Page last updated: 2024-09-03

rp 48740 and thiazoles

rp 48740 has been researched along with thiazoles in 21 studies

Compound Research Comparison

Studies
(rp 48740)
Trials
(rp 48740)
Recent Studies (post-2010)
(rp 48740)
Studies
(thiazoles)
Trials
(thiazoles)
Recent Studies (post-2010) (thiazoles)
240033,1792,10012,330

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19909 (42.86)18.7374
1990's11 (52.38)18.2507
2000's1 (4.76)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Claude, JR; Martin, C; Massicot, F; Pham Huy, C; Thevenin, M; Warnet, JM1
Bompart, F; Bruno, R; Clucas, A; Gaillot, J; Gregoire, J; Pinquier, JL; Sedivy, P; Strauch, G1
Braquet, P; Ferreira, MG; Fonteles, MC1
Burrell, R; Keller, GE; Lantz, RC1
Freiche, JC; Lang, J; Sedivy, P; Touraine, JL1
Breddin, HK; Weichert, W1
Benveniste, J; Coëffier, E; Desquand, S; Floch, A; Lefort, J; Maridonneau-Parini, I; Randon, J; Sedivy, P; Vargaftig, BB1
Bozza, PT; Cordeiro, RS; Dias, PM; Faria Neto, HC; Lima, MC; Martins, MA; Silva, PM; Vargaftig, BB1
Bureau, M; Joseph, D; Vargaftig, BB1
Adnot, S; Joseph, D; Vargaftig, BB1
Dechavanne, M; Hanss, M1
Myers, AK; Nakanishi, T; Ramwell, P1
Beijer, L; Burrell, R; Lantz, RC; Rylander, R; Sedivy, P1
Baggiolini, M; Dewald, B1
Bousseau, A; Clayette, P; Dormont, D; Henin, Y; Le Naour, R; Mabondzo, A; Raoul, H1
Bousseau, A; Fauci, AS; Poli, G; Weissman, D1
Imanishi, N; Koike, H; Morooka, S; Natsume, Y1
Bourgain, R; Decuyper, K; van Rossem, K; Vermariën, H1
Chignard, M; Paulin, D; Renesto, P; Vicart, P1
Clayette, P; Dereuddre-Bosquet, N; Dormont, D; Fretier, P; Martin, M1
Bensaid, O; Clayette, P; Dereuddre-Bosquet, N; Dong, CZ; Dormont, D; Godfroid, JJ; Heymans, F; Huet, J; Kan, E; Lamouri, A; Martin, M; Redeuilh, C; Serradji, N1

Other Studies

21 other study(ies) available for rp 48740 and thiazoles

ArticleYear
Inhibitory effects of a platelet activating factor-antagonist 48740RP in cyclosporin-induced nephrotoxicity in the rat as assessed by renal glutathione metabolism parameters.
    Archives of toxicology. Supplement. = Archiv fur Toxikologie. Supplement, 1991, Volume: 14

    Topics: Aminopeptidases; Animals; Blood Urea Nitrogen; CD13 Antigens; Creatinine; Cyclosporine; Glutathione; Kidney; Kidney Cortex; Platelet Activating Factor; Pyridines; Rats; Thiazoles

1991
Inhibition of ex-vivo PAF-induced platelet aggregation by the PAF-antagonist RP 48740: relationship to plasma concentrations in healthy volunteers.
    European journal of clinical pharmacology, 1991, Volume: 41, Issue:2

    Topics: Administration, Oral; Adult; Dose-Response Relationship, Drug; Humans; Male; Platelet Activating Factor; Platelet Aggregation Inhibitors; Pyridines; Reference Values; Thiazoles

1991
Effects of PAF antagonists on renal vascular escape and tachyphylaxis in perfused rabbit kidney.
    Lipids, 1991, Volume: 26, Issue:12

    Topics: Animals; Azepines; Diterpenes; Female; Gangliosides; Ginkgolides; In Vitro Techniques; Kidney; Kinetics; Lactones; Male; Perfusion; Platelet Activating Factor; Pyridines; Rabbits; Renal Circulation; Tachyphylaxis; Thiazoles; Time Factors; Triazoles

1991
The role of platelet-activating factor in the pulmonary response to inhaled bacterial endotoxin.
    The American review of respiratory disease, 1991, Volume: 144, Issue:1

    Topics: Animals; Blood Volume; Capillaries; Capillary Permeability; Cricetinae; Endothelium, Vascular; Endotoxins; Enterobacter; Leukocyte Count; Lung; Lung Volume Measurements; Male; Mesocricetus; Platelet Activating Factor; Platelet Count; Pulmonary Alveoli; Pulmonary Edema; Pyridines; Thiazoles

