Page last updated: 2024-08-07 17:59:38

SUMO-1-specific protease

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (46)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
ipriflavoneHomo sapiens (human)IC5057.200010
methyldimethylaminoazobenzeneHomo sapiens (human)IC504.400010
1-amino-2-methylanthraquinoneHomo sapiens (human)IC5042.300010
glaucineHomo sapiens (human)IC501.860010
witisolHomo sapiens (human)IC507.600010
papaveraldineHomo sapiens (human)IC500.805010
4',6-dihydroxyflavoneHomo sapiens (human)IC5087.700010
N-[2-(1-azepanyl)-1,3-benzothiazol-6-yl]carbamic acid ethyl esterHomo sapiens (human)IC5033.100010
6-bromoindirubin-3'-oximeHomo sapiens (human)IC50100.000010
2-[(4-nitrophenyl)methylthio]-1,3-benzoxazoleHomo sapiens (human)IC5023.300010
N-(1,3-benzothiazol-2-yl)-N-methylbenzamideHomo sapiens (human)IC5021.100010
N-(2-fluorophenyl)-4-phenylmethoxybenzamideHomo sapiens (human)IC5099.000010
vu0038882Homo sapiens (human)IC5015.000010
2-[(2-fluorophenyl)methylthio]-5-(4-methylphenyl)-1,3,4-oxadiazoleHomo sapiens (human)IC5014.600010
[4-[(2-fluorophenyl)methoxy]phenyl]-(1-pyrrolidinyl)methanethioneHomo sapiens (human)IC509.135020
4-methyl-N,5-diphenyl-3-thiophenecarboxamideHomo sapiens (human)IC506.640010
js 3Homo sapiens (human)IC5023.900010
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-4-methylbenzamideHomo sapiens (human)IC50100.000010
2-[[anilino(oxo)methyl]amino]-N-(phenylmethyl)benzamideHomo sapiens (human)IC50100.000010
5-[(4-methylphenoxy)methyl]-3-phenyl-1,2,4-oxadiazoleHomo sapiens (human)IC5047.100010
3-amino-2-(4-methylphenyl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-oneHomo sapiens (human)IC5018.200010
N-(3-methoxyphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamideHomo sapiens (human)IC5015.500010
N-(1-naphthalenyl)-5-pyridin-4-yl-1,3,4-thiadiazol-2-amineHomo sapiens (human)IC5010.100010
5-(2-chlorophenyl)-N-phenyl-2-furancarboxamideHomo sapiens (human)IC50100.000010
N-(4-methylphenyl)-4-benzofuro[3,2-d]pyrimidinamineHomo sapiens (human)IC50100.000010
4-(2-quinoxalinylamino)benzoic acid ethyl esterHomo sapiens (human)IC50100.000010
4-(3-chloro-2-thiophenyl)-2-(3-pyridinyl)thiazoleHomo sapiens (human)IC5011.300010
2-chloro-3-(prop-2-enylamino)naphthalene-1,4-dioneHomo sapiens (human)IC509.070010
fm19g11Homo sapiens (human)IC504.890010
5-bromo-N-(4,7-dimethoxy-1,3-benzothiazol-2-yl)-2-thiophenecarboxamideHomo sapiens (human)IC5099.000010
3-[[[3-[(3-nitrophenyl)sulfamoyl]phenyl]-oxomethyl]amino]benzoic acidHomo sapiens (human)IC509.020010
2,4-dithiophen-2-ylthiazoleHomo sapiens (human)IC5020.100010
4-(4-methylphenyl)-2-(3-nitrophenyl)-3-pyrazolamineHomo sapiens (human)IC50100.000010
N-[(2-chlorophenyl)methyl]-2-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-hydroxy-5-nitro-4-triazolimineHomo sapiens (human)IC50100.000010
5-(2-chlorophenyl)-N-(4-methoxyphenyl)-2-furancarboxamideHomo sapiens (human)IC504.210010
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-[(phenylmethyl)amino]ethyl] esterHomo sapiens (human)IC5012.800010
2-[4-(difluoromethylthio)anilino]benzoic acid [2-(dimethylamino)-2-oxoethyl] esterHomo sapiens (human)IC5012.800010
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-[[oxo-[(phenylmethyl)amino]methyl]amino]ethyl] esterHomo sapiens (human)IC504.590010
2'-hydroxy-4-methoxychalconeHomo sapiens (human)IC506.000010
5-chloro-N-[4-(2-thiazolo[5,4-b]pyridinyl)phenyl]-2-thiophenesulfonamideHomo sapiens (human)IC5025.000010
dihydroxanthohumolHomo sapiens (human)IC5010.000010
3-[3,5-dimethyl-1-[6-(1-piperidinyl)-3-pyridazinyl]-4-pyrazolyl]-N-(3-fluoro-4-methylphenyl)propanamideHomo sapiens (human)IC5024.400010
2-chloro-3-[2-(4-methylphenyl)-5-tetrazolyl]pyridineHomo sapiens (human)IC504.030010
3-chloro-N-propan-2-yl-5H-indazolo[2,3-a][3,1]benzoxazine-9-carboxamideHomo sapiens (human)IC5081.800010
1-(2,3-dihydro-1H-inden-5-yl)-3-(2-ethoxyphenyl)ureaHomo sapiens (human)IC509.820010
2-(4-methoxyphenyl)-1H-quinazolin-4-oneHomo sapiens (human)IC5017.300010