Page last updated: 2024-09-03

way 100135 and colforsin

way 100135 has been researched along with colforsin in 5 studies

Compound Research Comparison

Studies
(way 100135)
Trials
(way 100135)
Recent Studies (post-2010)
(way 100135)
Studies
(colforsin)
Trials
(colforsin)
Recent Studies (post-2010) (colforsin)
14303413,460461,298

Protein Interaction Comparison

ProteinTaxonomyway 100135 (IC50)colforsin (IC50)
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)1.729
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.041
Adenylate cyclase type 1Homo sapiens (human)0.0955

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (40.00)18.2507
2000's3 (60.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cadogan, AK; Kendall, DA; Marsden, CA1
Lima, L; Schmeer, C; Urbina, M1
AssiƩ, MB; Colpaert, FC; Cosi, C; Koek, W; Patoiseau, JF; Pauwels, PJ; Vacher, B1
Borsini, F; Cassano, GB; Giromella, A; Lucacchini, A; Marazziti, D; Mayer, N; Mazzoni, MR; Naccarato, AG; Palego, L1
Carreira, I; Lima, L; Mizrahi, C; Stojanovic, A; Urbina, M1

Other Studies

5 other study(ies) available for way 100135 and colforsin

ArticleYear
Serotonin 5-HT1A receptor activation increases cyclic AMP formation in the rat hippocampus in vivo.
    Journal of neurochemistry, 1994, Volume: 62, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Colforsin; Cyclic AMP; Hippocampus; Kinetics; Male; Microdialysis; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Time Factors

1994
5HT1A receptor agonist differentially increases cyclic AMP concentration in intact and lesioned goldfish retina. In vitro inhibition of outgrowth by forskolin.
    Neurochemistry international, 1996, Volume: 29, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Dopamine Antagonists; Goldfish; Nerve Crush; Nerve Regeneration; Optic Nerve; Piperazines; Retina; Serotonin Antagonists; Serotonin Receptor Agonists

1996
5-HT1A receptor activation and antidepressant-like effects: F 13714 has high efficacy and marked antidepressant potential.
    European journal of pharmacology, 2001, May-25, Volume: 420, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminopyridines; Animals; Antidepressive Agents; Binding, Competitive; Buspirone; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); HeLa Cells; Humans; Male; Motor Activity; Piperazines; Piperidines; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming

2001
Region-dependent effects of flibanserin and buspirone on adenylyl cyclase activity in the human brain.
    The international journal of neuropsychopharmacology, 2002, Volume: 5, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Aged; Aged, 80 and over; Benzimidazoles; Binding, Competitive; Brain; Buspirone; Colforsin; Dose-Response Relationship, Drug; Female; Hippocampus; Humans; Male; Middle Aged; Piperazines; Prefrontal Cortex; Raphe Nuclei; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2002
Differential cAMP levels and serotonin effects in blood peripheral mononuclear cells and lymphocytes from major depression patients.
    International immunopharmacology, 2004, Volume: 4, Issue:8

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adult; Colforsin; Cyclic AMP; Depressive Disorder, Major; Female; Humans; In Vitro Techniques; Leukocytes, Mononuclear; Lymphocytes; Male; Middle Aged; Norepinephrine; Piperazines; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists

2004