indazoles has been researched along with Emesis in 73 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 7 (9.59) | 18.7374 |
1990's | 57 (78.08) | 18.2507 |
2000's | 2 (2.74) | 29.6817 |
2010's | 6 (8.22) | 24.3611 |
2020's | 1 (1.37) | 2.80 |
Authors | Studies |
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Chin, S; Choi, JW; Kim, SG; Kim, YS; Yoo, JJ | 1 |
Gunderson, CC; Matulonis, U; Moore, KN | 1 |
O'Cearbhaill, RE | 1 |
Berardi, R; Burattini, L; Cascinu, S; Conti, A; De Giorgi, U; Iacovelli, R; Muzzonigro, G; Pantano, F; Santini, D; Santoni, M | 1 |
Arnold, JK; Edison, LA; Gerona, RR; Schwartz, MD; Steck, AR; Trecki, J | 1 |
Brown, AP; Courtney, CL; Criswell, KA; Evering, W; Holliman, CL; Jessen, BA | 1 |
Dowlati, A; Gibson, DM; Hodge, JP; Hurwitz, HI; Merkle, EM; Pandite, L; Saini, S; Savage, S; Suttle, AB | 1 |
Chowbay, B; Gao, F; Goh, BC; Ivy, P; Koh, TS; Leong, SS; Lim, WT; Ng, QS; Singh, O; Tan, DS; Tan, EH; Thng, CH; Toh, CK | 1 |
Andrews, L; Fishman, M; Gorbunova, V; Jonasch, E; Larkin, J; Negrier, S; Olivier, K; Pyle, L; Staehler, M; Wood, L | 1 |
Dott, CS; Joss, RA | 1 |
Smith, IE | 2 |
Angel, I; Garreau, M; Langer, SZ; Prouteau, M; Schoemaker, H | 1 |
de Wet, M; Falkson, G; Rapoport, BL | 1 |
Fukunaka, N; Ishioka, S; Itoh, E; Kitajima, Y; Kudo, R; Sagae, S; Sato, K | 1 |
Furue, H; Niitani, H; Ogawa, N; Ohta, K; Suminaga, M; Taguchi, T | 2 |
Gondo, H; Harada, M; Matsuishi, H; Omori, F; Otsuka, T; Shibuya, T; Taniguchi, S; Teshima, T; Yamano, Y; Yamazaki, K | 1 |
Aapro, MS | 1 |
Mori, K; Suga, Y; Takahashi, T; Tominaga, K | 1 |
Hiraoka, A; Kageyama, T; Kakishita, E; Masaoka, T; Matsuzawa, Y; Nagai, K; Okuda, K; Oshiba, S; Tatsumi, N; Uchino, H | 1 |
Cline, JM; Page, RL; Price, GS; Riviere, JE; Thrall, DE | 1 |
Endo, T; Hagihara, K; Hamaue, N; Hirafuji, M; Minami, M; Monma, Y; Ogawa, T; Tamakai, H; Yoshioka, M | 1 |
BaĆ¹, MG; Berruti, A; Bottini, A; Buniva, T; Danese, S; Dogliotti, L; Farris, A; Moro, G; Porcile, G; Richiardi, G; Zola, P | 1 |
Airey, JE; Campbell, HF; Darkes, P; Fitzpatrick, LR; Klein, S; Neuenschwander, K; Pendley, CE; Powers, M; Schnapper, M; Youssefyeh, RD | 1 |
Aguerri, MF; Alby, N; Giacchetti, S; Imbeaux, PH | 1 |
Bremer, K | 1 |
Marty, M | 2 |
Blijham, GH | 1 |
Andrews, PL; Bhandari, P; Bingham, S; Blower, PR; Davey, PT; Marr, HE | 1 |
Diehl, V | 1 |
Hacking, A | 1 |
Dilly, S | 1 |
Kamanabrou, D | 1 |
Andrews, PL; Bingham, S; Joel, SP; Patel, N; Slevin, ML; Thompson, PI | 1 |
Blijham, GH; Bots, MW; Dijkstra, HJ; Fehmers, MC; Keizer, HJ; Nortier, JW; Siegenbeek van Heukelom, L; Slee, PH; van der Wall, E; Veenhof, CH | 1 |
Kaizer, L; Laberge, F; Latreille, J; O'Connell, G; Osoba, D; Pater, J; Stewart, D; Venner, P; Warr, D; Wilan, A | 1 |
