Page last updated: 2024-08-07 23:06:59
Solute carrier family 22 member 3
A solute carrier family 22 member 3 that is encoded in the genome of rat. [OMA:O88446, PRO:DNx]
Synonyms
Organic cation transporter 3
Research
Bioassay Publications (3)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (66.67) | 18.2507 |
2000's | 1 (33.33) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (8)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
desipramine | Rattus norvegicus (Norway rat) | IC50 | 68.0000 | 1 | 1 |
amphetamine | Rattus norvegicus (Norway rat) | IC50 | 42.0000 | 1 | 1 |
corticosterone | Rattus norvegicus (Norway rat) | IC50 | 4.9000 | 1 | 1 |
desoxycorticosterone | Rattus norvegicus (Norway rat) | IC50 | 8.4000 | 1 | 1 |
methamphetamine | Rattus norvegicus (Norway rat) | IC50 | 248.0000 | 1 | 1 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
agmatine | Rattus norvegicus (Norway rat) | Km | 900.0000 | 1 | 1 |
tetraethylammonium | Rattus norvegicus (Norway rat) | Km | 4,350.0000 | 2 | 2 |
1-methyl-4-phenylpyridinium | Rattus norvegicus (Norway rat) | Km | 57.5000 | 2 | 2 |