Page last updated: 2024-08-21

thiazoles and Ache

thiazoles has been researched along with Ache in 165 studies

Research

Studies (165)

TimeframeStudies, this research(%)All Research%
pre-199015 (9.09)18.7374
1990's14 (8.48)18.2507
2000's51 (30.91)29.6817
2010's77 (46.67)24.3611
2020's8 (4.85)2.80

Authors

AuthorsStudies
Chandna, A; Devana, SK; Kumar, S; Mete, UK; Parmar, KM; Sharma, AP; Singh, SK1
Claessens, M; De Coninck, V; Keller, EX; Merckx, L; Pietropaolo, A; Somani, B; Tailly, T; Van Besien, J1
Akhtar, M; Akhtar, S; Haider, S; Saify, ZS; Shamim, S; Siddiqui, R1
Bai, L; Fu, Q; He, Y; Li, M; Liu, B; Liu, Y; Ma, L; Sui, X; Tian, B1
Gardhouse, SM; Hocker, SE; Kleinhenz, MD; Montgomery, SR; Rooney, TA; Sarvi, JY; Weeder, MM1
Arriaga-Gomez, E; Boo, B; Bush, S; Chatterjea, D; Emanuel, E; Kinnamon, R; Kline, J; Lim, J; Mengistu, H; Neamonitaki, N; Pasha, D; Shields-Cutler, R; Wattenberg, E; Yangdon, T; Zacheis, H1
Akhter, S; Ali, M; Haider, S; Mallick, TZ; Saify, ZS; Siddiqui, R1
Borgnia, MJ; He, Q; Hsu, AL; Ji, RR; Lee, SY; Suo, Y; Wang, Z; Zubcevic, L1
Kumar, G; Singh, NP1
Han, J; Huang, M; Luo, L; Ma, X; Shi, H; Su, C; Wang, A; Wang, H; Wang, W; Wu, K; Xu, T; Xu, X; Yuan, T1
Akasaka, R; Furukawa, A; Honda, K; Iwata, K; Kondo, M; Otsuki, K; Shimizu, K; Shinoda, M; Yonemoto, H1
Britti, D; Crupi, R; Cuzzocrea, S; Di Paola, R; Evangelista, M; Fusco, R; Gugliandolo, E; Impellizzeri, D; Morittu, VM; Schievano, C1
Wang, J1
Alves, D; de Oliveira, RL; Luchese, C; Pinz, MP; Reis, AS; Roehrs, JA; Sacramento, MD; Vogt, AG; Voss, GT; Wilhelm, EA1
Bradshaw, C; Flecknell, P; Lee, CCS; Lofgren, J; Miller, AL; Roughan, J1
Gellatly, D; Janzen, ED; Marti, S; Meléndez, DM; Moya, D; Pajor, EA; Schwartzkopf-Genswein, KS1
Hughes, HD; Powell, JG; Richeson, JT; Roberts, SL1
Ciotu, CI; Fischer, MJM; Gold-Binder, M; Heber, S; Kress, HG; Ninidze, N; Witek, M1
Heinonen, M; Larenza-Menzies, P; Oliviero, C; Ollila, A; Peltoniemi, O; Valros, A; Yun, J1
Allen, K; Badino, P; Bergamasco, L; Bertolotti, L; Coetzee, JF; Dockweiler, J; Edwards-Callaway, LN; Fraccaro, E; Glynn, H; Kukanich, B; Odore, R1
Chapinal, N; DeVries, TJ; Duffield, TF; Fitzpatrick, CE; Kelton, DF; Leslie, KE; Petersson-Wolfe, CS1
Duffield, TF; Leblanc, SJ; Leslie, KE; Newby, NC; Pearl, DL; von Keyserlingk, MA1
Abelson, KS; Fauerby, N; Hau, J; Jacobsen, KR; Johansen, FF; Kalliokoski, O; Raida, Z1
Gruet, P; King, JN; Seewald, W1
Ahola, JK; Bigler, BJ; Callan, RJ; Coetzee, JF; Engle, TE; Fox, JT; French, JT; Giles, RL; Peel, RK; Repenning, PE; Whittier, JC; Wulf, LW1
Akkas, G; Altikat, S; Cayci, MK; Deger, A; Inal, S; Kabay, S; Kuru, HI1
Asada, T; Hagiwara, M; Kawamoto, D; Kii, I; Kurihara, T; Miyata, A; Sakurai, E; Tanabe, T; Toyomoto, M; Yoshimura, M1
Aubriot, D; Colditz, IG; Hervault, G; Lee, C; Paull, DR1
Baycu, C; Bektur, E; Burukoglu, D; Sahin, E; Taplamacioglu, F1
Dorsey, K; Gustafson, DL; Hansen, RJ; Kang, S; Kendall, LV; Lunghofer, PJ1
Bauer, C; Frost, P; Kirschner, S1
Belson, S; Colditz, IG; Holm, M; Small, AH1
Bates, AJ; Eder, P; Laven, RA1
Alomrani, A; Badran, M; Shazly, G; Zoheir, K1
Ertan, M; Kazkayasi, I; Okay, G; Ozadali-Sari, K; Sarigol, D; Somuncuoglu, EI; Tel, BC; Tozkoparan, B; Unsal-Tan, O; Uzgoren-Baran, A1
Abell, CA; Coetzee, JF; Johnson, AK; Karriker, LA; Millman, ST; Pairis-Garcia, MD; Stalder, KJ1
Abe, K; Akagi, T; Matoba, M; Mawatari, H; Saito, O; Syuuto, C; Tagami, K; Takeno, N1
Burdick Sanchez, NC; Carroll, JA; Hubbell, DS; Hughes, HD; Powell, JG; Richeson, JT; Roberts, SL1
Babanouri, N; Oshagh, M; Salehi, P; Torkan, S; Zarif Najafi, H1
Altman, R; Gibofsky, A; Hochberg, M; Jaros, M; Young, C1
Dorsch, R; Hartmann, K; Sauter-Louis, C; Schulz, B; Zellner, F1
Brett, TJ; Feng, J; Hu, H; Liu, S; Luo, J; Yang, P1
Mainau, E; Manteca, X; Temple, D1
Mans, C; Martel-Arquette, A; Sladky, K1
Mejia, GL; Pasteris, RJ; Pember, SO; Price, TJ1
Eddicks, M; Numberger, J; Reese, S; Ritzmann, M; Übel, N; Zöls, S1
Chen, Y; Fan, P; Gooden, DM; Guilak, F; Kanju, P; Lee, SH; Lee, W; Liddle, RA; Liedtke, WB; Mook, RA; Romac, J; Shahid, R; Simon, SA; Spasojevic, I; Yeo, M1
Leung, V; Pang, DS; Zhang, E1
Doit, H; Wareham, K1
Betti, M; Borea, PA; Catarzi, D; Colotta, V; Falsini, M; Ravani, A; Varani, K; Varano, F; Vincenzi, F1
Bernardini, D; Contiero, B; De Benedictis, GM; Edwards, SA; Gottardo, F; Ravagnani, A; Scollo, A; Tavella, G1
Asiedu, MN; Dib-Hajj, SD; Dussor, G; Han, C; Price, TJ; Waxman, SG1
Bateman, SW; Dewey, C; Johnson, R; Kerr, C; Reimann, J1
Banse, H; Cribb, AE1
Atkinson, SJ; Fisher, AD; Lee, C; Paull, DR1
Carroll, GL; DeBoer, M; Kerwin, SC; Narbe, R; Peterson, K; Taylor, L1
Elzein, E; Zablocki, J1
Burbach, LR; Dong, L; Ford, AP; Guillon, MA; Hu, Y; Liu, X; Nunn, PA; Rong, W; Sun, B; Vilenski, O; Zhong, Y1
Dowling, SK; Rogers, AR; Schaefer, AL; Stafford, KJ; Stewart, M; Stookey, JM; Tucker, CB; Verkerk, GA; Webster, JR1
Bonnefous, C; Hassig, CA; Lee, TT; Massari, ME; Nguyen, PM; Noble, SA; Payne, JE; Rao, TS; Roppe, J; Rozenkrants, N; Sablad, M; Shiau, AK; Smith, ND; Symons, KT; Zhang, Y1
Horváth, C; Ji, G; Neugebauer, V1
Kimura, S; Kontani, H1
Bennett, D; Morton, C1
Abu-Hashem, AA; Badria, FA; Gouda, MA1
Baraka, MM; El-Sabbagh, OI; Ibrahim, SM; Kothayer, H1
Duffield, TF; Heinrich, A; Lissemore, KD; Millman, ST1
Kang, P; Li, J; Liu, G; Liu, W; Luo, R; Ma, X; Pei, F; Shen, B; Xie, Q; Zhou, Z1
Dolezal, T; Janovský, M; Krsiak, M; Procháizková, M; Slíva, J1
Carroll, WA; Chandran, P; Dart, MJ; Honore, P; Hooker, BA; Hsieh, GC; Meyer, MD; Pai, M; Salyers, AK; Wensink, EJ; Yao, BB; Zhan, C; Zhu, CZ1
Barron, GH; Budsberg, SC; Divers, SJ; Hernandez, SM; Koch, TF; McBride, M; Papich, M; Perpinan, D; Pethel, M; Stedman, NL1
Bondesson, U; Högberg, M; Ingvast-Larsson, C; Mengistu, U; Olsén, L; Olsson, K1
Ji, G; Li, Z; Neugebauer, V1
Grant, D; Johnston, L; Letellier, IM; Morton, CM; Narbe, R1
Hansson, M; Johansson, G; Lundeheim, N; Nyman, G1
Carroll, GL; Hartsfield, SM; Kerwin, SC; Narbe, R; Peterson, K; Taylor, L1
Chi, CS; Deng, JS; Huang, GJ; Huang, SS; Lin, TH; Shie, PH1
Baiuomy, AR; Elmegeed, GA; Eskander, EF; Mohareb, RM; William, MG1
Chen, G; de Groat, WC; Larson, JA; Ogagan, PD; Roppolo, JR; Shen, B; Tai, C; Wang, J1
Backer, RT; Barth, VN; Fisher, MJ; Garbison, KE; Gruber, JM; Heinz, BA; Hollinshead, SP; Iyengar, S; Kingston, A; Kuklish, SL; Li, L; Nisenbaum, ES; Peters, SC; Phebus, L; Simmons, RM; van der Aar, E1
Dalmau, A; Mainau, E; Manteca, X; Ruiz-de-la-Torre, JL; Salleras, JM1
Kang, PD; Li, J; Li, Q; Li, Y; Liu, G; Pei, FX; Shen, B; Tang, X; Zhao, XD; Zhou, ZK1
Colditz, IG; Lee, C; Palladin, P; Paull, DR; Small, AH1
Coetzee, JF; Cull, CA; Edwards, LN; Mosher, RA; Theurer, ME; White, BJ1
Coetzee, JF; Gehring, R; KuKanich, B; Mosher, RA; Reinbold, JB; Robert, B; White, BJ1
König, A; Schmidt, T; von Borell, E1
Hale, LP; Kim, CJ; Kolstad, AM; Rodriguiz, RM1
Schumacher, J; Seibert, R; Steeil, J; Tobias, K1
Flecknell, PA; Miller, AL; Roughan, JV; Wright-Williams, SL1
De Petrocellis, L; Schiano Moriello, A1
Behnke, CA; Igaki, S; Kawamura, T; Kiyota, Y; Kono, M; Kori, M; Matsumoto, T; Miyazaki, J; Nishimura, A; Oki, H; Shimojo, M1
Raghunath, A1
Akintola, M; Messerschmidt, C; Morewitz, J; Spiegel, DR1
Monteiro-Steagall, BP; Steagall, PV1
Atilla, P; Balkan, A; Cakar, AN; Caliş, U; Gören, Z; Urgun, H; Uzbay, T1
Jain, NK; Kulkarni, SK; Singh, A1
Fleischmann, R; Iqbal, I; Slobodin, G1
Huchkowsky, SL1
Ogino, K; Osugi, T; Saito, K; Satoh, H1
Atweh, SF; Bach, JF; Dardenne, M; Jabbur, SJ; Saadé, NE; Safieth-Garabedian, B1
Frendin, J; Viking Höglund, O1
Frye, CA; Walf, AA1
ERVENIUS, O1
HUGIN, W1
GLATZL, A1
Borer, LR; Peel, JE; Schawalder, P; Seewald, W; Spreng, DE1
Ertan, M; Gökhan, N; Küpeli, E; Tozkoparan, B; Yeşilada, E1
Davies, BR; Flecknell, PA; Roughan, JV1
Erol, K; Ito, S; Onkol, T; Sahin, MF; Yildirim, E1
Decker, MW; Gauvin, DM; Honore, P; Lynch, JJ; Mikusa, JP; Wade, CL; Wilson, SG; Wismer, CT; Zhu, CZ1
Castañeda-Hernández, G; Granados-Soto, V; Ortiz, MI1
Holman, AJ; Myers, RR1
Hanaoka, K; Sawamura, S; Sekiyama, H; Takeda, K; Tamai, H1
Hough, LB; Lu, Q; Montero, MJ; Nalwalk, JW; Shan, Z; Svokos, K; Wentland, MP1
Al'-Zamil', MKh1
Egger, CM; Gassel, AD; Rohrbach, BW; Tobias, KM1
Danysz, W; Sevostianova, N1
Büchler, MW; Ceyhan, GO; Erkan, M; Friess, H; Giese, NA; Giese, T; Kerscher, AG; Wente, MN1
Faden, AI; Lea, PM1
Clark, TP1
Calandre, EP; Hidalgo, J; Rico-Villademoros, F1
Hilário, MO; Len, CA; Terreri, MT1
Black, SR; Finn-Bodner, ST; Remedios, AM; Whiteside, DP1
Itahana, H; Kiso, T; Kohara, A; Nagakura, Y; Okada, M; Shitaka, Y; Tamura, S; Toya, T; Watabiki, T1
Arunadevi, R; Dudhgaonkar, SP; Kumar, D; Prakash, VR; Tandan, SK1
Barke, KE; Bodnar, RJ; Hough, LB; Koch, JE; Nalwalk, JW1
Hough, LB; Nalwalk, JW1
Fenech, G; Forestieri, AM; Giordano, A; Monforte, MT; Previtera, T; Vigorita, MG; Zappala, C1
Engelhardt, G; Homma, D; Schlegel, K; Schnitzler, C; Utzmann, R1
O'Neill, WM1
Ambrogi, V; Arenare, L; De Caprariis, P; Falcone, G; Filippelli, W; Grandolini, G; Palagiano, F; Perioli, L; Rossi, F1
Baumgartner, H; Björneboe, O; Bluhmki, E; Bolten, W; Burgos-Vargas, R; Distel, M; Franchimont, P; Hanft, G; Lemmel, EM; Nissilä, M; Platt, P; Sahlberg, D; Valat, JP1
Fox, SM; Johnston, SA1
Bosch, HC; Hettich, M; Sigmund, R1
Laird, JM; Lopez-Garcia, JA1
De Freitas, GA; Santos, AR; Vedana, EM1
Aguirre-Bañuelos, P; Granados-Soto, V1
Atweh, SF; Dardenne, M; Jabbur, SJ; Kanaan, SA; Saadé, NE; Safieh-Garabedian, B1
Frölich, JC; Stichtenoth, DO1
Chang, DM; Hsieh, TC; Hsu, CT; Kuo, SY; Young, TH1
Henry, JL; Pitcher, GM1
Bondavalli, F; Bruno, O; Falcone, G; Filippelli, W; Giordano, L; Ranise, A; Schenone, S; Vitelli, MR1
Cakir, B; Erol, K; Gökce, M; Sahin, MF1
Carter, AJ; Cervero, F; Grauert, M; Laird, JM1
Hackett, IJ; Henderson, AJ; Lascelles, BD1
Karczmarzyk, Z; Kleinrok, Z; Malinka, W; Sadowski, M; Sieklucka-Dziuba, M1
Miranda, HF; Pinardi, G; Sierralta, F1
Bergman, J; Hoeijmakers, M; Horspool, LJ; Nell, T; Van Laar, P1
Amoretti, L; Ballabeni, V; Barocelli, E; Incerti, M; Tognolini, M; Vicini, P1
Hui, KS1
Barocelli, E; Bordi, F; Chiavarini, M; Impicciatore, M; Mor, M; Morini, G; Plazzi, PV; Silva, C1
Cai, ZJ; Li, M; Liu, LN; Liu, YH; Zhang, JL; Zheng, JW1
Battles, AH; Hough, LB; Nalwalk, JW1
Reynolds, JC1
Miwa, T1
Barbara, L; Bianchi Porro, G; Blasi, A; Bovero, E; Carratelli, L; Cheli, R; Corinaldesi, R; Lazzaroni, M; Mangiameli, A; Wilkins, A1
Barbara, L; Bianchi Porro, G; Blasi, A; Carratelli, L; Cheli, R; Corinaldesi, R; Lazzaroni, M; Mangiameli, A; Paoluzi, P; Torsoli, A1
Hatcher, C; Levendoglu, H; Mehta, B; Reddy, G; Wait, C1
Bianchi Porro, G; Cook, T; Dicenta, C; Humphries, TJ1
Boero, A; Camarri, E; Crespi, M; De Pretis, G; Dobrilla, G; Fontana, G; Ideo, G; Manenti, F; Marenco, G; Piazzi, L1
Fölsch, UR; Hartmann, H1
Dammann, HG; Hentschel, E; Müller, P; Simon, B; Walter, TA1
Márquez, M; Roberts, DJ1
Fennessy, MR1