Bosanquet, N; Jones, AL; Lee, GJ | 1 |
Aapro, M; Diehl, V; Kaye, SB; Khayat, D | 1 |
Ito, T; Kato, S; Omoya, H; Yoshida, N | 1 |
Butler, M; Collis, C; Coumar, A; Gandhi, L; Hamon, M; Hunter, AE; Murdoch, R; Pothecary, K; Prentice, HG; Upward, J | 1 |
Davis, A; Erlichman, C; Fine, S; Laberge, F; Lofters, W; Osoba, D; Rusthoven, J; Warr, D; Willan, A; Wilson, K | 1 |
Hunter, RD; Logue, JP; Magee, B; Murdoch, RD | 1 |
Amaral, D; Lemerle, J; Murdoch, RD; Southall, DP; Upward, J | 1 |
Andrews, PL; Bhandari, P | 1 |
de Mulder, PH; Seynaeve, C; Verweij, J | 1 |
Goa, KL; Plosker, GL | 1 |
Gandara, DR; Hesketh, PJ | 1 |
Falkson, CI; Falkson, G; Falkson, HC | 1 |
Addelman, M; Erlichman, C; Fine, S; Murray, C; Warr, D | 1 |
Nakao, I | 1 |
King, GL | 1 |
Airey, JE; Bostwick, JS; Decktor, DL; Fitzpatrick, LR; Gessner, GW; Lambert, RM; Martin, GE; Pendleton, RG; Pendley, CE; Youssefyeh, RD | 1 |
Soukop, M | 1 |
Brand, BC; Buser, KS; Cerny, T; Joss, RA | 1 |
Caubel, M; Cupissol, DR; Serrou, B | 1 |
Chevallier, B | 1 |
Tabona, MV | 1 |
Blower, PR | 1 |
Pintens, H | 1 |
Brown, GW; Butcher, ME; Kidgell, AE | 1 |
Maher, M | 1 |
Button, D | 1 |
Falkson, G; van Zyl, AJ | 1 |
Bhandari, P; Gupta, YK; Seth, SD | 1 |
Brunner, K; Buser, K; Joss, R; Karde, C; Pirovino, M; Rohrbach, D | 1 |
Brunner, KW; Joss, RA; Pirovino, M; Richner, J; Rohrbach, D; Terrey, JP; Upward, J | 1 |
Bermudez, J; Boyle, EA; Miner, WD; Sanger, GJ | 1 |
Adams, L; Cassidy, J; Kaye, SB; Lewis, C; Raina, V; Rankin, EM; Rapeport, WG; Soukop, M; Zussman, BD | 1 |
10 review(s) available for indazoles and Emesis
Article | Year |
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Management of the toxicities of common targeted therapeutics for gynecologic cancers.
Topics: Anemia; Angiogenesis Inhibitors; Antineoplastic Agents, Immunological; Autoimmune Diseases; Bevacizumab; Diarrhea; Epistaxis; Fatigue; Female; Genital Neoplasms, Female; Headache; Hemorrhage; Humans; Hypertension; Indazoles; Intestinal Perforation; Molecular Targeted Therapy; Nausea; Neutropenia; Poly(ADP-ribose) Polymerase Inhibitors; Precision Medicine; Proteinuria; Pyrimidines; Risk Assessment; Sulfonamides; Vomiting; Water-Electrolyte Imbalance | 2018 |
Risk of gastrointestinal events with sorafenib, sunitinib and pazopanib in patients with solid tumors: a systematic review and meta-analysis of clinical trials.
Topics: Adverse Drug Reaction Reporting Systems; Carcinoma, Renal Cell; Clinical Trials as Topic; Diarrhea; Gastrointestinal Diseases; Gastrointestinal Tract; Humans; Incidence; Indazoles; Indoles; Liver Neoplasms; Neoplasms; Niacinamide; Phenylurea Compounds; Pyrimidines; Pyrroles; Sorafenib; Sulfonamides; Sunitinib; Vomiting | 2014 |
Review of experience with ondansetron and granisetron.
