Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
marimastat | Homo sapiens (human) | IC50 | 0.0184 | 2 | 0 |
2-(2,4-dioxo-3-phenyl-5-thiazolidinyl)-N-phenylacetamide | Homo sapiens (human) | IC50 | 46.6640 | 1 | 0 |
5-hydroxy-2-[[(4-methylphenyl)thio]methyl]-3-benzofurancarboxylic acid ethyl ester | Homo sapiens (human) | IC50 | 69.5550 | 1 | 0 |
4-ethoxy-N-(4-fluorophenyl)-2,3-dimethylbenzenesulfonamide | Homo sapiens (human) | IC50 | 69.5270 | 1 | 0 |
4-[[5-chloro-2-[(4-fluorophenyl)methoxy]phenyl]methylamino]benzenesulfonamide | Homo sapiens (human) | IC50 | 69.5130 | 1 | 0 |
4-[(2-bromophenoxy)methyl]-N-[4-[(3,5-dimethyl-1-pyrazolyl)methyl]phenyl]benzamide | Homo sapiens (human) | IC50 | 69.5200 | 1 | 0 |
5-bromo-N-[[4-[(3,5-dimethylphenyl)sulfamoyl]anilino]-sulfanylidenemethyl]-2-furancarboxamide | Homo sapiens (human) | IC50 | 69.5110 | 1 | 0 |
N-(9,9-dimethyl-7-oxo-8,10-dihydronaphtho[1,2-b]benzofuran-5-yl)-4-methoxybenzenesulfonamide | Homo sapiens (human) | IC50 | 69.5130 | 1 | 0 |
5-[3-[(2,4-dichlorophenyl)methoxy]-2-thiophenyl]-1,2-dihydro-1,2,4-triazole-3-thione | Homo sapiens (human) | IC50 | 69.5040 | 1 | 0 |
4-(4-chloro-2-methylphenoxy)-N-[3-(methylthio)phenyl]butanamide | Homo sapiens (human) | IC50 | 69.4980 | 1 | 0 |
3-[(2-methoxyphenyl)-prop-2-enylsulfamoyl]benzoic acid [2-(1H-indol-3-yl)-2-oxoethyl] ester | Homo sapiens (human) | IC50 | 69.4880 | 1 | 0 |
4-(1H-benzimidazol-2-ylthio)butanoic acid [2-oxo-2-(4-phenoxyanilino)ethyl] ester | Homo sapiens (human) | IC50 | 69.5130 | 1 | 0 |
4-[[3-methoxy-4-[(4-nitrophenyl)methoxy]phenyl]-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-5-methyl-1,2-dihydropyrazol-3-one | Homo sapiens (human) | IC50 | 69.5200 | 1 | 0 |
N-[2-[(2-furanylmethylamino)-oxomethyl]phenyl]-4-methyl-3-(1-piperidinylsulfonyl)benzamide | Homo sapiens (human) | IC50 | 69.4800 | 1 | 0 |
cb 7969312 | Homo sapiens (human) | IC50 | 9.1060 | 1 | 0 |
3-(6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-3-yl)-4-prop-2-enyl-1H-1,2,4-triazole-5-thione | Homo sapiens (human) | IC50 | 69.4490 | 1 | 0 |
5-chloro-7-[1-piperidinyl(2-pyridinyl)methyl]-8-quinolinol | Homo sapiens (human) | IC50 | 17.0040 | 1 | 0 |
2-(thiophen-2-ylsulfonylamino)benzoic acid [2-(3-acetylanilino)-2-oxo-1-phenylethyl] ester | Homo sapiens (human) | IC50 | 69.5340 | 2 | 0 |
4-[4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1-piperidinyl]-3-nitrobenzoic acid methyl ester | Homo sapiens (human) | IC50 | 69.5200 | 1 | 0 |
2-[(2,6-dichlorophenyl)sulfonylamino]-3-methylbutanoic acid [2-(1H-indol-3-yl)-2-oxoethyl] ester | Homo sapiens (human) | IC50 | 69.5130 | 1 | 0 |