Page last updated: 2024-08-07 15:40:52
Progesterone receptor
A progesterone receptor that is encoded in the genome of rabbit. [OMA:P06186, PRO:DNx]
Synonyms
PR;
Nuclear receptor subfamily 3 group C member 3
Research
Bioassay Publications (2)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 2 (100.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (2)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| bicalutamide | Oryctolagus cuniculus (rabbit) | IC50 | 5.6000 | 2 | 2 |
| dihydrotestosterone | Oryctolagus cuniculus (rabbit) | IC50 | 0.4400 | 2 | 2 |
Tetrahydroquinolines as a novel series of nonsteroidal selective androgen receptor modulators: structural requirements for better physicochemical and biological properties.Bioorganic & medicinal chemistry letters, , Nov-01, Volume: 21, Issue:21, 2011
Design and synthesis of tricyclic tetrahydroquinolines as a new series of nonsteroidal selective androgen receptor modulators (SARMs).Bioorganic & medicinal chemistry letters, , Mar-15, Volume: 21, Issue:6, 2011
Tetrahydroquinolines as a novel series of nonsteroidal selective androgen receptor modulators: structural requirements for better physicochemical and biological properties.Bioorganic & medicinal chemistry letters, , Nov-01, Volume: 21, Issue:21, 2011
Design and synthesis of tricyclic tetrahydroquinolines as a new series of nonsteroidal selective androgen receptor modulators (SARMs).Bioorganic & medicinal chemistry letters, , Mar-15, Volume: 21, Issue:6, 2011