Page last updated: 2024-08-17

carbostyril and HIV

carbostyril has been researched along with HIV in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (3.70)18.2507
2000's8 (29.63)29.6817
2010's17 (62.96)24.3611
2020's1 (3.70)2.80

Authors

AuthorsStudies
Ma, R; Tong, ZW; Xu, B; Zhang, Q; Zhang, YS; Zhao, CS; Zhao, RG1
Clark, MR; Deng, Y; Mohideen, M; Panse, G; Quijano, E; Saltzman, WM; Song, E; Zhang, W1
Chauhan, M; Chokkar, N; Kalra, S; Kumar, R1
Cassetti, I; Castillo, S; Cecchini, DM; Copertari, G; Lacal, V; Rodriguez, CG1
Ambrosioni, J; de Lazzari, E; García, F; Marcos, MÁ; Miró, JM; Mosquera, MM; Nicolás, D; Rico, JÁF1
Ayala-Sims, VA; Fulco, PP1
Debyser, Z; Schrijvers, R1
Arribas, JR; Di Perri, G; Ebrahimi, R; Gathe, J; Nguyen, T; Pialoux, G; Piontkowsky, D; Reynes, J; Tebas, P; White, K1
Antela, A; Domingo, P; Garner, W; Girard, PM; Guyer, B; Henry, K; Markowitz, M; Mills, A; Nguyen, T; Piontkowsky, D; Pozniak, A; Stellbrink, HJ; White, K1
Barreca, ML; Cecchetti, V; Corazza, G; Daelemans, D; Iraci, N; Manfroni, G; Marcello, A; Massari, S; Pannecouque, C; Sancineto, L; Tabarrini, O1
Grobler, JA; Hazuda, DJ1
Castagna, A; Chiappetta, S; Galli, L; Lazzarin, A; Nozza, S; Poli, A; Ripa, M; Rovelli, C; Spagnuolo, V; Tambussi, G1
Chen, FE; Chen, WX; Daelemans, D; De Clercq, E; He, QQ; Mao, TQ; Pannecouque, C; Tang, GF1
Hazuda, D; Iwamoto, M; Wenning, L1
Grant, P; Zolopa, A1
Cecchetti, V; Daelemans, D; Manfroni, G; Massari, S; Pannecouque, C; Sabatini, S; Tabarrini, O1
Christ, F; Debyser, Z; McNeely, M; Thys, W1
de Mendoza, C; Garrido, C; Soriano, V1
Cardona, C; Cauvin, C; Georges, B; Guiguen, A; Hevesi, L; Le Van, K; Mbemba, G; Michaux, C; Mouscadet, JF; Van Lint, C; Vandurm, P; Wouters, J1
Cecchetti, V; Ianni, F; Massari, S; Natalini, B; Sardella, R; Tabarrini, O1
Breeze, S1
Hutadilok-Towatana, N; Panthong, K; Rukachaisirikul, V; Srisud, Y; Tewtrakul, S; Voravuthikunchai, SP1
Bastow, KF; Chen, Y; Lee, KH; Morris-Natschke, SL; Xia, P; Xia, Y; Yang, ZY; Zhang, Q; Zheng, YQ1
Maurin, MB; Xie, M; Ziemba, TM1
Bringmann, G; Cai, P; Feineis, D; Heguy, A; Houck, D; Katz, B; Meyn, P; Michitsch, R; Pearce, C; Russo, S; Taylor, DL; Tyms, AS1
Cecchetti, V; Cruciani, G; Filipponi, E; Fravolini, A; Tabarrini, O1

Reviews

6 review(s) available for carbostyril and HIV

ArticleYear
A Review on Quinoline Derived Scaffolds as Anti-HIV Agents.
    Mini reviews in medicinal chemistry, 2019, Volume: 19, Issue:6

    Topics: Animals; Anti-HIV Agents; Drug Discovery; HIV; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; Humans; Models, Molecular; Quinolones

2019
Resistance to HIV integrase strand transfer inhibitors: in vitro findings and clinical consequences.
    Current opinion in virology, 2014, Volume: 8