Reviews

11 review(s) available for thiazoles and Ache

ArticleYear
Mirabegron for the Treatment of Ureteral Stent-related Symptoms: A Systematic Review and Meta-analysis.
    European urology focus, 2022, Volume: 8, Issue:4

    Topics: Acetanilides; Adult; Humans; Male; Pain; Quality of Life; Thiazoles; Ureter

2022
Low-dose meloxicam (Vivlodex) for osteoarthritis pain.
    The Medical letter on drugs and therapeutics, 2016, Mar-14, Volume: 58, Issue:1490

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Chemistry, Pharmaceutical; Drug Interactions; Female; Humans; Male; Meloxicam; Osteoarthritis; Pain; Randomized Controlled Trials as Topic; Thiazines; Thiazoles

2016
Can you reduce the dose of meloxicam in dogs with osteoarthritis?
    The Veterinary record, 2016, Dec-10, Volume: 179, Issue:23

    Topics: Animals; Dog Diseases; Dogs; Dose-Response Relationship, Drug; Meloxicam; Osteoarthritis; Pain; Randomized Controlled Trials as Topic; Thiazines; Thiazoles

2016
A1 adenosine receptor agonists and their potential therapeutic applications.
    Expert opinion on investigational drugs, 2008, Volume: 17, Issue:12

    Topics: Adenosine A1 Receptor Agonists; Aminopyridines; Angina Pectoris; Animals; Anti-Arrhythmia Agents; Humans; Insulin; Pain; Receptor, Adenosine A1; Thiazoles

2008
Meloxicam.
    Expert opinion on pharmacotherapy, 2002, Volume: 3, Issue:10

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Rheumatoid; Drug Interactions; Humans; Meloxicam; Osteoarthritis; Pain; Product Surveillance, Postmarketing; Spondylitis, Ankylosing; Thiazines; Thiazoles

2002
[Meloxicam (Mobic): a review of its pharmacological and clinical profile].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 2002, Volume: 120, Issue:6

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Experimental; Arthritis, Rheumatoid; Clinical Trials as Topic; Cyclooxygenase 2; Enzyme Inhibitors; Gastric Mucosa; Gastrointestinal Hemorrhage; Humans; Inflammation; Isoenzymes; Meloxicam; Membrane Proteins; Pain; Platelet Aggregation; Prostaglandin-Endoperoxide Synthases; Rats; Thiazines; Thiazoles

2002
Metabotropic glutamate receptor subtype 5 antagonists MPEP and MTEP.
    CNS drug reviews, 2006,Summer, Volume: 12, Issue:2

    Topics: Animals; Humans; Neurodegenerative Diseases; Pain; Pyridines; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Substance-Related Disorders; Thiazoles

2006
The clinical pharmacology of cyclooxygenase-2-selective and dual inhibitors.
    The Veterinary clinics of North America. Small animal practice, 2006, Volume: 36, Issue:5

    Topics: 4-Butyrolactone; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carbazoles; Cats; Cyclooxygenase 2 Inhibitors; Dogs; Etodolac; Meloxicam; Pain; Pain Measurement; Pyrazoles; Sulfones; Thiazines; Thiazoles

2006
Nonsteroidal anti-inflammatory drugs: cyclooxygenase 2 inhibitors.
    Jornal de pediatria, 2006, Volume: 82, Issue:5 Suppl

    Topics: Adolescent; Aspirin; Celecoxib; Child; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Drug Interactions; Etoricoxib; Fever; Humans; Hypersensitivity, Immediate; Inflammation; Leukotrienes; Meloxicam; Naproxen; Pain; Prostaglandins; Pyrazoles; Pyridines; Sulfonamides; Sulfones; Thiazines; Thiazoles; Treatment Outcome

2006
Use of carprofen for the treatment of pain and inflammation in dogs.
    Journal of the American Veterinary Medical Association, 1997, May-15, Volume: 210, Issue:10

    Topics: Acetaminophen; Analgesics, Non-Narcotic; Animals; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Carbazoles; Clonixin; Cyclooxygenase Inhibitors; Dog Diseases; Dogs; Ibuprofen; Indomethacin; Ketoprofen; Meclofenamic Acid; Meloxicam; Naproxen; Osteoarthritis; Pain; Phenylbutazone; Piroxicam; Thiazines; Thiazoles

1997
[Therapy with preferential and specific COX-2 inhibitors].
    Der Internist, 2001, Volume: 42, Issue:3

    Topics: Analgesics, Non-Narcotic; Anti-Inflammatory Agents, Non-Steroidal; Celecoxib; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Humans; Isoenzymes; Lactones; Meloxicam; Membrane Proteins; Pain; Prostaglandin-Endoperoxide Synthases; Pyrazoles; Randomized Controlled Trials as Topic; Sulfonamides; Sulfones; Thiazines; Thiazoles

2001

Trials

45 trial(s) available for thiazoles and Ache

ArticleYear
Comparison of stent related symptoms in patients taking mirabegron, solifenacin, or tamsulosin: A double blinded randomized clinical trial.
    Urologia, 2022, Volume: 89, Issue:4

    Topics: Acetanilides; Humans; Pain; Prospective Studies; Quality of Life; Solifenacin Succinate; Stents; Tamsulosin; Thiazoles; Treatment Outcome; Urological Agents

2022
Efficacy and safety of adalimumab by intra-articular injection for moderate to severe knee osteoarthritis: An open-label randomized controlled trial.
    The Journal of international medical research, 2018, Volume: 46, Issue:1

    Topics: Adalimumab; Aged; Antirheumatic Agents; Celecoxib; Diclofenac; Female; Humans; Hyaluronic Acid; Ibuprofen; Injections, Intra-Articular; Male; Meloxicam; Middle Aged; Osteoarthritis, Knee; Pain; Pain Measurement; Patient Safety; Pilot Projects; Severity of Illness Index; Thiazines; Thiazoles; Treatment Outcome

2018
A Human TRPA1-Specific Pain Model.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2019, 05-15, Volume: 39, Issue:20

    Topics: Acetamides; Adult; Cross-Over Studies; Dose-Response Relationship, Drug; Double-Blind Method; Female; Humans; Male; Models, Neurological; Oximes; Pain; Pain Measurement; Pain Perception; Psychophysics; Thiazoles; TRPA1 Cation Channel; Young Adult

2019
Behavioural alterations in piglets after surgical castration: Effects of analgesia and anaesthesia.
    Research in veterinary science, 2019, Volume: 125

