hydroxybut-2-enoic acid with the amino group of 2,5-dibromoaniline. It is a dual-function inhibitor of Bruton's tyrosine kinase (BTK) and Polo-like kinases (PLK) that exhibits anticancer properties. | LFM-A13 |
| n-(cyanomethyl)-4-(2-((4-(4-morpholinyl)phenyl)amino)-4-pyrimidinyl)benzamide | A benzamide obtained by formal condensation of the carboxy group of 4-{2-[4-(morpholin-4-yl)anilino]pyrimidin-4-yl}benzoic acid with the primary amino group of aminoacetonitrile. It is an ATP-competitive JAK1/JAK2 inhibitor with IC50 of 11 nM and 18 nM, respectively. Used for the treatment of patients with intermediate- or high-risk myelofibrosis. | momelotinib |
| pci 32765 | A member of the class of acrylamides that is (3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine in which the piperidine nitrogen is replaced by an acryloyl group. A selective and covalent inhibitor of the enzyme Bruton's tyrosine kinase, it is used for treatment of B-cell malignancies. | ibrutinib |
| pf 956980 | A pyrrolopyrimidine that is 7H-pyrrolo[2,3-d]pyrimidine substituted at position 4 by a methyl[(3R,4R)-4-methyl-1-(pyrrolidin-1-ylcarbonyl)piperidin-3-yl]nitrilo group. It is a potent JAK3-selective chemical probe. | PF-956980 |
| saracatinib | A member of the class of quinazolines that is quinazoline substituted by (5-chloro-2H-1,3-benzodioxol-4-yl)amino, (oxan-4-yl)oxy and 2-(4-methylpiperazin-1-yl)ethoxy groups at positions 4, 5 and 7, respectively. It is a dual inhibitor of the tyrosine kinases c-Src and Abl (IC50 = 2.7 and 30 nM, respectively). Saracatinib was originally developed by AstraZeneca for the treatment of cancer but in 2019 it was granted orphan drug designation by the US Food and Drug Administration for the treatment of idiopathic pulmonary fibrosis (IPF), a type of lung disease that results in scarring (fibrosis) of the lungs. | saracatinib |
| Src Inhibitor-1 | A member of the class of quinazolines that is quinazoline which is substituted at position 4 by a p-phenoxyanilino group and at positions 6 and 7 by methoxy groups. It is a potent, competitive dual site (both the ATP- and peptide-binding) Src kinase inhibitor. Src Inhibitor-1 is one of the 'gold standards' for Src kinase inhibition that has been shown to use PP1 or PP2 in parallel with Src-I1 to inhbit Src family kinases. | Src Inhibitor-1 |
| SU6656 | A member of the class of oxindoles that is 3-methyleneoxindole in which the hydrogeh at position 5 has been replaced by a dimethylaminosulfonyl group and in which one of the hydrogens of the methylene group has been replaced by a 4,5,6,7-tetrahydro-indol-2-yl group. It is a specific inhibitor of Src family kinase. | SU6656 |
| terreic acid | | terreic acid |
| tg101209 | A member of the class of pyrimidines that is 5-methylpyrimidine-2,4-diamine in which the amino group at position 2 is substituted by a p-(4-methylpiperazin-1-yl)phenyl group, while that at position 4 is substituted by a m-(tert-butylsulfamoyl)phenyl group. A Janus kinase 2 (JAK2) inhibitor. | TG101209 |
| tofacitinib | A pyrrolopyrimidine that is pyrrolo[2,3-d]pyrimidine substituted at position 4 by an N-methyl,N-(1-cyanoacetyl-4-methylpiperidin-3-yl)amino moiety. Used as its citrate salt to treat moderately to severely active rheumatoid arthritis. | tofacitinib |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | Homo sapiens (human) | Potency | 29.2954 | 1 | 4 |
| 15-lipoxygenase, partial | Homo sapiens (human) | Potency | 20.2096 | 1 | 4 |
| 67.9K protein | Vaccinia virus | Potency | 5.9658 | 2 | 4 |
| acetylcholinesterase | Homo sapiens (human) | Potency | 63.6740 | 3 | 4 |
| activating transcription factor 6 | Homo sapiens (human) | Potency | 35.6534 | 2 | 2 |
| aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 22.2653 | 1 | 8 |
| Alpha-synuclein | Homo sapiens (human) | Potency | 10.6147 | 1 | 4 |
| Amyloid-beta precursor protein | Homo sapiens (human) | Potency | 29.0929 | 1 | 1 |
| apical membrane antigen 1, AMA1 | Plasmodium falciparum 3D7 | Potency | 15.1052 | 1 | 3 |
| AR protein | Homo sapiens (human) | Potency | 23.9205 | 9 | 18 |
| aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 31.5725 | 3 | 6 |
| arylsulfatase A | Homo sapiens (human) | Potency | 5.3126 | 1 | 2 |
| ATAD5 protein, partial | Homo sapiens (human) | Potency | 20.8280 | 4 | 6 |
| Ataxin-2 | Homo sapiens (human) | Potency | 37.8086 | 2 | 3 |
| ATP-dependent phosphofructokinase | Trypanosoma brucei brucei TREU927 | Potency | 10.9389 | 1 | 3 |
| ATPase family AAA domain-containing protein 5 | Homo sapiens (human) | Potency | 48.3696 | 2 | 4 |
| Bloom syndrome protein isoform 1 | Homo sapiens (human) | Potency | 15.8364 | 2 | 6 |
| bromodomain adjacent to zinc finger domain 2B | Homo sapiens (human) | Potency | 30.7369 | 1 | 3 |
| caspase 7, apoptosis-related cysteine protease | Homo sapiens (human) | Potency | 27.4727 | 1 | 1 |
| caspase-1 isoform alpha precursor | Homo sapiens (human) | Potency | 23.7358 | 1 | 2 |
| caspase-3 | Homo sapiens (human) | Potency | 27.4727 | 1 | 1 |
| Caspase-7 | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 18.2861 | 3 | 7 |
| cellular tumor antigen p53 isoform a | Homo sapiens (human) | Potency | 28.1084 | 2 | 5 |
| Chain A, 2-oxoglutarate Oxygenase | Homo sapiens (human) | Potency | 26.1670 | 1 | 6 |
| Chain A, ATP-DEPENDENT DNA HELICASE Q1 | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| Chain A, Beta-lactamase | Escherichia coli K-12 | Potency | 2.8184 | 1 | 1 |
| Chain A, Breast cancer type 1 susceptibility protein | Homo sapiens (human) | Potency | 5.0119 | 1 | 3 |
| Chain A, Cruzipain | Trypanosoma cruzi | Potency | 31.6228 | 1 | 2 |
| Chain A, Ferritin light chain | Equus caballus (horse) | Potency | 30.0732 | 2 | 5 |
| Chain A, HADH2 protein | Homo sapiens (human) | Potency | 25.6611 | 2 | 7 |
| Chain A, JmjC domain-containing histone demethylation protein 3A | Homo sapiens (human) | Potency | 65.8363 | 1 | 4 |
| Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | Homo sapiens (human) | Potency | 12.2366 | 1 | 3 |
| Chain A, Putative fructose-1,6-bisphosphate aldolase | Giardia intestinalis | Potency | 17.7407 | 1 | 1 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 22.7880 | 1 | 8 |
| Chain B, HADH2 protein | Homo sapiens (human) | Potency | 25.6611 | 2 | 7 |
| chaperonin-containing TCP-1 beta subunit homolog | Homo sapiens (human) | Potency | 100.0000 | 1 | 1 |
| chromobox protein homolog 1 | Homo sapiens (human) | Potency | 37.6783 | 2 | 4 |
| ClpP | Bacillus subtilis | Potency | 28.1838 | 1 | 1 |
| cytochrome P450 2C19 precursor | Homo sapiens (human) | Potency | 25.1189 | 1 | 2 |
| cytochrome P450 2C9 precursor | Homo sapiens (human) | Potency | 15.9370 | 1 | 2 |
| cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 16.9330 | 1 | 1 |
| cytochrome P450 2D6 | Homo sapiens (human) | Potency | 20.3092 | 1 | 3 |
| cytochrome P450 2D6 isoform 1 | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| cytochrome P450 3A4 isoform 1 | Homo sapiens (human) | Potency | 12.6597 | 2 | 10 |
| cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 10.9906 | 1 | 3 |
| cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 34.4925 | 1 | 3 |
| D(1A) dopamine receptor | Homo sapiens (human) | Potency | 8.3492 | 2 | 2 |
| DNA dC->dU-editing enzyme APOBEC-3F isoform a | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
| DNA dC->dU-editing enzyme APOBEC-3G isoform 1 | Homo sapiens (human) | Potency | 27.2454 | 2 | 3 |
| DNA polymerase beta | Homo sapiens (human) | Potency | 44.6684 | 1 | 1 |
| DNA polymerase eta isoform 1 | Homo sapiens (human) | Potency | 11.2202 | 1 | 1 |
| DNA polymerase iota isoform a (long) | Homo sapiens (human) | Potency | 45.2644 | 1 | 5 |
| DNA polymerase kappa isoform 1 | Homo sapiens (human) | Potency | 29.6936 | 1 | 7 |
| endonuclease IV | Escherichia coli | Potency | 11.0299 | 1 | 3 |
| estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 42.9745 | 8 | 14 |
| estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 27.4727 | 2 | 2 |
| estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 16.4401 | 8 | 8 |
| euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 14.3918 | 1 | 11 |
| EWS/FLI fusion protein | Homo sapiens (human) | Potency | 11.9037 | 4 | 32 |
| eyes absent homolog 2 isoform a | Homo sapiens (human) | Potency | 199.5260 | 1 | 1 |
| farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 46.9792 | 4 | 4 |
| flap endonuclease 1 | Homo sapiens (human) | Potency | 41.1937 | 1 | 3 |
| Fumarate hydratase | Homo sapiens (human) | Potency | 31.0605 | 1 | 4 |
| G | Vesicular stomatitis virus | Potency | 16.9330 | 1 | 1 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Potency | 12.6597 | 1 | 5 |
| geminin | Homo sapiens (human) | Potency | 13.2668 | 4 | 11 |
| GLI family zinc finger 3 | Homo sapiens (human) | Potency | 14.7033 | 3 | 3 |
| glp-1 receptor, partial | Homo sapiens (human) | Potency | 6.3514 | 1 | 2 |
| GLS protein | Homo sapiens (human) | Potency | 15.0436 | 2 | 4 |
| glucocerebrosidase | Homo sapiens (human) | Potency | 31.0378 | 1 | 3 |
| glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 43.2943 | 3 | 4 |
| Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 77.4286 | 1 | 1 |
| GTP-binding nuclear protein Ran isoform 1 | Homo sapiens (human) | Potency | 40.0748 | 1 | 2 |
| Guanine nucleotide-binding protein G | Homo sapiens (human) | Potency | 35.4813 | 1 | 1 |
| guanine nucleotide-binding protein G(i) subunit alpha-1 isoform 1 | Homo sapiens (human) | Potency | 10.0000 | 1 | 1 |
| heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) | Homo sapiens (human) | Potency | 32.0286 | 1 | 5 |
| heat shock protein beta-1 | Homo sapiens (human) | Potency | 27.3162 | 2 | 2 |
| hemoglobin subunit beta | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| Histamine H2 receptor | Cavia porcellus (domestic guinea pig) | Potency | 16.4255 | 2 | 16 |
| histone acetyltransferase KAT2A isoform 1 | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| Histone H2A.x | Cricetulus griseus (Chinese hamster) | Potency | 101.3910 | 1 | 1 |
| histone-lysine N-methyltransferase 2A isoform 2 precursor | Homo sapiens (human) | Potency | 21.1546 | 1 | 2 |
| HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 16.9330 | 1 | 1 |
| huntingtin isoform 2 | Homo sapiens (human) | Potency | 3.5481 | 1 | 1 |
| hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 52.2970 | 2 | 2 |
| hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | Homo sapiens (human) | Potency | 15.9775 | 2 | 6 |
| IDH1 | Homo sapiens (human) | Potency | 19.2753 | 1 | 3 |
| importin subunit beta-1 isoform 1 | Homo sapiens (human) | Potency | 30.2794 | 2 | 4 |
| Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 16.9330 | 1 | 2 |
| Integrin alpha-IIb | Homo sapiens (human) | Potency | 32.4648 | 1 | 2 |
| Integrin beta-3 | Homo sapiens (human) | Potency | 32.4648 | 1 | 2 |
| Interferon beta | Homo sapiens (human) | Potency | 12.4720 | 2 | 31 |
| interleukin 8 | Homo sapiens (human) | Potency | 84.1267 | 1 | 1 |
| lamin isoform A-delta10 | Homo sapiens (human) | Potency | 16.8625 | 2 | 7 |
| lethal factor (plasmid) | Bacillus anthracis str. A2012 | Potency | 9.5059 | 1 | 3 |
| lethal(3)malignant brain tumor-like protein 1 isoform I | Homo sapiens (human) | Potency | 15.8489 | 1 | 1 |
| Luciferase | Photinus pyralis (common eastern firefly) | Potency | 31.5672 | 3 | 5 |
| lysosomal alpha-glucosidase preproprotein | Homo sapiens (human) | Potency | 39.5068 | 1 | 1 |
| M-phase phosphoprotein 8 | Homo sapiens (human) | Potency | 28.9050 | 1 | 4 |
| Microtubule-associated protein tau | Homo sapiens (human) | Potency | 14.0673 | 2 | 11 |
| mitogen-activated protein kinase 1 | Homo sapiens (human) | Potency | 31.7702 | 2 | 6 |
| muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | Potency | 11.4642 | 2 | 2 |
| muscleblind-like protein 1 isoform 1 | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| neuropeptide S receptor isoform A | Homo sapiens (human) | Potency | 12.6748 | 1 | 3 |
| NFKB1 protein, partial | Homo sapiens (human) | Potency | 8.7649 | 2 | 4 |
| nonstructural protein 1 | Influenza A virus (A/WSN/1933(H1N1)) | Potency | 38.6721 | 1 | 3 |
| NPC intracellular cholesterol transporter 1 precursor | Homo sapiens (human) | Potency | 115.8210 | 1 | 1 |
| Nrf2 | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 21.6407 | 4 | 4 |
| nuclear factor erythroid 2-related factor 2 isoform 2 | Homo sapiens (human) | Potency | 18.4782 | 1 | 2 |
| nuclear factor NF-kappa-B p105 subunit isoform 1 | Homo sapiens (human) | Potency | 50.1187 | 1 | 1 |
| nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 3.4895 | 1 | 1 |
| Nuclear receptor ROR-gamma | Homo sapiens (human) | Potency | 33.4915 | 1 | 1 |
| nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 22.1406 | 2 | 11 |
| nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 62.3531 | 3 | 3 |
| Ornithine decarboxylase | Rattus norvegicus (Norway rat) | Potency | 0.0063 | 1 | 1 |
| parathyroid hormone/parathyroid hormone-related peptide receptor precursor | Homo sapiens (human) | Potency | 82.8514 | 1 | 2 |
| Parkin | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
| peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens (human) | Potency | 15.9740 | 2 | 2 |
| peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 20.3148 | 1 | 1 |
| peripheral myelin protein 22 isoform 1 | Homo sapiens (human) | Potency | 21.6680 | 1 | 2 |
| peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 27.0962 | 5 | 8 |
| peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 29.5047 | 5 | 5 |
| phosphopantetheinyl transferase | Bacillus subtilis | Potency | 61.7433 | 1 | 6 |
| PINK1 | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
| plasminogen precursor | Mus musculus (house mouse) | Potency | 3.7646 | 1 | 2 |
| polyprotein | Zika virus | Potency | 31.0605 | 1 | 4 |
| polyunsaturated fatty acid lipoxygenase ALOX12 | Homo sapiens (human) | Potency | 22.5358 | 1 | 2 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | Potency | 16.7186 | 1 | 5 |
| potassium voltage-gated channel subfamily H member 2 isoform d | Homo sapiens (human) | Potency | 6.3076 | 1 | 4 |
| PPM1D protein | Homo sapiens (human) | Potency | 12.3233 | 1 | 20 |
| pregnane X nuclear receptor | Homo sapiens (human) | Potency | 37.3019 | 2 | 2 |
| pregnane X receptor | Rattus norvegicus (Norway rat) | Potency | 79.4328 | 1 | 1 |
| progesterone receptor | Homo sapiens (human) | Potency | 39.8396 | 2 | 2 |
| pyruvate kinase PKM isoform a | Homo sapiens (human) | Potency | 28.1838 | 2 | 2 |
| pyruvate kinase PKM isoform b | Homo sapiens (human) | Potency | 0.0063 | 2 | 2 |
| Rap guanine nucleotide exchange factor 4 | Homo sapiens (human) | Potency | 70.7946 | 1 | 1 |
| RAR-related orphan receptor gamma | Mus musculus (house mouse) | Potency | 53.8126 | 2 | 2 |
| ras-related protein Rab-9A | Homo sapiens (human) | Potency | 103.9103 | 1 | 2 |
| regulator of G-protein signaling 4 | Homo sapiens (human) | Potency | 23.1903 | 1 | 4 |
| retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 9.2176 | 2 | 2 |
| retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 30.7735 | 4 | 4 |
| RGS12 | Homo sapiens (human) | Potency | 10.0000 | 1 | 1 |
| serine/threonine-protein kinase mTOR isoform 1 | Homo sapiens (human) | Potency | 15.7922 | 1 | 2 |
| SMAD family member 2 | Homo sapiens (human) | Potency | 41.5410 | 2 | 2 |
| SMAD family member 3 | Homo sapiens (human) | Potency | 41.5410 | 2 | 2 |
| Smad3 | Homo sapiens (human) | Potency | 15.7482 | 1 | 6 |
| snurportin-1 | Homo sapiens (human) | Potency | 30.2794 | 2 | 4 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | Potency | 39.8107 | 1 | 2 |
| survival motor neuron protein isoform d | Homo sapiens (human) | Potency | 17.1859 | 1 | 6 |
| TAR DNA-binding protein 43 | Homo sapiens (human) | Potency | 24.5937 | 1 | 3 |
| TDP1 protein | Homo sapiens (human) | Potency | 18.1870 | 2 | 28 |
| thioredoxin glutathione reductase | Schistosoma mansoni | Potency | 39.8107 | 1 | 1 |
| thioredoxin reductase | Rattus norvegicus (Norway rat) | Potency | 26.8558 | 3 | 8 |
| Thrombopoietin | Homo sapiens (human) | Potency | 6.7946 | 2 | 4 |
| thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 26.2910 | 2 | 6 |
| thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 40.8685 | 4 | 4 |
| thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 25.4607 | 5 | 5 |
| thyrotropin-releasing hormone receptor | Homo sapiens (human) | Potency | 27.7247 | 1 | 1 |
| transcriptional regulator ERG isoform 3 | Homo sapiens (human) | Potency | 27.8298 | 1 | 2 |
| tumor susceptibility gene 101 protein | Homo sapiens (human) | Potency | 19.9526 | 1 | 1 |
| tyrosine-protein kinase Yes | Homo sapiens (human) | Potency | 1.7271 | 2 | 7 |
| urokinase plasminogen activator surface receptor precursor | Mus musculus (house mouse) | Potency | 3.7646 | 1 | 2 |
| urokinase-type plasminogen activator precursor | Mus musculus (house mouse) | Potency | 3.7646 | 1 | 2 |
| USP1 protein, partial | Homo sapiens (human) | Potency | 24.8798 | 2 | 4 |
| v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 13.9840 | 2 | 2 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 39.5969 | 5 | 5 |
| vitamin D3 receptor isoform VDRA | Homo sapiens (human) | Potency | 47.1636 | 1 | 5 |
| Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 77.4286 | 1 | 1 |
| WRN | Homo sapiens (human) | Potency | 50.1187 | 1 | 1 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| 1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform a | Homo sapiens (human) | IC50 | 9.6995 | 2 | 2 |
| 10 kDa chaperonin | Escherichia coli | IC50 | 3.0000 | 2 | 2 |
| 10 kDa heat shock protein, mitochondrial | Homo sapiens (human) | IC50 | 8.3000 | 1 | 1 |
| 17-beta-hydroxysteroid dehydrogenase type 2 | Homo sapiens (human) | IC50 | 1.7300 | 1 | 1 |
| 3-phosphoinositide-dependent protein kinase 1 | Homo sapiens (human) | IC50 | 5.0100 | 2 | 2 |
| 5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 1 | 1 |
| 60 kDa chaperonin | Escherichia coli K-12 | IC50 | 250.0000 | 1 | 1 |
| 60 kDa chaperonin | Escherichia coli | IC50 | 3.0000 | 2 | 2 |
| 60 kDa heat shock protein, mitochondrial | Homo sapiens (human) | IC50 | 8.3000 | 1 | 1 |
| Acetylcholinesterase | Electrophorus electricus (electric eel) | IC50 | 132.1300 | 2 | 2 |
| Acetylcholinesterase | Homo sapiens (human) | IC50 | 5.0000 | 1 | 1 |
| alkaline phosphatase, germ cell type preproprotein | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| alkaline phosphatase, intestinal | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| alkaline phosphatase, tissue-nonspecific isozyme isoform 1 preproprotein | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 5.4000 | 1 | 1 |
| Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 5.4000 | 1 | 1 |
| Alpha-1D adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 5.4000 | 1 | 1 |
| Alpha-synuclein | Homo sapiens (human) | IC50 | 81.0100 | 2 | 2 |
| Amine oxidase [flavin-containing] A | Homo sapiens (human) | IC50 | 3.5000 | 3 | 3 |
| Amine oxidase [flavin-containing] A | Homo sapiens (human) | Ki | 0.7100 | 1 | 1 |
| Amine oxidase [flavin-containing] B | Homo sapiens (human) | IC50 | 2.5733 | 3 | 3 |
| Amine oxidase [flavin-containing] B | Homo sapiens (human) | Ki | 21.5000 | 1 | 1 |
| Aminopeptidase N | Homo sapiens (human) | IC50 | 15.5000 | 1 | 1 |
| Aminopeptidase N | Sus scrofa (pig) | IC50 | 15.5000 | 1 | 1 |
| Amyloid-beta precursor protein | Homo sapiens (human) | IC50 | 9.8541 | 30 | 30 |
| Angiopoietin-1 receptor | Homo sapiens (human) | IC50 | 9.2575 | 4 | 4 |
| AP2-associated protein kinase 1 | Homo sapiens (human) | IC50 | 0.0585 | 1 | 2 |
| ATP-binding cassette sub-family C member 3 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 1 |
| Aurora kinase B | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Beta lactamase (plasmid) | Pseudomonas aeruginosa | IC50 | 7.7510 | 1 | 1 |
| Beta-secretase 1 | Homo sapiens (human) | IC50 | 343.0000 | 1 | 1 |
| Bile salt export pump | Homo sapiens (human) | IC50 | 133.0000 | 1 | 1 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | IC50 | 1.6300 | 1 | 1 |
| Bromodomain testis-specific protein | Homo sapiens (human) | IC50 | 0.2300 | 1 | 1 |
