Page last updated: 2024-09-02

sr 95531 and flumazenil

sr 95531 has been researched along with flumazenil in 8 studies

Compound Research Comparison

Studies
(sr 95531)
Trials
(sr 95531)
Recent Studies (post-2010)
(sr 95531)
Studies
(flumazenil)
Trials
(flumazenil)
Recent Studies (post-2010) (flumazenil)
61002094,673426981

Protein Interaction Comparison

ProteinTaxonomysr 95531 (IC50)flumazenil (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-1Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit beta-1Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit alpha-2Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit alpha-3Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-4Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit gamma-2Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0038
GABA theta subunitRattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0038

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19901 (12.50)18.7374
1990's3 (37.50)18.2507
2000's4 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Coale, A; Friedhoff, AJ; Gruen, RJ; Moghaddam, B1
Blasquez, C; Braquet, P; Delbende, C; Jégou, S; Tranchand Bunel, D; Vaudry, H1
Ikeda, M; Knapp, RJ; Malatynska, E; Yamamura, HI1
Cason, CR; Cheatham, G; Cook, JM; Gan, T; June, HL; Lui, R1
Abraini, JH; Balon, N; Kriem, B; Risso, JJ; Rostain, JC1
Jembrek, MJ; Pericić, D; Strac, DS; Vlainić, J1
Czajkowski, C; Sharkey, LM1
Anseloni, VC; Gold, MS1

Other Studies

8 other study(ies) available for sr 95531 and flumazenil

ArticleYear
Tonic inhibition of striatal dopamine transmission: effects of benzodiazepine and GABAA receptor antagonists on extracellular dopamine levels.
    Brain research, 1992, Dec-18, Volume: 599, Issue:1

    Topics: Animals; Corpus Striatum; Dialysis; Diazepam; Dopamine; Dose-Response Relationship, Drug; Extracellular Space; Flumazenil; GABA-A Receptor Antagonists; Male; Pyridazines; Rats; Rats, Sprague-Dawley; Synaptic Transmission

1992
Central-type benzodiazepines inhibit release of alpha-melanocyte-stimulating hormone from the rat hypothalamus.
    Neuroscience, 1991, Volume: 42, Issue:2

    Topics: Animals; Anti-Anxiety Agents; beta-Endorphin; Clonazepam; Diazepam; Flumazenil; GABA Antagonists; Hypothalamus; In Vitro Techniques; Male; Melanocyte-Stimulating Hormones; Perfusion; Pituitary Gland; Potassium Chloride; Pro-Opiomelanocortin; Pyridazines; Radioimmunoassay; Rats; Rats, Inbred Strains

1991
Amoxapine inhibition of GABA-stimulated chloride conductance: investigations of potential sites of activity.
    Life sciences, 1989, Volume: 45, Issue:20

    Topics: Amoxapine; Animals; Cerebral Cortex; Chlorides; Dibenzoxazepines; Dose-Response Relationship, Drug; Flumazenil; Flunitrazepam; GABA Antagonists; Ligands; Male; Pyridazines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1989
GABAA-benzodiazepine receptors in the striatum are involved in the sedation produced by a moderate, but not an intoxicating ethanol dose in outbred Wistar rats.
    Brain research, 1998, May-25, Volume: 794, Issue:1

    Topics: Alcoholic Intoxication; Analysis of Variance; Animals; Azides; Benzodiazepines; Corpus Striatum; Ethanol; Flumazenil; GABA Agents; GABA-A Receptor Agonists; Hypnotics and Sedatives; Male; Oocytes; Pyridazines; Rats; Rats, Wistar; Receptors, GABA-A; Xenopus

1998
Gamma-aminobutyric acid neuropharmacological investigations on narcosis produced by nitrogen, argon, or nitrous oxide.
    Anesthesia and analgesia, 2003, Volume: 96, Issue:3

    Topics: Anesthesia, Inhalation; Animals; Argon; Baclofen; Flumazenil; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Motor Activity; Nitrogen; Nitrous Oxide; Pyridazines; Rats; Rats, Sprague-Dawley

2003
Allosteric uncoupling and up-regulation of benzodiazepine and GABA recognition sites following chronic diazepam treatment of HEK 293 cells stably transfected with alpha1beta2gamma2S subunits of GABA (A) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:3

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Binding Sites; Binding, Competitive; Cell Line; Diazepam; Flumazenil; Flunitrazepam; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Muscimol; Picrotoxin; Protein Subunits; Pyridazines; Radioligand Assay; Rats; Receptors, GABA-A; Receptors, GABA-B; Transfection; Up-Regulation

2007
Individually monitoring ligand-induced changes in the structure of the GABAA receptor at benzodiazepine binding site and non-binding-site interfaces.
    Molecular pharmacology, 2008, Volume: 74, Issue:1

    Topics: Animals; Benzodiazepines; Binding Sites; Cysteine; Dose-Response Relationship, Drug; Electrophysiology; Female; Flumazenil; Flurazepam; GABA Agonists; GABA Antagonists; GABA Modulators; Inhibitory Concentration 50; Ligands; Microinjections; Muscimol; Mutagenesis, Site-Directed; Oocytes; Patch-Clamp Techniques; Pentobarbital; Pyridazines; Rats; Receptors, GABA-A; Xenopus

2008
Inflammation-induced shift in the valence of spinal GABA-A receptor-mediated modulation of nociception in the adult rat.
    The journal of pain, 2008, Volume: 9, Issue:8

    Topics: Animals; Antineoplastic Agents; Flumazenil; Freund's Adjuvant; GABA Agonists; GABA Antagonists; GABA Modulators; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Hyperalgesia; Inflammation; Injections, Spinal; Isoquinolines; Male; Midazolam; Muscimol; Nociceptors; Pain Measurement; Pain Threshold; Pyridazines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Signal Transduction; Spinal Cord

2008