Page last updated: 2024-08-07 21:19:12
Histamine H4 receptor
[no definition available]
Synonyms
Research
Bioassay Publications (2)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 2 (100.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (3)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| histamine | Cavia porcellus (domestic guinea pig) | Ki | 0.0060 | 1 | 1 |
| jnj 7777120 | Cavia porcellus (domestic guinea pig) | Ki | 1.0715 | 1 | 1 |
| pf-3893787 | Cavia porcellus (domestic guinea pig) | Ki | 0.1230 | 2 | 2 |
Functional Profiling of 2-Aminopyrimidine Histamine H4 Receptor Modulators.Journal of medicinal chemistry, , Sep-24, Volume: 58, Issue:18, 2015
Challenges of drug discovery in novel target space. The discovery and evaluation of PF-3893787: a novel histamine H4 receptor antagonist.Bioorganic & medicinal chemistry letters, , Nov-01, Volume: 21, Issue:21, 2011