Page last updated: 2024-08-08 00:06:59
Trace amine-associated receptor 1
A protein that is a translation product of the Taar1 gene in rat. [PRO:DNx, UniProtKB:Q923Y9]
Synonyms
TaR-1;
Trace amine receptor 1
Research
Bioassay Publications (7)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 2 (28.57) | 29.6817 |
2010's | 4 (57.14) | 24.3611 |
2020's | 1 (14.29) | 2.80 |
Compounds (16)
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
phenethylamine | Rattus norvegicus (Norway rat) | EC50 | 0.1842 | 5 | 5 |
tryptamine | Rattus norvegicus (Norway rat) | EC50 | 0.3100 | 1 | 1 |
n-methyl-3,4-methylenedioxyamphetamine | Rattus norvegicus (Norway rat) | EC50 | 1.7000 | 1 | 1 |
p-hydroxyamphetamine | Rattus norvegicus (Norway rat) | EC50 | 0.0505 | 2 | 2 |
octopamine | Rattus norvegicus (Norway rat) | EC50 | 1.3000 | 1 | 1 |
tyramine | Rattus norvegicus (Norway rat) | EC50 | 0.0495 | 2 | 2 |
dextroamphetamine | Rattus norvegicus (Norway rat) | EC50 | 0.5328 | 6 | 6 |
methamphetamine | Rattus norvegicus (Norway rat) | EC50 | 0.8173 | 4 | 4 |
l-amphetamine | Rattus norvegicus (Norway rat) | EC50 | 0.3847 | 6 | 6 |
desethylamiodarone | Rattus norvegicus (Norway rat) | EC50 | 0.0330 | 1 | 1 |
di-n-desethylamiodarone | Rattus norvegicus (Norway rat) | EC50 | 1.0000 | 1 | 1 |
3,3',5-triiodothyronamine | Rattus norvegicus (Norway rat) | EC50 | 0.0870 | 1 | 1 |
thyroxamine | Rattus norvegicus (Norway rat) | EC50 | 1.0000 | 1 | 1 |
thyronamine | Rattus norvegicus (Norway rat) | EC50 | 0.1310 | 1 | 1 |
3-iodothyronamine | Rattus norvegicus (Norway rat) | EC50 | 0.0224 | 1 | 1 |
ro5166017 | Rattus norvegicus (Norway rat) | EC50 | 0.0140 | 1 | 1 |