Page last updated: 2024-08-05 15:23:19

EC 2.7.1.137 (phosphatidylinositol 3-kinase) inhibitor

An inhibitor of phosphatidylinositol 3-kinase, EC 2.7.1.137, a family of related enzymes capable of phosphorylating the 3 position hydroxy group of the inositol ring of a phosphatidylinositol.

ChEBI ID: 50914

Members (21)

MemberDefinitionClass
2-(4-morpholinyl)-8-phenyl-4h-1-benzopyran-4-oneA chromone substituted with a phenyl group at position 8 and a morpholine group at position 2.LY294002
as 605240A quinoxaline derivative that is quinoxaline in which the hydrogen at position 6 is replaced by a (2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl group. It is a potent inhibitor of the PI3Kgamma, with an IC50 of 8 nM and inhibits the progression of joint inflammation and damage in both lymphocyte-independent and dependent mouse models of rheumatoid arthritis.(5Z)-5-(quinoxalin-6-ylmethylidene)-1,3-thiazolidine-2,4-dione
bgt226An imidazoquinoline that is 3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-c]quinoline substituted at position 1 by a 3-trifluoromethyl-4-(piperazin-1-yl)phenyl group and at position 8 by a 6-methoxypyridin-3-yl group. A dual PI3K/mTOR inhibitor.BGT226 free base
buparlisibAn aminopyridine that is 4-(trifluoromethyl)pyridin-2-amine substituted at position 5 by a 2,6-di(morpholin-4-yl)pyrimidin-4-y group. A selective PI3K inhibitor with anti-tumour properties.BKM120
dactolisibAn imidazoquinoline that is 3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-c]quinoline substituted at position 1 by a 4-(1-cyanoisopropyl)phenyl group and at position 8 by a quinolin-3-yl group. A dual PI3K/mTOR inhibitor used in cancer treatment.dactolisib
gdc 0941A sulfonamide composed of indazole, morpholine, and methylsulfonyl-substituted piperazine rings bound to a thienopyrimidine ring.pictrelisib
gsk 2126458A member of the class of quinolines that is quinoline which is substituted by pyridazin-4-yl and 5-[(2,4-difluorobenzene-1-sulfonyl)amino]-6-methoxypyridin-3-yl groups at positions 4 and 6, respectively. It is a highly potent inhibitor of PI3K and mTOR developed by GlaxoSmithKline and was previously in human phase 1 clinical trials for the treatment of idiopathic pulmonary fibrosis and solid tumors.omipalisib
GSK1059615A thiazolidinone that is the 5-{[4-(pyridin-4-yl)quinolin-6-yl]methylene} derivative of 1,3-thiazolidine-2,4-dione. A PI3K inhibitorGSK1059615
ic 87114A member of the class of quinazolines that is quinazolin-4(3H)-one carrying (6-amino-9H-purin-9-yl)methyl, 2-methylphenyl and methyl substituents at positions 2, 3 and 5 respectively.IC-87114
idelalisibA member of the class of quinazolines that is 5-fluoro-3-phenylquinazolin-4-one in which the hydrogen at position 2 is replaced by a (1S)-1-(3H-purin-6-ylamino)propyl group. used for for the treatment of refractory indolent non-Hodgkin's lymphoma and relapsed chronic lymphocytic leukemia.idelalisib
liphagalA meroterpenoid isolated from the marine sponge Aka coralliphaga and has been shown to exhibit inhibitory activity against phosphatidylinositol-3-OH kinase.liphagal
mk 2206An organic heterotricyclic compound that is [1,2,4]triazolo[3,4-f][1,6]naphthyridin-3(2H)-one substituted at positions 8 and 9 respectively by 4-(1-aminocyclobutyl)phenyl and phenyl groups.MK-2206
perifosineA phospholipid consisting of 1,1-dimethylpiperidinium-4-yl hydrogen phosphate in which the hydrogen is replaced by a stearyl (octadecyl) group.perifosine
pi103An organic heterotricyclic compound that is pyrido[3',2':4,5]furo[3,2-d]pyrimidine substituted at positions 2 and 4 by 3-hydroxyphenyl and morpholin-4-yl groups respectively. A dual-kinase inhibitor with anti-cancer properties.PI-103
PP121A pyrazolopyrimidine that is 1H-pyrazolo[3,4-d]pyrimidine which is substituted by a cyclopentyl, 1H-pyrrolo[2,3-b]pyridin-5-yl, and amino groups at positions 1, 3 and 4, respectively. It is a dual inhibitor of tyrosine and phosphoinositide kinases and exhibits anti-cancer properties.PP121
px-866An organic heterotetracyclic compound that is obtained from wortmanin via aminolysis of its furan ring by diallyl amine.PX-866
triciribineA nucleoside analogue in which the nucleobase portion is a 1,4,5,6,8-pentaazaacenaphthylene ring system substituted with an amino group at position 3, and a methyl group at position 5 and is bound to the beta-D-ribofuranosyl moiety by an N(1)-glycosidic linkage.triciribine
wortmanninwortmannin
xl147A sulfonamide that is the N-4-toluenesulfonyl (N-tosyl) derivative of N-(2,1,3-benzothiadiazol-5-yl)quinoxaline-2,3-diamine. A selective PI3K inhibitor used in cancer treatment.XL147
xl765A sulfonamide obtained by formal condensation of the sulfonic acid group of 4-[(3-methoxy-4-methylbenzoyl)amino]benzenesulfonic acid with the primary aromatic amino group of N-(3,5-dimethoxyphenyl)quinoxaline-2,3-diamine. A dual PI3K/mTOR inhibitor used in cancer treatment.XL765
zstk474A triamino-1,3,5-triazine that is 1,3,5-triazine in which two of the hydrogens have been replaced by morpholin-4-yl groups while the third hydrogen has been replaced by a 2-(difluoromethyl)benzimidazol-1-yl group. It is an inhibitor of phosphatidylinositol 3-kinase.ZSTK-474

Research

Studies (9,805)

TimeframeStudies, Drugs with This Role(%)All Drugs %
pre-19904 (0.04)18.7374
1990's1,165 (11.88)18.2507
2000's4,059 (41.40)29.6817
2010's4,043 (41.23)24.3611
2020's534 (5.45)2.80

Study Types

Publication TypeStudies, Drugs with this Role (%)All Drugs (%)
Trials203 (1.80%)5.53%
Reviews237 (2.10%)6.00%
Case Studies41 (0.36%)4.05%
Observational8 (0.07%)0.25%
Other10,818 (95.68%)84.16%

Protein Targets (707)

