Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
citric acid, anhydrous | Homo sapiens (human) | IC50 | 39.8690 | 1 | 0 |
ketotifen | Homo sapiens (human) | IC50 | 39.8410 | 1 | 0 |
alverine citrate | Homo sapiens (human) | IC50 | 39.8410 | 1 | 0 |
sufentanil citrate | Homo sapiens (human) | IC50 | 24.7890 | 1 | 0 |
carbetapentane citrate | Homo sapiens (human) | IC50 | 8.4485 | 2 | 0 |
butethamate citrate | Homo sapiens (human) | IC50 | 23.8730 | 1 | 0 |
mosapride | Homo sapiens (human) | IC50 | 12.7060 | 1 | 0 |
mosapride | Homo sapiens (human) | IC50 | 4.1800 | 1 | 0 |
1,5-bis(2-methoxyphenyl)penta-1,4-dien-3-one | Homo sapiens (human) | IC50 | 6.4640 | 1 | 0 |
[(1S,2R,3S,4S,6R,7R,8R)-4-ethenyl-3-hydroxy-2,4,7,14-tetramethyl-9-oxo-6-tricyclo[5.4.3.01,8]tetradecanyl] 2-[2-(diethylamino)ethylsulfanyl]acetate | Homo sapiens (human) | IC50 | 39.8410 | 1 | 0 |
toremifene citrate | Homo sapiens (human) | IC50 | 7.8660 | 1 | 0 |
zuclomifene citrate | Homo sapiens (human) | IC50 | 10.7550 | 1 | 0 |
ketotifen fumarate | Homo sapiens (human) | IC50 | 39.8410 | 1 | 0 |
2-[[5,6-bis(2-furanyl)-1,2,4-triazin-3-yl]thio]-N-(3-methylphenyl)acetamide | Homo sapiens (human) | IC50 | 1.4170 | 1 | 0 |
enclomiphene citrate | Homo sapiens (human) | IC50 | 5.0910 | 1 | 0 |
dibenzheptropine citrate | Homo sapiens (human) | IC50 | 10.0170 | 1 | 0 |
chlorhexidine | Homo sapiens (human) | IC50 | 26.3363 | 2 | 0 |
tiamulin fumarate (1:1), (3as-(3aalpha,4beta,5alpha,6alpha,8beta,9alpha,9abeta,10s*))-isomer | Homo sapiens (human) | IC50 | 39.8410 | 1 | 0 |
chlorhexidine hydrochloride | Homo sapiens (human) | IC50 | 21.4360 | 1 | 0 |
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamide | Homo sapiens (human) | IC50 | 21.5555 | 2 | 0 |
1-butyl-3-(5-methyl-6-oxo-3-benzo[b][1,4]benzothiazepinyl)urea | Homo sapiens (human) | IC50 | 39.8313 | 3 | 0 |
5-chloro-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(phenylmethyl)sulfonyl-4-pyrimidinecarboxamide | Homo sapiens (human) | IC50 | 5.9540 | 1 | 0 |
5-chloro-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[(4-fluorophenyl)methylsulfonyl]-4-pyrimidinecarboxamide | Homo sapiens (human) | IC50 | 5.5060 | 1 | 0 |