Topics: Antiemetics; Antineoplastic Agents; Granisetron; Humans; Indazoles; Nausea; Ondansetron; Serotonin Antagonists; Vomiting | 1993 |
Are granisetron and ondansetron equivalent in the clinic?
Topics: Antiemetics; Antineoplastic Agents; Cisplatin; Granisetron; Humans; Imidazoles; Indazoles; Nausea; Ondansetron; Serotonin Antagonists; Vomiting | 1992 |
5-HT3 receptor antagonists, a new approach in emesis: a review of ondansetron, granisetron and tropisetron.
Topics: Animals; Antiemetics; Granisetron; Humans; Imidazoles; Indazoles; Indoles; Ondansetron; Serotonin Antagonists; Tropisetron; Vomiting | 1991 |
Granisetron. A review of its pharmacological properties and therapeutic use as an antiemetic.
Topics: Animals; Antiemetics; Antineoplastic Agents; Female; Granisetron; Humans; Indazoles; Male; Nausea; Neoplasms; Serotonin Antagonists; Vomiting | 1991 |
[Gastrointestinal side effects of anticancer agents and their counter measures].
Topics: Antiemetics; Antineoplastic Agents; Cisplatin; Granisetron; Humans; Indazoles; Nausea; Vomiting | 1990 |
Granisetron (BRL 43694) in the treatment of cytostatic drug-induced emesis: a summary.
Topics: Animals; Antiemetics; Antineoplastic Agents; Cisplatin; Ferrets; Granisetron; Headache; Humans; Indazoles; Serotonin Antagonists; Vomiting | 1990 |
Antiemetic control: 5-HT3 antagonists: review of clinical results, with particular emphasis on ondansetron.
Topics: Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Cisplatin; Granisetron; Headache; Humans; Imidazoles; Indazoles; Indoles; Nausea; Ondansetron; Radiation Injuries; Radiotherapy; Serotonin Antagonists; Tropisetron; Vomiting | 1990 |
Recent developments in the management of emesis with the 5-HT3 antagonist granisetron.
Topics: Antiemetics; Granisetron; Humans; Indazoles; Serotonin Antagonists; Vomiting | 1990 |
25 trial(s) available for indazoles and Emesis
Article | Year |
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Phase I trial of pazopanib in patients with advanced cancer.
Topics: Administration, Oral; Adult; Aged; Angiogenesis Inhibitors; Anorexia; Cohort Studies; Diarrhea; Drug Administration Schedule; Fatigue; Female; Humans; Hypertension; Indazoles; Male; Middle Aged; Nausea; Neoplasms; Pyrimidines; Sulfonamides; Vomiting | 2009 |
A Phase II study of pazopanib in Asian patients with recurrent/metastatic nasopharyngeal carcinoma.
Topics: Adult; Aged; Angiogenesis Inhibitors; Anorexia; Asian People; Carcinoma; Diarrhea; Drug Administration Schedule; Fatigue; Female; Humans; Indazoles; Kaplan-Meier Estimate; Male; Middle Aged; Nasopharyngeal Carcinoma; Nasopharyngeal Neoplasms; Neoplasm Metastasis; Neoplasm Recurrence, Local; Neovascularization, Pathologic; Pyrimidines; Sulfonamides; Treatment Outcome; Vomiting | 2011 |
A dose-finding study of granisetron, a novel antiemetic, in patients receiving cytostatic chemotherapy. The Granisetron Study Group.
Topics: Antiemetics; Antineoplastic Agents; Double-Blind Method; Female; Granisetron; Humans; Indazoles; Infant, Newborn; Injections, Intravenous; Nausea; Vomiting | 1993 |
The antiemetic efficacy and safety of granisetron compared with metoclopramide plus dexamethasone in patients receiving fractionated chemotherapy over 5 days. The Granisetron Study Group.
Topics: Antiemetics; Antineoplastic Agents; Cisplatin; Dexamethasone; Drug Administration Schedule; Drug Therapy, Combination; Etoposide; Female; Granisetron; Humans; Ifosfamide; Indazoles; Male; Metoclopramide; Middle Aged; Vomiting | 1993 |
[Clinical evaluation of granisetron for nausea and vomiting induced by anticancer drugs--optimal dose-finding study].