    Topics: Analgesia; Anesthesia; Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Lidocaine; Male; Meloxicam; Orchiectomy; Pain; Pain Management; Pain Measurement; Swine; Thiazines; Thiazoles

2019
Effects of meloxicam on milk production, behavior, and feed intake in dairy cows following assisted calving.
    Journal of dairy science, 2013, Volume: 96, Issue:6

    Topics: 3-Hydroxybutyric Acid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Body Weight; Cattle; Cattle Diseases; Dystocia; Eating; Fatty Acids, Nonesterified; Feeding Behavior; Female; Lactation; Meloxicam; Milk; Pain; Parturition; Placebos; Pregnancy; Thiazines; Thiazoles

2013
Effects of buprenorphine and meloxicam analgesia on induced cerebral ischemia in C57BL/6 male mice.
    Comparative medicine, 2013, Volume: 63, Issue:2

    Topics: Analgesics; Animals; Brain Ischemia; Buprenorphine; Corticosterone; Infarction, Middle Cerebral Artery; Male; Meloxicam; Mice; Mice, Inbred C57BL; Pain; Pain Management; Research Design; Thiazines; Thiazoles

2013
Robenacoxib versus meloxicam for the management of pain and inflammation associated with soft tissue surgery in dogs: a randomized, non-inferiority clinical trial.
    BMC veterinary research, 2013, May-02, Volume: 9

    Topics: Animals; Cyclooxygenase 2 Inhibitors; Diphenylamine; Dogs; Double-Blind Method; Female; Hydrocortisone; Inflammation; Male; Meloxicam; Pain; Pain Measurement; Phenylacetates; Prospective Studies; Statistics, Nonparametric; Thiazines; Thiazoles

2013
Impact of oral meloxicam administration before and after band castration on feedlot performance and behavioral response in weanling beef bulls.
    Journal of animal science, 2013, Volume: 91, Issue:10

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Cattle; Cattle Diseases; Housing, Animal; Male; Meloxicam; Orchiectomy; Pain; Thiazines; Thiazoles; Time Factors; Weaning

2013
Efficacy of a buccal meloxicam formulation for pain relief in Merino lambs undergoing knife castration and tail docking in a randomised field trial.
    Australian veterinary journal, 2014, Volume: 92, Issue:10

    Topics: Administration, Buccal; Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Body Weight; Cohort Studies; Female; Male; Meloxicam; Orchiectomy; Pain; Sheep; Single-Blind Method; Statistics, Nonparametric; Thiazines; Thiazoles; Wound Healing

2014
Effect of analgesia and anti-inflammatory treatment on weight gain and milk intake of dairy calves after disbudding.
    New Zealand veterinary journal, 2015, Volume: 63, Issue:3

    Topics: Analgesia; Anesthetics, Local; Animal Husbandry; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cattle; Eating; Horns; Hypnotics and Sedatives; Lidocaine; Meloxicam; Pain; Thiazines; Thiazoles; Weight Gain; Xylazine

2015
Measuring the efficacy of flunixin meglumine and meloxicam for lame sows using a GAITFour pressure mat and an embedded microcomputer-based force plate system.
    Journal of animal science, 2015, Volume: 93, Issue:5

    Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Biomechanical Phenomena; Clonixin; Female; Foot; Gait; Lameness, Animal; Meloxicam; Microcomputers; Pain; Pregnancy; Pressure; Swine; Swine Diseases; Thiazines; Thiazoles; Weight-Bearing

2015
Effect of surgical castration with or without oral meloxicam on the acute inflammatory response in yearling beef bulls.
    Journal of animal science, 2015, Volume: 93, Issue:8

    Topics: Administration, Oral; Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cattle; Haptoglobins; Hydrocortisone; Inflammation; Male; Meloxicam; Orchiectomy; Pain; Pain, Postoperative; Thiazines; Thiazoles

2015
Comparison of the effects of preemptive acetaminophen, ibuprofen, and meloxicam on pain after separator placement: a randomized clinical trial.
    Progress in orthodontics, 2015, Volume: 16

    Topics: Acetaminophen; Adolescent; Adult; Analgesics, Non-Narcotic; Anti-Inflammatory Agents, Non-Steroidal; Cyclooxygenase Inhibitors; Dental Occlusion; Double-Blind Method; Female; Follow-Up Studies; Humans; Ibuprofen; Male; Mastication; Meloxicam; Orthodontic Appliances; Pain; Pain Measurement; Pain Perception; Premedication; Prospective Studies; Thiazines; Thiazoles; Young Adult

2015
Efficacy and safety of low-dose SoluMatrix meloxicam in the treatment of osteoarthritis pain: a 12-week, phase 3 study.
    Current medical research and opinion, 2015, Volume: 31, Issue:12

    Topics: Acetaminophen; Adult; Aged; Aged, 80 and over; Anti-Inflammatory Agents, Non-Steroidal; Double-Blind Method; Female; Humans; Male; Meloxicam; Middle Aged; Osteoarthritis, Hip; Osteoarthritis, Knee; Pain; Pain Measurement; Thiazines; Thiazoles; Treatment Outcome

2015
Evaluation of meloxicam for the treatment of obstructive feline idiopathic cystitis.
    Journal of feline medicine and surgery, 2016, Volume: 18, Issue:11

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cat Diseases; Cats; Cystitis; Double-Blind Method; Drug Administration Schedule; Female; Humans; Male; Meloxicam; Ownership; Pain; Pain Measurement; Surveys and Questionnaires; Thiazines; Thiazoles; Treatment Outcome; Urethral Obstruction

2016
Experimental study on the effect of oral meloxicam administration in sows on pre-weaning mortality and growth and immunoglobulin G transfer to piglets.
    Preventive veterinary medicine, 2016, Apr-01, Volume: 126

    Topics: Animals; Animals, Newborn; Anti-Inflammatory Agents, Non-Steroidal; Female; Immunity, Maternally-Acquired; Immunoglobulin G; Male; Meloxicam; Pain; Parturition; Pregnancy; Survival Rate; Swine; Thiazines; Thiazoles; Weaning

2016
Ear tagging in piglets: the cortisol response with and without analgesia in comparison with castration and tail docking.
    Animal : an international journal of animal bioscience, 2016, Volume: 10, Issue:11

    Topics: Analgesia; Animal Husbandry; Animal Identification Systems; Animals; Ear; Hydrocortisone; Male; Meloxicam; Orchiectomy; Pain; Stress, Psychological; Swine; Tail; Thiazines; Thiazoles; Time Factors

2016
Efficacy of celecoxib, meloxicam and paracetamol in elderly Kashin-Beck disease (KBD) patients.
    International orthopaedics, 2011, Volume: 35, Issue:9

    Topics: Acetaminophen; Adolescent; Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Celecoxib; Female; Health Status; Humans; Joints; Kashin-Beck Disease; Male; Meloxicam; Middle Aged; Pain; Pain Measurement; Pyrazoles; Sulfonamides; Thiazines; Thiazoles; Treatment Outcome; Young Adult

2011
Pharmacokinetics of meloxicam in adult goats and its analgesic effect in disbudded kids.
    Journal of veterinary pharmacology and therapeutics, 2011, Volume: 34, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Area Under Curve; Blood Glucose; Goat Diseases; Goats; Half-Life; Hydrocortisone; Meloxicam; Pain; Surgical Procedures, Operative; Thiazines; Thiazoles

2011
Clinical evaluation of meloxicam versus ketoprofen in cats suffering from painful acute locomotor disorders.
    Journal of feline medicine and surgery, 2011, Volume: 13, Issue:4

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cat Diseases; Cats; Female; Ketoprofen; Lameness, Animal; Male; Meloxicam; Pain; Pain Measurement; Taste; Thiazines; Thiazoles; Treatment Outcome

2011
Dose range finding study for the efficacy of meloxicam administered prior to sodium urate-induced synovitis in cats.
    Veterinary anaesthesia and analgesia, 2011, Volume: 38, Issue:4

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cats; Cross-Over Studies; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Male; Meloxicam; Pain; Pain Measurement; Single-Blind Method; Synovitis; Thiazines; Thiazoles; Treatment Outcome; Uric Acid

2011
Effects of meloxicam (Metacam®) on post-farrowing sow behaviour and piglet performance.
    Animal : an international journal of animal bioscience, 2012, Volume: 6, Issue:3

    Topics: Animal Husbandry; Animal Welfare; Animals; Anti-Inflammatory Agents, Non-Steroidal; Female; Inflammation; Meloxicam; Motor Activity; Pain; Parity; Parturition; Swine; Swine Diseases; Thiazines; Thiazoles

2012
A randomized, single-blind comparison of the efficacy and tolerability of hyaluronate acid and meloxicam in adult patients with Kashin-Beck disease of the knee.
    Clinical rheumatology, 2012, Volume: 31, Issue:7

    Topics: Administration, Oral; Adolescent; Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Female; Humans; Hyaluronic Acid; Injections, Intra-Articular; Kashin-Beck Disease; Knee Joint; Male; Meloxicam; Middle Aged; Pain; Pain Measurement; Single-Blind Method; Thiazines; Thiazoles; Treatment Outcome; Viscosupplements

2012
Evaluating a novel analgesic strategy for ring castration of ram lambs.
    Veterinary anaesthesia and analgesia, 2012, Volume: 39, Issue:5

    Topics: Analgesics; Animals; Behavior, Animal; Body Temperature; Clonixin; Drug Administration Schedule; Hydrocortisone; Male; Meloxicam; Orchiectomy; Pain; Sheep; Sheep Diseases; Thiazines; Thiazoles; Weight Gain

2012
Assessment of behavioral changes associated with oral meloxicam administration at time of dehorning in calves using a remote triangulation device and accelerometers.
    BMC veterinary research, 2012, Apr-30, Volume: 8

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Cattle; Horns; Male; Meloxicam; Pain; Remote Sensing Technology; Thiazines; Thiazoles

2012
Pharmacokinetics and effect of intravenous meloxicam in weaned Holstein calves following scoop dehorning without local anesthesia.
    BMC veterinary research, 2012, Sep-01, Volume: 8

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cattle; Cattle Diseases; Heart Rate; Horns; Hydrocortisone; Meloxicam; Pain; Substance P; Thiazines; Thiazoles; Weight Gain

2012
A comparison of abdominal and scrotal approach methods of vasectomy and the influence of analgesic treatment in laboratory mice.
    Laboratory animals, 2012, Volume: 46, Issue:4

    Topics: Abdomen; Acetaminophen; Analgesics, Non-Narcotic; Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Drug Combinations; Image Processing, Computer-Assisted; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Meloxicam; Mice; Pain; Pain Measurement; Pilot Projects; Scrotum; Surgery, Veterinary; Thiazines; Thiazoles; Time Factors; Vasectomy; Videotape Recording

2012
Analgesic effect of meloxicam in canine acute dermatitis--a pilot study.
    Acta veterinaria Scandinavica, 2002, Volume: 43, Issue:4

    Topics: Acute Disease; Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cephalexin; Dermatitis; Dog Diseases; Dogs; Double-Blind Method; Meloxicam; Pain; Pain Measurement; Pilot Projects; Severity of Illness Index; Thiazines; Thiazoles; Treatment Outcome

2002
A randomized, double-blind, placebo-controlled trial of pramipexole, a dopamine agonist, in patients with fibromyalgia receiving concomitant medications.
    Arthritis and rheumatism, 2005, Volume: 52, Issue:8

    Topics: Adult; Analgesics, Opioid; Benzothiazoles; Disabled Persons; Dopamine Agonists; Double-Blind Method; Drug Therapy, Combination; Fatigue; Female; Fibromyalgia; Humans; Male; Middle Aged; Pain; Pramipexole; Thiazoles; Treatment Outcome

2005
Use of ziprasidone in patients with fibromyalgia: a case series.
    Rheumatology international, 2007, Volume: 27, Issue:5