| Bromodomain-containing protein 4 | Homo sapiens (human) | IC50 | 0.1300 | 4 | 4 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit beta | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit gamma | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 1 |
| Casein kinase I isoform delta | Homo sapiens (human) | IC50 | 0.0410 | 1 | 1 |
| CDGSH iron-sulfur domain-containing protein 1 | Homo sapiens (human) | IC50 | 2.3600 | 1 | 1 |
| CDGSH iron-sulfur domain-containing protein 1 | Homo sapiens (human) | Ki | 0.1010 | 1 | 1 |
| Chain A, Lck Kinase | Homo sapiens (human) | IC50 | 0.0200 | 1 | 1 |
| Chain A, Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | IC50 | 0.0027 | 1 | 1 |
| Chain A, Tyrosine-protein kinase | Homo sapiens (human) | IC50 | 0.0116 | 1 | 4 |
| Chain A, Tyrosine-protein kinase BTK | Homo sapiens (human) | IC50 | 0.0007 | 1 | 1 |
| Chain A, Tyrosine-protein kinase JAK2 | Homo sapiens (human) | IC50 | 0.0116 | 1 | 2 |
| Chain A, Tyrosine-protein kinase Lyn | Mus musculus (house mouse) | IC50 | 0.0090 | 1 | 2 |
| Cholinesterase | Equus caballus (horse) | IC50 | 300.0000 | 1 | 1 |
| Cholinesterase | Homo sapiens (human) | IC50 | 5.0000 | 1 | 1 |
| CREB-binding protein | Homo sapiens (human) | IC50 | 25.0000 | 4 | 4 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | IC50 | 275.0000 | 2 | 2 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | IC50 | 93.0500 | 6 | 6 |
| Cyclin-dependent kinase 3 | Homo sapiens (human) | IC50 | 500.0000 | 1 | 1 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Cyclin-G-associated kinase | Homo sapiens (human) | IC50 | 0.1280 | 1 | 2 |
| Cysteine protease | Trypanosoma brucei rhodesiense | IC50 | 7.7500 | 1 | 1 |
| Cytochrome P450 1A2 | Homo sapiens (human) | IC50 | 33.3397 | 3 | 3 |
| Cytochrome P450 2A6 | Homo sapiens (human) | IC50 | 0.0120 | 1 | 1 |
| Cytochrome P450 2B6 | Homo sapiens (human) | IC50 | 5.6005 | 2 | 2 |
| Cytochrome P450 2C19 | Homo sapiens (human) | IC50 | 13.1446 | 4 | 4 |
| Cytochrome P450 2C8 | Homo sapiens (human) | IC50 | 2.6401 | 3 | 3 |
| Cytochrome P450 2C9 | Homo sapiens (human) | IC50 | 6.0643 | 3 | 3 |
| Cytochrome P450 2D6 | Homo sapiens (human) | IC50 | 33.3602 | 3 | 3 |
| Cytochrome P450 3A4 | Homo sapiens (human) | IC50 | 10.3986 | 5 | 5 |
| Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens (human) | GI50 | 0.0090 | 1 | 1 |
| Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens (human) | IC50 | 12.8346 | 13 | 22 |
| D-amino-acid oxidase | Sus scrofa (pig) | IC50 | 1.0700 | 2 | 2 |
| Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens (human) | IC50 | 38.0533 | 3 | 3 |
| Dual specificity mitogen-activated protein kinase kinase 2 | Homo sapiens (human) | IC50 | 8.0533 | 3 | 3 |
| Dual specificity mitogen-activated protein kinase kinase 7 | Homo sapiens (human) | IC50 | 0.0815 | 1 | 8 |
| Ephrin type-A receptor 2 | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Ephrin type-B receptor 2 | Homo sapiens (human) | IC50 | 69.0000 | 1 | 2 |
| Epidermal growth factor receptor | Homo sapiens (human) | GI50 | 2.0493 | 7 | 7 |
| Epidermal growth factor receptor | Homo sapiens (human) | IC50 | 0.8473 | 47 | 57 |
| Epidermal growth factor receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Fibroblast growth factor receptor 1 | Homo sapiens (human) | IC50 | 5.7400 | 2 | 2 |
| Fibroblast growth factor receptor 2 | Homo sapiens (human) | IC50 | 1.2100 | 2 | 2 |
| Fibroblast growth factor receptor 3 | Homo sapiens (human) | IC50 | 1.4800 | 1 | 1 |
| Fibroblast growth factor receptor 4 | Homo sapiens (human) | IC50 | 1.4800 | 1 | 1 |
| G1/S-specific cyclin-E1 | Homo sapiens (human) | IC50 | 25.0000 | 1 | 1 |
| G2/mitotic-specific cyclin-B1 | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| G2/mitotic-specific cyclin-B2 | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| G2/mitotic-specific cyclin-B3 | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 1 | Rattus norvegicus (Norway rat) | IC50 | 54.6667 | 3 | 3 |
| Glutamate receptor ionotropic, NMDA 2A | Rattus norvegicus (Norway rat) | IC50 | 19.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2B | Rattus norvegicus (Norway rat) | IC50 | 22.5003 | 2 | 2 |
| Glutamate receptor ionotropic, NMDA 2C | Rattus norvegicus (Norway rat) | IC50 | 100.0000 | 1 | 1 |
| Glutathione S-transferase P | Homo sapiens (human) | IC50 | 69.0000 | 1 | 1 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | IC50 | 12.6500 | 3 | 3 |
| Glycogen synthase kinase-3 beta | Rattus norvegicus (Norway rat) | IC50 | 0.0660 | 1 | 1 |
| Heme oxygenase 1 | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 1 | 1 |
| Heme oxygenase 2 | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 1 | 1 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | IC50 | 215.0000 | 1 | 1 |
| Histone acetyltransferase p300 | Homo sapiens (human) | IC50 | 21.9167 | 6 | 6 |
| Histone deacetylase 1 | Homo sapiens (human) | IC50 | 187.0000 | 1 | 1 |
| Histone deacetylase 1 | Homo sapiens (human) | Ki | 50.7900 | 1 | 1 |
| Histone deacetylase 11 | Homo sapiens (human) | IC50 | 187.0000 | 1 | 1 |
| Histone deacetylase 2 | Homo sapiens (human) | IC50 | 187.0000 | 1 | 1 |
| Histone deacetylase 2 | Homo sapiens (human) | Ki | 97.6700 | 1 | 1 |
| Histone deacetylase 3 | Homo sapiens (human) | IC50 | 187.0000 | 1 | 1 |
| Histone deacetylase 4 | Homo sapiens (human) | IC50 | 187.0000 | 1 | 1 |
| Histone deacetylase 5 | Homo sapiens (human) | IC50 | 187.0000 | 1 | 1 |
| Histone deacetylase 6 | Homo sapiens (human) | IC50 | 93.5075 | 2 | 2 |
| Histone deacetylase 7 | Homo sapiens (human) | IC50 | 187.0000 | 1 | 1 |
| Histone deacetylase 8 | Homo sapiens (human) | IC50 | 187.0000 | 1 | 1 |
| Histone deacetylase 8 | Homo sapiens (human) | Ki | 64.9800 | 1 | 1 |
| Histone deacetylase 9 | Homo sapiens (human) | IC50 | 187.0000 | 1 | 1 |
| hypothetical protein SA1422 | Staphylococcus aureus subsp. aureus N315 | IC50 | 42.9000 | 2 | 2 |
| Inhibitor of nuclear factor kappa-B kinase subunit alpha | Homo sapiens (human) | IC50 | 500.0000 | 1 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit beta | Homo sapiens (human) | IC50 | 166.8667 | 3 | 3 |
| Insulin receptor | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | IC50 | 500.0000 | 1 | 1 |
| intestinal alkaline phosphatase precursor | Mus musculus (house mouse) | IC50 | 18.7000 | 1 | 1 |
| Lactoylglutathione lyase | Homo sapiens (human) | Ki | 0.0050 | 1 | 1 |
| large T antigen | Betapolyomavirus macacae | IC50 | 14.6100 | 1 | 1 |
| Lysine-specific histone demethylase 1A | Homo sapiens (human) | IC50 | 9.6000 | 1 | 1 |
| Macrophage colony-stimulating factor 1 receptor | Homo sapiens (human) | IC50 | 3.2725 | 2 | 2 |
| MAP kinase-activated protein kinase 2 | Homo sapiens (human) | IC50 | 10.0000 | 2 | 2 |
| MAP kinase-activated protein kinase 5 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | IC50 | 125.1500 | 4 | 4 |
| Maternal embryonic leucine zipper kinase | Homo sapiens (human) | IC50 | 0.3300 | 1 | 1 |
| Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase | Homo sapiens (human) | IC50 | 5.2090 | 2 | 2 |
| Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase | Homo sapiens (human) | Ki | 2.6199 | 2 | 2 |
| Microtubule-associated protein tau | Homo sapiens (human) | IC50 | 54.8750 | 4 | 4 |
| Mitogen-activated protein kinase 1 | Homo sapiens (human) | IC50 | 250.8900 | 2 | 2 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase 11 | Homo sapiens (human) | IC50 | 10.5000 | 2 | 2 |
| Mitogen-activated protein kinase 12 | Homo sapiens (human) | IC50 | 10.5000 | 2 | 2 |
| Mitogen-activated protein kinase 13 | Homo sapiens (human) | IC50 | 10.5000 | 2 | 2 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | IC50 | 131.3075 | 4 | 4 |
| Mitogen-activated protein kinase 3 | Homo sapiens (human) | IC50 | 1.7800 | 1 | 1 |
| Mitogen-activated protein kinase 8 | Homo sapiens (human) | IC50 | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase 9 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Multidrug resistance-associated protein 4 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 1 |
| NACHT, LRR and PYD domains-containing protein 3 | Homo sapiens (human) | IC50 | 24.2000 | 1 | 1 |
| Neuronal proto-oncogene tyrosine-protein kinase Src | Mus musculus (house mouse) | IC50 | 2.2000 | 1 | 1 |
| NF-kappa-B essential modulator | Homo sapiens (human) | IC50 | 500.0000 | 1 | 1 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | GI50 | 1.5240 | 1 | 1 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | IC50 | 6.4634 | 62 | 95 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | Ki | 0.0037 | 8 | 9 |
| Nuclear receptor subfamily 4 group A member 3 | Homo sapiens (human) | IC50 | 0.0780 | 1 | 1 |
| Oxysterols receptor LXR-beta | Homo sapiens (human) | Ki | 45.0000 | 1 | 1 |
| perilipin-1 | Homo sapiens (human) | IC50 | 9.1670 | 1 | 1 |
| perilipin-5 | Homo sapiens (human) | IC50 | 10.2320 | 1 | 1 |
| Peroxiredoxin-like 2A | Homo sapiens (human) | IC50 | 0.9000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | Homo sapiens (human) | IC50 | 500.0000 | 1 | 1 |
| Phospholipase A2 | Homo sapiens (human) | IC50 | 11.1000 | 1 | 1 |
| Platelet glycoprotein VI | Homo sapiens (human) | IC50 | 0.6650 | 1 | 2 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | IC50 | 170.4967 | 3 | 3 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | IC50 | 126.8725 | 4 | 4 |
| Polyamine deacetylase HDAC10 | Homo sapiens (human) | IC50 | 187.0000 | 1 | 1 |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens (human) | IC50 | 30.0000 | 1 | 1 |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | IC50 | 4.4000 | 2 | 2 |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | Ki | 1.1000 | 1 | 1 |
| Prostaglandin E synthase | Homo sapiens (human) | IC50 | 3.8500 | 4 | 4 |
| Prostaglandin G/H synthase 1 | Ovis aries (sheep) | IC50 | 63.8350 | 1 | 2 |
| Prostaglandin G/H synthase 2 | Homo sapiens (human) | IC50 | 63.8350 | 1 | 2 |
| Proteasome subunit beta type-5 | Homo sapiens (human) | IC50 | 10.0000 | 2 | 2 |
| Protein kinase C alpha type | Homo sapiens (human) | IC50 | 14.7333 | 3 | 3 |
| Protein kinase C beta type | Homo sapiens (human) | IC50 | 33.0000 | 1 | 1 |