Topics: Administration, Oral; Adult; Aged; Antiemetics; Cisplatin; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Nausea; Neoplasms; Vomiting | 1993 |
[Clinical evaluation of granisetron for nausea and vomiting induced by anticancer drugs--multi-centered placebo-controlled double-blind comparative study].
Topics: Administration, Oral; Antiemetics; Cisplatin; Double-Blind Method; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Nausea; Tablets; Vomiting | 1993 |
[Study on the inhibitory effect of oral granisetron against nausea/vomiting induced by cytosine arabinoside containing chemotherapy for tumors in the hematopoietic organs].
Topics: Administration, Oral; Adult; Aged; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Cytarabine; Daunorubicin; Etoposide; Female; Granisetron; Humans; Indazoles; Lymphoma; Male; Middle Aged; Mitoxantrone; Nausea; Vomiting | 1993 |
[Granisetron oral phase III clinical trial--study on the inhibitory effect of granisetron for nausea/vomiting induced by chemotherapy for tumors in the hematopoietic organs].
Topics: Administration, Oral; Adolescent; Adult; Aged; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Drug Administration Schedule; Female; Granisetron; Hodgkin Disease; Humans; Indazoles; Leukemia; Lymphoma, Non-Hodgkin; Male; Middle Aged; Nausea; Vomiting | 1993 |
Cisplatin, epirubicin, and lonidamine combination regimen as first-line chemotherapy for metastatic breast cancer: a pilot study.
Topics: Administration, Oral; Adult; Aged; Anemia; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Cisplatin; Epirubicin; Female; Humans; Indazoles; Infusions, Intravenous; Middle Aged; Nausea; Pilot Projects; Thrombocytopenia; Treatment Outcome; Vomiting | 1998 |
A single-blind study of the efficacy and safety of intravenous granisetron compared with alizapride plus dexamethasone in the prophylaxis and control of emesis in patients receiving 5-day cytostatic therapy. The Granisetron Study Group.
Topics: Adult; Antiemetics; Antineoplastic Agents; Dexamethasone; Drug Therapy, Combination; Female; Granisetron; Humans; Indazoles; Infusions, Intravenous; Male; Middle Aged; Nausea; Pyrrolidines; Single-Blind Method; Vomiting | 1992 |
A comparison of granisetron as a single agent with conventional combination antiemetic therapies in the treatment of cytostatic-induced emesis. The Granisetron Study Group.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Agents; Cisplatin; Drug Therapy, Combination; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Nausea; Single-Blind Method; Vomiting | 1992 |
Fractionated chemotherapy--granisetron or conventional antiemetics? The Granisetron Study Group.
Topics: Adult; Antiemetics; Antineoplastic Agents; Dexamethasone; Drug Administration Schedule; Drug Therapy, Combination; Female; Granisetron; Humans; Indazoles; Male; Metoclopramide; Middle Aged; Nausea; Pyrrolidines; Single-Blind Method; Vomiting | 1992 |
Oral granisetron--simple and effective: a preliminary report. The Granisetron Study Group.
Topics: Administration, Oral; Adult; Antiemetics; Antineoplastic Agents; Double-Blind Method; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Nausea; Vomiting | 1992 |
Intravenous granisetron--establishing the optimal dose. The Granisetron Study Group.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Agents; Double-Blind Method; Drug Administration Schedule; Female; Granisetron; Humans; Indazoles; Infusions, Intravenous; Male; Middle Aged; Nausea; Vomiting | 1992 |
A randomized trial of two doses of granisetron in the treatment of chemotherapy-induced emesis. Dutch results within a multinational study.
Topics: Adult; Aged; Aged, 80 and over; Antiemetics; Antineoplastic Agents; Cisplatin; Dose-Response Relationship, Drug; Double-Blind Method; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Nausea; Netherlands; Serotonin Antagonists; Vomiting | 1992 |
A randomised, double-blind comparison of granisetron with high-dose metoclopramide, dexamethasone and diphenhydramine for cisplatin-induced emesis. An NCI Canada Clinical Trials Group Phase III Trial.
Topics: Antiemetics; Cisplatin; Dexamethasone; Diphenhydramine; Double-Blind Method; Drug Therapy, Combination; Female; Granisetron; Humans; Indazoles; Male; Metoclopramide; Middle Aged; Nausea; Vomiting | 1992 |
Superiority of granisetron to dexamethasone plus prochlorperazine in the prevention of chemotherapy-induced emesis.