Potency Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
15-lipoxygenase, partialHomo sapiens (human)Potency39.810711
67.9K proteinVaccinia virusPotency27.246328
acetylcholinesteraseHomo sapiens (human)Potency17.950822
aldehyde dehydrogenase 1 family, member A1Homo sapiens (human)Potency39.090613
Alpha-synucleinHomo sapiens (human)Potency5.011911
AR proteinHomo sapiens (human)Potency9.5867810
aryl hydrocarbon receptorHomo sapiens (human)Potency14.930323
arylsulfatase AHomo sapiens (human)Potency0.301311
ATAD5 protein, partialHomo sapiens (human)Potency24.245723
Ataxin-2Homo sapiens (human)Potency17.743422
ATP-dependent phosphofructokinaseTrypanosoma brucei brucei TREU927Potency0.012011
ATPase family AAA domain-containing protein 5Homo sapiens (human)Potency33.491511
Cellular tumor antigen p53Homo sapiens (human)Potency9.044412
cellular tumor antigen p53 isoform aHomo sapiens (human)Potency10.000011
Chain A, 2-oxoglutarate OxygenaseHomo sapiens (human)Potency39.810711
Chain A, ATP-DEPENDENT DNA HELICASE Q1Homo sapiens (human)Potency35.481311
Chain A, CruzipainTrypanosoma cruziPotency28.183811
Chain A, Ferritin light chainEquus caballus (horse)Potency31.622811
Chain A, HADH2 proteinHomo sapiens (human)Potency39.810711
Chain B, HADH2 proteinHomo sapiens (human)Potency39.810711
chromobox protein homolog 1Homo sapiens (human)Potency26.679511
cytochrome P450 2C19 precursorHomo sapiens (human)Potency10.000011
cytochrome P450 2C9 precursorHomo sapiens (human)Potency39.810711
cytochrome P450 2C9, partialHomo sapiens (human)Potency7.749914
cytochrome P450 2D6Homo sapiens (human)Potency38.901811
cytochrome P450 2D6 isoform 1Homo sapiens (human)Potency25.118911
cytochrome P450 3A4 isoform 1Homo sapiens (human)Potency7.506024
cytochrome P450 family 3 subfamily A polypeptide 4Homo sapiens (human)Potency7.796124
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_aHomo sapiens (human)Potency1.333311
D(1A) dopamine receptorSus scrofa (pig)Potency7.551612
DNA dC->dU-editing enzyme APOBEC-3G isoform 1Homo sapiens (human)Potency17.782811
DNA polymerase iota isoform a (long)Homo sapiens (human)Potency89.125111
estrogen nuclear receptor alphaHomo sapiens (human)Potency13.1496810
estrogen receptor 2 (ER beta)Homo sapiens (human)Potency1.188311
estrogen-related nuclear receptor alphaHomo sapiens (human)Potency5.619277
euchromatic histone-lysine N-methyltransferase 2Homo sapiens (human)Potency15.544913
EWS/FLI fusion proteinHomo sapiens (human)Potency5.0785460
farnesoid X nuclear receptorHomo sapiens (human)Potency33.488922
flap endonuclease 1Homo sapiens (human)Potency38.713212
Fumarate hydrataseHomo sapiens (human)Potency7.6124111
GVesicular stomatitis virusPotency7.749914
GABA theta subunitRattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)Potency7.506012
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)Potency7.506012
gemininHomo sapiens (human)Potency5.804811
GLI family zinc finger 3Homo sapiens (human)Potency3.424034
GLS proteinHomo sapiens (human)Potency3.548111
glucocorticoid receptor [Homo sapiens]Homo sapiens (human)Potency1.068211
Glutamate receptor 2Rattus norvegicus (Norway rat)Potency2.113211
GTP-binding nuclear protein Ran isoform 1Homo sapiens (human)Potency28.183811
Guanine nucleotide-binding protein GHomo sapiens (human)Potency11.220211
Histamine H2 receptorCavia porcellus (domestic guinea pig)Potency33.934025
histone deacetylase 9 isoform 3Homo sapiens (human)Potency14.960111
Histone H2A.xCricetulus griseus (Chinese hamster)Potency49.520412
HLA class I histocompatibility antigen, B alpha chain Homo sapiens (human)Potency7.749914
hypoxia-inducible factor 1 alpha subunitHomo sapiens (human)Potency6.007011
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor)Homo sapiens (human)Potency7.943322
IDH1Homo sapiens (human)Potency12.995311
importin subunit beta-1 isoform 1Homo sapiens (human)Potency28.183811
Inositol hexakisphosphate kinase 1Homo sapiens (human)Potency7.749918
Inositol monophosphatase 1Rattus norvegicus (Norway rat)Potency28.183811
Integrin alpha-IIbHomo sapiens (human)Potency10.000011
Integrin beta-3Homo sapiens (human)Potency10.000011
Interferon betaHomo sapiens (human)Potency5.2276335
M-phase phosphoprotein 8Homo sapiens (human)Potency37.685811
Microtubule-associated protein tauHomo sapiens (human)Potency19.622222
NFKB1 protein, partialHomo sapiens (human)Potency7.079522
NPC intracellular cholesterol transporter 1 precursorHomo sapiens (human)Potency10.322511
Nrf2Homo sapiens (human)Potency22.387211
nuclear factor erythroid 2-related factor 2 isoform 1Homo sapiens (human)Potency16.836423
nuclear factor erythroid 2-related factor 2 isoform 2Homo sapiens (human)Potency2.291322
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_aHomo sapiens (human)Potency1.899611
nuclear receptor subfamily 1, group I, member 2Rattus norvegicus (Norway rat)Potency0.281811
nuclear receptor subfamily 1, group I, member 3Homo sapiens (human)Potency11.908323
parathyroid hormone/parathyroid hormone-related peptide receptor precursorHomo sapiens (human)Potency56.234111
ParkinHomo sapiens (human)Potency15.358923
peptidyl-prolyl cis-trans isomerase NIMA-interacting 1Homo sapiens (human)Potency67.455511
peroxisome proliferator activated receptor gammaHomo sapiens (human)Potency9.438411
peroxisome proliferator-activated receptor deltaHomo sapiens (human)Potency25.136622
phosphopantetheinyl transferaseBacillus subtilisPotency35.481311
polyproteinZika virusPotency7.6124111
Polyunsaturated fatty acid lipoxygenase ALOX15BHomo sapiens (human)Potency25.118911
PPM1D proteinHomo sapiens (human)Potency4.6717120
pregnane X nuclear receptorHomo sapiens (human)Potency5.588223
RAR-related orphan receptor gammaMus musculus (house mouse)Potency0.517224
ras-related protein Rab-9AHomo sapiens (human)Potency3.264311
regulator of G-protein signaling 4Homo sapiens (human)Potency14.214413
retinoic acid nuclear receptor alpha variant 1Homo sapiens (human)Potency5.429236
retinoid X nuclear receptor alphaHomo sapiens (human)Potency2.007122
serine/threonine-protein kinase mTOR isoform 1Homo sapiens (human)Potency10.758547
SMAD family member 2Homo sapiens (human)Potency8.130222
SMAD family member 3Homo sapiens (human)Potency8.130222
Smad3Homo sapiens (human)Potency6.047613
snurportin-1Homo sapiens (human)Potency28.183811
Spike glycoproteinSevere acute respiratory syndrome-related coronavirusPotency1.412511
survival motor neuron protein isoform dHomo sapiens (human)Potency9.874412
TAR DNA-binding protein 43Homo sapiens (human)Potency1.000011
TDP1 proteinHomo sapiens (human)Potency5.2844220
thioredoxin reductaseRattus norvegicus (Norway rat)Potency52.766025
ThrombopoietinHomo sapiens (human)Potency10.000022
thyroid hormone receptor beta isoform 2Rattus norvegicus (Norway rat)Potency7.778824
thyroid hormone receptor beta isoform aHomo sapiens (human)Potency40.074822
thyroid stimulating hormone receptorHomo sapiens (human)Potency23.846446
transcriptional regulator ERG isoform 3Homo sapiens (human)Potency22.387211
tyrosine-protein kinase YesHomo sapiens (human)Potency34.651913
USP1 protein, partialHomo sapiens (human)Potency89.125111
v-jun sarcoma virus 17 oncogene homolog (avian)Homo sapiens (human)Potency21.313811
vitamin D (1,25- dihydroxyvitamin D3) receptorHomo sapiens (human)Potency16.163222
vitamin D3 receptor isoform VDRAHomo sapiens (human)Potency60.456612
Voltage-dependent calcium channel gamma-2 subunitMus musculus (house mouse)Potency2.113211
VprHuman immunodeficiency virus 1Potency17.782811
WRNHomo sapiens (human)Potency14.125411