| Protein kinase C delta type | Homo sapiens (human) | IC50 | 33.0000 | 1 | 1 |
| Protein kinase C epsilon type | Homo sapiens (human) | IC50 | 33.0000 | 1 | 1 |
| Protein kinase C eta type | Homo sapiens (human) | IC50 | 33.0000 | 1 | 1 |
| Protein kinase C gamma type | Homo sapiens (human) | IC50 | 33.0000 | 1 | 1 |
| Protein kinase C iota type | Homo sapiens (human) | IC50 | 33.0000 | 1 | 1 |
| Protein kinase C theta type | Homo sapiens (human) | IC50 | 33.0000 | 1 | 1 |
| Protein kinase C zeta type | Homo sapiens (human) | IC50 | 33.0000 | 1 | 1 |
| Protein-tyrosine kinase 6 | Homo sapiens (human) | IC50 | 133.5090 | 2 | 2 |
| Proto-oncogene tyrosine-protein kinase LCK | Mus musculus (house mouse) | IC50 | 0.0310 | 1 | 1 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | IC50 | 0.0262 | 3 | 3 |
| Proto-oncogene tyrosine-protein kinase Src | Gallus gallus (chicken) | IC50 | 0.1080 | 1 | 2 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | IC50 | 1.3613 | 27 | 29 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | Ki | 0.5000 | 2 | 2 |
| RAC-alpha serine/threonine-protein kinase | Homo sapiens (human) | IC50 | 5.0140 | 2 | 2 |
| RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens (human) | IC50 | 55.0000 | 2 | 2 |
| Receptor tyrosine-protein kinase erbB-2 | Homo sapiens (human) | IC50 | 2.0583 | 13 | 21 |
| Receptor tyrosine-protein kinase erbB-3 | Homo sapiens (human) | GI50 | 0.0040 | 1 | 1 |
| Receptor tyrosine-protein kinase erbB-4 | Homo sapiens (human) | IC50 | 0.0429 | 9 | 17 |
| Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | IC50 | 0.0225 | 1 | 2 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | GI50 | 0.1200 | 1 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | IC50 | 0.3660 | 3 | 3 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | IC50 | 31.7500 | 1 | 2 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | IC50 | 31.7500 | 1 | 2 |
| Rho-associated protein kinase 2 | Homo sapiens (human) | IC50 | 3.4000 | 2 | 2 |
| Ribosomal protein S6 kinase alpha-1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Ribosomal protein S6 kinase alpha-3 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Ribosomal protein S6 kinase alpha-5 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Ribosomal protein S6 kinase beta-1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 | Oryctolagus cuniculus (rabbit) | IC50 | 3.0000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 | Oryctolagus cuniculus (rabbit) | Ki | 5.8000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 2 | Homo sapiens (human) | IC50 | 7.0000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 2 | Homo sapiens (human) | Ki | 53.0000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 2 | Rattus norvegicus (Norway rat) | Ki | 5.8000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 3 | Homo sapiens (human) | IC50 | 7.0000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 3 | Homo sapiens (human) | Ki | 8.6000 | 1 | 1 |
| Serine/threonine-protein kinase Chk1 | Homo sapiens (human) | IC50 | 255.0000 | 2 | 2 |
| Serine/threonine-protein kinase D1 | Homo sapiens (human) | IC50 | 33.0000 | 1 | 1 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | IC50 | 33.0000 | 1 | 1 |
| Serine/threonine-protein kinase PAK 1 | Homo sapiens (human) | IC50 | 16.0000 | 1 | 1 |
| Serine/threonine-protein kinase PLK1 | Xenopus laevis (African clawed frog) | IC50 | 21.4000 | 2 | 2 |
| Serine/threonine-protein kinase PLK3 | Homo sapiens (human) | IC50 | 97.0250 | 8 | 8 |
| Serine/threonine-protein kinase Sgk1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase TBK1 | Homo sapiens (human) | IC50 | 5.7600 | 1 | 1 |
| Serine/threonine-protein kinase/endoribonuclease IRE1 | Homo sapiens (human) | IC50 | 3.5000 | 1 | 1 |
| Sigma intracellular receptor 2 | Rattus norvegicus (Norway rat) | IC50 | 0.5072 | 1 | 2 |
| Solute carrier family 22 member 3 | Homo sapiens (human) | IC50 | 7.9000 | 1 | 1 |
| Sortase A | Streptococcus mutans | IC50 | 10.2000 | 1 | 1 |
| Synaptic vesicular amine transporter | Rattus norvegicus (Norway rat) | IC50 | 0.0031 | 1 | 1 |
| Testosterone 17-beta-dehydrogenase 3 | Rattus norvegicus (Norway rat) | IC50 | 0.0028 | 2 | 3 |
| Thioredoxin reductase 1, cytoplasmic | Homo sapiens (human) | IC50 | 40.4667 | 3 | 3 |
| Thioredoxin reductase 2, mitochondrial | Homo sapiens (human) | IC50 | 40.4667 | 3 | 3 |
| Thioredoxin reductase 3 | Homo sapiens (human) | IC50 | 40.4667 | 3 | 3 |
| Thiosulfate sulfurtransferase | Homo sapiens (human) | IC50 | 56.0000 | 1 | 1 |
| Tissue factor | Homo sapiens (human) | IC50 | 0.0132 | 1 | 1 |
| toll-like receptor 9 | Homo sapiens (human) | IC50 | 8.3620 | 1 | 1 |
| TPA: protein transporter TIM10 | Saccharomyces cerevisiae S288C | IC50 | 19.7000 | 1 | 1 |
| Tyrosinase | Homo sapiens (human) | IC50 | 5.0000 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | IC50 | 125.0225 | 4 | 4 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | Ki | 0.5000 | 1 | 1 |
| Tyrosine-protein kinase Blk | Homo sapiens (human) | IC50 | 0.1034 | 8 | 16 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | IC50 | 0.3307 | 108 | 126 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | Ki | 0.2149 | 2 | 2 |
| Tyrosine-protein kinase BTK | Mus musculus (house mouse) | IC50 | 2.5000 | 1 | 1 |
| Tyrosine-protein kinase CSK | Homo sapiens (human) | IC50 | 2.5378 | 8 | 8 |
| Tyrosine-protein kinase Fgr | Homo sapiens (human) | IC50 | 0.0021 | 2 | 2 |
| Tyrosine-protein kinase FRK | Homo sapiens (human) | IC50 | 0.0541 | 2 | 2 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | IC50 | 34.4618 | 7 | 7 |
| Tyrosine-protein kinase HCK | Homo sapiens (human) | IC50 | 1.9310 | 4 | 4 |
| Tyrosine-protein kinase ITK/TSK | Homo sapiens (human) | IC50 | 1.3860 | 14 | 24 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | GI50 | 4.5112 | 2 | 2 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | IC50 | 0.1449 | 112 | 156 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | Ki | 0.0005 | 9 | 9 |
| Tyrosine-protein kinase JAK1 | Mus musculus (house mouse) | IC50 | 0.0150 | 2 | 2 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | GI50 | 3.7420 | 3 | 3 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | IC50 | 270.3062 | 134 | 187 |
| Tyrosine-protein kinase JAK2 | Rattus norvegicus (Norway rat) | IC50 | 3.5700 | 2 | 2 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | Ki | 0.0006 | 8 | 8 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | GI50 | 0.5030 | 1 | 1 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | IC50 | 584,064,706.1816 | 102 | 136 |
| Tyrosine-protein kinase JAK3 | Mus musculus (house mouse) | IC50 | 0.6640 | 5 | 5 |
| Tyrosine-protein kinase JAK3 | Rattus norvegicus (Norway rat) | IC50 | 1.2000 | 1 | 1 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | Ki | 0.0014 | 9 | 9 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | IC50 | 1.2847 | 17 | 18 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | Ki | 0.0008 | 1 | 1 |
| Tyrosine-protein kinase Lyn | Homo sapiens (human) | IC50 | 0.2051 | 4 | 4 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Tyrosine-protein kinase Tec | Homo sapiens (human) | IC50 | 0.0491 | 11 | 20 |
| Tyrosine-protein kinase TXK | Homo sapiens (human) | IC50 | 0.0998 | 6 | 14 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | IC50 | 71.4322 | 7 | 7 |
| Tyrosine-protein kinase ZAP-70 | Homo sapiens (human) | IC50 | 50,025.0000 | 2 | 2 |
| Tyrosyl-DNA phosphodiesterase 1 | Homo sapiens (human) | IC50 | 333.0000 | 1 | 1 |
| Vascular endothelial growth factor receptor 1 | Homo sapiens (human) | IC50 | 50.7600 | 2 | 2 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | IC50 | 8.9728 | 7 | 8 |
| Vascular endothelial growth factor receptor 3 | Homo sapiens (human) | IC50 | 5.3450 | 2 | 2 |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Rattus norvegicus (Norway rat) | IC50 | 100.0000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1D | Rattus norvegicus (Norway rat) | IC50 | 100.0000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1S | Rattus norvegicus (Norway rat) | IC50 | 100.0000 | 1 | 1 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 26S proteasome regulatory subunit 6B | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| 3-phosphoinositide-dependent protein kinase 1 | Homo sapiens (human) | EC50 | 0.0010 | 1 | 1 |
| 3-phosphoinositide-dependent protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| 5-hydroxytryptamine receptor 4 | Homo sapiens (human) | EC50 | 10.0000 | 1 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| 5'-AMP-activated protein kinase subunit gamma-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| 5'-AMP-activated protein kinase subunit gamma-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| AarF domain-containing protein kinase 1 | Homo sapiens (human) | Kd | 25.0362 | 1 | 6 |
| Actin-related protein 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Actin-related protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Activated CDC42 kinase 1 | Homo sapiens (human) | Kd | 14.9909 | 3 | 10 |
| Activin receptor type-1 | Homo sapiens (human) | Kd | 21.0004 | 3 | 10 |
| Activin receptor type-1B | Homo sapiens (human) | Kd | 20.0158 | 3 | 9 |
| Activin receptor type-2A | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Activin receptor type-2B | Homo sapiens (human) | Kd | 20.4309 | 3 | 9 |
| Acyl-CoA dehydrogenase family member 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Acyl-CoA dehydrogenase family member 11 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Adenine phosphoribosyltransferase | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Adenosine kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Adenylate kinase 2, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| ADP/ATP translocase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| ADP/ATP translocase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | Kd | 7.1667 | 2 | 3 |
| Alpha-synuclein | Homo sapiens (human) | Kd | 3.5000 | 4 | 4 |
| amino acid transporter AGP1 | Saccharomyces cerevisiae S288C | EC50 | 10.8000 | 1 | 1 |