Topics: Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Nausea; Prochlorperazine; Serotonin Antagonists; Vomiting | 1991 |
The antiemetic effect of granisetron in lower hemibody radiotherapy.
Topics: Aged; Antiemetics; Bone Neoplasms; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Prospective Studies; Radiotherapy; Vomiting | 1991 |
Granisetron. A review of its pharmacological properties and therapeutic use as an antiemetic.
Topics: Animals; Antiemetics; Antineoplastic Agents; Female; Granisetron; Humans; Indazoles; Male; Nausea; Neoplasms; Serotonin Antagonists; Vomiting | 1991 |
High versus low dose granisetron, a selective 5HT3 antagonist, for the prevention of chemotherapy-induced nausea and vomiting.
Topics: Antineoplastic Agents; Double-Blind Method; Drugs, Investigational; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Nausea; Random Allocation; Serotonin Antagonists; Vomiting | 1990 |
A comparison of two dose levels of granisetron in patients receiving high-dose cisplatin. The Granisetron Study Group.
Topics: Cisplatin; Double-Blind Method; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Nausea; Neoplasms; Serotonin Antagonists; Time Factors; Vomiting | 1990 |
A comparison of two dose levels of granisetron in patients receiving moderately emetogenic cytostatic chemotherapy. The Granisetron Study Group.
Topics: Antineoplastic Agents; Double-Blind Method; Female; Granisetron; Headache; Humans; Indazoles; Male; Middle Aged; Nausea; Serotonin Antagonists; Time Factors; Vomiting | 1990 |
The efficacy of granisetron as a prophylactic anti-emetic and intervention agent in high-dose cisplatin-induced emesis.
Topics: Adult; Aged; Cisplatin; Double-Blind Method; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Nausea; Neoplasms; Serotonin Antagonists; Sex Factors; Time Factors; Vomiting | 1990 |
A comparative study of the use of granisetron, a selective 5-HT3 antagonist, versus a standard anti-emetic regimen of chlorpromazine plus dexamethasone in the treatment of cytostatic-induced emesis. The Granisetron Study Group.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antineoplastic Agents; Chlorpromazine; Dexamethasone; Double-Blind Method; Drug Therapy, Combination; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Serotonin Antagonists; Time Factors; Vomiting | 1990 |
Efficacy and safety of granisetron compared with high-dose metoclopramide plus dexamethasone in patients receiving high-dose cisplatin in a single-blind study. The Granisetron Study Group.
Topics: Cisplatin; Dexamethasone; Drug Therapy, Combination; Female; Granisetron; Headache; Humans; Indazoles; Male; Metoclopramide; Middle Aged; Neoplasms; Serotonin Antagonists; Single-Blind Method; Vomiting | 1990 |
39 other study(ies) available for indazoles and Emesis
Article | Year |
---|---|
Pazopanib-induced severe acute liver injury: A case report.
Topics: Bilirubin; Biopsy; Carcinoma, Renal Cell; Chemical and Drug Induced Liver Injury; Female; Hepatitis B; Humans; Indazoles; Jaundice; Kidney Neoplasms; Middle Aged; Nausea; Pyrimidines; Steroids; Sulfonamides; Tomography, X-Ray Computed; Ultrasonography; United States; Vomiting | 2021 |
Using PARP Inhibitors in Advanced Ovarian Cancer.
Topics: Anemia; Creatinine; Drug Administration Schedule; Drug Interactions; Exanthema; Fatigue; Female; Genes, BRCA1; Genes, BRCA2; Heart Rate; Humans; Hypertension; Indazoles; Leukopenia; Mutation; Myelodysplastic Syndromes; Nasopharyngitis; Nausea; Ovarian Neoplasms; Piperidines; Pneumonia; Poly(ADP-ribose) Polymerase Inhibitors; Thrombocytopenia; Transaminases; Vomiting | 2018 |
A Common Source Outbreak of Severe Delirium Associated with Exposure to the Novel Synthetic Cannabinoid ADB-PINACA.