    Topics: Adult; Aged; Antipsychotic Agents; Female; Fibromyalgia; Humans; Male; Middle Aged; Pain; Piperazines; Severity of Illness Index; Thiazoles; Treatment Outcome

2007
The cognitive and psychomotor effects of opioid drugs in cancer pain management.
    Cancer surveys, 1994, Volume: 21

    Topics: Adult; Amphetamines; Analgesics, Opioid; Buprenorphine; Central Nervous System Stimulants; Chronic Disease; Cocaine; Codeine; Cognition; Dextropropoxyphene; Dopamine Uptake Inhibitors; Humans; Methylphenidate; Morphine; Neoplasms; Pain; Psychomotor Performance; Randomized Controlled Trials as Topic; Reaction Time; Thiazoles

1994
Efficacy and safety of meloxicam in patients with rheumatoid arthritis.
    The Journal of rheumatology, 1997, Volume: 24, Issue:2

    Topics: Aged; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Rheumatoid; Demography; Double-Blind Method; Female; Humans; Joints; Male; Meloxicam; Middle Aged; Pain; Safety; Thiazines; Thiazoles; Treatment Outcome

1997
Efficacy and tolerability of intramuscular and oral meloxicam in patients with acute lumbago: a comparison with intramuscular and oral piroxicam.
    Current medical research and opinion, 1997, Volume: 14, Issue:1

    Topics: Activities of Daily Living; Acute Disease; Administration, Oral; Adult; Anti-Inflammatory Agents, Non-Steroidal; Chi-Square Distribution; Drug Administration Schedule; Female; Humans; Injections, Intramuscular; Low Back Pain; Male; Meloxicam; Middle Aged; Movement; Pain; Pain Measurement; Piroxicam; Thiazines; Thiazoles

1997
Endoscopic comparison of the gastroduodenal safety and the effects on arachidonic acid products between meloxicam and piroxicam in the treatment of osteoarthritis.
    Clinical rheumatology, 2001, Volume: 20, Issue:2

    Topics: Adult; Aged; Arachidonic Acid; Cyclooxygenase Inhibitors; Digestive System; Dinoprostone; Double-Blind Method; Endoscopy, Digestive System; Female; Gastric Juice; Humans; Leukotriene B4; Male; Meloxicam; Middle Aged; Osteoarthritis, Knee; Pain; Pain Measurement; Piroxicam; Safety; Thiazines; Thiazoles; Thromboxane B2

2001
Evaluation of the clinical efficacy of meloxicam in cats with painful locomotor disorders.
    The Journal of small animal practice, 2001, Volume: 42, Issue:12

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cat Diseases; Cats; Female; Ketoprofen; Lameness, Animal; Male; Meloxicam; Pain; Pain Measurement; Thiazines; Thiazoles; Treatment Outcome

2001
Comparison of vedaprofen and meloxicam in dogs with musculoskeletal pain and inflammation.
    The Journal of small animal practice, 2002, Volume: 43, Issue:5

    Topics: Acute Disease; Animals; Anti-Inflammatory Agents, Non-Steroidal; Chronic Disease; Dog Diseases; Dogs; Female; Inflammation; Male; Meloxicam; Musculoskeletal Diseases; Naphthalenes; Pain; Propionates; Thiazines; Thiazoles; Treatment Outcome

2002
Famotidine therapy for active duodenal ulcers. A multivariate analysis of factors affecting early healing.
    Annals of internal medicine, 1989, Jul-01, Volume: 111, Issue:1

    Topics: Adult; Aged; Aged, 80 and over; Alcohol Drinking; Anti-Inflammatory Agents, Non-Steroidal; Duodenal Ulcer; Duodenoscopy; Factor Analysis, Statistical; Famotidine; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Multicenter Studies as Topic; Pain; Prospective Studies; Recurrence; Risk Factors; Thiazoles; Time Factors

1989
Clinical evaluation of 20 mg/day famotidine in the treatment of acute gastric mucosal lesions.
    The Journal of international medical research, 1989, Volume: 17 Suppl 1

    Topics: Adult; Aged; Anti-Ulcer Agents; Clinical Trials as Topic; Dose-Response Relationship, Drug; Famotidine; Gastric Mucosa; Humans; Middle Aged; Pain; Random Allocation; Stomach Ulcer; Thiazoles

1989
Famotidine in the management of duodenal ulcer: experience in Italy.
    Digestion, 1985, Volume: 32 Suppl 1

    Topics: Adult; Circadian Rhythm; Clinical Trials as Topic; Double-Blind Method; Duodenal Ulcer; Famotidine; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Pain; Random Allocation; Thiazoles

1985
Famotidine (MK-208) in the treatment of gastric ulcer. Results of a multicenter double-blind controlled study.
    Digestion, 1985, Volume: 32 Suppl 1

    Topics: Adolescent; Adult; Aged; Antacids; Circadian Rhythm; Clinical Trials as Topic; Double-Blind Method; Endoscopy; Famotidine; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Pain; Random Allocation; Stomach Ulcer; Thiazoles

1985
Nizatidine: a new histamine receptor blocker in the treatment of active duodenal ulcers.
    The American journal of gastroenterology, 1986, Volume: 81, Issue:12

    Topics: Clinical Trials as Topic; Double-Blind Method; Duodenal Ulcer; Histamine H2 Antagonists; Humans; Nizatidine; Pain; Placebos; Random Allocation; Thiazoles; Time Factors

1986
Review of an extensive worldwide study of a new H2-receptor antagonist, famotidine, as compared to ranitidine in the treatment of acute duodenal ulcer.
    Journal of clinical gastroenterology, 1987, Volume: 9 Suppl 2

    Topics: Acute Disease; Adult; Antacids; Duodenal Ulcer; Famotidine; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Pain; Ranitidine; Thiazoles

1987
Comparison of once-daily bedtime administration of famotidine and ranitidine in the short-term treatment of duodenal ulcer. A multicenter, double-blind, controlled study.
    Scandinavian journal of gastroenterology. Supplement, 1987, Volume: 134

    Topics: Adolescent; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Duodenal Ulcer; Duodenoscopy; Famotidine; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Pain; Random Allocation; Ranitidine; Thiazoles

1987
Famotidine versus cimetidine in the treatment of acute duodenal ulcer. Double-blind, randomized clinical trial comparing nocturnal administration of 40 mg famotidine to 800 mg cimetidine.
    Digestion, 1988, Volume: 39, Issue:3

    Topics: Acute Disease; Adult; Aged; Anti-Ulcer Agents; Cimetidine; Clinical Trials as Topic; Double-Blind Method; Duodenal Ulcer; Famotidine; Female; Humans; Male; Middle Aged; Pain; Random Allocation; Thiazoles

1988
Famotidine: nocturnal administration for gastric ulcer healing. Results of multicenter trials in Austria and Germany.
    Digestion, 1985, Volume: 32 Suppl 1

    Topics: Adolescent; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Endoscopy; Famotidine; Female; Humans; Male; Middle Aged; Pain; Random Allocation; Stomach Ulcer; Thiazoles; Time Factors

1985

Other Studies

109 other study(ies) available for thiazoles and Ache

ArticleYear
New series of hydrazinyl thiazole derivatives of piperidin-4-one: Synthesis, structural elucidation, analgesic activity and comparative structure activity relationship.
    Pakistan journal of pharmaceutical sciences, 2021, Volume: 34, Issue:4

    Topics: Analgesics; Animals; Molecular Structure; Pain; Piperidines; Structure-Activity Relationship; Thiazoles

2021
Preclinical studies of a high drug-loaded meloxicam nanocrystals injection for analgesia.
    Colloids and surfaces. B, Biointerfaces, 2022, Volume: 218

    Topics: Acetates; Analgesia; Animals; Anti-Inflammatory Agents, Non-Steroidal; Meloxicam; Nanoparticles; Pain; Pain Management; Rats; Thiazines; Thiazoles; Water

2022
Measurement of Cyclooxygenase Products in Plasma as Markers for Inhibition of Cyclooxygenase Isoforms by Oral Meloxicam in New Zealand White Rabbits (
    Journal of the American Association for Laboratory Animal Science : JAALAS, 2023, 05-01, Volume: 62, Issue:3

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cat Diseases; Cats; Cyclooxygenase 2; Dinoprostone; Dog Diseases; Dogs; Meloxicam; Pain; Protein Isoforms; Rabbits; Thiazines; Thiazoles

2023
Repeated Vaginal Exposures to the Common Cosmetic and Household Preservative Methylisothiazolinone Induce Persistent, Mast Cell-Dependent Genital Pain in ND4 Mice.
    International journal of molecular sciences, 2019, Oct-28, Volume: 20, Issue:21

    Topics: Allergens; Animals; Cosmetics; Dermatitis, Allergic Contact; Dronabinol; Female; Humans; Immunoglobulin E; Mast Cells; Mice; Mucous Membrane; Pain; Preservatives, Pharmaceutical; Skin; Thiazoles; Vagina

2019
Synthesis, characterization and analgesic studies of novel thiazole derivatives of 4-piperidone.
    Pakistan journal of pharmaceutical sciences, 2019, Volume: 32, Issue:5

    Topics: Analgesics; Animals; Female; Male; Mice; Pain; Piperidones; Structure-Activity Relationship; Thiazoles

2019
Structural Insights into Electrophile Irritant Sensing by the Human TRPA1 Channel.
    Neuron, 2020, 03-04, Volume: 105, Issue:5

    Topics: Acetamides; Cryoelectron Microscopy; Cysteine; HEK293 Cells; Humans; Irritants; Isothiocyanates; Models, Molecular; Nociceptors; Pain; Patch-Clamp Techniques; Phospholipids; Protein Domains; Protein Structure, Tertiary; Pruritus; Thiazoles; TRPA1 Cation Channel

2020
Synthesis, anti-inflammatory and analgesic evaluation of thiazole/oxazole substituted benzothiazole derivatives.
    Bioorganic chemistry, 2021, Volume: 107

    Topics: Analgesics; Animals; Anti-Inflammatory Agents; Antioxidants; Benzothiazoles; Edema; Mice; Molecular Conformation; Oxazoles; Pain; Rats; Structure-Activity Relationship; Thiazoles

2021
mGluR5-Mediated eCB Signaling in the Nucleus Accumbens Controls Vulnerability to Depressive-Like Behaviors and Pain After Chronic Social Defeat Stress.
    Molecular neurobiology, 2021, Volume: 58, Issue:10

    Topics: Animals; Cannabinoid Receptor Antagonists; Chronic Disease; Depressive Disorder, Major; Endocannabinoids; Male; Mice; Mice, Inbred C57BL; Microinjections; Nucleus Accumbens; Pain; Piperidines; Pyrazoles; Pyridines; Receptor, Metabotropic Glutamate 5; Signal Transduction; Social Defeat; Stress, Psychological; Thiazoles

2021
Sensitization of TRPV1 and TRPA1 via peripheral mGluR5 signaling contributes to thermal and mechanical hypersensitivity.
    Pain, 2017, Volume: 158, Issue:9

    Topics: Acetanilides; Animals; Disease Models, Animal; Enzyme Inhibitors; Freund's Adjuvant; Glutamic Acid; Glycine; Hyperalgesia; Male; Neurons; Pain; Pain Threshold; Phenylacetates; Physical Stimulation; Purines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Signal Transduction; Skin; Thiazoles; Trigeminal Ganglion; TRPA1 Cation Channel; TRPV Cation Channels

2017
A novel composite formulation of palmitoylethanolamide and quercetin decreases inflammation and relieves pain in inflammatory and osteoarthritic pain models.
    BMC veterinary research, 2017, Aug-02, Volume: 13, Issue:1

    Topics: Administration, Oral; Amides; Animals; Anti-Inflammatory Agents; Carrageenan; Drug Combinations; Edema; Ethanolamines; Hyperalgesia; Inflammation; Male; Meloxicam; Osteoarthritis; Pain; Palmitic Acids; Quercetin; Rats, Sprague-Dawley; Thiazines; Thiazoles

