Page last updated: 2024-08-07 12:30:06

electroneutral potassium-chloride cotransporter KCC2

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (22)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
n-(4-methylthiazol-2-yl)-2-(6-phenylpyridazin-3-ylthio)acetamideHomo sapiens (human)IC500.560010

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
diflunisalHomo sapiens (human)EC503.250010
phenolphthaleinHomo sapiens (human)EC501.800010
3,3',5-triiodothyropropionic acidHomo sapiens (human)EC504.250010
physodic acidHomo sapiens (human)EC508.190010
2-[[5-[(2,3-dimethylphenoxy)methyl]-4-methyl-1,2,4-triazol-3-yl]thio]-1-thiophen-2-ylethanoneHomo sapiens (human)EC509.240010
3-[[4-(1-benzotriazolyl)-1-piperidinyl]sulfonyl]-N-cyclopentylbenzenesulfonamideHomo sapiens (human)EC504.050010
r 59949Homo sapiens (human)EC5074.000030
2-(2-furanyl)-5-[4-(phenylmethyl)-1-piperazinyl]-4-oxazolecarbonitrileHomo sapiens (human)EC5012.000010
1-(2-chlorophenyl)-3-[(2-chlorophenyl)methyl]thioureaHomo sapiens (human)EC505.740010
(E)-4-Phenyl-2-(3-(thiophen-2-yl)acrylamido)thiophene-3-carboxylic acidHomo sapiens (human)EC5029.000010
N-[(3-bromoanilino)-sulfanylidenemethyl]-3-phenylpropanamideHomo sapiens (human)EC50296.000010
2-[[2-[[5-(4-ethylanilino)-1,3,4-thiadiazol-2-yl]thio]-1-oxoethyl]amino]-3-thiophenecarboxamideHomo sapiens (human)EC503.540010
6-(2,3-dihydrobenzofuran-5-yl)-1H-pyrimidine-2-thioneHomo sapiens (human)EC5012.410020
N-[2-(tert-butylamino)-2-oxo-1-thiophen-2-ylethyl]-N-(2-oxolanylmethyl)-5-phenyl-1H-pyrrole-2-carboxamideHomo sapiens (human)EC502.310010
N-[2-(tert-butylamino)-2-oxo-1-pyridin-4-ylethyl]-N-(2-furanylmethyl)-5-phenyl-1H-pyrrole-2-carboxamideHomo sapiens (human)EC5019.100010
5-nitro-2-[(phenylmethyl)amino]benzoic acid [2-(cyclohexylamino)-2-oxoethyl] esterHomo sapiens (human)EC500.481010
[4-(3-chlorophenyl)sulfonyl-3-nitrophenyl]-[4-(2-pyridinyl)-1-piperazinyl]methanoneHomo sapiens (human)EC502.550010
4-methyl-N-[[4-[oxo-[4-(phenylmethyl)-1-piperazinyl]methyl]phenyl]methyl]benzenesulfonamideHomo sapiens (human)EC506.590010
calcimycinHomo sapiens (human)EC5012.680020
2',3'-dihydroxy-4',6'-dimethoxychalconeHomo sapiens (human)EC50486.000010
dafadine CHomo sapiens (human)EC5017.900010