Topics: Acidosis; Adolescent; Adult; Aggression; Anxiety; Cannabinoids; Delirium; Disease Outbreaks; Female; Georgia; Humans; Hyperglycemia; Hypokalemia; Indazoles; Male; Middle Aged; Nausea; Seizures; Tachycardia; Vomiting; Young Adult | 2015 |
Toxicity and toxicokinetics of the cyclin-dependent kinase inhibitor AG-024322 in cynomolgus monkeys following intravenous infusion.
Topics: Animals; Anorexia; Antineoplastic Agents; Ataxia; Benzimidazoles; Blood Vessels; Bone Marrow; Cyclin-Dependent Kinases; Dose-Response Relationship, Drug; Female; Gastrointestinal Tract; Hematologic Diseases; Indazoles; Infusions, Intravenous; Kidney Tubules; Lethargy; Macaca fascicularis; Male; Protein Kinase Inhibitors; Self Mutilation; Stereotyped Behavior; Vomiting | 2008 |
Axitinib for the treatment of metastatic renal cell carcinoma: recommendations for therapy management to optimize outcomes.
Topics: Axitinib; Carcinoma, Renal Cell; Diarrhea; Dysphonia; Fatigue; Humans; Hypertension; Imidazoles; Indazoles; Kidney Neoplasms; Nausea; Protein Kinase Inhibitors; Proteinuria; Vomiting | 2014 |
Clinical studies with granisetron, a new 5-HT3 receptor antagonist for the treatment of cancer chemotherapy-induced emesis. The Granisetron Study Group.
Topics: Adult; Aged; Antiemetics; Antineoplastic Agents; Constipation; Dose-Response Relationship, Drug; Female; Granisetron; Headache; Humans; Indazoles; Male; Middle Aged; Serotonin Antagonists; Vomiting | 1993 |
Litoxetine: a selective 5-HT uptake inhibitor with concomitant 5-HT3 receptor antagonist and antiemetic properties.
Topics: Animals; Antiemetics; Binding, Competitive; Cerebral Cortex; Cisplatin; Dose-Response Relationship, Drug; Ferrets; Fluoxetine; Granisetron; Indazoles; Male; Piperidines; Quipazine; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Vomiting | 1993 |
Repeated use of granisetron in patients receiving cytostatic agents.
Topics: Adult; Age Factors; Aged; Antiemetics; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Cisplatin; Constipation; Female; Granisetron; Headache; Humans; Indazoles; Infusions, Intravenous; Male; Middle Aged; Nausea; Remission Induction; Serotonin Antagonists; Vomiting | 1993 |
[The prevention of CDDP-induced emesis with granisetron].
Topics: Antiemetics; Cisplatin; Female; Granisetron; Humans; Indazoles; Infusions, Intravenous; Nausea; Ovarian Neoplasms; Uterine Neoplasms; Vomiting | 1993 |
[Antiemetic efficacy of granisetron in patients receiving 5-day continuous infusion of cisplatin].
Topics: Adenocarcinoma; Aged; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Carcinoma, Small Cell; Carcinoma, Squamous Cell; Cisplatin; Drug Administration Schedule; Etoposide; Female; Granisetron; Humans; Indazoles; Infusions, Intra-Arterial; Lung Neoplasms; Male; Middle Aged; Nausea; Vindesine; Vomiting | 1993 |
Pharmacokinetics and toxicity of oral and intravenous lonidamine in dogs.
Topics: Administration, Oral; Animals; Antineoplastic Agents; Dogs; Indazoles; Injections, Intravenous; Kinetics; Liver; Male; Testis; Vomiting | 1996 |
Antiemetic effects of N-3389, a newly synthesized 5-HT3 and 5-HT4 receptor antagonist, in ferrets.
Topics: 5-Methoxytryptamine; Animals; Antiemetics; Antineoplastic Agents; Bridged Bicyclo Compounds, Heterocyclic; Cisplatin; Copper Sulfate; Cyclophosphamide; Emetics; Ferrets; Indazoles; Male; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Vagus Nerve; Vomiting | 1997 |
Development of high-affinity 5-HT3 receptor antagonists. 1. Initial structure-activity relationship of novel benzamides.
Topics: Animals; Antiemetics; Benzamides; Benzofurans; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cisplatin; Ferrets; Granisetron; Imidazoles; Indazoles; Indoles; Male; Metoclopramide; Molecular Structure; Ondansetron; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Vomiting | 1992 |
[Nausea and vomiting in chemotherapy].
