Page last updated: 2024-08-07 23:26:23
Glucagon-like peptide 1 receptor
A glucagon-like peptide 1 receptor that is encoded in the genome of rat. [OMA:P32301, PRO:DNx]
Synonyms
GLP-1 receptor;
GLP-1-R;
GLP-1R
Research
Bioassay Publications (2)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 1 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (2)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
glucagon-like peptide 1 (1-37) | Rattus norvegicus (Norway rat) | IC50 | 1.0000 | 1 | 1 |
exenatide | Rattus norvegicus (Norway rat) | IC50 | 0.0001 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
glucagon-like peptide 1 (1-37) | Rattus norvegicus (Norway rat) | EC50 | 0.0001 | 1 | 1 |