Page last updated: 2024-08-07 13:20:53
Translocator protein
A translocator protein that is encoded in the genome of mouse. [PRO:DNx, UniProtKB:P50637]
Synonyms
Mitochondrial benzodiazepine receptor;
PKBS;
Peripheral-type benzodiazepine receptor;
PBR
Research
Bioassay Publications (3)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (33.33) | 18.2507 |
2000's | 2 (66.67) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (5)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
ro 5-4864 | Mus musculus (house mouse) | IC50 | 0.0100 | 1 | 1 |
n,n-di-n-hexyl-2-(4-fluorophenyl)indole-3-acetamide | Mus musculus (house mouse) | IC50 | 0.0100 | 1 | 1 |
arginine vasopressin | Mus musculus (house mouse) | Ki | 0.0004 | 1 | 2 |
deamino arginine vasopressin | Mus musculus (house mouse) | Ki | 0.0003 | 1 | 2 |
vasopressin, 1-deamino-4-val-8-arg- | Mus musculus (house mouse) | Ki | 0.0003 | 1 | 2 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
ro 5-4864 | Mus musculus (house mouse) | Activity | 0.0002 | 1 | 1 |
arginine vasopressin | Mus musculus (house mouse) | Kact | 0.0023 | 1 | 1 |