Topics: Antineoplastic Agents; Clinical Protocols; Granisetron; Humans; Indazoles; Nausea; Vomiting | 1992 |
Dose granisetron remain effective over multiple cycles? The Granisetron Study Group.
Topics: Adult; Aged; Antiemetics; Antineoplastic Agents; Drug Administration Schedule; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Nausea; Serotonin Antagonists; Sex Factors; Vomiting | 1992 |
Are all 5-HT3 receptor antagonists the same?
Topics: Animals; Antiemetics; Cisplatin; Dose-Response Relationship, Drug; Ferrets; Granisetron; Imidazoles; Indazoles; Ondansetron; Serotonin Antagonists; Vomiting; Whole-Body Irradiation | 1992 |
Morphine 6-glucuronide: a metabolite of morphine with greater emetic potency than morphine in the ferret.
Topics: Animals; Cyclophosphamide; Dose-Response Relationship, Drug; Emetics; Ferrets; Granisetron; Imidazoles; Indazoles; Injections, Subcutaneous; Morphine; Morphine Derivatives; Naloxone; Ondansetron; Vomiting | 1992 |
The budgetary impact of 5-HT3 receptor antagonists in the management of chemotherapy-induced emesis.
Topics: Antiemetics; Antineoplastic Agents; Drug Costs; Granisetron; Humans; Indazoles; Models, Theoretical; Nausea; Ondansetron; Serotonin Antagonists; Vomiting | 1992 |
Caring for the cancer patient: managing emesis now. An interactive workshop. Proceedings of a satellite symposium to the 6th European Conference on Clinical Oncology. Florence, October 1991.
Topics: Antiemetics; Antineoplastic Agents; Granisetron; Humans; Indazoles; Nausea; Vomiting | 1992 |
Who should receive a 5-HT3 antagonist?
Topics: Acute Disease; Antineoplastic Agents; Granisetron; Humans; Indazoles; Nausea; Ondansetron; Serotonin Antagonists; Vomiting | 1992 |
5-HT3 receptor antagonist effects of DAT-582, (R) enantiomer of AS-5370.
Topics: Animals; Azepines; Bradycardia; Cisplatin; Ferrets; Guinea Pigs; Ileum; In Vitro Techniques; Indazoles; Male; Muscle Contraction; Muscle, Smooth; Rats; Serotonin Antagonists; Stereoisomerism; Vomiting | 1992 |
Granisetron, a selective 5-HT3 receptor antagonist, for the prevention of radiation induced emesis during total body irradiation.
Topics: Adolescent; Adult; Bone Marrow Transplantation; Female; Granisetron; Humans; Indazoles; Injections, Intravenous; Male; Middle Aged; Serotonin Antagonists; Vomiting; Whole-Body Irradiation | 1991 |
Efficacy and safety of granisetron in the prevention of chemotherapy-induced emesis in paediatric patients.
Topics: Adolescent; Antineoplastic Agents; Child; Child, Preschool; Female; Granisetron; Humans; Indazoles; Male; Nausea; Prognosis; Serotonin Antagonists; Time Factors; Vomiting | 1991 |
Preliminary evidence for the involvement of the putative 5-HT4 receptor in zacopride- and copper sulphate-induced vomiting in the ferret.
Topics: Analysis of Variance; Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Copper; Copper Sulfate; Female; Ferrets; Granisetron; Imidazoles; Indazoles; Indoles; Loperamide; Male; Ondansetron; Receptors, Serotonin; Serotonin Antagonists; Tropisetron; Vomiting | 1991 |
Serotonin antagonists: a new class of antiemetic agents.
Topics: Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Granisetron; Humans; Imidazoles; Indazoles; Indoles; Metoclopramide; Ondansetron; Quinolizines; Receptors, Serotonin; Serotonin Antagonists; Tropanes; Tropisetron; Vomiting | 1991 |
Phase I/II trial of granisetron: a novel 5-hydroxytryptamine antagonist for the prevention of chemotherapy-induced nausea and vomiting.
