Page last updated: 2024-08-07 23:00:25
Solute carrier family 22 member 1
A solute carrier family 22 member 1 that is encoded in the genome of mouse. [OMA:O08966, PRO:DNx]
Synonyms
Organic cation transporter 1;
mOCT1
Research
Bioassay Publications (5)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (20.00) | 18.2507 |
2000's | 3 (60.00) | 29.6817 |
2010's | 1 (20.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (11)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
choline | Mus musculus (house mouse) | IC50 | 55.0000 | 1 | 1 |
cimetidine | Mus musculus (house mouse) | IC50 | 0.5900 | 1 | 1 |
procainamide | Mus musculus (house mouse) | IC50 | 3.9000 | 1 | 1 |
pyrimethamine | Mus musculus (house mouse) | Ki | 3.6000 | 1 | 1 |
tetraethylammonium | Mus musculus (house mouse) | IC50 | 0.5400 | 1 | 1 |
tetraethylammonium | Mus musculus (house mouse) | Ki | 128.0000 | 1 | 1 |
tetramethylammonium chloride | Mus musculus (house mouse) | Ki | 2,040.0000 | 1 | 1 |
tetrapropylammonium | Mus musculus (house mouse) | Ki | 19.8000 | 1 | 1 |
tetrabutylammonium | Mus musculus (house mouse) | Ki | 7.3000 | 1 | 1 |
n-methylnicotinamide | Mus musculus (house mouse) | IC50 | 7,337.0000 | 1 | 1 |
quinine | Mus musculus (house mouse) | IC50 | 0.2800 | 1 | 1 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
choline | Mus musculus (house mouse) | Km | 42.0000 | 1 | 1 |
tetraethylammonium | Mus musculus (house mouse) | Km | 38.0000 | 1 | 1 |
tetrabutylammonium | Mus musculus (house mouse) | Km | 43.0000 | 1 | 1 |
1-methyl-4-phenylpyridinium | Mus musculus (house mouse) | Km | 10.0000 | 1 | 1 |