    Topics: Drug Resistance, Viral; Heterocyclic Compounds, 3-Ring; HIV; HIV Integrase; HIV Integrase Inhibitors; Humans; Mutation, Missense; Oxazines; Piperazines; Pyridones; Pyrrolidinones; Quinolones; Raltegravir Potassium; Virulence; Virus Replication

2014
Emerging pharmacology: inhibitors of human immunodeficiency virus integration.
    Annual review of pharmacology and toxicology, 2009, Volume: 49

    Topics: Animals; HIV; HIV Integrase Inhibitors; Humans; Models, Theoretical; Molecular Structure; Pharmacology, Clinical; Pyrrolidinones; Quinolones; Raltegravir Potassium; Virus Integration

2009
Integrase inhibitors: a clinical review of raltegravir and elvitegravir.
    Journal of HIV therapy, 2008, Volume: 13, Issue:2

    Topics: Clinical Trials, Phase III as Topic; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance, Viral; Drug Therapy, Combination; HIV; HIV Infections; HIV Integrase; HIV Protease Inhibitors; Humans; Pyrrolidinones; Quinolones; Raltegravir Potassium

2008
Targeting the HIV integration process in antiviral therapy.
    Journal of HIV therapy, 2008, Volume: 13, Issue:4

    Topics: HIV; HIV Infections; HIV Integrase Inhibitors; Humans; Pyrrolidinones; Quinolones; Raltegravir Potassium; Virus Integration

2008
[Resistance to integrase inhibitors].
    Enfermedades infecciosas y microbiologia clinica, 2008, Volume: 26 Suppl 12

    Topics: Amino Acid Substitution; Clinical Trials as Topic; Drug Resistance, Multiple, Viral; Drug Resistance, Viral; Genetic Variation; HIV; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; Humans; Models, Molecular; Mutation, Missense; Point Mutation; Protein Conformation; Pyrrolidinones; Quinolones; Raltegravir Potassium

2008

Trials

2 trial(s) available for carbostyril and HIV

ArticleYear
Simplification to coformulated elvitegravir, cobicistat, emtricitabine, and tenofovir versus continuation of ritonavir-boosted protease inhibitor with emtricitabine and tenofovir in adults with virologically suppressed HIV (STRATEGY-PI): 48 week results o
    The Lancet. Infectious diseases, 2014, Volume: 14, Issue:7

    Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Drug Therapy, Combination; Emtricitabine; Female; HIV; HIV Infections; Humans; Male; Middle Aged; Organophosphonates; Protease Inhibitors; Quinolones; Ritonavir; Tenofovir; Thiazoles; Viral Load

2014
Switching to coformulated elvitegravir, cobicistat, emtricitabine, and tenofovir versus continuation of non-nucleoside reverse transcriptase inhibitor with emtricitabine and tenofovir in virologically suppressed adults with HIV (STRATEGY-NNRTI): 48 week r
    The Lancet. Infectious diseases, 2014, Volume: 14, Issue:7

    Topics: Adenine; Adult; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Emtricitabine; Female; HIV; HIV Infections; Humans; Male; Middle Aged; Organophosphonates; Quinolones; Reverse Transcriptase Inhibitors; Tenofovir; Thiazoles; Viral Load

2014

Other Studies

19 other study(ies) available for carbostyril and HIV

ArticleYear
Preoperative rapid suppression of viral load by elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide regimen in human immunodeficiency virus-positive fracture patients significantly reduces postoperative complications.
    Chinese medical journal, 2020, Dec-05, Volume: 133, Issue:23

    Topics: Adenine; Alanine; Anti-HIV Agents; Cobicistat; Drug Combinations; Emtricitabine; HIV; HIV Infections; Humans; Postoperative Complications; Quinolones; Tenofovir; Viral Load

2020
Degradable bioadhesive nanoparticles for prolonged intravaginal delivery and retention of elvitegravir.
    Biomaterials, 2017, Volume: 144

    Topics: Administration, Intravaginal; Animals; Anti-HIV Agents; Delayed-Action Preparations; Female; HIV; HIV Infections; Humans; Mice, Inbred C57BL; Nanoparticles; Quinolones; Vagina

2017
Resistance to HIV integrase strand transfer inhibitors in Argentina: first interim survey.
    Revista espanola de quimioterapia : publicacion oficial de la Sociedad Espanola de Quimioterapia, 2019, Volume: 32, Issue:3