Topics: Antiemetics; Antineoplastic Agents; Aspartate Aminotransferases; Chromatography, High Pressure Liquid; Cisplatin; Doxorubicin; Drug Evaluation; Drug Tolerance; Granisetron; Humans; Indazoles; Nausea; Pyrazoles; Serotonin Antagonists; Vomiting | 1990 |
Emesis and defecations induced by the 5-hydroxytryptamine (5-HT3) receptor antagonist zacopride in the ferret.
Topics: Administration, Oral; Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Defecation; Dose-Response Relationship, Drug; Ferrets; Granisetron; Indazoles; Injections, Intravenous; Male; Metoclopramide; Pyrazoles; Serotonin; Serotonin Antagonists; Vagotomy; Vomiting | 1990 |
RG 12915: a potent 5-hydroxytryptamine-3 antagonist that is an orally effective inhibitor of cytotoxic drug-induced emesis in the ferret and dog.
Topics: Administration, Oral; Animals; Antiemetics; Antineoplastic Agents; Benzofurans; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cisplatin; Dogs; Dopamine; Ferrets; Gastric Emptying; Granisetron; Imidazoles; Indazoles; Ondansetron; Receptors, Serotonin; Serotonin Antagonists; Vomiting | 1990 |
The symptomatic control of cytostatic drug-induced emesis. A recent history and review.
Topics: Antiemetics; Antineoplastic Agents; Granisetron; Humans; Indazoles; Serotonin Antagonists; Vomiting | 1990 |
An overview on the use of granisetron in the treatment of emesis associated with cytostatic chemotherapy.
Topics: Antineoplastic Agents; Constipation; Granisetron; Headache; Humans; Indazoles; Serotonin Antagonists; Time Factors; Vomiting | 1990 |
The role of specific 5-HT3 receptor antagonism in the control of cytostatic drug-induced emesis.
Topics: Animals; Antineoplastic Agents; Brain; Dose-Response Relationship, Drug; Ferrets; Granisetron; Heart Rate; Indazoles; Male; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Vomiting | 1990 |
The conduct of clinical trials in the area of emesis control.
Topics: Antiemetics; Clinical Trials as Topic; Drug Evaluation; Granisetron; Humans; Indazoles; Oncology Nursing; Vomiting | 1990 |
A phase I study of a new 5HT3-receptor antagonist, BRL43694A, an agent for the prevention of chemotherapy-induced nausea and vomiting.
Topics: Adult; Aged; Antiemetics; Antineoplastic Combined Chemotherapy Protocols; Drug Evaluation; Drug Tolerance; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Nausea; Neoplasms; Pyrazoles; Serotonin Antagonists; Vomiting | 1989 |
BRL 43694, a new 5HT3 receptor antagonist, prevents cisplatin-induced emesis in dogs.
Topics: Animals; Cisplatin; Dogs; Female; Granisetron; Indazoles; Male; Pyrazoles; Serotonin Antagonists; Vomiting | 1989 |
[BRL 43694A--a 5-hydroxytryptamine receptor blocker as an antiemetic in cytostatic therapy].
Topics: Adult; Aged; Antiemetics; Antineoplastic Agents; Drug Evaluation; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Pyrazoles; Serotonin Antagonists; Vomiting | 1989 |
BRL 43694.
Topics: Antineoplastic Agents; Granisetron; Humans; Indazoles; Pyrazoles; Serotonin Antagonists; Vomiting | 1989 |
BRL 43694: a novel antiemetic to prevent nausea and vomiting induced by chemotherapy.
Topics: Adult; Aged; Antiemetics; Antineoplastic Agents; Female; Granisetron; Humans; Indazoles; Male; Middle Aged; Nausea; Pyrazoles; Vomiting | 1988 |
The anti-emetic potential of the 5-hydroxytryptamine3 receptor antagonist BRL 43694.
Topics: Animals; Apomorphine; Cisplatin; Cyclophosphamide; Dogs; Doxorubicin; Ferrets; Granisetron; Indazoles; Male; Pyrazoles; Triazines; Vomiting; Whole-Body Irradiation | 1988 |
Pharmacokinetics and anti-emetic efficacy of BRL43694, a new selective 5HT-3 antagonist.
Topics: Adolescent; Adult; Aged; Antineoplastic Agents; Drug Tolerance; Female; Granisetron; Half-Life; Humans; Indazoles; Male; Middle Aged; Pilot Projects; Pyrazoles; Vomiting | 1988 |