Inhibition Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
5-hydroxytryptamine receptor 2AHomo sapiens (human)IC502.796011
5-hydroxytryptamine receptor 2AHomo sapiens (human)Ki0.799011
5-hydroxytryptamine receptor 2BHomo sapiens (human)IC5036.707011
5-hydroxytryptamine receptor 2BHomo sapiens (human)Ki23.359011
5-hydroxytryptamine receptor 2CHomo sapiens (human)IC501.002011
5-hydroxytryptamine receptor 2CHomo sapiens (human)Ki0.525011
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)IC501.002011
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)Ki0.525011
AcetylcholinesteraseRattus norvegicus (Norway rat)IC500.003012
AcetylcholinesteraseRattus norvegicus (Norway rat)Ki0.010212
Aldehyde oxidaseHomo sapiens (human)IC500.130011
Aldo-keto reductase family 1 member C3Homo sapiens (human)IC508.700022
Aldo-keto reductase family 1 member C3Homo sapiens (human)Ki14.000011
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)IC500.006112
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)IC500.006112
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)IC500.006112
Amine oxidase [flavin-containing] AHomo sapiens (human)IC50165.800011
Amine oxidase [flavin-containing] BHomo sapiens (human)IC5013.000022
ATP-binding cassette sub-family C member 3Homo sapiens (human)IC50133.000012
Bile salt export pumpHomo sapiens (human)IC5011.700023
Breakpoint cluster region proteinHomo sapiens (human)IC500.018011
Bromodomain-containing protein 2Homo sapiens (human)IC5010.300011
Bromodomain-containing protein 3Homo sapiens (human)IC5013.700011
Bromodomain-containing protein 4Homo sapiens (human)IC5012.400011
Canalicular multispecific organic anion transporter 1Homo sapiens (human)IC5089.550012
Casein kinase II subunit alphaHomo sapiens (human)IC503.460022
Casein kinase II subunit alpha'Homo sapiens (human)IC503.460022
Casein kinase II subunit betaHomo sapiens (human)IC503.460022
CDGSH iron-sulfur domain-containing protein 1Homo sapiens (human)IC503.260011
cGMP-dependent 3',5'-cyclic phosphodiesteraseHomo sapiens (human)IC5040.000011
cGMP-inhibited 3',5'-cyclic phosphodiesterase AHomo sapiens (human)IC50100.000011
cGMP-inhibited 3',5'-cyclic phosphodiesterase BHomo sapiens (human)IC50100.000011
cGMP-specific 3',5'-cyclic phosphodiesteraseHomo sapiens (human)IC509.614011
Chain A, Methyltransferase WbddEscherichia coliIC5068.000011
Chain A, PHOSPHATIDYLINOSITOL-4,5-BISPHOSPHATE 3-KINASE CATALYTIC SUBUNIT DELTA ISOFORMMus musculus (house mouse)IC500.0673126
Chain A, Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma isoformHomo sapiens (human)IC500.262011
Chain A, Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoformHomo sapiens (human)IC500.008012
Chain A, PHOSPHOTIDYLINOSITOL 3 KINASE 59FDrosophila melanogaster (fruit fly)IC502.300014
Chain A, Proto-oncogene serine/threonine-protein kinase Pim-1Homo sapiens (human)IC504.000012
Cholesteryl ester transfer proteinHomo sapiens (human)IC500.032011
Cytochrome P450 1A2Homo sapiens (human)IC500.210948
Cytochrome P450 2B6Homo sapiens (human)IC500.011011
Cytochrome P450 2C19Homo sapiens (human)IC500.379034
Cytochrome P450 2C8Homo sapiens (human)IC500.040011
Cytochrome P450 2D6Homo sapiens (human)IC500.325012
Cytochrome P450 3A4Homo sapiens (human)IC500.010659
DNA-dependent protein kinase catalytic subunitHomo sapiens (human)IC501.87561820
DNA-dependent protein kinase catalytic subunitHomo sapiens (human)Ki3.648055
Dual specificity protein kinase CLK1Homo sapiens (human)IC500.070011
Dual specificity tyrosine-phosphorylation-regulated kinase 1AHomo sapiens (human)IC500.815022
Dual specificity tyrosine-phosphorylation-regulated kinase 1BHomo sapiens (human)IC500.080011
Dual specificity tyrosine-phosphorylation-regulated kinase 2Homo sapiens (human)IC500.100011
Ephrin type-B receptor 4Homo sapiens (human)IC500.190011
Epidermal growth factor receptorHomo sapiens (human)IC505.130022
Glycogen synthase kinase-3 betaHomo sapiens (human)IC508.100011
High affinity nerve growth factor receptorHomo sapiens (human)IC502.850011
Histone deacetylase 6Homo sapiens (human)IC500.002011
Metabotropic glutamate receptor 1Rattus norvegicus (Norway rat)IC500.008522
Mitogen-activated protein kinase 14Homo sapiens (human)IC501.200011
Mu-type opioid receptorCavia porcellus (domestic guinea pig)IC501.600011
Multidrug resistance-associated protein 4Homo sapiens (human)IC5098.100012
Myosin light chain kinase, smooth muscleGallus gallus (chicken)IC500.260011
Myosin light chain kinase, smooth muscleHomo sapiens (human)IC502.356733
Neuronal acetylcholine receptor subunit alpha-4Rattus norvegicus (Norway rat)IC501.600011
Neuronal acetylcholine receptor subunit beta-2Rattus norvegicus (Norway rat)IC501.600011
Phosphatidylinositol 3-kinase catalytic subunit type 3Homo sapiens (human)IC5070.7326817
Phosphatidylinositol 3-kinase regulatory subunit alphaHomo sapiens (human)IC501,690.36866787
Phosphatidylinositol 3-kinase regulatory subunit alphaHomo sapiens (human)Ki0.006645
Phosphatidylinositol 4-kinase alphaHomo sapiens (human)IC506.760023
Phosphatidylinositol 4-kinase betaHomo sapiens (human)IC509.100045
Phosphatidylinositol 4-kinase type 2-alphaHomo sapiens (human)IC5030.000011
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alphaHomo sapiens (human)IC5039.341449
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit betaHomo sapiens (human)IC501.49361235
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformHomo sapiens (human)GI500.028011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformBos taurus (cattle)IC503.753333
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformHomo sapiens (human)IC50631.8549183234
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformRattus norvegicus (Norway rat)IC500.058113
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformHomo sapiens (human)Ki0.879077
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform Mus musculus (house mouse)IC500.336233
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformHomo sapiens (human)GI500.028011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformHomo sapiens (human)IC50932.6040114158
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformRattus norvegicus (Norway rat)IC500.226313
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformHomo sapiens (human)Ki0.000322
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformHomo sapiens (human)GI500.028011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformHomo sapiens (human)IC50821.5890133179
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformHomo sapiens (human)Ki0.013956
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)GI500.028011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)IC50898.5568117164
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Mus musculus (house mouse)IC501.302011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)Ki0.000733
Phosphoinositide 3-kinase regulatory subunit 5Homo sapiens (human)IC500.371056
Polyunsaturated fatty acid 5-lipoxygenaseHomo sapiens (human)IC501.200011
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)IC5052.666733
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)IC500.001011
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)IC500.014022
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)IC505.421499
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)IC500.012011
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)IC500.065011
Rapamycin-insensitive companion of mTORHomo sapiens (human)IC500.041622
Regulatory-associated protein of mTORHomo sapiens (human)IC500.028033
Reverse transcriptase/RNaseH Human immunodeficiency virus 1IC500.035034
Serine-protein kinase ATMHomo sapiens (human)IC5052.501844
Serine/threonine-protein kinase ATRHomo sapiens (human)IC5052.855044
Serine/threonine-protein kinase mTORHomo sapiens (human)IC500.95906684
Serine/threonine-protein kinase mTORRattus norvegicus (Norway rat)IC501.272522
Serine/threonine-protein kinase mTORHomo sapiens (human)Ki0.283679
Serine/threonine-protein kinase mTOR Mus musculus (house mouse)IC500.832011
Serine/threonine-protein kinase pim-1Homo sapiens (human)IC504.470066
Serine/threonine-protein kinase pim-3Homo sapiens (human)IC501.400011
Serine/threonine-protein kinase PLK1Homo sapiens (human)IC501.086035
Serine/threonine-protein kinase PLK1Homo sapiens (human)Ki10.766719
Serine/threonine-protein kinase PLK2Homo sapiens (human)Ki10.766719
Serine/threonine-protein kinase PLK3Homo sapiens (human)IC5018.263435
Serine/threonine-protein kinase PLK3Homo sapiens (human)Ki10.766719
Serine/threonine-protein kinase PLK4Homo sapiens (human)Ki10.766719
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)IC502.300011
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)Ki6.000011
Target of rapamycin complex 2 subunit MAPKAP1Homo sapiens (human)IC500.041622
Target of rapamycin complex subunit LST8Homo sapiens (human)IC500.033455
Type-1 angiotensin II receptorOryctolagus cuniculus (rabbit)IC500.500011
Tyrosine-protein kinase ABL1Homo sapiens (human)IC500.012733
Tyrosine-protein kinase HCKHomo sapiens (human)IC500.008011
Tyrosine-protein kinase JAK3Homo sapiens (human)IC501.000011
Ubiquitin carboxyl-terminal hydrolase isozyme L3Homo sapiens (human)IC500.050011
Vascular endothelial growth factor receptor 2Homo sapiens (human)IC500.021733