1991
Prolonged survival of renal transplants in nonimmunized and hyperimmunized rats receiving a platelet-activating factor antagonist.
    Transplantation, 1990, Volume: 50, Issue:1

    Topics: Animals; Cyclosporins; Cytotoxicity, Immunologic; Graft Rejection; Immunization; Kidney Transplantation; Male; Platelet Activating Factor; Pyridines; Rats; Rats, Inbred BN; Rats, Inbred Lew; Survival Rate; Thiazoles

1990
A PAF-acether antagonist (N 48740 RP/Rhône-Poulenc) and laser-induced thrombi in rat mesenteric vessels.
    Haemostasis, 1989, Volume: 19, Issue:4

    Topics: Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Fibrinolytic Agents; Lasers; Male; Mesenteric Arteries; Platelet Activating Factor; Platelet Aggregation Inhibitors; Pyridines; Rats; Rats, Inbred Strains; Thiazoles; Thrombosis

1989
Pharmacological profile of 48740 R.P., a PAF-acether antagonist.
    European journal of pharmacology, 1988, Jun-10, Volume: 150, Issue:3

    Topics: Animals; Blood Cell Count; Blood Platelets; Bronchodilator Agents; Guinea Pigs; Humans; In Vitro Techniques; Macrophages; Male; Muscle Contraction; Muscle, Smooth; N-Formylmethionine Leucyl-Phenylalanine; Perfusion; Platelet Activating Factor; Platelet Aggregation; Pulmonary Alveoli; Pyridines; Rabbits; Radioimmunoassay; Superoxides; Thiazoles; Thromboxane B2

1988
Pharmacological modulation of Paf-induced rat pleurisy and its role in inflammation by zymosan.
    British journal of pharmacology, 1989, Volume: 96, Issue:2

    Topics: Animals; Azepines; Carrageenan; Leukocyte Count; Male; Platelet Activating Factor; Pleurisy; Pyridines; Rats; Rats, Inbred Strains; Thiazoles; Triazines; Triazoles; Zymosan

1989
Desensitization and antagonism of rat polymorphonuclear leukocytes stimulated with PAF acether.
    Prostaglandins, 1987, Volume: 33, Issue:1

    Topics: Animals; Cells, Cultured; Cytochalasin B; Diterpenes; Exocytosis; Ginkgolides; Glucuronidase; Lactones; Leukotriene B4; Male; Muramidase; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Plant Extracts; Platelet Activating Factor; Pyridines; Rats; Rats, Inbred Strains; Thiazoles

1987
Antagonists of PAF-acether do not suppress thrombin-induced aggregation of ADP-deprived and aspirin-treated human platelets.
    Agents and actions, 1987, Volume: 21, Issue:1-2

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Aspirin; Blood Platelets; Crotalid Venoms; Cyclooxygenase Inhibitors; Diterpenes; Ginkgolides; Glyceryl Ethers; Humans; Lactones; Lectins, C-Type; Phospholipid Ethers; Plant Extracts; Platelet Activating Factor; Platelet Aggregation; Pyridines; Thiazoles; Thrombin

1987
48740 RP, an antagonist of PAF, does not affect human plasma fibrinolysis before and after venous occlusion.
    Thrombosis research, 1988, Jan-01, Volume: 49, Issue:1

    Topics: Adult; Constriction; Fibrinolysis; Humans; In Vitro Techniques; Male; Platelet Activating Factor; Pyridines; Thiazoles; Tissue Plasminogen Activator; Veins

1988
Antagonism of PAF-induced death in mice.
    Prostaglandins, 1988, Volume: 35, Issue:3

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Arachidonic Acid; Arachidonic Acids; Bridged Bicyclo Compounds, Heterocyclic; Collagen; Diterpenes; Epinephrine; Fatty Acids, Unsaturated; Furans; Ginkgolides; Hydrazines; Lactones; Male; Mice; Platelet Activating Factor; Platelet Aggregation Inhibitors; Prostaglandin Endoperoxides, Synthetic; Pyridines; Thiazoles; Thromboxane A2

1988
Modulation of pulmonary inflammation after endotoxin inhalation with a platelet-activating factor antagonist (48740 RP).
    International archives of allergy and applied immunology, 1988, Volume: 86, Issue:3

    Topics: Administration, Inhalation; Animals; Capillary Permeability; Cricetinae; Endothelium, Vascular; Endotoxins; Female; Guinea Pigs; Male; Platelet Activating Factor; Pneumonia; Pyridines; Thiazoles

1988
Evaluation of PAF antagonists using human neutrophils in a microtiter plate assay.
    Biochemical pharmacology, 1987, Aug-01, Volume: 36, Issue:15

