Page last updated: 2024-08-07 23:36:19
Sodium/glucose cotransporter 2
A sodium/glucose cotransporter 2 that is encoded in the genome of rat. [OMA:P53792, PRO:DNx]
Synonyms
Na(+)/glucose cotransporter 2;
Low affinity sodium-glucose cotransporter;
Solute carrier family 5 member 2
Research
Bioassay Publications (4)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 2 (50.00) | 29.6817 |
2010's | 2 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (3)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
phlorhizin | Rattus norvegicus (Norway rat) | IC50 | 0.0960 | 1 | 1 |
pf 04971729 | Rattus norvegicus (Norway rat) | IC50 | 0.0012 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
dapagliflozin | Rattus norvegicus (Norway rat) | EC50 | 0.0030 | 2 | 2 |