Activation Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
26S proteasome regulatory subunit 6BHomo sapiens (human)Kd30.0000110
3-phosphoinositide-dependent protein kinase 1Homo sapiens (human)Kd10.000023
5'-AMP-activated protein kinase catalytic subunit alpha-1Homo sapiens (human)Kd25.3846313
5'-AMP-activated protein kinase catalytic subunit alpha-2Homo sapiens (human)Kd10.000023
5'-AMP-activated protein kinase subunit gamma-1Homo sapiens (human)Kd30.0000110
5'-AMP-activated protein kinase subunit gamma-2Homo sapiens (human)Kd30.0000110
AarF domain-containing protein kinase 1Homo sapiens (human)Kd30.0000110
Actin-related protein 2Homo sapiens (human)Kd30.000019
Actin-related protein 3Homo sapiens (human)Kd30.0000111
Activated CDC42 kinase 1Homo sapiens (human)Kd25.7143314
Activin receptor type-1Homo sapiens (human)Kd25.3846313
Activin receptor type-1BHomo sapiens (human)Kd25.3846313
Activin receptor type-2AHomo sapiens (human)Kd10.000023
Activin receptor type-2BHomo sapiens (human)Kd25.3846313
Acyl-CoA dehydrogenase family member 10Homo sapiens (human)Kd30.000019
Acyl-CoA dehydrogenase family member 11Homo sapiens (human)Kd30.0000110
Adenine phosphoribosyltransferaseHomo sapiens (human)Kd30.000016
Adenosine kinaseHomo sapiens (human)Kd30.0000110
Adenylate kinase 2, mitochondrialHomo sapiens (human)Kd30.0000111
ADP/ATP translocase 2Homo sapiens (human)Kd30.0000111
ADP/ATP translocase 3Homo sapiens (human)Kd30.0000110
ALK tyrosine kinase receptorHomo sapiens (human)Kd18.000035
Angiopoietin-1 receptorHomo sapiens (human)Kd10.000023
Ankyrin repeat and protein kinase domain-containing protein 1Homo sapiens (human)Kd10.000023
AP2-associated protein kinase 1Homo sapiens (human)Kd25.6500314
ATP-dependent 6-phosphofructokinase, platelet typeHomo sapiens (human)Kd30.0000110
ATP-dependent RNA helicase DDX1Homo sapiens (human)Kd30.000019
ATP-dependent RNA helicase DDX3XHomo sapiens (human)Kd30.0000110
ATP-dependent RNA helicase DDX42Homo sapiens (human)Kd30.000017
ATP-dependent RNA helicase DHX30Homo sapiens (human)Kd30.000014
Atypical kinase COQ8A, mitochondrialHomo sapiens (human)Kd25.7143314
Atypical kinase COQ8B, mitochondrialHomo sapiens (human)Kd10.000023
Aurora kinase AHomo sapiens (human)Kd25.3846313
Aurora kinase BHomo sapiens (human)Kd25.3846313
Aurora kinase CHomo sapiens (human)Kd10.000023
BDNF/NT-3 growth factors receptorHomo sapiens (human)Kd10.000023
Beta-adrenergic receptor kinase 1Homo sapiens (human)Kd30.0000111
BMP-2-inducible protein kinaseHomo sapiens (human)Kd25.3846313
Bone morphogenetic protein receptor type-1AHomo sapiens (human)Kd25.3846313
Bone morphogenetic protein receptor type-1BHomo sapiens (human)Kd26.9231213
Bone morphogenetic protein receptor type-2Homo sapiens (human)Kd25.3846313
Breakpoint cluster region proteinHomo sapiens (human)Kd30.0000110
Calcium-dependent protein kinase 1Plasmodium falciparum 3D7Kd10.000012
Calcium/calmodulin-dependent protein kinase kinase 1Homo sapiens (human)Kd10.000023
Calcium/calmodulin-dependent protein kinase kinase 2Homo sapiens (human)Kd25.7143314
Calcium/calmodulin-dependent protein kinase type 1Homo sapiens (human)Kd8.233323
Calcium/calmodulin-dependent protein kinase type 1DHomo sapiens (human)Kd10.000023
Calcium/calmodulin-dependent protein kinase type 1GHomo sapiens (human)Kd8.933323
Calcium/calmodulin-dependent protein kinase type II subunit alphaHomo sapiens (human)Kd10.000023
Calcium/calmodulin-dependent protein kinase type II subunit betaHomo sapiens (human)Kd10.000023
Calcium/calmodulin-dependent protein kinase type II subunit deltaHomo sapiens (human)Kd25.3846313
Calcium/calmodulin-dependent protein kinase type II subunit gammaHomo sapiens (human)Kd25.7143314
Calcium/calmodulin-dependent protein kinase type IVHomo sapiens (human)Kd25.3846313
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)Kd25.3846313
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)Kd25.3846313
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)Kd27.5006112
cAMP-dependent protein kinase catalytic subunit PRKXHomo sapiens (human)Kd10.000023
cAMP-dependent protein kinase type II-alpha regulatory subunitHomo sapiens (human)Kd30.0000110
Casein kinase I isoform alphaHomo sapiens (human)Kd26.9231213
Casein kinase I isoform alpha-likeHomo sapiens (human)Kd10.000023
Casein kinase I isoform deltaHomo sapiens (human)Kd24.7077313
Casein kinase I isoform epsilonHomo sapiens (human)Kd24.7077313
Casein kinase I isoform gamma-1Homo sapiens (human)Kd25.0000312
Casein kinase I isoform gamma-2Homo sapiens (human)Kd23.333339
Casein kinase I isoform gamma-3Homo sapiens (human)Kd25.3846313
Casein kinase II subunit alphaHomo sapiens (human)Kd8.466723
Casein kinase II subunit alpha'Homo sapiens (human)Kd20.5545313
Cell division control protein 2 homologPlasmodium falciparum 3D7Kd10.000012
Cell division cycle 7-related protein kinaseHomo sapiens (human)Kd30.000015
cGMP-dependent protein kinase 1 Homo sapiens (human)Kd26.0000315
cGMP-dependent protein kinase 2Homo sapiens (human)Kd10.000023
Choline-phosphate cytidylyltransferase AHomo sapiens (human)Kd30.000014
Chromodomain-helicase-DNA-binding protein 4Homo sapiens (human)Kd30.0000110
Citron Rho-interacting kinaseHomo sapiens (human)Kd25.7143314
Cyclin-dependent kinase 1Homo sapiens (human)Kd30.0000111
Cyclin-dependent kinase 10Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 11AHomo sapiens (human)Kd10.000023
Cyclin-dependent kinase 11BHomo sapiens (human)Kd10.000023
Cyclin-dependent kinase 12Homo sapiens (human)Kd30.0000110
Cyclin-dependent kinase 13Homo sapiens (human)Kd26.9231213
Cyclin-dependent kinase 14Homo sapiens (human)Kd10.000023
Cyclin-dependent kinase 15Homo sapiens (human)Kd10.000012
Cyclin-dependent kinase 16Homo sapiens (human)Kd25.0786314
Cyclin-dependent kinase 17Homo sapiens (human)Kd25.3846313
Cyclin-dependent kinase 18Homo sapiens (human)Kd8.200023
Cyclin-dependent kinase 19Homo sapiens (human)Kd10.000023
Cyclin-dependent kinase 2Homo sapiens (human)Kd25.3846313
Cyclin-dependent kinase 3Homo sapiens (human)Kd25.3846313
Cyclin-dependent kinase 4Homo sapiens (human)Kd25.0000316
Cyclin-dependent kinase 6Homo sapiens (human)Kd30.0000112
Cyclin-dependent kinase 7Homo sapiens (human)Kd25.5143314
Cyclin-dependent kinase 8Homo sapiens (human)Kd10.000023
Cyclin-dependent kinase 9Homo sapiens (human)Kd25.7143314
Cyclin-dependent kinase-like 1Homo sapiens (human)Kd10.000012
Cyclin-dependent kinase-like 2Homo sapiens (human)Kd10.000012
Cyclin-dependent kinase-like 3Homo sapiens (human)Kd10.000012
Cyclin-dependent kinase-like 5Homo sapiens (human)Kd23.333326
Cyclin-dependent-like kinase 5 Homo sapiens (human)Kd25.3846313
Cyclin-G-associated kinaseHomo sapiens (human)Kd24.8231313
Cysteine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000017
Cytochrome c1, heme protein, mitochondrialHomo sapiens (human)Kd30.0000111
Cytoplasmic tyrosine-protein kinase BMXHomo sapiens (human)Kd10.000023
dCTP pyrophosphatase 1Homo sapiens (human)Kd30.0000113
Death-associated protein kinase 1Homo sapiens (human)Kd2.933323
Death-associated protein kinase 2Homo sapiens (human)Kd5.133323