| Angiopoietin-1 receptor | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Angiotensin-converting enzyme 2 | Homo sapiens (human) | EC50 | 2.9000 | 1 | 1 |
| Ankyrin repeat and protein kinase domain-containing protein 1 | Homo sapiens (human) | Kd | 6.7967 | 2 | 3 |
| AP2-associated protein kinase 1 | Homo sapiens (human) | Kd | 9.3164 | 8 | 16 |
| ATP-dependent 6-phosphofructokinase, platelet type | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| ATP-dependent RNA helicase DDX1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| ATP-dependent RNA helicase DDX3X | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| ATP-dependent RNA helicase DDX42 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| ATP-dependent RNA helicase DHX30 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Atypical kinase COQ8A, mitochondrial | Homo sapiens (human) | Kd | 21.0275 | 3 | 10 |
| Atypical kinase COQ8B, mitochondrial | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Aurora kinase A | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| Aurora kinase B | Homo sapiens (human) | Kd | 21.0525 | 3 | 10 |
| Aurora kinase C | Homo sapiens (human) | Kd | 9.5667 | 2 | 3 |
| BDNF/NT-3 growth factors receptor | Homo sapiens (human) | Kd | 6.7867 | 2 | 3 |
| Beta-adrenergic receptor kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| BMP-2-inducible protein kinase | Homo sapiens (human) | Kd | 11.9888 | 5 | 12 |
| Bone morphogenetic protein receptor type-1A | Homo sapiens (human) | Kd | 20.0067 | 3 | 9 |
| Bone morphogenetic protein receptor type-1B | Homo sapiens (human) | Kd | 20.2286 | 2 | 8 |
| Bone morphogenetic protein receptor type-2 | Homo sapiens (human) | Kd | 22.3256 | 3 | 9 |
| Breakpoint cluster region protein | Homo sapiens (human) | Kd | 20.2458 | 1 | 6 |
| Bromodomain-containing protein 4 | Homo sapiens (human) | Kd | 0.1230 | 1 | 1 |
| Calcium-dependent protein kinase 1 | Plasmodium falciparum 3D7 | Kd | 10.0000 | 1 | 2 |
| Calcium/calmodulin-dependent protein kinase kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Calcium/calmodulin-dependent protein kinase kinase 2 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Calcium/calmodulin-dependent protein kinase type 1 | Homo sapiens (human) | Kd | 2.9175 | 3 | 4 |
| Calcium/calmodulin-dependent protein kinase type 1D | Homo sapiens (human) | Kd | 3.9067 | 2 | 3 |
| Calcium/calmodulin-dependent protein kinase type 1G | Homo sapiens (human) | Kd | 20.3143 | 3 | 7 |
| Calcium/calmodulin-dependent protein kinase type II subunit alpha | Homo sapiens (human) | Kd | 4.5153 | 2 | 3 |
| Calcium/calmodulin-dependent protein kinase type II subunit beta | Homo sapiens (human) | Kd | 6.7700 | 2 | 3 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta | Homo sapiens (human) | Kd | 11.5642 | 3 | 9 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma | Homo sapiens (human) | Kd | 12.3554 | 3 | 9 |
| Calcium/calmodulin-dependent protein kinase type IV | Homo sapiens (human) | Kd | 20.0218 | 3 | 9 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | Kd | 20.3997 | 3 | 9 |
| cAMP-dependent protein kinase catalytic subunit beta | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| cAMP-dependent protein kinase catalytic subunit gamma | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| cAMP-dependent protein kinase catalytic subunit PRKX | Homo sapiens (human) | Kd | 15.0000 | 3 | 4 |
| cAMP-dependent protein kinase type II-alpha regulatory subunit | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Casein kinase I isoform alpha | Homo sapiens (human) | Kd | 23.1143 | 2 | 7 |
| Casein kinase I isoform alpha-like | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Casein kinase I isoform delta | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Casein kinase I isoform epsilon | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Casein kinase I isoform gamma-1 | Homo sapiens (human) | Kd | 15.3255 | 3 | 8 |
| Casein kinase I isoform gamma-2 | Homo sapiens (human) | Kd | 20.0294 | 3 | 9 |
| Casein kinase I isoform gamma-3 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Casein kinase II subunit alpha | Homo sapiens (human) | Kd | 8.0667 | 2 | 3 |
| Casein kinase II subunit alpha' | Homo sapiens (human) | Kd | 16.3776 | 3 | 9 |
| Cell division control protein 2 homolog | Plasmodium falciparum 3D7 | Kd | 10.0000 | 1 | 2 |
| Cell division cycle 7-related protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| cGMP-dependent protein kinase 1 | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| cGMP-dependent protein kinase 2 | Homo sapiens (human) | Kd | 6.8967 | 2 | 3 |
| Choline-phosphate cytidylyltransferase A | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Chromodomain-helicase-DNA-binding protein 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Citron Rho-interacting kinase | Homo sapiens (human) | Kd | 15.6299 | 3 | 9 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Cyclin-dependent kinase 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 11A | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Cyclin-dependent kinase 11B | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Cyclin-dependent kinase 12 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Cyclin-dependent kinase 13 | Homo sapiens (human) | Kd | 25.0000 | 2 | 8 |
| Cyclin-dependent kinase 14 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Cyclin-dependent kinase 15 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Cyclin-dependent kinase 16 | Homo sapiens (human) | Kd | 20.1291 | 3 | 9 |
| Cyclin-dependent kinase 17 | Homo sapiens (human) | Kd | 20.1536 | 3 | 9 |
| Cyclin-dependent kinase 18 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Cyclin-dependent kinase 19 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | Kd | 21.2113 | 3 | 10 |
| Cyclin-dependent kinase 3 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Cyclin-dependent kinase 4 | Homo sapiens (human) | Kd | 22.0000 | 3 | 10 |
| Cyclin-dependent kinase 6 | Homo sapiens (human) | Kd | 25.5593 | 1 | 6 |
| Cyclin-dependent kinase 7 | Homo sapiens (human) | Kd | 22.5889 | 3 | 9 |
| Cyclin-dependent kinase 8 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Cyclin-dependent kinase 9 | Homo sapiens (human) | Kd | 20.0823 | 3 | 9 |
| Cyclin-dependent kinase-like 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Cyclin-dependent kinase-like 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Cyclin-dependent kinase-like 3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Cyclin-dependent kinase-like 5 | Homo sapiens (human) | Kd | 20.0000 | 2 | 4 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| Cyclin-G-associated kinase | Homo sapiens (human) | Kd | 9.5979 | 7 | 14 |
| Cysteine--tRNA ligase, cytoplasmic | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Cytochrome c1, heme protein, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens (human) | Kd | 4.3760 | 4 | 7 |
| dCTP pyrophosphatase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Death-associated protein kinase 1 | Homo sapiens (human) | Kd | 6.6907 | 2 | 3 |
| Death-associated protein kinase 2 | Homo sapiens (human) | Kd | 6.6990 | 2 | 3 |
| Death-associated protein kinase 3 | Homo sapiens (human) | Kd | 7.5222 | 3 | 4 |
| Delta(24)-sterol reductase | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Deoxycytidine kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Discoidin domain-containing receptor 2 | Homo sapiens (human) | Kd | 24.6978 | 3 | 9 |
| DNA replication licensing factor MCM4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| DNA topoisomerase 2-alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| DNA topoisomerase 2-beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| DnaJ homolog subfamily A member 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Dual serine/threonine and tyrosine protein kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens (human) | Kd | 19.1477 | 3 | 9 |
| Dual specificity mitogen-activated protein kinase kinase 2 | Homo sapiens (human) | Kd | 24.0000 | 3 | 11 |
| Dual specificity mitogen-activated protein kinase kinase 3 | Homo sapiens (human) | Kd | 22.2744 | 3 | 9 |
| Dual specificity mitogen-activated protein kinase kinase 4 | Homo sapiens (human) | Kd | 12.9500 | 3 | 4 |
| Dual specificity mitogen-activated protein kinase kinase 5 | Homo sapiens (human) | Kd | 21.2804 | 2 | 8 |
| Dual specificity mitogen-activated protein kinase kinase 6 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Dual specificity mitogen-activated protein kinase kinase 7 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Dual specificity protein kinase CLK1 | Homo sapiens (human) | Kd | 15.4929 | 3 | 10 |
| Dual specificity protein kinase CLK2 | Homo sapiens (human) | Kd | 17.1295 | 4 | 10 |
| Dual specificity protein kinase CLK3 | Homo sapiens (human) | Kd | 21.4286 | 3 | 7 |
| Dual specificity protein kinase CLK4 | Homo sapiens (human) | Kd | 16.2000 | 4 | 7 |
| Dual specificity protein kinase TTK | Homo sapiens (human) | Kd | 20.0686 | 3 | 7 |
| Dual specificity testis-specific protein kinase 1 | Homo sapiens (human) | Kd | 20.0000 | 3 | 6 |
| Dual specificity testis-specific protein kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | Kd | 21.5337 | 2 | 9 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B | Homo sapiens (human) | Kd | 15.0000 | 3 | 4 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 2 | Homo sapiens (human) | Kd | 6.8500 | 1 | 2 |
| Dynamin-like 120 kDa protein, mitochondrial | Homo sapiens (human) | Kd | 25.1175 | 1 | 6 |
| eIF-2-alpha kinase GCN2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| EKC/KEOPS complex subunit TP53RK | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Electron transfer flavoprotein subunit beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Elongation factor Tu, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Ephrin type-A receptor 1 | Homo sapiens (human) | Kd | 18.7512 | 3 | 8 |
| Ephrin type-A receptor 2 | Homo sapiens (human) | Kd | 18.1067 | 4 | 10 |
| Ephrin type-A receptor 3 | Homo sapiens (human) | Kd | 56.5250 | 3 | 4 |
