u 101958 has been researched along with piperidines in 9 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 8 (88.89) | 18.2507 |
2000's | 1 (11.11) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Dinh, DM; Duncan, JN; Lajiness, ME; Lawson, CF; Poel, TJ; Rees, SA; Romero, AG; Schlachter, SK; Smith, MW | 1 |
Bakthavachalam, V; Baldessarini, RJ; Kebabian, JW; Kula, NS; Xu, L | 1 |
Hsu, SF; Jackson, MB; Wilke, RA | 1 |
Bobirnac, I; Bruinvels, AT; Danzeisen, M; Gazi, L; Geisse, S; Hoyer, D; Schoeffter, P; Schüpbach, E; Sommer, B; Tricklebank, M | 1 |
Bakthavachalam, V; Baldessarini, RJ; Kula, NS; Pounds, S; Tarazi, FI; True, CD; Xu, L | 1 |
Helmeste, DM; Mitsuhashi, M; Shioiri, T; Tang, SW | 1 |
Chari, S; Deth, RC; DuRand, CJ; Kotb, M; Kramer, ML; Liu, D; Nagata, M; Ouellette, D; Sharma, A; Shim, S; Tan, W; Wick, PF | 1 |
Bobirnac, I; Danzeisen, M; Gazi, L; Hoyer, D; Langenegger, D; Schoeffter, P; Schüpbach, E; Sommer, B; Tricklebank, M | 1 |
De La Garza, R; Madras, BK | 1 |
9 other study(ies) available for u 101958 and piperidines
Article | Year |
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Substituted 4-aminopiperidines having high in vitro affinity and selectivity for the cloned human dopamine D4 receptor.
Topics: Aminopyridines; Animals; CHO Cells; Cricetinae; Humans; Mitosis; Piperidines; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Signal Transduction | 1997 |
RBI-257: a highly potent dopamine D4 receptor-selective ligand.
Topics: Aminopyridines; Animals; Brain Chemistry; Cricetinae; Dopamine Agents; Guinea Pigs; Humans; In Vitro Techniques; Isomerism; Ligands; Membranes; Piperidines; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Dopamine D4 | 1997 |
Dopamine D4 receptor mediated inhibition of potassium current in neurohypophysial nerve terminals.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aminopyridines; Animals; Dopamine Agonists; Dopamine Antagonists; Electric Conductivity; Female; Kinetics; Male; Membrane Potentials; Nerve Endings; Patch-Clamp Techniques; Phenethylamines; Piperidines; Pituitary Gland, Posterior; Potassium; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4; Salicylamides | 1998 |
The agonist activities of the putative antipsychotic agents, L-745,870 and U-101958 in HEK293 cells expressing the human dopamine D4.4 receptor.
Topics: Aminopyridines; Antipsychotic Agents; Cell Line; Clozapine; Colforsin; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Humans; Kidney; Piperidines; Pyridines; Pyrroles; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone | 1998 |
Neuropharmacological assessment of potential dopamine D4 receptor-selective radioligands.
Topics: Aminopyridines; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Dopamine Agents; Dopamine Antagonists; Haloperidol; Humans; In Vitro Techniques; Ligands; Male; Piperidines; Prosencephalon; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4; Spiperone; Tritium | 1999 |
Binding of [3H]U-101958 to sigma1 receptor-like sites in human cerebellum and neuroblastoma cells.
Topics: Aminopyridines; Binding, Competitive; Cerebellum; Culture Techniques; Dopamine Agents; Humans; Neuroblastoma; Piperidines; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, sigma; Reverse Transcriptase Polymerase Chain Reaction; Sigma-1 Receptor | 1999 |
D4 dopamine receptor-mediated phospholipid methylation and its implications for mental illnesses such as schizophrenia.
Topics: Amino Acid Sequence; Aminopyridines; Animals; Benzazepines; Binding Sites; Carbon Radioisotopes; CHO Cells; Clozapine; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Formates; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Methionine; Mutagenesis, Site-Directed; Neuroblastoma; Phospholipids; Phosphorylation; Piperidines; Psychotic Disorders; Pyridines; Pyrroles; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; S-Adenosylmethionine; Salicylamides; Schizophrenia; Transfection; Tumor Cells, Cultured | 1999 |
Receptor density as a factor governing the efficacy of the dopamine D4 receptor ligands, L-745,870 and U-101958 at human recombinant D4.4 receptors expressed in CHO cells.
Topics: Aminopyridines; Animals; Butyrates; CHO Cells; Cricetinae; Cyclic AMP; Dopamine Agents; Humans; Ligands; Piperidines; Pyridines; Pyrroles; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Spiperone | 1999 |
[(3)H]PNU-101958, a D(4) dopamine receptor probe, accumulates in prefrontal cortex and hippocampus of non-human primate brain.
Topics: Aminopyridines; Animals; Autoradiography; Brain; Hippocampus; Macaca mulatta; Molecular Probes; Piperidines; Prefrontal Cortex; Pyridines; Pyrroles; Receptors, Dopamine D2; Receptors, Dopamine D4; Tissue Distribution; Tritium | 2000 |