Death-associated protein kinase 3Homo sapiens (human)Kd3.370034
Delta(24)-sterol reductaseHomo sapiens (human)Kd30.0000111
Deoxycytidine kinaseHomo sapiens (human)Kd30.0000111
Discoidin domain-containing receptor 2Homo sapiens (human)Kd25.3846313
DNA replication licensing factor MCM4Homo sapiens (human)Kd30.0000111
DNA topoisomerase 2-alphaHomo sapiens (human)Kd30.000018
DNA topoisomerase 2-betaHomo sapiens (human)Kd30.0000110
DNA-dependent protein kinase catalytic subunitHomo sapiens (human)Kd1.550012
DnaJ homolog subfamily A member 1Homo sapiens (human)Kd30.0000112
Dual serine/threonine and tyrosine protein kinaseHomo sapiens (human)Kd10.000012
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)Kd25.3846313
Dual specificity mitogen-activated protein kinase kinase 2Homo sapiens (human)Kd25.3846313
Dual specificity mitogen-activated protein kinase kinase 3Homo sapiens (human)Kd25.3846313
Dual specificity mitogen-activated protein kinase kinase 4Homo sapiens (human)Kd18.000035
Dual specificity mitogen-activated protein kinase kinase 5Homo sapiens (human)Kd26.6667212
Dual specificity mitogen-activated protein kinase kinase 6Homo sapiens (human)Kd25.3846313
Dual specificity mitogen-activated protein kinase kinase 7Homo sapiens (human)Kd10.000012
Dual specificity protein kinase CLK1Homo sapiens (human)Kd20.7622312
Dual specificity protein kinase CLK2Homo sapiens (human)Kd23.2818311
Dual specificity protein kinase CLK3Homo sapiens (human)Kd13.975034
Dual specificity protein kinase CLK4Homo sapiens (human)Kd22.388939
Dual specificity protein kinase TTKHomo sapiens (human)Kd23.4300310
Dual specificity testis-specific protein kinase 1Homo sapiens (human)Kd25.7143314
Dual specificity testis-specific protein kinase 2Homo sapiens (human)Kd30.000014
Dual specificity tyrosine-phosphorylation-regulated kinase 1AHomo sapiens (human)Kd24.2435212
Dual specificity tyrosine-phosphorylation-regulated kinase 1BHomo sapiens (human)Kd18.250036
Dual specificity tyrosine-phosphorylation-regulated kinase 2Homo sapiens (human)Kd5.850012
Dynamin-like 120 kDa protein, mitochondrialHomo sapiens (human)Kd30.0000111
eIF-2-alpha kinase GCN2Homo sapiens (human)Kd10.000023
EKC/KEOPS complex subunit TP53RKHomo sapiens (human)Kd27.3645111
Electron transfer flavoprotein subunit betaHomo sapiens (human)Kd30.000017
Elongation factor Tu, mitochondrialHomo sapiens (human)Kd30.0000110
endoribonuclease toxin MazFEscherichia coli str. K-12 substr. MG1655EC5099.000022
Ephrin type-A receptor 1Homo sapiens (human)Kd25.0000312
Ephrin type-A receptor 2Homo sapiens (human)Kd25.7143314
Ephrin type-A receptor 3Homo sapiens (human)Kd10.000023
Ephrin type-A receptor 4Homo sapiens (human)Kd25.3846313
Ephrin type-A receptor 5Homo sapiens (human)Kd25.7143314
Ephrin type-A receptor 6Homo sapiens (human)Kd10.000023
Ephrin type-A receptor 7Homo sapiens (human)Kd25.0000312
Ephrin type-A receptor 8Homo sapiens (human)Kd10.000023
Ephrin type-B receptor 1Homo sapiens (human)Kd10.000023
Ephrin type-B receptor 2Homo sapiens (human)Kd25.3846313
Ephrin type-B receptor 3Homo sapiens (human)Kd25.3846313
Ephrin type-B receptor 4Homo sapiens (human)Kd25.7143314
Ephrin type-B receptor 6Homo sapiens (human)Kd25.9667212
Epidermal growth factor receptorHomo sapiens (human)Kd14.54552344
Epithelial discoidin domain-containing receptor 1Homo sapiens (human)Kd25.3846313
Eukaryotic peptide chain release factor GTP-binding subunit ERF3BHomo sapiens (human)Kd30.000011
Eukaryotic translation initiation factor 2-alpha kinase 1Homo sapiens (human)Kd27.1429214
Eukaryotic translation initiation factor 5BHomo sapiens (human)Kd30.000017
Exosome RNA helicase MTR4Homo sapiens (human)Kd30.0000110
Ferrochelatase, mitochondrialHomo sapiens (human)Kd22.5070211
Fibroblast growth factor receptor 1Homo sapiens (human)Kd25.7143314
Fibroblast growth factor receptor 2Homo sapiens (human)Kd10.000023
Fibroblast growth factor receptor 3Homo sapiens (human)Kd10.000046
Fibroblast growth factor receptor 4Homo sapiens (human)Kd10.000023
Focal adhesion kinase 1Homo sapiens (human)Kd26.0000315
G protein-coupled receptor kinase 4Homo sapiens (human)Kd10.000012
G protein-coupled receptor kinase 6Homo sapiens (human)Kd30.000015
General transcription and DNA repair factor IIH helicase subunit XPDHomo sapiens (human)Kd30.0000111
Glycine--tRNA ligaseHomo sapiens (human)Kd30.0000110
Glycogen phosphorylase, brain formHomo sapiens (human)Kd30.0000110
Glycogen phosphorylase, liver formHomo sapiens (human)Kd30.0000110
Glycogen synthase kinase-3 alphaHomo sapiens (human)Kd23.3387313
Glycogen synthase kinase-3 betaHomo sapiens (human)Kd25.7143314
GTP-binding nuclear protein RanHomo sapiens (human)Kd30.0000110
Guanine nucleotide-binding protein G(i) subunit alpha-2Homo sapiens (human)Kd30.000016
Heme oxygenase 2Homo sapiens (human)Kd30.000019
Hepatocyte growth factor receptorHomo sapiens (human)Kd20.0000514
High affinity nerve growth factor receptorHomo sapiens (human)Kd24.0000310
Histone deacetylase 6Homo sapiens (human)EC5030.000011
Homeodomain-interacting protein kinase 1Homo sapiens (human)Kd2.200012
Homeodomain-interacting protein kinase 2Homo sapiens (human)Kd0.405012
Homeodomain-interacting protein kinase 3Homo sapiens (human)Kd0.455012
Homeodomain-interacting protein kinase 4Homo sapiens (human)Kd7.500012
Hormonally up-regulated neu tumor-associated kinaseHomo sapiens (human)Kd10.000012
Inhibitor of nuclear factor kappa-B kinase subunit alphaHomo sapiens (human)Kd5.850012
Inhibitor of nuclear factor kappa-B kinase subunit betaHomo sapiens (human)Kd10.000012
Inhibitor of nuclear factor kappa-B kinase subunit epsilonHomo sapiens (human)Kd25.7143314
Inosine-5'-monophosphate dehydrogenase 2Homo sapiens (human)Kd30.0000110
Insulin receptorHomo sapiens (human)Kd25.7143314
Insulin receptor-related proteinHomo sapiens (human)Kd10.000023
Insulin-like growth factor 1 receptorHomo sapiens (human)Kd25.7143314
Integrin-linked protein kinaseHomo sapiens (human)Kd30.000018
Interferon-induced, double-stranded RNA-activated protein kinaseHomo sapiens (human)Kd10.000023
Interleukin-1 receptor-associated kinase 1Homo sapiens (human)Kd26.6667212
Interleukin-1 receptor-associated kinase 3Homo sapiens (human)Kd23.1952314
Interleukin-1 receptor-associated kinase 4Homo sapiens (human)Kd26.9231213
Isoleucine--tRNA ligase, mitochondrialHomo sapiens (human)Kd30.000017
Leucine-rich repeat serine/threonine-protein kinase 2Homo sapiens (human)Kd10.000024
Leukocyte tyrosine kinase receptorHomo sapiens (human)Kd10.000023
Leukotriene C4 synthaseCavia porcellus (domestic guinea pig)Kd10.000012
LIM domain kinase 1Homo sapiens (human)Kd25.3846313
LIM domain kinase 2Homo sapiens (human)Kd24.3846313
Long-chain-fatty-acid--CoA ligase 5Homo sapiens (human)Kd30.000016
Macrophage colony-stimulating factor 1 receptorHomo sapiens (human)Kd10.000023
Macrophage-stimulating protein receptorHomo sapiens (human)Kd26.6667212
MAP kinase-activated protein kinase 2Homo sapiens (human)Kd25.7143314
MAP kinase-activated protein kinase 3Homo sapiens (human)Kd30.000014
MAP kinase-activated protein kinase 5Homo sapiens (human)Kd25.3846313