2017
7-Chloro-4-phenylsulfonyl quinoline, a new antinociceptive and anti-inflammatory molecule: Structural improvement of a quinoline derivate with pharmacological activity.
    Regulatory toxicology and pharmacology : RTP, 2017, Volume: 90

    Topics: Acetic Acid; Analgesics; Animals; Anti-Inflammatory Agents; Croton Oil; Edema; Hot Temperature; Humans; Male; Meloxicam; Mice; Nociception; Pain; Quinolines; Stomach Ulcer; Thiazines; Thiazoles

2017
Analgesics promote welfare and sustain tumour growth in orthotopic 4T1 and B16 mouse cancer models.
    Laboratory animals, 2018, Volume: 52, Issue:4

    Topics: Analgesics; Animal Welfare; Animals; Breast Neoplasms; Buprenorphine; Cell Line, Tumor; Disease Models, Animal; Female; Lung Neoplasms; Mammary Neoplasms, Experimental; Melanoma, Experimental; Meloxicam; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Neoplasm Metastasis; Pain; Thiazines; Thiazoles; Xenograft Model Antitumor Assays

2018
Effect of timing of subcutaneous meloxicam administration on indicators of pain after knife castration of weaned calves.
    Journal of animal science, 2017, Volume: 95, Issue:12

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Canada; Cattle; Female; Haptoglobins; Hydrocortisone; Inflammation; Injections; Male; Meloxicam; Orchiectomy; Pain; Random Allocation; Substance P; Thiazines; Thiazoles; Weaning

2017
Effect of castration method and analgesia on inflammation, behavior, growth performance, and carcass traits in feedlot cattle.
    Journal of animal science, 2018, Feb-15, Volume: 96, Issue:1

    Topics: Analgesia; Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Cattle; Haptoglobins; Inflammation; Male; Meloxicam; Orchiectomy; Pain; Pain Management; Random Allocation; Thiazines; Thiazoles

2018
A study to compare circulating flunixin, meloxicam and gabapentin concentrations with prostaglandin E₂ levels in calves undergoing dehorning.
    Research in veterinary science, 2013, Volume: 95, Issue:1

    Topics: Amines; Analgesics; Animals; Area Under Curve; Cattle; Clonixin; Cyclohexanecarboxylic Acids; Dinoprostone; Gabapentin; gamma-Aminobutyric Acid; Half-Life; Horns; Male; Meloxicam; Pain; Random Allocation; Statistics, Nonparametric; Thiazines; Thiazoles

2013
The effect of meloxicam on pain sensitivity, rumination time, and clinical signs in dairy cows with endotoxin-induced clinical mastitis.
    Journal of dairy science, 2013, Volume: 96, Issue:5

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cattle; Digestion; Female; Lipopolysaccharides; Mastitis, Bovine; Meloxicam; Pain; Pain Management; Pain Measurement; Thiazines; Thiazoles

2013
Comparison of the effects of dexketoprofen trometamol, meloxicam and diclofenac sodium on fibular fracture healing, kidney and liver: an experimental rat model.
    Injury, 2014, Volume: 45, Issue:3

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Biomechanical Phenomena; Diclofenac; Fibula; Fracture Healing; Fractures, Bone; Inflammation; Ketoprofen; Kidney; Liver; Male; Meloxicam; Oxidative Stress; Pain; Rats; Rats, Sprague-Dawley; Thiazines; Thiazoles; Tromethamine

2014
Alleviation of behavioral hypersensitivity in mouse models of inflammatory pain with two structurally different casein kinase 1 (CK1) inhibitors.
    Molecular pain, 2014, Mar-10, Volume: 10

    Topics: Animals; Carrageenan; Casein Kinase I; Cells, Cultured; Disease Models, Animal; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Humans; Hyperalgesia; Indoles; Inflammation; Male; Membrane Potentials; Mice; Mice, Inbred C57BL; Pain; Pain Measurement; Pain Threshold; Phloroglucinol; Protein Transport; Spinal Cord; Thiazoles

2014
Development of a lameness model in sheep for assessing efficacy of analgesics.
    Australian veterinary journal, 2011, Volume: 89, Issue:8

    Topics: Analysis of Variance; Animals; Anti-Inflammatory Agents, Non-Steroidal; Body Temperature; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Combinations; Irritants; Lameness, Animal; Meloxicam; Pain; Sheep; Sheep Diseases; Thiazines; Thiazoles; Turpentine

2011
Effects of nonsteroidal anti-inflammatory meloxicam on stomach, kidney, and liver of rats.
    Toxicology and industrial health, 2016, Volume: 32, Issue:6

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Chemical and Drug Induced Liver Injury; Cyclooxygenase 2; Disease Models, Animal; Dose-Response Relationship, Drug; Inflammation; Kidney; Kidney Diseases; Liver; Meloxicam; Metaplasia; Pain; Rats; Rats, Sprague-Dawley; Stomach; Stomach Diseases; Thiazines; Thiazoles; Toxicity Tests

2016
Pharmacokinetics of sustained-release analgesics in mice.
    Journal of the American Association for Laboratory Animal Science : JAALAS, 2014, Volume: 53, Issue:5

    Topics: Analgesics; Animals; Buprenorphine; Butorphanol; Carbazoles; Delayed-Action Preparations; Female; Meloxicam; Mice; Pain; Thiazines; Thiazoles

2014
Pharmacokinetics of 3 formulations of meloxicam in cynomolgus macaques (Macaca fascicularis).
    Journal of the American Association for Laboratory Animal Science : JAALAS, 2014, Volume: 53, Issue:5

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Female; Humans; Injections, Intramuscular; Macaca fascicularis; Male; Meloxicam; Pain; Thiazines; Thiazoles

2014
Utilization of spray drying technique for improvement of dissolution and anti-inflammatory effect of Meloxicam.
    Pakistan journal of pharmaceutical sciences, 2015, Volume: 28, Issue:1

    Topics: Aerosols; Animals; Anti-Inflammatory Agents, Non-Steroidal; Buffers; Calorimetry, Differential Scanning; Chemistry, Pharmaceutical; Crystallography, X-Ray; Desiccation; Disease Models, Animal; Excipients; Formaldehyde; Hydrogen-Ion Concentration; Kinetics; Male; Meloxicam; Microscopy, Electron, Scanning; Pain; Particle Size; Rats, Wistar; Solubility; Spectroscopy, Fourier Transform Infrared; Technology, Pharmaceutical; Thiazines; Thiazoles; Water

2015
Novel thiazolo[3,2-b]-1,2,4-triazoles derived from naproxen with analgesic/anti-inflammatory properties: Synthesis, biological evaluation and molecular modeling studies.
    Bioorganic & medicinal chemistry, 2015, May-15, Volume: 23, Issue:10

    Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Disease Models, Animal; Drug Design; Edema; Humans; Inflammation; Mice; Molecular Docking Simulation; Molecular Dynamics Simulation; Naproxen; Nociception; Pain; Pain Measurement; Structure-Activity Relationship; Thiazoles; Thiones; Triazoles

2015
Perospirone Exhibits Antiemetic Efficacy against Opioid-Induced Nausea in Patients with Advanced Cancer.
    Journal of palliative medicine, 2015, Volume: 18, Issue:10

    Topics: Analgesics, Opioid; Antiemetics; Antipsychotic Agents; Female; Humans; Isoindoles; Japan; Male; Nausea; Neoplasms; Pain; Retrospective Studies; Thiazoles

2015
Eact, a small molecule activator of TMEM16A, activates TRPV1 and elicits pain- and itch-related behaviours.
    British journal of pharmacology, 2016, Volume: 173, Issue:7

    Topics: Animals; Anoctamin-1; Behavior, Animal; Benzamides; Cells, Cultured; Chloride Channel Agonists; Chloride Channels; Ganglia, Spinal; Humans; Mice, Congenic; Nociceptors; Pain; Pruritus; Rats; Thiazoles; TRPV Cation Channels

2016
Management of Severe Frostbite in a Grey-Headed Parrot (Poicephalus fuscicollis suahelicus).
    Journal of avian medicine and surgery, 2016, Volume: 30, Issue:1

    Topics: Animals; Anti-Bacterial Agents; Anti-Inflammatory Agents, Non-Steroidal; Antifungal Agents; Bird Diseases; Enrofloxacin; Female; Fluoroquinolones; Frostbite; Itraconazole; Meloxicam; Pain; Pentoxifylline; Psittaciformes; Thiazines; Thiazoles; Vasodilator Agents

2016
Piperidinyl thiazole isoxazolines: A new series of highly potent, slowly reversible FAAH inhibitors with analgesic properties.
    Bioorganic & medicinal chemistry letters, 2016, 06-15, Volume: 26, Issue:12

    Topics: Amidohydrolases; Analgesics; Animals; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Isoxazoles; Kinetics; Male; Mice; Mice, Inbred ICR; Molecular Docking Simulation; Molecular Structure; Pain; Pain Measurement; Piperidines; Structure-Activity Relationship; Thiazoles

2016
Small molecule dual-inhibitors of TRPV4 and TRPA1 for attenuation of inflammation and pain.
    Scientific reports, 2016, 06-01, Volume: 6

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Astrocytes; Cell Line, Tumor; Ceruletide; Chondrocytes; Disease Models, Animal; Humans; Inflammation; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Nociception; Pain; Pancreatitis, Acute Necrotizing; Primary Cell Culture; Rats; Swine; Thiazoles; Trigeminal Ganglion; TRPA1 Cation Channel; TRPV Cation Channels

2016
Real-time application of the Rat Grimace Scale as a welfare refinement in laboratory rats.
    Scientific reports, 2016, 08-17, Volume: 6

    Topics: Analgesia; Animal Welfare; Animals; Buprenorphine; Carrageenan; Computer Systems; Facial Expression; Feasibility Studies; Female; Male; Meloxicam; Pain; Pain Measurement; Rats; Rats, Sprague-Dawley; Retrospective Studies; Thiazines; Thiazoles; Video Recording

2016
Design, Synthesis, and Pharmacological Characterization of 2-(2-Furanyl)thiazolo[5,4-d]pyrimidine-5,7-diamine Derivatives: New Highly Potent A
    Journal of medicinal chemistry, 2016, 12-08, Volume: 59, Issue:23

    Topics: Acetic Acid; Adenosine A2 Receptor Agonists; Analgesics; Animals; CHO Cells; Cricetulus; Cyclic AMP; Diamines; Dose-Response Relationship, Drug; Drug Design; Female; Humans; Mice; Molecular Structure; Pain; Pyrimidines; Receptor, Adenosine A2A; Structure-Activity Relationship; Thiazoles

2016
Pain alleviation during castration of piglets: a comparative study of different farm options.
    Journal of animal science, 2016, Volume: 94, Issue:12

    Topics: Anesthesia, Local; Animal Husbandry; Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Hydrocortisone; Ketoprofen; Male; Meloxicam; Orchiectomy; ortho-Aminobenzoates; Pain; Pain Management; Swine; Thiazines; Thiazoles

2016
The AMPK Activator A769662 Blocks Voltage-Gated Sodium Channels: Discovery of a Novel Pharmacophore with Potential Utility for Analgesic Development.
    PloS one, 2017, Volume: 12, Issue:1

    Topics: AMP-Activated Protein Kinases; Analgesics; Anesthetics, Local; Animals; Binding Sites; Biphenyl Compounds; Drug Evaluation, Preclinical; HEK293 Cells; Hot Temperature; Humans; Male; meta-Aminobenzoates; Metformin; NAV1.7 Voltage-Gated Sodium Channel; Neural Conduction; Pain; Patch-Clamp Techniques; Pyrones; Rats; Rats, Sprague-Dawley; Reaction Time; Recombinant Fusion Proteins; Resveratrol; Sensory Receptor Cells; Sodium Channel Blockers; Stilbenes; Thiazoles; Thiophenes; Trigeminal Ganglion

2017
Perioperative analgesic use by Ontario veterinarians, 2012.
    The Canadian veterinary journal = La revue veterinaire canadienne, 2017, Volume: 58, Issue:2

    Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Castration; Cats; Dogs; Female; Hysterectomy; Male; Meloxicam; Ontario; Ovariectomy; Pain; Pain, Postoperative; Surveys and Questionnaires; Thiazines; Thiazoles; Veterinarians

2017
Comparative efficacy of oral meloxicam and phenylbutazone in 2 experimental pain models in the horse.
    The Canadian veterinary journal = La revue veterinaire canadienne, 2017, Volume: 58, Issue:2

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Female; Horses; Lameness, Animal; Lipopolysaccharides; Male; Meloxicam; Pain; Phenylbutazone; Skin Temperature; Synovitis; Thiazines; Thiazoles; Treatment Outcome

2017
Effects of meloxicam or tolfenamic acid administration on the pain and stress responses of Merino lambs to mulesing.
    Australian veterinary journal, 2008, Volume: 86, Issue:8

    Topics: Analgesics; Animal Welfare; Animals; Animals, Newborn; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; beta-Endorphin; Female; Haptoglobins; Hydrocortisone; Male; Meloxicam; ortho-Aminobenzoates; Pain; Posture; Random Allocation; Sheep; Sheep Diseases; Thiazines; Thiazoles; Time Factors; Treatment Outcome; Wound Healing

2008
A pilot study: sodium urate synovitis as an acute model of inflammatory response using objective and subjective criteria to evaluate arthritic pain in cats.
    Journal of veterinary pharmacology and therapeutics, 2008, Volume: 31, Issue:5

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Antioxidants; Area Under Curve; Cats; Female; Inflammation; Lameness, Animal; Meloxicam; Osteoarthritis; Pain; Pain Measurement; Pilot Projects; Severity of Illness Index; Synovitis; Thiazines; Thiazoles; Uric Acid

2008
The role of metabotropic glutamate receptor mGlu5 in control of micturition and bladder nociception.
    Neuroscience letters, 2009, Jan-23, Volume: 450, Issue:1

    Topics: Action Potentials; Analysis of Variance; Animals; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Jejunum; Mice; Models, Biological; Pain; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Reflex; Reflex, Stretch; Thiazoles; Urinary Bladder; Urination

2009
Effects of local anesthetic and a nonsteroidal antiinflammatory drug on pain responses of dairy calves to hot-iron dehorning.
    Journal of dairy science, 2009, Volume: 92, Issue:4

    Topics: Anesthetics, Local; Animals; Anti-Inflammatory Agents, Non-Steroidal; Body Temperature; Cattle; Dairying; Female; Heart Rate; Horns; Hot Temperature; Lidocaine; Male; Meloxicam; Ocular Physiological Phenomena; Pain; Random Allocation; Thiazines; Thiazoles; Time Factors

2009
KLYP956 is a non-imidazole-based orally active inhibitor of nitric-oxide synthase dimerization.
    Molecular pharmacology, 2009, Volume: 76, Issue:1

    Topics: Administration, Oral; Animals; Cells, Cultured; Dimerization; Enzyme Inhibitors; Fluoroquinolones; Humans; Mice; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type II; Pain; Species Specificity; Thiazoles

2009
NR2B receptor blockade inhibits pain-related sensitization of amygdala neurons.
    Molecular pain, 2009, Apr-28, Volume: 5

    Topics: Amygdala; Animals; Arthritis; Dose-Response Relationship, Drug; Male; Neurons; Pain; Rats; Receptors, N-Methyl-D-Aspartate; Thiazoles; Time Factors

2009
Demonstration of antiallodynic effects of the cyclooxygenase-2 inhibitor meloxicam on established diabetic neuropathic pain in mice.
    Journal of pharmacological sciences, 2009, Volume: 110, Issue:2

    Topics: Analgesics; Animals; Cyclooxygenase 2 Inhibitors; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Injections, Intraperitoneal; Injections, Spinal; Male; Meloxicam; Mice; Pain; Pain Measurement; Thiazines; Thiazoles

2009
A study of owner observed behavioural and lifestyle changes in cats with musculoskeletal disease before and after analgesic therapy.
    Journal of feline medicine and surgery, 2009, Volume: 11, Issue:12

    Topics: Analgesics; Animals; Behavior, Animal; Cat Diseases; Cats; Chronic Disease; Dogs; Female; Human-Animal Bond; Male; Meloxicam; Musculoskeletal Diseases; Pain; Pain Measurement; Severity of Illness Index; Thiazines; Thiazoles; Time Factors; Treatment Outcome

2009
Synthesis of some new pyrimido[2',1':2,3]thiazolo[4,5-b]quinoxaline derivatives as anti-inflammatory and analgesic agents.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:5

    Topics: Acetic Acid; Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Drug Evaluation, Preclinical; Edema; Female; Male; Mice; Molecular Structure; Pain; Pain Measurement; Pyrimidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Stereoisomerism; Thiazoles

2010
Synthesis of new 2,3-dihydroquinazolin-4(1H)-one derivatives for analgesic and anti-inflammatory evaluation.
    Archiv der Pharmazie, 2010, Volume: 343, Issue:5

    Topics: Acetic Acid; Analgesics; Animals; Anti-Inflammatory Agents; Carrageenan; Chalcones; Drug Evaluation, Preclinical; Edema; Male; Mice; Molecular Structure; Pain; Pain Measurement; Pyrazoles; Quinazolinones; Rats; Stomach Ulcer; Structure-Activity Relationship; Thiazoles

2010
The effect of meloxicam on behavior and pain sensitivity of dairy calves following cautery dehorning with a local anesthetic.
    Journal of dairy science, 2010, Volume: 93, Issue:6

    Topics: Anesthesia, Local; Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Cattle; Dairying; Drinking; Eating; Female; Horns; Meloxicam; Pain; Thiazines; Thiazoles; Video Recording

2010
Influence on analgesic activity and serum levels after meloxicam complexation with beta-cyclodextrin in mice and rats.
    Arzneimittel-Forschung, 2010, Volume: 60, Issue:6

    Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; beta-Cyclodextrins; Carrageenan; Hyperalgesia; Male; Meloxicam; Mice; Pain; Pain Measurement; Rats; Rats, Wistar; Thiazines; Thiazoles; Veins

2010
Central and peripheral sites of action for CB₂ receptor mediated analgesic activity in chronic inflammatory and neuropathic pain models in rats.
    British journal of pharmacology, 2011, Volume: 162, Issue:2

    Topics: Analgesia; Analgesics; Animals; Brain; Cannabinoids; Disease Models, Animal; Ganglia, Spinal; Inflammation; Male; Neuralgia; Opioid Peptides; Pain; Pain Perception; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB2; RNA, Messenger; Spinal Cord; Thiazoles

2011
Pharmacokinetics of meloxicam following intravenous and oral administration in green iguanas (Iguana iguana).
    American journal of veterinary research, 2010, Volume: 71, Issue:11

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Area Under Curve; Blood Cells; Body Weight; Female; Iguanas; Injections, Intravenous; Kidney; Male; Meloxicam; Pain; Stomach; Thiazines; Thiazoles

2010
Mitochondrial reactive oxygen species are activated by mGluR5 through IP3 and activate ERK and PKA to increase excitability of amygdala neurons and pain behavior.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Jan-19, Volume: 31, Issue:3

    Topics: Amygdala; Analysis of Variance; Animals; Antioxidants; Benzoates; Cyclic AMP-Dependent Protein Kinases; Cyclic N-Oxides; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Extracellular Signal-Regulated MAP Kinases; Glycine; Inositol 1,4,5-Trisphosphate; Macrocyclic Compounds; Mitochondria; Neurons; NG-Nitroarginine Methyl Ester; Oxazoles; Pain; Pain Measurement; Pain Perception; Patch-Clamp Techniques; Pyridines; Reactive Oxygen Species; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Signal Transduction; Spin Labels; Superoxides; Thiazoles; Vocalization, Animal

2011
Effect of local anaesthesia and/or analgesia on pain responses induced by piglet castration.
    Acta veterinaria Scandinavica, 2011, May-31, Volume: 53

    Topics: Analgesia; Anesthesia, Local; Anesthetics, Local; Animal Welfare; Animals; Animals, Newborn; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Lidocaine; Male; Meloxicam; Orchiectomy; Pain; Random Allocation; Serum Amyloid A Protein; Skin Temperature; Sus scrofa; Sweden; Thiazines; Thiazoles; Vocalization, Animal; Wounds and Injuries

2011
Antioxidant, analgesic, and anti-inflammatory activities of the ethanolic extracts of Taxillus liquidambaricola.
    Journal of ethnopharmacology, 2011, Oct-11, Volume: 137, Issue:3

    Topics: Acetic Acid; Analgesics; Animals; Anti-Inflammatory Agents; Antioxidants; Benzothiazoles; Biphenyl Compounds; Carrageenan; Catalase; Cell Line; Chromatography, High Pressure Liquid; Cyclooxygenase 2; Disease Models, Animal; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Edema; Endotoxins; Ethanol; Formaldehyde; Glutathione Peroxidase; Loranthaceae; Macrophages; Male; Malondialdehyde; Mice; Mice, Inbred ICR; Nitric Oxide; Nitric Oxide Synthase Type II; Pain; Picrates; Plants, Medicinal; Solvents; Sulfonic Acids; Superoxide Dismutase; Thiazoles; Time Factors; Tumor Necrosis Factor-alpha

2011
Evaluation of anti-inflammatory, anti-nociceptive, and anti-ulcerogenic activities of novel synthesized thiazolyl and pyrrolyl steroids.
    Archiv der Pharmazie, 2011, Volume: 344, Issue:9

    Topics: Analgesics; Animals; Anti-Inflammatory Agents; Anti-Ulcer Agents; Carrageenan; Disease Models, Animal; Edema; Inflammation; Pain; Pyrroles; Rats; Rats, Sprague-Dawley; Steroids; Stomach Ulcer; Thiazoles; Ulcer

2011
Involvement of metabotropic glutamate receptor 5 in pudendal inhibition of nociceptive bladder activity in cats.
    The Journal of physiology, 2011, Dec-01, Volume: 589, Issue:Pt 23

    Topics: Acetic Acid; Animals; Cats; Disease Models, Animal; Female; Pain; Pudendal Nerve; Pyridines; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Thiazoles; Urinary Bladder; Urinary Bladder Diseases; Urination

2011
3-Phenyl-5-isothiazole carboxamides with potent mGluR1 antagonist activity.
    Bioorganic & medicinal chemistry letters, 2012, Apr-01, Volume: 22, Issue:7

    Topics: Administration, Oral; Amides; Analgesics; Animals; Biological Availability; Brain; Excitatory Amino Acid Antagonists; Humans; Pain; Pain Measurement; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Stereoisomerism; Structure-Activity Relationship; Thiazoles

2012
Impact of general injection anaesthesia and analgesia on post-castration behaviour and teat order of piglets.
    Animal : an international journal of animal bioscience, 2012, Volume: 6, Issue:12

    Topics: Anesthetics, General; Animal Welfare; Animals; Animals, Newborn; Animals, Suckling; Anti-Inflammatory Agents, Non-Steroidal; Azaperone; Behavior, Animal; Drug Combinations; Injections, Subcutaneous; Ketamine; Male; Meloxicam; Orchiectomy; Pain; Postoperative Period; Sus scrofa; Thiazines; Thiazoles

2012
Effect of pain management on immunization efficacy in mice.
    Journal of the American Association for Laboratory Animal Science : JAALAS, 2012, Volume: 51, Issue:4

    Topics: Acetaminophen; Analgesia; Analgesics; Animals; Animals, Laboratory; Antibody Formation; Behavior, Animal; Buprenorphine; Freund's Adjuvant; Immunization; Lipids; Meloxicam; Mice; Pain; Pain Management; Thiazines; Thiazoles

2012
Cefovecin (Convenia) for the treatment of septic peritonitis in a female lion (Panthera leo).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2012, Volume: 43, Issue:3

    Topics: Animals; Anti-Bacterial Agents; Anti-Inflammatory Agents, Non-Steroidal; Cephalosporins; Female; Hysterectomy; Lions; Meloxicam; Pain; Peritonitis; Pyometra; Sepsis; Thiazines; Thiazoles