| Ephrin type-A receptor 4 | Homo sapiens (human) | Kd | 20.1019 | 3 | 9 |
| Ephrin type-A receptor 5 | Homo sapiens (human) | Kd | 20.2646 | 3 | 9 |
| Ephrin type-A receptor 6 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Ephrin type-A receptor 7 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Ephrin type-A receptor 8 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Ephrin type-B receptor 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Ephrin type-B receptor 2 | Homo sapiens (human) | Kd | 25.8468 | 4 | 11 |
| Ephrin type-B receptor 3 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Ephrin type-B receptor 4 | Homo sapiens (human) | Kd | 20.4309 | 3 | 9 |
| Ephrin type-B receptor 6 | Homo sapiens (human) | Kd | 20.8378 | 2 | 8 |
| Epidermal growth factor receptor | Homo sapiens (human) | EC50 | 1.4548 | 2 | 4 |
| Epidermal growth factor receptor | Homo sapiens (human) | Kd | 11.6850 | 25 | 45 |
| Epithelial discoidin domain-containing receptor 1 | Homo sapiens (human) | Kd | 20.4890 | 3 | 9 |
| Eukaryotic peptide chain release factor GTP-binding subunit ERF3B | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Eukaryotic translation initiation factor 2-alpha kinase 1 | Homo sapiens (human) | Kd | 20.0479 | 2 | 7 |
| Eukaryotic translation initiation factor 5B | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Exosome RNA helicase MTR4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Ferrochelatase, mitochondrial | Homo sapiens (human) | Kd | 26.2000 | 2 | 7 |
| Fibroblast growth factor receptor 1 | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| Fibroblast growth factor receptor 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Fibroblast growth factor receptor 3 | Homo sapiens (human) | Kd | 10.0000 | 4 | 6 |
| Fibroblast growth factor receptor 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Focal adhesion kinase 1 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| G protein-coupled receptor kinase 4 | Homo sapiens (human) | Kd | 8.0500 | 1 | 2 |
| G protein-coupled receptor kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| General transcription and DNA repair factor IIH helicase subunit XPD | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Glycine--tRNA ligase | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Glycogen phosphorylase, brain form | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Glycogen phosphorylase, liver form | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Glycogen synthase kinase-3 alpha | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| GTP-binding nuclear protein Ran | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Guanine nucleotide-binding protein G(i) subunit alpha-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Heme oxygenase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | Kd | 20.0000 | 5 | 14 |
| High affinity nerve growth factor receptor | Homo sapiens (human) | Kd | 21.4375 | 3 | 8 |
| Homeodomain-interacting protein kinase 1 | Homo sapiens (human) | Kd | 5.6000 | 1 | 2 |
| Homeodomain-interacting protein kinase 2 | Homo sapiens (human) | Kd | 5.5000 | 1 | 2 |
| Homeodomain-interacting protein kinase 3 | Homo sapiens (human) | Kd | 5.6000 | 1 | 2 |
| Homeodomain-interacting protein kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Hormonally up-regulated neu tumor-associated kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Inhibitor of nuclear factor kappa-B kinase subunit alpha | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Inhibitor of nuclear factor kappa-B kinase subunit beta | Homo sapiens (human) | Kd | 6.1500 | 1 | 2 |
| Inhibitor of nuclear factor kappa-B kinase subunit epsilon | Homo sapiens (human) | Kd | 20.1400 | 3 | 10 |
| Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Insulin receptor | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Insulin receptor-related protein | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Integrin-linked protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Interferon-induced, double-stranded RNA-activated protein kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Interleukin-1 receptor-associated kinase 1 | Homo sapiens (human) | Kd | 23.7863 | 2 | 8 |
| Interleukin-1 receptor-associated kinase 3 | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| Interleukin-1 receptor-associated kinase 4 | Homo sapiens (human) | Kd | 25.0000 | 2 | 8 |
| Isoleucine--tRNA ligase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| LAP4 | Saccharomyces cerevisiae (brewer's yeast) | EC50 | 4.8230 | 1 | 1 |
| Leucine-rich repeat serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 0.5575 | 2 | 4 |
| Leukocyte tyrosine kinase receptor | Homo sapiens (human) | Kd | 6.8133 | 2 | 3 |
| Leukotriene C4 synthase | Cavia porcellus (domestic guinea pig) | Kd | 10.0000 | 1 | 2 |
| LIM domain kinase 1 | Homo sapiens (human) | Kd | 22.3432 | 3 | 9 |
| LIM domain kinase 2 | Homo sapiens (human) | Kd | 24.5455 | 3 | 11 |
| Long-chain-fatty-acid--CoA ligase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Lymphocyte antigen 96 | Homo sapiens (human) | Kd | 379.0000 | 1 | 1 |
| Macrophage colony-stimulating factor 1 receptor | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Macrophage-stimulating protein receptor | Homo sapiens (human) | Kd | 25.0000 | 2 | 8 |
| MAP kinase-activated protein kinase 2 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| MAP kinase-activated protein kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| MAP kinase-activated protein kinase 5 | Homo sapiens (human) | Kd | 20.3464 | 3 | 9 |
| MAP kinase-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| MAP kinase-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 3.9333 | 2 | 3 |
| MAP/microtubule affinity-regulating kinase 3 | Homo sapiens (human) | Kd | 12.9034 | 3 | 9 |
| MAP/microtubule affinity-regulating kinase 4 | Homo sapiens (human) | Kd | 22.5000 | 3 | 8 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | Kd | 9.5522 | 15 | 23 |
| Maternal embryonic leucine zipper kinase | Homo sapiens (human) | Kd | 22.4667 | 3 | 9 |
| Megakaryocyte-associated tyrosine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Membrane-associated progesterone receptor component 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase | Homo sapiens (human) | Kd | 21.2817 | 4 | 10 |
| Microtubule-associated serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 5.2600 | 1 | 2 |
| Midasin | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Misshapen-like kinase 1 | Homo sapiens (human) | Kd | 23.3333 | 2 | 6 |
| Mitogen-activated protein kinase 1 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | Kd | 21.1191 | 3 | 10 |
| Mitogen-activated protein kinase 11 | Homo sapiens (human) | Kd | 22.5000 | 3 | 8 |
| Mitogen-activated protein kinase 12 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Mitogen-activated protein kinase 13 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| Mitogen-activated protein kinase 15 | Homo sapiens (human) | Kd | 24.5455 | 3 | 11 |
| Mitogen-activated protein kinase 3 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Mitogen-activated protein kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Mitogen-activated protein kinase 6 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Mitogen-activated protein kinase 7 | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| Mitogen-activated protein kinase 8 | Homo sapiens (human) | Kd | 20.5399 | 3 | 10 |
| Mitogen-activated protein kinase 9 | Homo sapiens (human) | Kd | 21.1137 | 3 | 10 |
| Mitogen-activated protein kinase kinase kinase 1 | Homo sapiens (human) | Kd | 20.7614 | 2 | 8 |
| Mitogen-activated protein kinase kinase kinase 10 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Mitogen-activated protein kinase kinase kinase 11 | Homo sapiens (human) | Kd | 20.2111 | 3 | 9 |
| Mitogen-activated protein kinase kinase kinase 12 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Mitogen-activated protein kinase kinase kinase 13 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Mitogen-activated protein kinase kinase kinase 15 | Homo sapiens (human) | Kd | 5.5500 | 1 | 2 |
| Mitogen-activated protein kinase kinase kinase 19 | Homo sapiens (human) | Kd | 5.1350 | 1 | 2 |
| Mitogen-activated protein kinase kinase kinase 2 | Homo sapiens (human) | Kd | 24.4490 | 2 | 9 |
| Mitogen-activated protein kinase kinase kinase 20 | Homo sapiens (human) | Kd | 17.1878 | 3 | 9 |
| Mitogen-activated protein kinase kinase kinase 3 | Homo sapiens (human) | Kd | 23.7688 | 2 | 8 |
| Mitogen-activated protein kinase kinase kinase 4 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Mitogen-activated protein kinase kinase kinase 5 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Mitogen-activated protein kinase kinase kinase 6 | Homo sapiens (human) | Kd | 25.0000 | 2 | 8 |
| Mitogen-activated protein kinase kinase kinase 7 | Homo sapiens (human) | Kd | 5.3650 | 1 | 2 |
| Mitogen-activated protein kinase kinase kinase 9 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Mitogen-activated protein kinase kinase kinase kinase 1 | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| Mitogen-activated protein kinase kinase kinase kinase 2 | Homo sapiens (human) | Kd | 23.3500 | 2 | 8 |
| Mitogen-activated protein kinase kinase kinase kinase 3 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Mitogen-activated protein kinase kinase kinase kinase 4 | Homo sapiens (human) | Kd | 21.1121 | 3 | 10 |
| Mitogen-activated protein kinase kinase kinase kinase 5 | Homo sapiens (human) | Kd | 23.0098 | 3 | 9 |
| Mitotic checkpoint serine/threonine-protein kinase BUB1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Multifunctional protein ADE2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Muscle, skeletal receptor tyrosine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Myosin light chain kinase 2, skeletal/cardiac muscle | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Myosin light chain kinase 3 | Homo sapiens (human) | Kd | 25.5556 | 2 | 9 |
