Page last updated: 2024-08-07 15:10:33

Sphingosine-1-phosphate receptor 4

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (22)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
9,10-phenanthrenequinoneHomo sapiens (human)IC502.029010
isovelleralHomo sapiens (human)IC500.253010
2-phenyl-4,5-dichloro-3-pyridazinoneHomo sapiens (human)IC501.860010
2-methyl-4-nitroquinoline 1-oxideHomo sapiens (human)IC500.220010
8-(4-tolylsulfonylamino)quinolineHomo sapiens (human)IC500.590120
2,3-dichloro-5,8-dimethoxy-1,4-naphthoquinoneHomo sapiens (human)IC502.016010
6-methoxy-3-nitro-2-(phenylsulfonyl)pyridineHomo sapiens (human)IC501.057020
nsc 105827Homo sapiens (human)IC500.420010
(3E,9E)-5,6-Dihydroxy-9,13,14-trimethyl-16-(2-methylpropyl)-17-azatricyclo[9.7.0.01,15]octadeca-3,9,12-triene-2,18-dioneHomo sapiens (human)IC500.648010
5-(2,5-difluorophenyl)-N-(2,6-dimethylphenyl)-2-furancarboxamideHomo sapiens (human)IC500.308010
5-(2,5-dichlorophenyl)-N-(2,6-dimethoxyphenyl)-2-furancarboxamideHomo sapiens (human)IC500.417010
5-(2,5-dichlorophenyl)-N-[2,6-di(propan-2-yl)phenyl]-2-furancarboxamideHomo sapiens (human)IC500.105010
5-(2,5-dichlorophenyl)-N-(2,6-diethylphenyl)-2-furancarboxamideHomo sapiens (human)IC500.089010
N-(2,6-dimethylphenyl)-5-(4-methyl-3-thiophenyl)-2-furancarboxamideHomo sapiens (human)IC500.286010

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
pinafideHomo sapiens (human)EC505.530010
2-(3-formyl-2,5-dimethyl-1-pyrrolyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid methyl esterHomo sapiens (human)EC5049.800010
2-[2,5-dimethyl-3-[(2,4,6-trioxo-1,3-diazinan-5-ylidene)methyl]-1-pyrrolyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid ethyl esterHomo sapiens (human)EC5016.600010
3-[2-(2,4-dichlorophenoxy)ethoxy]-6-methyl-2-nitropyridineHomo sapiens (human)EC500.345520
N-cyclohexyl-5-propyl-3-isoxazolecarboxamideHomo sapiens (human)EC5050.000010
N,N-dicyclohexyl-5-propyl-3-isoxazolecarboxamideHomo sapiens (human)EC5050.000010
(2S)-2-[[oxo-[5-[oxo-[(phenylmethyl)amino]methyl]-1H-imidazol-4-yl]methyl]amino]-3-phenylpropanoic acid (phenylmethyl) esterHomo sapiens (human)EC5090.200010
(2S)-4-methyl-2-[[oxo-[5-[oxo-[(phenylmethyl)amino]methyl]-1H-imidazol-4-yl]methyl]amino]pentanoic acid (phenylmethyl) esterHomo sapiens (human)EC5014.400010