MAP kinase-interacting serine/threonine-protein kinase 1Homo sapiens (human)Kd10.000023
MAP kinase-interacting serine/threonine-protein kinase 2Homo sapiens (human)Kd10.000023
MAP/microtubule affinity-regulating kinase 3Homo sapiens (human)Kd25.7143314
MAP/microtubule affinity-regulating kinase 4Homo sapiens (human)Kd24.5455311
Mast/stem cell growth factor receptor KitHomo sapiens (human)Kd10.83331624
Maternal embryonic leucine zipper kinaseHomo sapiens (human)Kd23.5558314
Megakaryocyte-associated tyrosine-protein kinaseHomo sapiens (human)Kd10.000012
Membrane-associated progesterone receptor component 1Homo sapiens (human)Kd30.000018
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinaseHomo sapiens (human)Kd25.3846313
Microtubule-associated serine/threonine-protein kinase 1Homo sapiens (human)Kd10.000012
MidasinHomo sapiens (human)Kd30.0000111
Misshapen-like kinase 1Homo sapiens (human)Kd25.000028
Mitogen-activated protein kinase 1Homo sapiens (human)Kd25.3846313
Mitogen-activated protein kinase 10Homo sapiens (human)Kd24.2133312
Mitogen-activated protein kinase 11Homo sapiens (human)Kd25.7143314
Mitogen-activated protein kinase 12Homo sapiens (human)Kd10.000023
Mitogen-activated protein kinase 13Homo sapiens (human)Kd10.000012
Mitogen-activated protein kinase 14Homo sapiens (human)Kd26.0000315
Mitogen-activated protein kinase 15Homo sapiens (human)Kd26.2500316
Mitogen-activated protein kinase 3 Homo sapiens (human)Kd26.2500316
Mitogen-activated protein kinase 4Homo sapiens (human)Kd10.000023
Mitogen-activated protein kinase 6Homo sapiens (human)Kd10.000023
Mitogen-activated protein kinase 7Homo sapiens (human)Kd25.3846313
Mitogen-activated protein kinase 8Homo sapiens (human)Kd24.7308313
Mitogen-activated protein kinase 9Homo sapiens (human)Kd24.7538313
Mitogen-activated protein kinase kinase kinase 1Homo sapiens (human)Kd26.6667212
Mitogen-activated protein kinase kinase kinase 10Homo sapiens (human)Kd10.000023
Mitogen-activated protein kinase kinase kinase 11Homo sapiens (human)Kd25.3846313
Mitogen-activated protein kinase kinase kinase 12Homo sapiens (human)Kd10.000012
Mitogen-activated protein kinase kinase kinase 13Homo sapiens (human)Kd10.000012
Mitogen-activated protein kinase kinase kinase 15Homo sapiens (human)Kd10.000012
Mitogen-activated protein kinase kinase kinase 19Homo sapiens (human)Kd2.465012
Mitogen-activated protein kinase kinase kinase 2Homo sapiens (human)Kd26.6667212
Mitogen-activated protein kinase kinase kinase 20Homo sapiens (human)Kd25.3846313
Mitogen-activated protein kinase kinase kinase 3Homo sapiens (human)Kd26.6667212
Mitogen-activated protein kinase kinase kinase 4Homo sapiens (human)Kd25.7143314
Mitogen-activated protein kinase kinase kinase 5Homo sapiens (human)Kd25.3846313
Mitogen-activated protein kinase kinase kinase 6Homo sapiens (human)Kd26.6667212
Mitogen-activated protein kinase kinase kinase 7Homo sapiens (human)Kd10.000012
Mitogen-activated protein kinase kinase kinase 9Homo sapiens (human)Kd10.000023
Mitogen-activated protein kinase kinase kinase kinase 1Homo sapiens (human)Kd25.3846313
Mitogen-activated protein kinase kinase kinase kinase 2Homo sapiens (human)Kd26.6667212
Mitogen-activated protein kinase kinase kinase kinase 3Homo sapiens (human)Kd25.3846313
Mitogen-activated protein kinase kinase kinase kinase 4Homo sapiens (human)Kd25.7143314
Mitogen-activated protein kinase kinase kinase kinase 5Homo sapiens (human)Kd25.7143314
Mitotic checkpoint serine/threonine-protein kinase BUB1Homo sapiens (human)Kd30.000018
Multifunctional protein ADE2Homo sapiens (human)Kd30.0000110
Muscle, skeletal receptor tyrosine-protein kinaseHomo sapiens (human)Kd10.000023
Myosin light chain kinase 2, skeletal/cardiac muscleHomo sapiens (human)Kd10.000023
Myosin light chain kinase 3Homo sapiens (human)Kd23.7368211
Myosin light chain kinase family member 4Homo sapiens (human)Kd6.926723
Myosin light chain kinase, smooth muscleGallus gallus (chicken)Kd10.000011
Myosin light chain kinase, smooth muscleHomo sapiens (human)Kd24.8667315
Myosin-10Homo sapiens (human)Kd30.000019
Myosin-14Homo sapiens (human)Kd30.000018
Myosin-IIIaHomo sapiens (human)Kd10.000023
Myosin-IIIbHomo sapiens (human)Kd10.000023
Myotonin-protein kinaseHomo sapiens (human)Kd10.000023
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13Homo sapiens (human)Kd30.0000110
Non-receptor tyrosine-protein kinase TNK1Homo sapiens (human)Kd25.3846313
Non-receptor tyrosine-protein kinase TYK2Homo sapiens (human)Kd22.5133415
NT-3 growth factor receptorHomo sapiens (human)Kd10.000023
NUAK family SNF1-like kinase 1Homo sapiens (human)Kd10.000023
NUAK family SNF1-like kinase 2Homo sapiens (human)Kd25.3846313
Nucleolar GTP-binding protein 1Homo sapiens (human)Kd30.0000110
Nucleoside diphosphate kinase BHomo sapiens (human)Kd30.000014
Obg-like ATPase 1Homo sapiens (human)Kd30.000019
PAS domain-containing serine/threonine-protein kinaseHomo sapiens (human)Kd30.000018
Peripheral plasma membrane protein CASKHomo sapiens (human)Kd10.000012
Peroxisomal acyl-coenzyme A oxidase 1Homo sapiens (human)Kd30.000016
Peroxisomal acyl-coenzyme A oxidase 3Homo sapiens (human)Kd30.0000110
Phenylalanine--tRNA ligase beta subunitHomo sapiens (human)Kd30.0000110
Phosphatidylethanolamine-binding protein 1Homo sapiens (human)Kd30.000018
Phosphatidylinositol 3-kinase catalytic subunit type 3Homo sapiens (human)Kd0.200011
Phosphatidylinositol 3-kinase regulatory subunit alphaHomo sapiens (human)EC500.046723
Phosphatidylinositol 4-kinase betaHomo sapiens (human)Kd23.375024
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit betaHomo sapiens (human)Kd0.464035
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gammaHomo sapiens (human)Kd0.170512
Phosphatidylinositol 4-phosphate 5-kinase type-1 alphaHomo sapiens (human)Kd10.000023
Phosphatidylinositol 4-phosphate 5-kinase type-1 gammaHomo sapiens (human)Kd10.000012
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformHomo sapiens (human)EC500.054357
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformHomo sapiens (human)Kd0.00241526
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformHomo sapiens (human)EC500.029524
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformHomo sapiens (human)Kd0.010946
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformHomo sapiens (human)EC500.042835
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformHomo sapiens (human)Kd0.049046
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)EC500.059024
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)Kd0.037446
Phosphatidylinositol 5-phosphate 4-kinase type-2 alphaHomo sapiens (human)Kd30.000017
Phosphatidylinositol 5-phosphate 4-kinase type-2 betaHomo sapiens (human)Kd10.000023
Phosphatidylinositol 5-phosphate 4-kinase type-2 gammaHomo sapiens (human)Kd22.0605213
Phosphorylase b kinase gamma catalytic chain, liver/testis isoformHomo sapiens (human)Kd25.3846313
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoformHomo sapiens (human)Kd10.000023
Platelet-derived growth factor receptor alphaHomo sapiens (human)Kd10.000023
Platelet-derived growth factor receptor betaHomo sapiens (human)Kd25.7143314
