Page last updated: 2024-09-05

zm 241385 and psb603

zm 241385 has been researched along with psb603 in 6 studies

Compound Research Comparison

Studies
(zm 241385)
Trials
(zm 241385)
Recent Studies (post-2010)
(zm 241385)
Studies
(psb603)
Trials
(psb603)
Recent Studies (post-2010) (psb603)
401312414013

Protein Interaction Comparison

ProteinTaxonomyzm 241385 (IC50)psb603 (IC50)
Adenosine receptor A1Rattus norvegicus (Norway rat)0.0005
Adenosine receptor A3Rattus norvegicus (Norway rat)0.0007
Adenosine receptor A2bHomo sapiens (human)0.0052

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (66.67)24.3611
2020's2 (33.33)2.80

Authors

AuthorsStudies
French, SW; Khachatoorian, R; Micewicz, ED; Ruchala, P1
Behrenswerth, A; Fiene, A; Gollos, S; Heisig, F; Karcz, T; Kieć-Kononowicz, K; Köse, M; Müller, CE; Namasivayam, V1
Alispahic, B; Åqvist, J; Azuaje, J; Brea, J; Caamaño, O; Crespo, A; El Maatougui, A; Fernandez-Masaguer, C; Freire-Garabal, M; García-Mera, X; Garcia-Santiago, C; Gioé, C; Gutiérrez-de-Terán, H; Jespers, W; Loza, MI; Majellaro, M; Mallo-Abreu, A; Novio, S; Núñez, MJ; Prieto-Díaz, R; Rodríguez-García, C; Sardina, JF; Sotelo, E; Stefanachi, A1
Gaba, S; Gupta, GD; Monga, V; Patel, R; Saini, A; Singh, G1
Christopoulos, A; Gregory, KJ; May, LT; Tan, CY; Vecchio, EA; White, PJ1
Adam, RM; Chung, YG; Cristofaro, V; Doyle, C; Lukianov, SN; Sack, BS; Schäfer, M; Sullivan, MP1

Reviews

1 review(s) available for zm 241385 and psb603

ArticleYear
Adenosine receptor antagonists: Recent advances and therapeutic perspective.
    European journal of medicinal chemistry, 2022, Jan-05, Volume: 227

    Topics: Dose-Response Relationship, Drug; Humans; Molecular Structure; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Structure-Activity Relationship

2022

Other Studies

5 other study(ies) available for zm 241385 and psb603

ArticleYear
Identification of novel small-molecule inhibitors of Zika virus infection.
    Bioorganic & medicinal chemistry letters, 2018, 02-01, Volume: 28, Issue:3

    Topics: A549 Cells; Antiviral Agents; Cell Survival; Dose-Response Relationship, Drug; Humans; Molecular Structure; Small Molecule Libraries; Structure-Activity Relationship; Zika Virus; Zika Virus Infection

2018
Fluorescent-Labeled Selective Adenosine A
    Journal of medicinal chemistry, 2018, 05-24, Volume: 61, Issue:10

    Topics: Adenosine A2 Receptor Antagonists; Animals; Binding, Competitive; Cell Proliferation; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Flow Cytometry; Fluorescent Dyes; Humans; Mice; Models, Molecular; Molecular Structure; Protein Binding; Protein Conformation; Radioligand Assay; Rats; Receptor, Adenosine A2B

2018
3,4-Dihydropyrimidin-2(1
    Journal of medicinal chemistry, 2021, 01-14, Volume: 64, Issue:1

    Topics: Adenosine A2 Receptor Antagonists; Animals; CHO Cells; Cricetulus; Cyclic AMP; HEK293 Cells; HeLa Cells; Humans; Models, Molecular; Neoplasm Metastasis; Pyrimidines; Radioligand Assay; Receptor, Adenosine A2B; Stereoisomerism; Structure-Activity Relationship

2021
Ligand-Independent Adenosine A2B Receptor Constitutive Activity as a Promoter of Prostate Cancer Cell Proliferation.
    The Journal of pharmacology and experimental therapeutics, 2016, Volume: 357, Issue:1

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine Deaminase; Animals; Cell Line, Tumor; Cell Proliferation; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Drug Design; Humans; Inositol Phosphates; Ligands; Male; MAP Kinase Signaling System; Prostatic Neoplasms; Receptor, Adenosine A2B; Signal Transduction; Sulfonamides; Triazines; Triazoles; Xanthines

2016
Inosine attenuates spontaneous activity in the rat neurogenic bladder through an A
    Scientific reports, 2017, 03-15, Volume: 7

    Topics: Adenosine A2 Receptor Antagonists; Animals; Disease Models, Animal; Humans; Inosine; Potassium Channels; Rats; Receptor, Adenosine A2A; Spinal Cord Injuries; Sulfonamides; Triazines; Triazoles; Urinary Bladder, Neurogenic; Urinary Bladder, Overactive; Xanthines

2017