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szl 49 and prazosin

szl 49 has been researched along with prazosin in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19905 (29.41)18.7374
1990's10 (58.82)18.2507
2000's2 (11.76)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Buchowiecki, W; Kusiak, JW; Pitha, J; Szabo, L; Szurmai, Z1
Elhawary, AM; Pettinger, WA; Wolff, DW1
Piascik, MT; Pruitt, TA; Sparks, MS1
Piascik, MT; Pruitt, TA; Soltis, EE; Sparks, MS1
Mante, S; Minneman, KP1
Butler, BT; Kusiak, JW; Piascik, MT; Pruitt, TA1
Barron, KW; Kusiak, JW; Piascik, MT1
Kusiak, JW; Piascik, MT; Pitha, J1
Butler, BT; Holtman, JR; Kusiak, JW; Piascik, MT; Pitha, J1
Babich, M; Butler, BT; Kusiak, JW; Le, HT; Piascik, MT; Pitha, J1
Baum, BJ; Helman, J; Kusiak, JW; Pitha, J1
Lupichuk, SM; Tabrizchi, R1
Graham, D; Langer, SZ; Pimoule, C1
Daniel, EE; Hoo, KH; Kwan, CY1
Oriowo, MA1
Amobi, NI; Guillebaud, J; Kaisary, AV; Smith, IC; Turner, E1
Amobi, N; Guillebaud, J; Kaisary, A; Lloyd-Davies, RW; Smith, IC; Turner, E1

Other Studies

17 other study(ies) available for szl 49 and prazosin

ArticleYear
Alkylating prazosin analogue: irreversible label for alpha 1-adrenoceptors.
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:1

    Topics: Acylation; Animals; Binding, Competitive; Chemical Phenomena; Chemistry; Prazosin; Quinazolines; Radioligand Assay; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship

1989
Subtype-selective alpha-1 adrenoceptor alkylation in the rat kidney and its effect on the vascular pressor response.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:2

    Topics: Adrenergic alpha-Antagonists; Alkylation; Animals; Clonidine; Imidazoles; Kidney; Male; Methoxamine; Phenylephrine; Prazosin; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Renal Artery

1992
Interaction of imidazolines with alkylation-sensitive and -resistant alpha-1 adrenoceptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 1991, Jul-01, Volume: 258, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Clonidine; Drug Interactions; Imidazoles; Injections, Intraperitoneal; Male; Muscle, Smooth, Vascular; Phentolamine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1991
Evidence for a complex interaction between the subtypes of the alpha 1-adrenoceptor.
    European journal of pharmacology, 1991, Jul-09, Volume: 199, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Clonidine; Dioxanes; In Vitro Techniques; Kinetics; Male; Methoxamine; Muscle, Smooth, Vascular; Phenoxybenzamine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1991
The alkylating prazosin analog SZL 49 inactivates both alpha 1A- and alpha 1B-adrenoceptors.
    European journal of pharmacology, 1991, Oct-14, Volume: 208, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Drug Synergism; Hippocampus; Liver; Male; Membranes; Phenethylamines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones

1991
Agonist interaction with alkylation-sensitive and -resistant alpha-1 adrenoceptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Clonidine; Diltiazem; Dioxanes; Drug Interactions; Heart; Inositol Phosphates; Male; Muscle, Smooth, Vascular; Myocardium; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1990
Alpha 1-adrenoceptor subtypes and the regulation of peripheral hemodynamics in the conscious rat.
    European journal of pharmacology, 1990, Sep-21, Volume: 186, Issue:2-3

    Topics: Adrenergic alpha-Antagonists; Anesthesia; Animals; Blood Pressure; Cardiac Output; Chlorisondamine; Dose-Response Relationship, Drug; Hemodynamics; Male; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vascular Resistance

1990
Interaction of a chemically reactive prazosin analog with alpha-1 adrenoceptors of rat tissues.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 249, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Dose-Response Relationship, Drug; Male; Phenoxybenzamine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1989
Effect of an alkylating analog of prazosin on alpha-1 adrenoceptor subtypes and arterial blood pressure.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:3

    Topics: Adrenergic alpha-Antagonists; Alkylation; Animals; Blood Pressure; Dose-Response Relationship, Drug; Male; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1989
Alkylation of alpha-1 receptors with a chemically reactive analog of prazosin reveals low affinity sites for norepinephrine in rabbit aorta.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:3

    Topics: Alkylation; Animals; Dose-Response Relationship, Drug; Microsomes; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Yohimbine

1988
Inhibition of alpha 1-adrenergic responsiveness in intact cells by a new, irreversible receptor antagonist.
    Biochemical and biophysical research communications, 1987, Jan-30, Volume: 142, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Calcium; Cell Aggregation; Dose-Response Relationship, Drug; Epinephrine; In Vitro Techniques; Male; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1987
The effects of losartan and captopril on vasopressor actions of cirazoline in the absence and presence of SZL-49 and nifedipine.
    Journal of cardiovascular pharmacology, 1995, Volume: 26, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Antihypertensive Agents; Biphenyl Compounds; Blood Pressure; Captopril; Decerebrate State; Dose-Response Relationship, Drug; Imidazoles; Infusions, Intra-Arterial; Infusions, Intravenous; Losartan; Male; Nifedipine; Prazosin; Rats; Rats, Sprague-Dawley; Tetrazoles; Vasoconstriction; Vasodilator Agents

1995
Further evidence that the classical alpha 1A- and cloned alpha 1c-adrenoceptors are the same subtype.
    European journal of pharmacology, 1995, Jun-23, Volume: 290, Issue:1

    Topics: Animals; Binding Sites; Cattle; Clonidine; HeLa Cells; Humans; Prazosin; Rats; Receptors, Adrenergic, alpha-1; Recombinant Proteins

1995
Investigation of alpha 1-adrenoceptor subtypes in canine aorta, using alkylating agents.
    Canadian journal of physiology and pharmacology, 1994, Volume: 72, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Alkylating Agents; Animals; Aorta; Binding, Competitive; Clonidine; Dioxanes; Dogs; Female; In Vitro Techniques; Male; Mesenteric Veins; Muscle, Smooth, Vascular; Oxymetazoline; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha-1

1994
Alpha 1-adrenoceptor subtype(s) mediating noradrenaline-induced contractions of the guinea-pig aorta.
    Fundamental & clinical pharmacology, 1994, Volume: 8, Issue:3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Bridged Bicyclo Compounds; Bridged-Ring Compounds; Clonidine; Dioxanes; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Oxazines; Prazosin; Receptors, Adrenergic, alpha-1

1994
Discrimination by SZL49 between contractions evoked by noradrenaline in longitudinal and circular muscle of human vas deferens.
    British journal of pharmacology, 2002, Volume: 136, Issue:1

    Topics: Adrenergic alpha-Antagonists; Cystamine; Dibenzylchlorethamine; Humans; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Prazosin; Receptors, Adrenergic, alpha-1; Vas Deferens; Vasoconstrictor Agents

2002
Contractile actions of imidazoline alpha-adrenoceptor agonists and effects of noncompetitive alpha1-adrenoceptor antagonists in human vas deferens.
    European journal of pharmacology, 2003, Feb-21, Volume: 462, Issue:1-3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Dibenzylchlorethamine; Dose-Response Relationship, Drug; Humans; Imidazoles; Male; Muscle Contraction; Norepinephrine; Oxymetazoline; Phenoxybenzamine; Prazosin; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes; Vas Deferens

2003
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