Probable ATP-dependent RNA helicase DDX6Homo sapiens (human)Kd30.000019
Prostaglandin G/H synthase 2Homo sapiens (human)Kd10.000012
Protein kinase C alpha typeHomo sapiens (human)Kd30.0000112
Protein kinase C beta typeHomo sapiens (human)Kd30.0000111
Protein kinase C delta typeHomo sapiens (human)Kd25.3846313
Protein kinase C epsilon typeHomo sapiens (human)Kd10.000023
Protein kinase C eta typeHomo sapiens (human)Kd10.000023
Protein kinase C iota typeHomo sapiens (human)Kd26.6667212
Protein kinase C theta typeHomo sapiens (human)Kd25.0000312
Protein kinase C zeta typeHomo sapiens (human)Kd30.000016
Protein-tyrosine kinase 2-betaHomo sapiens (human)Kd25.3846313
Protein-tyrosine kinase 6Homo sapiens (human)Kd25.3846313
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)Kd20.0000720
Proto-oncogene tyrosine-protein kinase ROSHomo sapiens (human)Kd10.000023
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)Kd25.3846313
Putative heat shock protein HSP 90-beta 2Homo sapiens (human)Kd30.0000111
Putative nucleoside diphosphate kinaseHomo sapiens (human)Kd30.000012
Pyridoxal kinaseHomo sapiens (human)Kd30.0000110
Rab-like protein 3Homo sapiens (human)Kd30.0000110
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)Kd21.4358414
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)Kd23.5729314
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)Kd23.5866314
RAF proto-oncogene serine/threonine-protein kinaseHomo sapiens (human)Kd5.800023
Ras-related C3 botulinum toxin substrate 1Homo sapiens (human)Kd30.000011
Ras-related protein Rab-10Homo sapiens (human)Kd30.0000110
Ras-related protein Rab-27AHomo sapiens (human)Kd30.000019
Ras-related protein Rab-6AHomo sapiens (human)Kd30.000018
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)Kd10.000023
Receptor tyrosine-protein kinase erbB-3Homo sapiens (human)Kd10.000012
Receptor tyrosine-protein kinase erbB-4Homo sapiens (human)Kd10.000012
Receptor-interacting serine/threonine-protein kinase 1Homo sapiens (human)Kd10.000023
Receptor-interacting serine/threonine-protein kinase 2Homo sapiens (human)Kd26.0000315
Receptor-interacting serine/threonine-protein kinase 3Homo sapiens (human)Kd30.0000110
Receptor-interacting serine/threonine-protein kinase 4Homo sapiens (human)Kd10.000012
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)Kd14.80381329
Rho-associated protein kinase 1Homo sapiens (human)Kd27.1429214
Rho-associated protein kinase 2Homo sapiens (human)Kd27.1429214
Rhodopsin kinase GRK1Homo sapiens (human)Kd10.000012
Rhodopsin kinase GRK7Homo sapiens (human)Kd10.000012
Ribosomal protein S6 kinase alpha-1Homo sapiens (human)Kd22.5000516
Ribosomal protein S6 kinase alpha-2Homo sapiens (human)Kd10.000046
Ribosomal protein S6 kinase alpha-3Homo sapiens (human)Kd24.8462313
Ribosomal protein S6 kinase alpha-4Homo sapiens (human)Kd22.5000516
Ribosomal protein S6 kinase alpha-5Homo sapiens (human)Kd22.9412517
Ribosomal protein S6 kinase alpha-6Homo sapiens (human)Kd22.6706517
Ribosomal protein S6 kinase beta-1Homo sapiens (human)Kd26.0000210
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiens (human)Kd27.1028110
RNA cytidine acetyltransferaseHomo sapiens (human)Kd30.0000111
S-adenosylmethionine synthase isoform type-2Homo sapiens (human)Kd30.000019
Septin-9Homo sapiens (human)Kd30.0000112
Serine/threonine-protein kinase 10Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase 16Homo sapiens (human)Kd25.0786314
Serine/threonine-protein kinase 17AHomo sapiens (human)Kd10.000023
Serine/threonine-protein kinase 17BHomo sapiens (human)Kd10.000023
Serine/threonine-protein kinase 24Homo sapiens (human)Kd25.0000312
Serine/threonine-protein kinase 25Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase 26Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase 3Homo sapiens (human)Kd25.7143314
Serine/threonine-protein kinase 32AHomo sapiens (human)Kd10.000012
Serine/threonine-protein kinase 32BHomo sapiens (human)Kd10.000023
Serine/threonine-protein kinase 32CHomo sapiens (human)Kd10.000023
Serine/threonine-protein kinase 33Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase 35Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase 36Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase 38Homo sapiens (human)Kd23.333326
Serine/threonine-protein kinase 38-likeHomo sapiens (human)Kd23.333339
Serine/threonine-protein kinase 4Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase A-RafHomo sapiens (human)Kd30.000019
Serine/threonine-protein kinase ATRHomo sapiens (human)Kd30.000014
Serine/threonine-protein kinase B-rafHomo sapiens (human)Kd20.6500516
Serine/threonine-protein kinase BRSK1Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase BRSK2Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase Chk1Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase Chk2Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase D1Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase D2Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase D3Homo sapiens (human)Kd25.7143314
Serine/threonine-protein kinase DCLK1Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase DCLK2Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase DCLK3Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase ICKHomo sapiens (human)Kd26.6083212
Serine/threonine-protein kinase LATS1Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase LATS2Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase MAKHomo sapiens (human)Kd10.000012
Serine/threonine-protein kinase MARK1Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase MARK2Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase MRCK alphaHomo sapiens (human)Kd24.5429314
Serine/threonine-protein kinase MRCK betaHomo sapiens (human)Kd25.7143314
Serine/threonine-protein kinase MRCK gammaHomo sapiens (human)Kd24.0000310
Serine/threonine-protein kinase mTORHomo sapiens (human)Kd1.587846
Serine/threonine-protein kinase N1Homo sapiens (human)Kd25.7143314
Serine/threonine-protein kinase N2Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase N3Homo sapiens (human)Kd30.000016
Serine/threonine-protein kinase Nek1Homo sapiens (human)Kd25.7143314
Serine/threonine-protein kinase Nek11Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase Nek2Homo sapiens (human)Kd25.7143314
Serine/threonine-protein kinase Nek3Homo sapiens (human)Kd26.9231213
Serine/threonine-protein kinase Nek4Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase Nek5Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase Nek6Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase Nek7Homo sapiens (human)Kd23.333339
Serine/threonine-protein kinase Nek9Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase NIM1Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase NLKHomo sapiens (human)Kd26.0000315
Serine/threonine-protein kinase OSR1Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase PAK 1Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase PAK 2Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase PAK 3Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase PAK 4Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase PAK 5Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase PAK 6Homo sapiens (human)Kd23.333339