    Topics: Benzofurans; Diterpenes; Exocytosis; Fluorescence; Ginkgolides; Humans; Lactones; Lignans; Methods; Neutrophils; Pancreatic Elastase; Phospholipid Ethers; Plant Extracts; Platelet Activating Factor; Pyridines; Thiazoles

1987
Infection of human macrophages with an endogenous tumour necrosis factor-alpha (TNF-alpha)-independent human immunodeficiency virus type 1 isolate is unresponsive to the TNF-alpha synthesis inhibitor RP 55778.
    The Journal of general virology, 1994, Volume: 75 ( Pt 6)

    Topics: Cells, Cultured; Gene Expression; HIV Reverse Transcriptase; HIV-1; Humans; Immunophenotyping; In Vitro Techniques; Interleukin-1; Interleukin-6; Macrophages; Pyridines; RNA-Directed DNA Polymerase; RNA, Messenger; Thiazoles; Tumor Necrosis Factor-alpha; Virus Replication

1994
A platelet-activating factor antagonist, RP 55778, inhibits cytokine-dependent induction of human immunodeficiency virus expression in chronically infected promonocytic cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Mar-15, Volume: 90, Issue:6

    Topics: Cell Line; Chloramphenicol O-Acetyltransferase; Cytokines; Fluorescent Antibody Technique; Granulocyte-Macrophage Colony-Stimulating Factor; HIV Reverse Transcriptase; HIV-1; Humans; Interleukin-6; Kinetics; Monocytes; Platelet Activating Factor; Pyridines; Recombinant Proteins; RNA Processing, Post-Transcriptional; RNA-Directed DNA Polymerase; RNA, Messenger; RNA, Viral; Tetradecanoylphorbol Acetate; Thiazoles; Transcription, Genetic; Transfection; Tumor Necrosis Factor-alpha

1993
Effects of platelet activating factor receptor antagonists on intracellular platelet activating factor function in neutrophils.
    European journal of pharmacology, 1994, Nov-15, Volume: 269, Issue:3

    Topics: Animals; Azepines; Binding, Competitive; Calcium; Cell Count; Cell Degranulation; Chemotaxis, Leukocyte; Free Radical Scavengers; Inositol 1,4,5-Trisphosphate; Male; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Platelet Activating Factor; Platelet Aggregation Inhibitors; Platelet Membrane Glycoproteins; Pyridines; Rats; Rats, Wistar; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Reference Standards; Signal Transduction; Structure-Activity Relationship; Superoxides; Thiazoles; Thiazolidines; Triazoles; Vitamin E

1994
The role of PAF and the effect of a specific PAF antagonist on local tissue PO2 and neuronal integrity during and after photothrombotic brain infarction in unanesthetised rabbits.
    Advances in experimental medicine and biology, 1996, Volume: 388

    Topics: Animals; Brain; Cerebral Infarction; Disease Models, Animal; Evoked Potentials, Somatosensory; Male; Neurons; Oxygen Consumption; Photobiology; Platelet Activating Factor; Pyridines; Rabbits; Thiazoles; Time Factors

1996
Protective effect of platelet activating factor antagonists on cultured endothelial cell lysis induced by elastase or activated neutrophils.
    British journal of pharmacology, 1996, Volume: 117, Issue:5

    Topics: Azepines; Cells, Cultured; Diterpenes; Dose-Response Relationship, Drug; Endothelium, Vascular; Ginkgolides; Humans; Lactones; Leukocyte Elastase; Neutrophils; Platelet Activating Factor; Platelet Membrane Glycoproteins; Pyridines; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Thiazoles; Triazoles

1996
Effects of RP 55778, a tumor necrosis factor alpha synthesis inhibitor, on antiviral activity of dideoxynucleosides.
    Antimicrobial agents and chemotherapy, 1997, Volume: 41, Issue:4

    Topics: Anti-HIV Agents; Dideoxynucleosides; HIV-1; Humans; Microbial Sensitivity Tests; Pyridines; Thiazoles; Tumor Necrosis Factor-alpha; Virus Replication; Zidovudine

1997
Structure-activity relationships in platelet-activating factor (PAF). 10. From PAF antagonism to inhibition of HIV-1 replication.
    Journal of medicinal chemistry, 2000, Jun-01, Volume: 43, Issue:11

    Topics: Anti-HIV Agents; Cells, Cultured; HIV; Humans; In Vitro Techniques; Inhibitory Concentration 50; Macrophages; Microbial Sensitivity Tests; Piperazines; Platelet Activating Factor; Platelet Membrane Glycoproteins; Pyridines; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Structure-Activity Relationship; Thiazoles; Virus Replication

2000