2012
2-Amino-4-arylthiazole compounds as TRPA1 antagonists (WO 2012085662): a patent evaluation.
    Expert opinion on therapeutic patents, 2013, Volume: 23, Issue:1

    Topics: Animals; Calcium Channels; Drug Design; Humans; Inflammation; Nerve Tissue Proteins; Pain; Patents as Topic; Thiazoles; Transient Receptor Potential Channels; TRPA1 Cation Channel

2013
Synthesis, SAR study, and biological evaluation of a series of piperazine ureas as fatty acid amide hydrolase (FAAH) inhibitors.
    Bioorganic & medicinal chemistry, 2013, Jan-01, Volume: 21, Issue:1

    Topics: Amidohydrolases; Analgesics; Animals; Humans; Mice; Molecular Docking Simulation; Pain; Piperazine; Piperazines; Rats; Structure-Activity Relationship; Thiazoles; Urea

2013
Gingival pain: an unusual side effect of ziprasidone.
    BMJ case reports, 2013, Jan-02, Volume: 2013

    Topics: Antipsychotic Agents; Gingiva; Humans; Male; Middle Aged; Pain; Piperazines; Thiazoles

2013
A case of recurrent psychosis during sickle cell disease crisis treated successfully with ziprasidone.
    Clinical schizophrenia & related psychoses, 2013, Volume: 6, Issue:4

    Topics: Adult; Analgesics, Opioid; Anemia, Sickle Cell; Antipsychotic Agents; Blood Transfusion; Diagnosis, Differential; Fluid Therapy; Hospitalization; Humans; Male; Pain; Pain Management; Piperazines; Psychotic Disorders; Recurrence; Thiazoles

2013
Multimodal analgesia for perioperative pain in three cats.
    Journal of feline medicine and surgery, 2013, Volume: 15, Issue:8

    Topics: Analgesics, Opioid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cat Diseases; Cats; Male; Meloxicam; Pain; Perioperative Period; Thiazines; Thiazoles

2013
Evaluation of the analgesic and anti-inflammatory activities of some thiazolo[4,5-d]pyrimidines.
    Arzneimittel-Forschung, 2002, Volume: 52, Issue:6

    Topics: Acetic Acid; Analgesics, Non-Narcotic; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Edema; Gastric Mucosa; Mice; Pain; Pyrimidines; Rats; Rats, Wistar; Stomach Ulcer; Structure-Activity Relationship; Thiazoles

2002
Modulation of NSAID-induced antinociceptive and anti-inflammatory effects by alpha2-adrenoceptor agonists with gastroprotective effects.
    Life sciences, 2002, May-03, Volume: 70, Issue:24

    Topics: Adrenergic alpha-Agonists; Animals; Anti-Inflammatory Agents, Non-Steroidal; Clonidine; Drug Synergism; Drug Therapy, Combination; Meloxicam; Mice; Naproxen; Pain; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Stomach Ulcer; Sulfonamides; Thiazines; Thiazoles; Yohimbine

2002
Craniomandibular osteopathy in a bullmastiff.
    The Canadian veterinary journal = La revue veterinaire canadienne, 2002, Volume: 43, Issue:11

    Topics: Analgesics, Non-Narcotic; Animals; Bone Diseases, Developmental; Craniomandibular Disorders; Dog Diseases; Dogs; Female; Mandible; Meloxicam; Pain; Radiography; Thiazines; Thiazoles

2002
A thymulin analogue peptide with powerful inhibitory effects on pain of neurogenic origin.
    Neuroscience, 2003, Volume: 119, Issue:1

    Topics: Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Capsaicin; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Hot Temperature; Hyperalgesia; Ligation; Male; Meloxicam; Morphine; Pain; Pain Threshold; Peptides; Peripheral Nervous System Diseases; Rats; Rats, Sprague-Dawley; Reaction Time; Thiazines; Thiazoles; Thymic Factor, Circulating; Time Factors

2003
Anti-nociception following exposure to trimethylthiazoline, peripheral or intra-amygdala estrogen and/or progesterone.
    Behavioural brain research, 2003, Sep-15, Volume: 144, Issue:1-2

    Topics: Amygdala; Animals; Corticosterone; Drug Administration Routes; Drug Administration Schedule; Drug Interactions; Estrogens; Female; Naloxone; Narcotic Antagonists; Odorants; Ovariectomy; Pain; Pain Measurement; Progesterone; Rats; Rats, Long-Evans; Reaction Time; Thiazoles

2003
[Treatment of severe pain with morphine in combination with fenamizol].
    Svensk farmaceutisk tidskrift, 1955, Nov-30, Volume: 59, Issue:33

    Topics: Analgesia; Anesthesia; Anesthesia and Analgesia; Morphine; Pain; Pain Management; Thiazoles

1955
[Intensive analgesia with daptazol-morphine combination].
    Schweizerische medizinische Wochenschrift, 1956, Sep-22, Volume: 86, Issue:38

    Topics: Analgesia; Morphine; Pain; Pain Management; Thiazoles

1956
[Clinical experience in the treatment of pain with a combination of amiphenazol and morphine during the surgery of accident injuries].
    Der Anaesthesist, 1958, Volume: 7, Issue:11

    Topics: Accidents; Humans; Morphine; Pain; Psychotherapy; Thiazoles; Wounds and Injuries

1958
Effect of carprofen, etodolac, meloxicam, or butorphanol in dogs with induced acute synovitis.
    American journal of veterinary research, 2003, Volume: 64, Issue:11

    Topics: Acute Disease; Animals; Anti-Inflammatory Agents, Non-Steroidal; Butorphanol; Carbazoles; Dog Diseases; Dogs; Female; Male; Meloxicam; Narcotic Antagonists; Pain; Synovitis; Thiazines; Thiazoles

2003
Synthesis, characterization and antiinflammatory-analgesic properties of 6-(alpha-amino-4-chlorobenzyl)thiazolo [3,2-b]-1,2,4-triazol-5-ols.
    Arzneimittel-Forschung, 2004, Volume: 54, Issue:1

    Topics: Acetic Acid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Benzoquinones; Capillary Permeability; Carrageenan; Chemical Phenomena; Chemistry, Physical; Edema; Foot; Indicators and Reagents; Magnetic Resonance Spectroscopy; Male; Mice; Models, Molecular; Molecular Conformation; Naproxen; Pain; Spectroscopy, Fourier Transform Infrared; Stomach Ulcer; Structure-Activity Relationship; Thiazoles; Triazoles

2004
Behavioural assessment of the effects of tumour growth in rats and the influence of the analgesics carprofen and meloxicam.
    Laboratory animals, 2004, Volume: 38, Issue:3

    Topics: Analysis of Variance; Animals; Behavior, Animal; Carbazoles; Disease Models, Animal; Male; Meloxicam; Pain; Pain Measurement; Pain, Postoperative; Rats; Rats, Inbred F344; Thiazines; Thiazoles; Urinary Bladder Neoplasms

2004
Synthesis and antinociceptive activity of (5-chloro-2(3H)-benzothiazolon-3-yl)propanamide derivatives.
    Archiv der Pharmazie, 2004, Volume: 337, Issue:9

    Topics: Analgesics, Non-Narcotic; Animals; Mice; Molecular Structure; Pain; Structure-Activity Relationship; Thiazoles

2004
Assessing the role of metabotropic glutamate receptor 5 in multiple nociceptive modalities.
    European journal of pharmacology, 2004, Dec-15, Volume: 506, Issue:2

    Topics: Acetic Acid; Animals; Carrageenan; Central Nervous System; Constriction, Pathologic; Edema; Formaldehyde; Hyperalgesia; Male; Mice; Mice, Inbred ICR; Motor Activity; Pain; Pain Measurement; Pain, Postoperative; Psychomotor Performance; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Spinal Nerves; Thiazoles; Vincristine

2004
Pharmacological evidence for the activation of Ca2+-activated K+ channels by meloxicam in the formalin test.
    Pharmacology, biochemistry, and behavior, 2005, Volume: 81, Issue:4

    Topics: 4-Aminopyridine; Analgesics, Non-Narcotic; Analysis of Variance; Animals; Apamin; Behavior, Animal; Charybdotoxin; Dose-Response Relationship, Drug; Female; Formaldehyde; Glyburide; Meloxicam; Pain; Pain Measurement; Potassium Channel Blockers; Potassium Channels, Calcium-Activated; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Tetraethylammonium; Thiazines; Thiazoles; Tolbutamide

2005
Role for cyclooxygenase 2 in the development and maintenance of neuropathic pain and spinal glial activation.
    Anesthesiology, 2005, Volume: 103, Issue:4

    Topics: Animals; Cyclooxygenase 2; Male; Meloxicam; Neuroglia; Pain; Peripheral Nervous System Diseases; Rats; Rats, Sprague-Dawley; Spinal Cord; Thiazines; Thiazoles

2005
Antinociceptive, brain-penetrating derivatives related to improgan, a non-opioid analgesic.
    European journal of pharmacology, 2005, Oct-17, Volume: 522, Issue:1-3

    Topics: Algorithms; Analgesics; Animals; Behavior, Animal; Benzothiazoles; Brain; Cimetidine; Dose-Response Relationship, Drug; Histamine H2 Antagonists; Injections, Intraventricular; Male; Mice; Molecular Structure; Pain; Pain Measurement; Phenoxypropanolamines; Piperidines; Quinazolines; Quinazolinones; Rats; Rats, Sprague-Dawley; Thiazoles; Time Factors; Triazoles

2005
[Efficacy of movalis in marked neurological manifestations of lumbar osteochondrosis].
    Zhurnal nevrologii i psikhiatrii imeni S.S. Korsakova, 2005, Volume: 105, Issue:9

    Topics: Adult; Anti-Inflammatory Agents, Non-Steroidal; Female; Humans; Lumbar Vertebrae; Male; Meloxicam; Middle Aged; Osteochondritis; Pain; Severity of Illness Index; Thiazines; Thiazoles

2005
Comparison of oral and subcutaneous administration of buprenorphine and meloxicam for preemptive analgesia in cats undergoing ovariohysterectomy.
    Journal of the American Veterinary Medical Association, 2005, Dec-15, Volume: 227, Issue:12

    Topics: Administration, Oral; Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Behavior, Animal; Buprenorphine; Cats; Drug Administration Routes; Female; Hysterotomy; Injections, Subcutaneous; Meloxicam; Ovariectomy; Pain; Postoperative Care; Thiazines; Thiazoles; Time Factors; Treatment Outcome

2005
Parkinson's drug may relieve fibromyalgia pain.
    Health news (Waltham, Mass.), 2005, Volume: 11, Issue:12

    Topics: Antiparkinson Agents; Benzothiazoles; Fibromyalgia; Humans; Pain; Pramipexole; Thiazoles

2005
Analgesic effects of mGlu1 and mGlu5 receptor antagonists in the rat formalin test.
    Neuropharmacology, 2006, Volume: 51, Issue:3

    Topics: Analgesics; Analysis of Variance; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Drug Interactions; Drug Tolerance; Formaldehyde; Male; Morphine; Pain; Pain Measurement; Pain Threshold; Pyridines; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Thiazoles

2006
The neurotrophic factor artemin promotes pancreatic cancer invasion.
    Annals of surgery, 2006, Volume: 244, Issue:2

    Topics: Adenocarcinoma; Blotting, Western; Cell Line, Tumor; Cell Proliferation; Coloring Agents; Glial Cell Line-Derived Neurotrophic Factor Receptors; Humans; Hypertrophy; Immunohistochemistry; Neoplasm Invasiveness; Nerve Growth Factors; Nerve Regeneration; Nerve Tissue Proteins; Neurons; Pain; Pancreas; Pancreatic Neoplasms; Polymerase Chain Reaction; Prospective Studies; Tetrazolium Salts; Thiazoles

