Page last updated: 2024-09-04

ym 09151-2 and mazindol

ym 09151-2 has been researched along with mazindol in 8 studies

Compound Research Comparison

Studies
(ym 09151-2)
Trials
(ym 09151-2)
Recent Studies (post-2010)
(ym 09151-2)
Studies
(mazindol)
Trials
(mazindol)
Recent Studies (post-2010) (mazindol)
2496136317331

Protein Interaction Comparison

ProteinTaxonomyym 09151-2 (IC50)mazindol (IC50)
Sodium-dependent noradrenaline transporter Homo sapiens (human)0.0029
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)0.0454
Sodium-dependent serotonin transporterHomo sapiens (human)0.074
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.231
Sodium-dependent dopamine transporter Homo sapiens (human)0.0275
Sodium-dependent dopamine transporterMus musculus (house mouse)0.013
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.2344

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (62.50)18.2507
2000's3 (37.50)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Boja, JW; Carroll, FI; Kuhar, MJ; Lewin, AH; Philip, A; Rahman, MA1
Arregui, A; Hollingsworth, Z; Penney, JB; Young, AB1
Araki, T; Fujiwara, T; Itoyama, Y; Kato, H; Kogure, K; Shuto, K1
Araki, T; Fujiwara, T; Itoyama, Y; Kato, H; Shuto, K1
Araki, T; Itoyama, Y; Kato, H; Tanji, H1
Augood, SJ; Emson, PC; Hollingsworth, ZR; Penney, JB; Standaert, DG1
Albers, DS; Augood, SJ; Breakefield, XO; Hollingsworth, Z; Leung, J; Standaert, DG; Yang, L1
Charlton, CG; Chen, H; Lamango, NS; Lee, ES; Shepherd, KR; Soliman, KF1

Other Studies

8 other study(ies) available for ym 09151-2 and mazindol

ArticleYear
Isothiocyanate derivatives of cocaine: irreversible inhibition of ligand binding at the dopamine transporter.
    Molecular pharmacology, 1991, Volume: 39, Issue:3

    Topics: Animals; Benzamides; Binding, Competitive; Brain Stem; Carrier Proteins; Cerebral Cortex; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Ligands; Male; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Paroxetine; Phencyclidine; Piperidines; Rats; Rats, Inbred Strains; Thiocyanates

1991
Autoradiographic evidence for increased dopamine uptake sites in striatum of hypoxic mice.
    Neuroscience letters, 1994, Feb-14, Volume: 167, Issue:1-2

    Topics: Animals; Autoradiography; Benzamides; Benzazepines; Binding Sites; Corpus Striatum; Desipramine; Dopamine; Dopamine D2 Receptor Antagonists; Hypoxia; Male; Mazindol; Mice; Mice, Inbred BALB C; Receptors, Dopamine D1; Receptors, Dopamine D2; Time Factors

1994
Effects of cerebral ischemia on dopamine receptors in the gerbil striatum.
    European journal of pharmacology, 1996, Jun-13, Volume: 306, Issue:1-3

    Topics: Animals; Benzamides; Benzazepines; Brain Ischemia; Cerebral Cortex; Corpus Striatum; Dopamine Antagonists; Dopamine Uptake Inhibitors; Gerbillinae; Male; Mazindol; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone

1996
Effect of aging on dopaminergic receptors and uptake sites in the rat brain studied by receptor autoradiography.
    Journal of the neurological sciences, 1997, May-29, Volume: 148, Issue:2

    Topics: Aging; Animals; Autoradiography; Benzamides; Benzazepines; Brain Chemistry; Dopamine Antagonists; Dopamine Uptake Inhibitors; Male; Mazindol; Rats; Rats, Inbred F344; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Tritium

1997
Sequential changes of dopaminergic receptors in the rat brain after 6-hydroxydopamine lesions of the medial forebrain bundle.
    Journal of the neurological sciences, 1998, Oct-08, Volume: 160, Issue:2

    Topics: Adrenergic Agents; Animals; Autoradiography; Benzamides; Benzazepines; Brain Diseases; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Male; Mazindol; Medial Forebrain Bundle; Oxidopamine; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Time Factors

1998
Localization of dopaminergic markers in the human subthalamic nucleus.
    The Journal of comparative neurology, 2000, May-29, Volume: 421, Issue:2

    Topics: Benzamides; Benzazepines; Biomarkers; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Humans; Mazindol; Parkinson Disease; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Subthalamic Nucleus; Tyrosine 3-Monooxygenase

2000
Dopamine transmission in DYT1 dystonia.
    Advances in neurology, 2004, Volume: 94

    Topics: 3,4-Dihydroxyphenylacetic Acid; Autoradiography; Basal Ganglia; Benzamides; Benzazepines; Binding Sites; Carrier Proteins; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dystonia; Family Health; Homovanillic Acid; Humans; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Chaperones; Neuropeptides; Synaptic Transmission; Tetrabenazine; Tritium; Vesicular Biogenic Amine Transport Proteins

2004
The inhibitory role of methylation on the binding characteristics of dopamine receptors and transporter.
    Neuroscience research, 2004, Volume: 48, Issue:3

    Topics: Analysis of Variance; Animals; Benzamides; Benzazepines; Binding, Competitive; Brain; Brain Chemistry; Dizocilpine Maleate; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Injections, Intraventricular; Male; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Methylation; Nerve Tissue Proteins; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; S-Adenosylmethionine; Tissue Distribution; Tritium

2004