    Topics: Adult; Argentina; Drug Resistance, Viral; Female; Heterocyclic Compounds, 3-Ring; HIV; HIV Infections; HIV Integrase Inhibitors; Humans; Male; Middle Aged; Oxazines; Pilot Projects; Piperazines; Prevalence; Pyridones; Quinolones; Raltegravir Potassium; Retrospective Studies; Surveys and Questionnaires; Urban Population; Viral Load; Young Adult

2019
E157Q integrase strand-transfer inhibitor substitution in patients with acute/recent HIV infection.
    AIDS (London, England), 2019, 08-01, Volume: 33, Issue:10

    Topics: Adult; Amino Acid Substitution; Disease Transmission, Infectious; Drug Resistance, Viral; Female; Gene Frequency; Genotype; Genotyping Techniques; High-Throughput Nucleotide Sequencing; HIV; HIV Infections; HIV Integrase; HIV Integrase Inhibitors; Humans; Male; Molecular Epidemiology; Mutation, Missense; Phylogeny; Prevalence; Prospective Studies; Quinolones; Raltegravir Potassium; Sexual and Gender Minorities; Viral Load

2019
Sustained virological response after taking crushed elvitegravir-cobicistat-emtricitabine-tenofovir tablets.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 2014, May-15, Volume: 71, Issue:10

    Topics: Adenine; Adult; Antiretroviral Therapy, Highly Active; Carbamates; Cobicistat; Deoxycytidine; Emtricitabine; Female; HIV; HIV Infections; Humans; Organophosphonates; Powders; Quinolones; Tablets; Tenofovir; Thiazoles; Viral Load

2014
Switching STRATEGIES in HIV treatment.
    The Lancet. Infectious diseases, 2014, Volume: 14, Issue:7

    Topics: Adenine; Anti-HIV Agents; Carbamates; Cobicistat; Deoxycytidine; Emtricitabine; Female; HIV; HIV Infections; Humans; Male; Organophosphonates; Protease Inhibitors; Quinolones; Reverse Transcriptase Inhibitors; Ritonavir; Tenofovir; Thiazoles

2014
Exploiting the anti-HIV 6-desfluoroquinolones to design multiple ligands.
    Bioorganic & medicinal chemistry, 2014, Sep-01, Volume: 22, Issue:17

    Topics: Anti-HIV Agents; Cell Line; Dose-Response Relationship, Drug; HIV; Humans; Ligands; Microbial Sensitivity Tests; Models, Molecular; Molecular Structure; Quinolones; Structure-Activity Relationship; Virus Replication

2014
Efficacy of elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate as treatment for primary or recent HIV infection.
    The Journal of antimicrobial chemotherapy, 2017, Volume: 72, Issue:2

    Topics: Adult; Anti-HIV Agents; CD4 Lymphocyte Count; Cobicistat; Emtricitabine; HIV; HIV Infections; Humans; Male; Middle Aged; Quinolones; Retrospective Studies; Tenofovir; Treatment Outcome; Viral Load

2017
Structural Modifications of Diarylpyrimidine-quinolone Hybrids as Potent HIV-1 NNRTIs with an Improved Drug Resistance Profile.
    Current pharmaceutical design, 2016, Volume: 22, Issue:46

    Topics: Anti-HIV Agents; Cell Line, Tumor; Dose-Response Relationship, Drug; Drug Resistance, Viral; HIV; HIV Reverse Transcriptase; Humans; Microbial Sensitivity Tests; Models, Molecular; Molecular Structure; Pyrimidines; Quinolones; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Virus Replication

2016
Studies on anti-HIV quinolones: new insights on the C-6 position.
    Bioorganic & medicinal chemistry, 2009, Jan-15, Volume: 17, Issue:2

    Topics: Anti-HIV Agents; HIV; Humans; Quinolones; Structure-Activity Relationship; Transcription, Genetic; Virus Replication

2009
Synthesis, biological evaluation and molecular modeling studies of quinolonyl diketo acid derivatives: new structural insight into the HIV-1 integrase inhibition.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:5

