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Translocator protein
A translocator protein that is encoded in the genome of mouse. [PRO:DNx, UniProtKB:P50637]
Synonyms
Mitochondrial benzodiazepine receptor;
PKBS;
Peripheral-type benzodiazepine receptor;
PBR
Research
Bioassay Publications (3)
Timeframe | Studies on this Protein(%) | All Drugs % |
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (33.33) | 18.2507 |
2000's | 2 (66.67) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (5)
Drugs with Inhibition Measurements
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
ro 5-4864 | Mus musculus (house mouse) | Activity | 0.0002 | 1 | 1 |
arginine vasopressin | Mus musculus (house mouse) | Kact | 0.0023 | 1 | 1 |
The translocator protein (18 kDa): central nervous system disease and drug design.Journal of medicinal chemistry, , Feb-12, Volume: 52, Issue:3, 2009
(S)-(-)-4-[4-[2-(isochroman-1-yl)ethyl]-piperazin-1-yl] benzenesulfonamide, a selective dopamine D4 antagonist.Journal of medicinal chemistry, , Jun-21, Volume: 39, Issue:13, 1996