2006
Meloxicam and surgical denervation of the coxofemoral joint for the treatment of degenerative osteoarthritis in a Bengal tiger (Panthera tigris tigris).
    Journal of zoo and wildlife medicine : official publication of the American Association of Zoo Veterinarians, 2006, Volume: 37, Issue:3

    Topics: Animals; Animals, Wild; Anti-Inflammatory Agents, Non-Steroidal; Combined Modality Therapy; Denervation; Hip Joint; Male; Meloxicam; Osteoarthritis; Pain; Thiazines; Thiazoles; Tigers; Treatment Outcome

2006
Antinociceptive profile of a selective metabotropic glutamate receptor 1 antagonist YM-230888 in chronic pain rodent models.
    European journal of pharmacology, 2007, Sep-24, Volume: 571, Issue:1

    Topics: Analgesics; Animals; Arthritis, Experimental; Benzimidazoles; Binding, Competitive; Cell Line; Cells, Cultured; Chronic Disease; Cycloheptanes; Dose-Response Relationship, Drug; Humans; Kinetics; Ligation; Molecular Structure; Motor Activity; Pain; Pain Measurement; Pyrimidines; Radioligand Assay; Rats; Rats, Inbred Lew; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Metabotropic Glutamate; Spinal Nerves; Thiazoles; Tritium

2007
Synergistic interaction between meloxicam and aminoguanidine in formalin-induced nociception in mice.
    European journal of pain (London, England), 2008, Volume: 12, Issue:3

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cyclooxygenase 2 Inhibitors; Drug Evaluation, Preclinical; Drug Synergism; Drug Therapy, Combination; Formaldehyde; Guanidines; Male; Meloxicam; Mice; Nitric Oxide Synthase Type II; Nociceptors; Pain; Pain Measurement; Thiazines; Thiazoles

2008
Modulation of morphine antinociception by the brain-penetrating H2 antagonist zolantidine: detailed characterization in five nociceptive test systems.
    Pharmacology, biochemistry, and behavior, 1995, Volume: 50, Issue:3

    Topics: Animals; Benzothiazoles; Blood-Brain Barrier; Histamine H2 Antagonists; Hot Temperature; Male; Morphine; Pain; Pain Measurement; Phenoxypropanolamines; Piperidines; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Thiazoles

1995
Importance of histamine H2 receptors in restraint-morphine interactions.
    Life sciences, 1995, Volume: 57, Issue:13

    Topics: Analysis of Variance; Animals; Benzothiazoles; Histamine; Histamine H2 Antagonists; Male; Morphine; Pain; Phenoxypropanolamines; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2; Restraint, Physical; Thiazoles; Time Factors

1995
3,3'-Bi-[1,3-thiazolidine-4-one] system. VII. Synthesis and SARS of some 2-heteroaryl derivatives with antiinflammatory and related activities.
    Farmaco (Societa chimica italiana : 1989), 1994, Volume: 49, Issue:1

    Topics: Acetates; Acetic Acid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Experimental; Carrageenan; Edema; Magnetic Resonance Spectroscopy; Male; Mice; Pain; Pain Measurement; Rats; Rats, Wistar; Spectrophotometry, Infrared; Stomach Ulcer; Structure-Activity Relationship; Thiazoles

1994
Anti-inflammatory, analgesic, antipyretic and related properties of meloxicam, a new non-steroidal anti-inflammatory agent with favourable gastrointestinal tolerance.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1995, Volume: 44, Issue:10

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Bronchial Spasm; Chemotaxis, Leukocyte; Fever; Guinea Pigs; In Vitro Techniques; Inflammation; Male; Meloxicam; Mice; Pain; Pain Measurement; Rats; Stomach Ulcer; Thiazines; Thiazoles; Uricosuric Agents

1995
Synthesis and SAR study of imidazo[2,1-b]benzothiazole acids and some related compounds with anti-inflammatory and analgesic activities.
    Farmaco (Societa chimica italiana : 1989), 1996, Volume: 51, Issue:7

    Topics: Acetates; Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Edema; Female; Imidazoles; Pain; Pain Measurement; Pregnancy; Rats; Stomach Ulcer; Structure-Activity Relationship; Thiazoles

1996
Central antinociceptive effects of meloxicam on rat spinal cord in vitro.
    Neuroreport, 1998, Mar-09, Volume: 9, Issue:4

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Cyclooxygenase 1; Cyclooxygenase 2; Electric Stimulation; Female; Hindlimb; Hyperalgesia; In Vitro Techniques; Indomethacin; Isoenzymes; Male; Meloxicam; Membrane Proteins; Pain; Perfusion; Prostaglandin-Endoperoxide Synthases; Rats; Rats, Wistar; Spinal Cord; Spinal Nerve Roots; Thiazines; Thiazoles

1998
Antinociceptive effect of meloxicam, in neurogenic and inflammatory nociceptive models in mice.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1998, Volume: 47, Issue:7

    Topics: Abdominal Muscles; Acetic Acid; Analgesics; Analgesics, Opioid; Animals; Capsaicin; Cyclooxygenase Inhibitors; Diclofenac; Formaldehyde; Inflammation; Male; Meloxicam; Mice; Morphine; Muscle Contraction; Pain; Pain Measurement; Reaction Time; Thiazines; Thiazoles

1998
Evidence for the participation of the nitric oxide-cyclic GMP pathway in the antinociceptive action of meloxicam in the formalin test.
    European journal of pharmacology, 2000, Apr-21, Volume: 395, Issue:1

    Topics: Analgesics, Non-Narcotic; Animals; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Formaldehyde; Guanylate Cyclase; Meloxicam; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Pain; Pain Measurement; Quinoxalines; Rats; Rats, Wistar; Thiazines; Thiazoles

2000
The role of cytokines and prostaglandin-E(2) in thymulin induced hyperalgesia.
    Neuropharmacology, 2000, Jul-10, Volume: 39, Issue:9

    Topics: Analgesics, Non-Narcotic; Animals; Cytokines; Dinoprostone; Dose-Response Relationship, Drug; Hyperalgesia; Immune Sera; Interleukin 1 Receptor Antagonist Protein; Interleukin-1; Male; Meloxicam; Nerve Growth Factor; Pain; Pain Measurement; Rats; Rats, Sprague-Dawley; Sialoglycoproteins; Thiazines; Thiazoles; Thymic Factor, Circulating; Time Factors; Tumor Necrosis Factor-alpha

2000
Meloxicam selectively depresses the afterdischarge of rat spinal dorsal horn neurones in response to noxious stimulation.
    Neuroscience letters, 2001, Jun-01, Volume: 305, Issue:1

    Topics: Analgesics, Non-Narcotic; Animals; Male; Meloxicam; Neurons; Pain; Physical Stimulation; Rats; Rats, Sprague-Dawley; Spinal Cord; Thiazines; Thiazoles

2001
3-Arylsulphonyl-5-arylamino-1,3,4-thiadiazol-2(3H)ones as anti-inflammatory and analgesic agents.
    Bioorganic & medicinal chemistry, 2001, Volume: 9, Issue:8

    Topics: Analgesics; Animals; Anti-Inflammatory Agents; Disease Models, Animal; Edema; Female; Male; Mice; Pain; Rats; Sulfur Compounds; Thiazoles

2001
Synthesis and antinociceptive activity of [(2-oxobenzothiazolin-3-yl)methyl]-4-alkyl/aryl-1,2,4-triazoline-5-thiones.
    Archiv der Pharmazie, 2001, Volume: 334, Issue:8-9

    Topics: Analgesics; Animals; Mice; Pain; Structure-Activity Relationship; Thiazoles

2001
Analgesic activity of a novel use-dependent sodium channel blocker, crobenetine, in mono-arthritic rats.
    British journal of pharmacology, 2001, Volume: 134, Issue:8

    Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Experimental; Benzomorphans; Dose-Response Relationship, Drug; Female; Freund's Adjuvant; Hyperalgesia; Inflammation; Meloxicam; Mexiletine; Pain; Pain Measurement; Posture; Rats; Rats, Wistar; Sodium Channel Blockers; Thiazines; Thiazoles

2001
Synthesis and in vivo pharmacology of new derivatives of isothiazolo[5,4-b]pyridine of Mannich base type.
    Farmaco (Societa chimica italiana : 1989), 2001, Volume: 56, Issue:12

    Topics: Analgesics, Non-Narcotic; Animals; Crystallography, X-Ray; Drug Evaluation, Preclinical; Injections, Intraperitoneal; Mice; Molecular Structure; Motor Activity; Pain; Pyridines; Rats; Serotonin Agents; Structure-Activity Relationship; Thiazoles

2001
Neostigmine interactions with non steroidal anti-inflammatory drugs.
    British journal of pharmacology, 2002, Volume: 135, Issue:7

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cholinesterase Inhibitors; Diclofenac; Disease Models, Animal; Drug Synergism; Ketoprofen; Meloxicam; Mice; Neostigmine; Pain; Pain Measurement; Prostaglandin-Endoperoxide Synthases; Thiazines; Thiazoles

2002
Synthesis and pharmacological properties of benzisothiazole/benzimidazole derivatives with acidic groups.
    Farmaco (Societa chimica italiana : 1989), 2002, Volume: 57, Issue:5

    Topics: Acetaminophen; Acetic Acid; Analgesics; Animals; Benzimidazoles; Escherichia coli; Female; Guinea Pigs; Ileum; Lethal Dose 50; Lipopolysaccharides; Male; Mice; Pain; Pain Measurement; Parasympatholytics; Platelet Aggregation Inhibitors; Rats; Rats, Wistar; Stereoisomerism; Structure-Activity Relationship; Thiazoles

2002
The effect of thiazol-4-yimethoxyamine, a histidine decarboxylase inhibitor, on the development of morphine tolerance and physical dependance in mice.
    Experientia, 1976, Oct-15, Volume: 32, Issue:10

    Topics: Animals; Behavior, Animal; Brain; Carboxy-Lyases; Drug Tolerance; Female; Histamine; Histidine Decarboxylase; Humans; Hydroxylamines; Male; Mice; Morphine; Pain; Substance-Related Disorders; Thiazoles

1976
4-(1,2-Benzisothiazol-3-yl)alkanoic and phenylalkanoic acids: synthesis and anti-inflammatory, analgesic and antipyretic activities.
    Farmaco (Societa chimica italiana : 1989), 1992, Volume: 47, Issue:5

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Edema; Escherichia coli; Ibuprofen; Male; Mice; Pain; Phenylbutazone; Pyrogens; Rats; Rats, Wistar; Thiazoles

1992
[Experimental study on the principal effects and dependence potential of thiofentanil].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1991, Volume: 26, Issue:4

    Topics: Analgesics, Opioid; Animals; Dogs; Female; Immobilization; Macaca mulatta; Male; Mice; Pain; Piperidines; Rabbits; Rats; Sensory Thresholds; Substance Withdrawal Syndrome; Substance-Related Disorders; Thiazoles

1991
Zolantidine-induced attenuation of morphine antinociception in rhesus monkeys.
    Brain research, 1990, Aug-27, Volume: 526, Issue:1

    Topics: Animals; Benzothiazoles; Dose-Response Relationship, Drug; Double-Blind Method; Female; Histamine H2 Antagonists; Macaca mulatta; Morphine; Pain; Phenoxypropanolamines; Piperidines; Thiazoles

1990
Pharmacological properties of thiazolinobutazone (LAS 11871). II. Analgesic and antipyretic effects.
    Arzneimittel-Forschung, 1974, Volume: 24, Issue:11

    Topics: Acetates; Administration, Oral; Animals; Bradykinin; Drug Evaluation, Preclinical; Inflammation; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Mice; Pain; Phenylbutazone; Pressure; Rats; Reaction Time; Tail; Thiazoles

1974
The analgesic action of morphine-n-oxide.
    British journal of pharmacology, 1968, Volume: 34, Issue:2

    Topics: Acridines; Analgesia; Animals; Cyclic N-Oxides; Hot Temperature; Injections, Intraperitoneal; Injections, Subcutaneous; Mice; Morphine; Pain; Rats; Tail; Thiazoles

1968