    Topics: Anti-HIV Agents; Catalytic Domain; Dose-Response Relationship, Drug; Drug Design; HIV; HIV Integrase; HIV Integrase Inhibitors; Keto Acids; Models, Molecular; Molecular Structure; Quinolones; Stereoisomerism; Structure-Activity Relationship

2011
Synthesis and chromatographic enantioresolution of anti-HIV quinolone derivatives.
    Talanta, 2011, Sep-15, Volume: 85, Issue:3

    Topics: Acetic Acid; Amylose; Anti-HIV Agents; Cellulose; Chloroform; Chromatography, High Pressure Liquid; Ethanol; HIV; Humans; Mesylates; Methanol; Models, Chemical; Molecular Structure; Phenylcarbamates; Quinolones; Stereoisomerism; Trifluoroacetic Acid

2011
A 4-drug combination (Stribild) for HIV.
    The Medical letter on drugs and therapeutics, 2012, Nov-26, Volume: 54, Issue:1404

    Topics: Adenine; Anti-HIV Agents; Carbamates; Clinical Trials as Topic; Cobicistat; Deoxycytidine; Double-Blind Method; Drug Approval; Drug Combinations; Drug Interactions; Drug Resistance, Multiple, Viral; Emtricitabine; HIV; HIV Infections; Humans; Organophosphonates; Quinolones; Randomized Controlled Trials as Topic; Tenofovir; Thiazoles; United States; United States Food and Drug Administration

2012
Novel HIV-1 treatment Stribild™ gains regulatory approval.
    Expert review of clinical pharmacology, 2012, Volume: 5, Issue:6

    Topics: Adenine; Anti-HIV Agents; Carbamates; Deoxycytidine; Drug Approval; Drug Combinations; Elvitegravir, Cobicistat, Emtricitabine, Tenofovir Disoproxil Fumarate Drug Combination; HIV; HIV Infections; Humans; Organophosphonates; Quinolones; Thiazoles

2012
Benzene, coumarin and quinolinone derivatives from roots of Citrus hystrix.
    Phytochemistry, 2013, Volume: 88

    Topics: Anti-Bacterial Agents; Anti-HIV Agents; Antioxidants; Bacteria; Benzene; Cells, Cultured; Citrus; Coumarins; HIV; Humans; Magnetic Resonance Spectroscopy; Molecular Structure; Plant Roots; Quinolones

2013
Synthesis and bioactivity of 4,10-dimethyl-pyridino[2,3-h]quinolin-2(1H)-one-9-carboxylic acid and its esters.
    Bioorganic & medicinal chemistry, 2003, Mar-20, Volume: 11, Issue:6

    Topics: Anti-HIV Agents; Antineoplastic Agents; Cell Survival; Drug Evaluation, Preclinical; Drug Screening Assays, Antitumor; HIV; Humans; Indicators and Reagents; Magnetic Resonance Spectroscopy; Quinolones; Tumor Cells, Cultured

2003
Sublimation characterization and vapor pressure estimation of an HIV nonnucleoside reverse transcriptase inhibitor using thermogravimetric analysis.
    AAPS PharmSciTech, 2003, Volume: 4, Issue:2

    Topics: Chemical Phenomena; Chemistry, Pharmaceutical; Chemistry, Physical; HIV; Quinolones; Reverse Transcriptase Inhibitors; Technology, Pharmaceutical; Thermodynamics; Thermogravimetry; Volatilization

2003
Isolation and characterization of the fungal metabolite 3-O-methylviridicatin as an inhibitor of tumour necrosis factor alpha-induced human immunodeficiency virus replication.
    Antiviral chemistry & chemotherapy, 1998, Volume: 9, Issue:2

    Topics: Anti-HIV Agents; Fungi; HeLa Cells; HIV; HIV Long Terminal Repeat; Humans; Hydroxyquinolines; Microbial Sensitivity Tests; Quinolones; Tumor Necrosis Factor-alpha; Virus Replication

1998
QSAR study and VolSurf characterization of anti-HIV quinolone library.
    Journal of computer-aided molecular design, 2001, Volume: 15, Issue:3

    Topics: Anti-HIV Agents; Computer-Aided Design; Databases, Factual; Drug Design; HIV; HIV Infections; Humans; Models, Chemical; Multivariate Analysis; Quantitative Structure-Activity Relationship; Quinolones; Software

2001