| Myosin light chain kinase family member 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Myosin light chain kinase, smooth muscle | Gallus gallus (chicken) | Kd | 10.0000 | 1 | 1 |
| Myosin light chain kinase, smooth muscle | Homo sapiens (human) | Kd | 22.2622 | 3 | 9 |
| Myosin-10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Myosin-14 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Myosin-IIIa | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Myosin-IIIb | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Myotonin-protein kinase | Homo sapiens (human) | Kd | 4.9000 | 2 | 3 |
| NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Non-receptor tyrosine-protein kinase TNK1 | Homo sapiens (human) | Kd | 14.8823 | 4 | 11 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | EC50 | 0.3375 | 3 | 4 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | Kd | 12.5613 | 6 | 13 |
| NPYLR7B | Aedes aegypti (yellow fever mosquito) | EC50 | 20.0000 | 1 | 2 |
| NT-3 growth factor receptor | Homo sapiens (human) | Kd | 6.7767 | 2 | 3 |
| NUAK family SNF1-like kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| NUAK family SNF1-like kinase 2 | Homo sapiens (human) | Kd | 16.8222 | 4 | 9 |
| Nuclear factor erythroid 2-related factor 2 | Homo sapiens (human) | EC50 | 21.0000 | 1 | 1 |
| Nucleolar GTP-binding protein 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Nucleoside diphosphate kinase B | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Obg-like ATPase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| PAS domain-containing serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Peripheral plasma membrane protein CASK | Homo sapiens (human) | Kd | 5.7500 | 1 | 2 |
| Peroxisomal acyl-coenzyme A oxidase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Peroxisomal acyl-coenzyme A oxidase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Phenylalanine--tRNA ligase beta subunit | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Phosphatidylethanolamine-binding protein 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Phosphatidylinositol 4-kinase beta | Homo sapiens (human) | Kd | 6.7000 | 1 | 2 |
| Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | Homo sapiens (human) | Kd | 10.0000 | 12 | 22 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 4 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 beta | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma | Homo sapiens (human) | Kd | 25.0000 | 2 | 8 |
| Phosphorylase b kinase gamma catalytic chain, liver/testis isoform | Homo sapiens (human) | Kd | 20.5404 | 3 | 10 |
| Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform | Homo sapiens (human) | Kd | 8.5667 | 2 | 3 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | Kd | 20.0701 | 3 | 9 |
| Probable ATP-dependent RNA helicase DDX6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Procathepsin L | Homo sapiens (human) | EC50 | 2.9000 | 1 | 1 |
| Prostaglandin G/H synthase 2 | Homo sapiens (human) | Kd | 6.2500 | 1 | 2 |
| Protein kinase C alpha type | Homo sapiens (human) | Kd | 22.7772 | 1 | 6 |
| Protein kinase C beta type | Homo sapiens (human) | Kd | 29.3873 | 1 | 6 |
| Protein kinase C delta type | Homo sapiens (human) | Kd | 16.9201 | 3 | 9 |
| Protein kinase C epsilon type | Homo sapiens (human) | Kd | 6.8433 | 2 | 3 |
| Protein kinase C eta type | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Protein kinase C iota type | Homo sapiens (human) | Kd | 25.0000 | 2 | 8 |
| Protein kinase C theta type | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Protein kinase C zeta type | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Protein-tyrosine kinase 2-beta | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Protein-tyrosine kinase 6 | Homo sapiens (human) | Kd | 16.7330 | 3 | 9 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | Kd | 8.4924 | 7 | 16 |
| Proto-oncogene tyrosine-protein kinase ROS | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Proto-oncogene tyrosine-protein kinase Src | Gallus gallus (chicken) | Kd | 0.2960 | 1 | 1 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | Kd | 16.6921 | 3 | 9 |
| Putative heat shock protein HSP 90-beta 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Putative nucleoside diphosphate kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Pyridoxal kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Rab-like protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| RAC-alpha serine/threonine-protein kinase | Homo sapiens (human) | Kd | 24.5455 | 3 | 11 |
| RAC-beta serine/threonine-protein kinase | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| RAC-gamma serine/threonine-protein kinase | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Ras-related protein Rab-10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 7 |
| Ras-related protein Rab-27A | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Ras-related protein Rab-6A | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Receptor tyrosine-protein kinase erbB-2 | Homo sapiens (human) | Kd | 4.3371 | 4 | 7 |
| Receptor tyrosine-protein kinase erbB-3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Receptor tyrosine-protein kinase erbB-4 | Homo sapiens (human) | Kd | 3.3672 | 3 | 6 |
| Receptor-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 16.6732 | 3 | 9 |
| Receptor-interacting serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 20.3088 | 1 | 6 |
| Receptor-interacting serine/threonine-protein kinase 4 | Homo sapiens (human) | Kd | 6.0500 | 1 | 2 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | Kd | 13.1430 | 13 | 26 |
| Replicase polyprotein 1a | Severe acute respiratory syndrome-related coronavirus | EC50 | 2.9000 | 1 | 1 |
| Replicase polyprotein 1ab | Betacoronavirus England 1 | EC50 | 2.9000 | 1 | 1 |
| Replicase polyprotein 1ab | Human coronavirus 229E | EC50 | 2.9000 | 1 | 1 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | EC50 | 6.4500 | 2 | 2 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | EC50 | 6.4500 | 2 | 2 |
| Rho-associated protein kinase 1 | Homo sapiens (human) | Kd | 8.2404 | 2 | 8 |
| Rho-associated protein kinase 2 | Homo sapiens (human) | Kd | 8.7964 | 2 | 8 |
| Rhodopsin kinase GRK1 | Homo sapiens (human) | Kd | 5.3650 | 1 | 2 |
| Rhodopsin kinase GRK7 | Homo sapiens (human) | Kd | 2.4200 | 1 | 2 |
| Ribosomal protein S6 kinase alpha-1 | Homo sapiens (human) | Kd | 16.6733 | 5 | 12 |
| Ribosomal protein S6 kinase alpha-2 | Homo sapiens (human) | Kd | 4.7929 | 5 | 7 |
| Ribosomal protein S6 kinase alpha-3 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Ribosomal protein S6 kinase alpha-4 | Homo sapiens (human) | Kd | 19.1950 | 5 | 12 |
| Ribosomal protein S6 kinase alpha-5 | Homo sapiens (human) | Kd | 19.1783 | 5 | 12 |
| Ribosomal protein S6 kinase alpha-6 | Homo sapiens (human) | Kd | 16.7493 | 6 | 14 |
| Ribosomal protein S6 kinase beta-1 | Homo sapiens (human) | Kd | 25.0000 | 2 | 8 |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens (human) | Kd | 30.0000 | 1 | 8 |
| RNA cytidine acetyltransferase | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| RPL19A | Saccharomyces cerevisiae (brewer's yeast) | EC50 | 0.8525 | 2 | 2 |
| S-adenosylmethionine synthase isoform type-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Septin-9 | Homo sapiens (human) | Kd | 25.0140 | 1 | 6 |
| Serine/threonine-protein kinase 10 | Homo sapiens (human) | Kd | 21.2979 | 3 | 9 |
| Serine/threonine-protein kinase 16 | Homo sapiens (human) | Kd | 19.0857 | 3 | 9 |
| Serine/threonine-protein kinase 17A | Homo sapiens (human) | Kd | 8.7333 | 2 | 3 |
| Serine/threonine-protein kinase 17B | Homo sapiens (human) | Kd | 7.8333 | 2 | 3 |
| Serine/threonine-protein kinase 24 | Homo sapiens (human) | Kd | 21.4286 | 3 | 7 |
| Serine/threonine-protein kinase 25 | Homo sapiens (human) | Kd | 8.7667 | 2 | 3 |
| Serine/threonine-protein kinase 26 | Homo sapiens (human) | Kd | 23.3100 | 3 | 10 |
| Serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 21.6909 | 4 | 11 |
| Serine/threonine-protein kinase 32A | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Serine/threonine-protein kinase 32B | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase 32C | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase 33 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase 35 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Serine/threonine-protein kinase 36 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase 38 | Homo sapiens (human) | Kd | 20.0000 | 2 | 4 |
| Serine/threonine-protein kinase 38-like | Homo sapiens (human) | Kd | 15.0000 | 3 | 4 |
| Serine/threonine-protein kinase 4 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Serine/threonine-protein kinase A-Raf | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Serine/threonine-protein kinase ATR | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | Kd | 18.8667 | 5 | 12 |
| Serine/threonine-protein kinase BRSK1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase BRSK2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase Chk1 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Serine/threonine-protein kinase Chk2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Serine/threonine-protein kinase D1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase D2 | Homo sapiens (human) | Kd | 20.0590 | 3 | 9 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | Kd | 21.0650 | 3 | 10 |
| Serine/threonine-protein kinase DCLK1 | Homo sapiens (human) | Kd | 5.5893 | 2 | 3 |
| Serine/threonine-protein kinase DCLK2 | Homo sapiens (human) | Kd | 6.9200 | 2 | 3 |
| Serine/threonine-protein kinase DCLK3 | Homo sapiens (human) | Kd | 0.0703 | 3 | 4 |
| Serine/threonine-protein kinase ICK | Homo sapiens (human) | Kd | 21.3400 | 2 | 8 |
| Serine/threonine-protein kinase LATS1 | Homo sapiens (human) | Kd | 20.2093 | 3 | 9 |
| Serine/threonine-protein kinase LATS2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase MAK | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Serine/threonine-protein kinase MARK1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase MARK2 | Homo sapiens (human) | Kd | 11.0142 | 3 | 9 |