Serine/threonine-protein kinase pim-1Homo sapiens (human)EC505.005022
Serine/threonine-protein kinase pim-1Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase pim-2Homo sapiens (human)EC505.005022
Serine/threonine-protein kinase pim-2Homo sapiens (human)Kd20.000036
Serine/threonine-protein kinase pim-3Homo sapiens (human)EC505.005022
Serine/threonine-protein kinase pim-3Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase PknBMycobacterium tuberculosis H37RvKd10.000012
Serine/threonine-protein kinase PLK1Homo sapiens (human)Kd22.500038
Serine/threonine-protein kinase PLK2Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase PLK3Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase PLK4Homo sapiens (human)Kd24.8154313
Serine/threonine-protein kinase PRP4 homologHomo sapiens (human)Kd10.000012
Serine/threonine-protein kinase receptor R3Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase RIO1Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase RIO2Homo sapiens (human)Kd0.720012
Serine/threonine-protein kinase RIO3Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase SBK1Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase Sgk3Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase SIK1Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase SIK2Homo sapiens (human)Kd25.3846313
Serine/threonine-protein kinase SIK3Homo sapiens (human)Kd25.0008214
Serine/threonine-protein kinase STK11Homo sapiens (human)Kd25.0000312
Serine/threonine-protein kinase TAO1Homo sapiens (human)Kd26.9231213
Serine/threonine-protein kinase TAO2Homo sapiens (human)Kd26.6667212
Serine/threonine-protein kinase TAO3Homo sapiens (human)Kd26.6667212
Serine/threonine-protein kinase TBK1Homo sapiens (human)Kd27.1429214
Serine/threonine-protein kinase TNNI3KHomo sapiens (human)Kd10.000023
Serine/threonine-protein kinase tousled-like 1Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase tousled-like 2Homo sapiens (human)Kd10.000023
Serine/threonine-protein kinase ULK1Homo sapiens (human)Kd26.6667212
Serine/threonine-protein kinase ULK2Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase ULK3Homo sapiens (human)Kd26.6667212
Serine/threonine-protein kinase VRK2Homo sapiens (human)Kd10.000012
Serine/threonine-protein kinase/endoribonuclease IRE1Homo sapiens (human)Kd26.6667212
Serine/threonine-protein kinase/endoribonuclease IRE2Homo sapiens (human)Kd30.0000110
Signal recognition particle receptor subunit alphaHomo sapiens (human)Kd30.000018
SNF-related serine/threonine-protein kinaseHomo sapiens (human)Kd10.000012
SRSF protein kinase 1Homo sapiens (human)Kd10.000023
SRSF protein kinase 2Homo sapiens (human)Kd10.000023
SRSF protein kinase 3Homo sapiens (human)Kd10.000012
STE20-like serine/threonine-protein kinase Homo sapiens (human)Kd25.3846313
STE20-related kinase adapter protein alphaHomo sapiens (human)Kd30.0000111
STE20/SPS1-related proline-alanine-rich protein kinaseHomo sapiens (human)Kd10.000012
Structural maintenance of chromosomes protein 1AHomo sapiens (human)Kd30.000019
Structural maintenance of chromosomes protein 2Homo sapiens (human)Kd30.0000110
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrialHomo sapiens (human)Kd30.0000110
Testis-specific serine/threonine-protein kinase 1Homo sapiens (human)Kd10.000023
TGF-beta receptor type-1Homo sapiens (human)Kd25.3846313
TGF-beta receptor type-2Homo sapiens (human)Kd24.5455311
Thyroid hormone receptor-associated protein 3Homo sapiens (human)Kd30.000017
TRAF2 and NCK-interacting protein kinaseHomo sapiens (human)Kd25.3846313
Transient receptor potential cation channel subfamily M member 6Homo sapiens (human)Kd10.000012
Tubulin alpha-1A chainRattus norvegicus (Norway rat)Kd10.000011
Tyrosine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000019
Tyrosine-protein kinase ABL1Homo sapiens (human)Kd14.25532347
Tyrosine-protein kinase ABL2Homo sapiens (human)Kd25.7143314
Tyrosine-protein kinase BlkHomo sapiens (human)Kd10.000023
Tyrosine-protein kinase BTKHomo sapiens (human)Kd25.7143314
Tyrosine-protein kinase CSKHomo sapiens (human)Kd25.3846313
Tyrosine-protein kinase FerHomo sapiens (human)Kd25.3846313
Tyrosine-protein kinase Fes/FpsHomo sapiens (human)Kd25.7143314
Tyrosine-protein kinase FgrHomo sapiens (human)Kd21.428637
Tyrosine-protein kinase FRKHomo sapiens (human)Kd25.3846313
Tyrosine-protein kinase FynHomo sapiens (human)Kd25.7143314
Tyrosine-protein kinase HCKHomo sapiens (human)Kd25.3846313
Tyrosine-protein kinase ITK/TSKHomo sapiens (human)Kd10.000023
Tyrosine-protein kinase JAK1Homo sapiens (human)Kd22.6519416
Tyrosine-protein kinase JAK2Homo sapiens (human)Kd15.000034
Tyrosine-protein kinase JAK3Homo sapiens (human)Kd10.000023
Tyrosine-protein kinase LckHomo sapiens (human)Kd25.3846313
Tyrosine-protein kinase LynHomo sapiens (human)Kd25.3846313
Tyrosine-protein kinase MerHomo sapiens (human)Kd18.000035
Tyrosine-protein kinase receptor Tie-1Homo sapiens (human)Kd10.000023
Tyrosine-protein kinase receptor TYRO3Homo sapiens (human)Kd10.000023
Tyrosine-protein kinase receptor UFOHomo sapiens (human)Kd10.000023
Tyrosine-protein kinase SrmsHomo sapiens (human)Kd10.000023
Tyrosine-protein kinase SYKHomo sapiens (human)Kd25.3846313
Tyrosine-protein kinase TecHomo sapiens (human)Kd25.3846313
Tyrosine-protein kinase TXKHomo sapiens (human)Kd10.000023
Tyrosine-protein kinase YesHomo sapiens (human)Kd25.3846313
Tyrosine-protein kinase ZAP-70Homo sapiens (human)Kd10.000023
U5 small nuclear ribonucleoprotein 200 kDa helicaseHomo sapiens (human)Kd30.0000110
UMP-CMP kinase Homo sapiens (human)Kd30.000015
Uncharacterized aarF domain-containing protein kinase 5Homo sapiens (human)Kd30.000015
Uncharacterized protein FLJ45252Homo sapiens (human)Kd30.0000110
Uncharacterized serine/threonine-protein kinase SBK3Homo sapiens (human)Kd10.000012
Vascular endothelial growth factor receptor 1 Homo sapiens (human)Kd10.000023
Vascular endothelial growth factor receptor 2Homo sapiens (human)Kd10.000023
Vascular endothelial growth factor receptor 3Homo sapiens (human)Kd10.000023
Very long-chain specific acyl-CoA dehydrogenase, mitochondrialHomo sapiens (human)Kd30.0000111
Wee1-like protein kinaseHomo sapiens (human)Kd26.0000315
Wee1-like protein kinase 2Homo sapiens (human)Kd10.000012

Other Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
heat shock protein 90, putativePlasmodium falciparum 3D7AC500.215011
heat shock protein HSP 90-alpha isoform 2Homo sapiens (human)AC500.363011
Phosphatidylinositol 3-kinase regulatory subunit alphaHomo sapiens (human)INH0.016011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformHomo sapiens (human)INH0.008911
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformHomo sapiens (human)Imax16.750023
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformHomo sapiens (human)INH0.017011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformHomo sapiens (human)INH0.016011
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)INH0.053011
Proteinase-activated receptor 1Homo sapiens (human)Imax13.187524