Compounds > u 101958
Page last updated: 2024-08-16

u 101958 and piperidines

u 101958 has been researched along with piperidines in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (88.89)18.2507
2000's1 (11.11)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dinh, DM; Duncan, JN; Lajiness, ME; Lawson, CF; Poel, TJ; Rees, SA; Romero, AG; Schlachter, SK; Smith, MW1
Bakthavachalam, V; Baldessarini, RJ; Kebabian, JW; Kula, NS; Xu, L1
Hsu, SF; Jackson, MB; Wilke, RA1
Bobirnac, I; Bruinvels, AT; Danzeisen, M; Gazi, L; Geisse, S; Hoyer, D; Schoeffter, P; Schüpbach, E; Sommer, B; Tricklebank, M1
Bakthavachalam, V; Baldessarini, RJ; Kula, NS; Pounds, S; Tarazi, FI; True, CD; Xu, L1
Helmeste, DM; Mitsuhashi, M; Shioiri, T; Tang, SW1
Chari, S; Deth, RC; DuRand, CJ; Kotb, M; Kramer, ML; Liu, D; Nagata, M; Ouellette, D; Sharma, A; Shim, S; Tan, W; Wick, PF1
Bobirnac, I; Danzeisen, M; Gazi, L; Hoyer, D; Langenegger, D; Schoeffter, P; Schüpbach, E; Sommer, B; Tricklebank, M1
De La Garza, R; Madras, BK1

Other Studies

9 other study(ies) available for u 101958 and piperidines

ArticleYear
Substituted 4-aminopiperidines having high in vitro affinity and selectivity for the cloned human dopamine D4 receptor.
    European journal of pharmacology, 1997, Mar-19, Volume: 322, Issue:2-3

    Topics: Aminopyridines; Animals; CHO Cells; Cricetinae; Humans; Mitosis; Piperidines; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Signal Transduction

1997
RBI-257: a highly potent dopamine D4 receptor-selective ligand.
    European journal of pharmacology, 1997, Jul-23, Volume: 331, Issue:2-3

    Topics: Aminopyridines; Animals; Brain Chemistry; Cricetinae; Dopamine Agents; Guinea Pigs; Humans; In Vitro Techniques; Isomerism; Ligands; Membranes; Piperidines; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Dopamine D4

1997
Dopamine D4 receptor mediated inhibition of potassium current in neurohypophysial nerve terminals.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Aminopyridines; Animals; Dopamine Agonists; Dopamine Antagonists; Electric Conductivity; Female; Kinetics; Male; Membrane Potentials; Nerve Endings; Patch-Clamp Techniques; Phenethylamines; Piperidines; Pituitary Gland, Posterior; Potassium; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4; Salicylamides

1998
The agonist activities of the putative antipsychotic agents, L-745,870 and U-101958 in HEK293 cells expressing the human dopamine D4.4 receptor.
    British journal of pharmacology, 1998, Volume: 124, Issue:5

    Topics: Aminopyridines; Antipsychotic Agents; Cell Line; Clozapine; Colforsin; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Humans; Kidney; Piperidines; Pyridines; Pyrroles; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone

1998
Neuropharmacological assessment of potential dopamine D4 receptor-selective radioligands.
    European journal of pharmacology, 1999, Feb-12, Volume: 367, Issue:1

    Topics: Aminopyridines; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Dopamine Agents; Dopamine Antagonists; Haloperidol; Humans; In Vitro Techniques; Ligands; Male; Piperidines; Prosencephalon; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4; Spiperone; Tritium

1999
Binding of [3H]U-101958 to sigma1 receptor-like sites in human cerebellum and neuroblastoma cells.
    European journal of pharmacology, 1999, Apr-09, Volume: 370, Issue:2

    Topics: Aminopyridines; Binding, Competitive; Cerebellum; Culture Techniques; Dopamine Agents; Humans; Neuroblastoma; Piperidines; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, sigma; Reverse Transcriptase Polymerase Chain Reaction; Sigma-1 Receptor

1999
D4 dopamine receptor-mediated phospholipid methylation and its implications for mental illnesses such as schizophrenia.
    Molecular psychiatry, 1999, Volume: 4, Issue:3

    Topics: Amino Acid Sequence; Aminopyridines; Animals; Benzazepines; Binding Sites; Carbon Radioisotopes; CHO Cells; Clozapine; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Formates; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Methionine; Mutagenesis, Site-Directed; Neuroblastoma; Phospholipids; Phosphorylation; Piperidines; Psychotic Disorders; Pyridines; Pyrroles; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; S-Adenosylmethionine; Salicylamides; Schizophrenia; Transfection; Tumor Cells, Cultured

1999
Receptor density as a factor governing the efficacy of the dopamine D4 receptor ligands, L-745,870 and U-101958 at human recombinant D4.4 receptors expressed in CHO cells.
    British journal of pharmacology, 1999, Volume: 128, Issue:3

    Topics: Aminopyridines; Animals; Butyrates; CHO Cells; Cricetinae; Cyclic AMP; Dopamine Agents; Humans; Ligands; Piperidines; Pyridines; Pyrroles; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Spiperone

1999
[(3)H]PNU-101958, a D(4) dopamine receptor probe, accumulates in prefrontal cortex and hippocampus of non-human primate brain.
    Synapse (New York, N.Y.), 2000, Sep-01, Volume: 37, Issue:3

    Topics: Aminopyridines; Animals; Autoradiography; Brain; Hippocampus; Macaca mulatta; Molecular Probes; Piperidines; Prefrontal Cortex; Pyridines; Pyrroles; Receptors, Dopamine D2; Receptors, Dopamine D4; Tissue Distribution; Tritium

2000