| Serine/threonine-protein kinase MRCK alpha | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Serine/threonine-protein kinase MRCK beta | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| Serine/threonine-protein kinase MRCK gamma | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Serine/threonine-protein kinase mTOR | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Serine/threonine-protein kinase N1 | Homo sapiens (human) | Kd | 10.3782 | 4 | 10 |
| Serine/threonine-protein kinase N2 | Homo sapiens (human) | Kd | 19.0521 | 3 | 9 |
| Serine/threonine-protein kinase N3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Serine/threonine-protein kinase Nek1 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Serine/threonine-protein kinase Nek11 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Serine/threonine-protein kinase Nek2 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Serine/threonine-protein kinase Nek3 | Homo sapiens (human) | Kd | 20.1566 | 2 | 8 |
| Serine/threonine-protein kinase Nek4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Serine/threonine-protein kinase Nek5 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase Nek6 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase Nek7 | Homo sapiens (human) | Kd | 21.8625 | 3 | 8 |
| Serine/threonine-protein kinase Nek9 | Homo sapiens (human) | Kd | 20.0527 | 3 | 9 |
| Serine/threonine-protein kinase NIM1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Serine/threonine-protein kinase NLK | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Serine/threonine-protein kinase OSR1 | Homo sapiens (human) | Kd | 6.3500 | 1 | 2 |
| Serine/threonine-protein kinase PAK 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase PAK 2 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Serine/threonine-protein kinase PAK 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase PAK 4 | Homo sapiens (human) | Kd | 23.1600 | 3 | 10 |
| Serine/threonine-protein kinase PAK 5 | Homo sapiens (human) | Kd | 7.1000 | 2 | 3 |
| Serine/threonine-protein kinase PAK 6 | Homo sapiens (human) | Kd | 21.6125 | 3 | 8 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Serine/threonine-protein kinase pim-2 | Homo sapiens (human) | Kd | 18.0000 | 3 | 5 |
| Serine/threonine-protein kinase pim-3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase PknB | Mycobacterium tuberculosis H37Rv | Kd | 3.1000 | 1 | 2 |
| Serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Kd | 13.5528 | 3 | 6 |
| Serine/threonine-protein kinase PLK2 | Homo sapiens (human) | Kd | 5.7500 | 1 | 2 |
| Serine/threonine-protein kinase PLK3 | Homo sapiens (human) | Kd | 6.9033 | 2 | 3 |
| Serine/threonine-protein kinase PLK4 | Homo sapiens (human) | Kd | 20.0819 | 3 | 10 |
| Serine/threonine-protein kinase PRP4 homolog | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Serine/threonine-protein kinase receptor R3 | Homo sapiens (human) | Kd | 18.0000 | 3 | 5 |
| Serine/threonine-protein kinase RIO1 | Homo sapiens (human) | Kd | 7.5000 | 2 | 3 |
| Serine/threonine-protein kinase RIO2 | Homo sapiens (human) | Kd | 5.6000 | 1 | 2 |
| Serine/threonine-protein kinase RIO3 | Homo sapiens (human) | Kd | 5.1991 | 3 | 5 |
| Serine/threonine-protein kinase SBK1 | Homo sapiens (human) | Kd | 5.6500 | 1 | 2 |
| Serine/threonine-protein kinase Sgk3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Serine/threonine-protein kinase SIK1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase SIK2 | Homo sapiens (human) | Kd | 16.9108 | 3 | 9 |
| Serine/threonine-protein kinase SIK3 | Homo sapiens (human) | Kd | 17.1262 | 2 | 8 |
| Serine/threonine-protein kinase STK11 | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| Serine/threonine-protein kinase TAO1 | Homo sapiens (human) | Kd | 22.3433 | 2 | 9 |
| Serine/threonine-protein kinase TAO2 | Homo sapiens (human) | Kd | 21.6565 | 2 | 8 |
| Serine/threonine-protein kinase TAO3 | Homo sapiens (human) | Kd | 23.8238 | 2 | 8 |
| Serine/threonine-protein kinase TBK1 | Homo sapiens (human) | Kd | 20.2828 | 2 | 8 |
| Serine/threonine-protein kinase TNNI3K | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase tousled-like 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase tousled-like 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Serine/threonine-protein kinase ULK1 | Homo sapiens (human) | Kd | 21.2344 | 2 | 9 |
| Serine/threonine-protein kinase ULK2 | Homo sapiens (human) | Kd | 5.0950 | 1 | 2 |
| Serine/threonine-protein kinase ULK3 | Homo sapiens (human) | Kd | 19.8864 | 2 | 8 |
| Serine/threonine-protein kinase VRK2 | Homo sapiens (human) | Kd | 7.0000 | 1 | 2 |
| Serine/threonine-protein kinase/endoribonuclease IRE1 | Homo sapiens (human) | Kd | 24.0625 | 2 | 8 |
| Serine/threonine-protein kinase/endoribonuclease IRE2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Signal recognition particle receptor subunit alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| SNF-related serine/threonine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Sodium/bile acid cotransporter | Homo sapiens (human) | Kd | 64.3000 | 1 | 1 |
| Spike glycoprotein | Betacoronavirus England 1 | EC50 | 2.9000 | 1 | 1 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | EC50 | 2.9000 | 1 | 1 |
| SRSF protein kinase 1 | Homo sapiens (human) | Kd | 7.3667 | 2 | 3 |
| SRSF protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| SRSF protein kinase 3 | Homo sapiens (human) | Kd | 6.6500 | 1 | 2 |
| STE20-like serine/threonine-protein kinase | Homo sapiens (human) | Kd | 23.5237 | 3 | 9 |
| STE20-related kinase adapter protein alpha | Homo sapiens (human) | Kd | 24.7344 | 1 | 5 |
| STE20/SPS1-related proline-alanine-rich protein kinase | Homo sapiens (human) | Kd | 5.9500 | 1 | 2 |
| Structural maintenance of chromosomes protein 1A | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Structural maintenance of chromosomes protein 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| Testis-specific serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| TGF-beta receptor type-1 | Homo sapiens (human) | Kd | 20.0219 | 3 | 9 |
| TGF-beta receptor type-2 | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Thyroid hormone receptor-associated protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 5 |
| TRAF2 and NCK-interacting protein kinase | Homo sapiens (human) | Kd | 18.9219 | 3 | 8 |
| Transient receptor potential cation channel subfamily M member 6 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |
| Transmembrane protease serine 2 | Homo sapiens (human) | EC50 | 2.9000 | 1 | 1 |
| Tubulin alpha-1A chain | Rattus norvegicus (Norway rat) | Kd | 10.0000 | 1 | 1 |
| Tyrosine--tRNA ligase, cytoplasmic | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | Kd | 9.8964 | 23 | 43 |
| Tyrosine-protein kinase ABL2 | Homo sapiens (human) | Kd | 16.7789 | 3 | 9 |
| Tyrosine-protein kinase Blk | Homo sapiens (human) | Kd | 6.0037 | 3 | 5 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | EC50 | 0.0383 | 2 | 3 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | Kd | 12.3222 | 5 | 13 |
| Tyrosine-protein kinase CSK | Homo sapiens (human) | Kd | 21.1058 | 3 | 9 |
| Tyrosine-protein kinase Fer | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Tyrosine-protein kinase Fes/Fps | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| Tyrosine-protein kinase Fgr | Homo sapiens (human) | Kd | 12.1912 | 3 | 5 |
| Tyrosine-protein kinase FRK | Homo sapiens (human) | Kd | 18.2919 | 3 | 10 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | Kd | 17.1503 | 3 | 10 |
| Tyrosine-protein kinase HCK | Homo sapiens (human) | Kd | 16.6824 | 3 | 9 |
| Tyrosine-protein kinase ITK/TSK | Homo sapiens (human) | Kd | 7.4457 | 4 | 7 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | EC50 | 0.0573 | 6 | 8 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | Kd | 16.9236 | 6 | 13 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | EC50 | 0.5571 | 6 | 8 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | Kd | 6.6717 | 6 | 9 |
| Tyrosine-protein kinase JAK2 | Mus musculus (house mouse) | EC50 | 0.1860 | 1 | 1 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | EC50 | 0.0165 | 2 | 2 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | Kd | 1.4517 | 6 | 9 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | Kd | 14.7080 | 3 | 9 |
| Tyrosine-protein kinase Lyn | Homo sapiens (human) | Kd | 16.6957 | 3 | 9 |
| Tyrosine-protein kinase Mer | Homo sapiens (human) | Kd | 15.0000 | 3 | 4 |
| Tyrosine-protein kinase receptor Tie-1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Tyrosine-protein kinase receptor TYRO3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Tyrosine-protein kinase receptor UFO | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Tyrosine-protein kinase Srms | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | Kd | 23.3333 | 3 | 9 |
| Tyrosine-protein kinase Tec | Homo sapiens (human) | Kd | 15.0034 | 5 | 14 |
| Tyrosine-protein kinase TXK | Homo sapiens (human) | Kd | 6.0049 | 3 | 5 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | Kd | 18.0122 | 3 | 10 |
| Tyrosine-protein kinase ZAP-70 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| U5 small nuclear ribonucleoprotein 200 kDa helicase | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| UMP-CMP kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Uncharacterized aarF domain-containing protein kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 3 |
| Uncharacterized protein FLJ45252 | Homo sapiens (human) | Kd | 15.0462 | 1 | 6 |
| Uncharacterized serine/threonine-protein kinase SBK3 | Homo sapiens (human) | Kd | 7.9000 | 1 | 2 |
| Vascular endothelial growth factor receptor 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Vascular endothelial growth factor receptor 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 3 |
| Very long-chain specific acyl-CoA dehydrogenase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 6 |
| Wee1-like protein kinase | Homo sapiens (human) | Kd | 24.0000 | 3 | 10 |
| Wee1-like protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 2 |