Page last updated: 2024-08-23

quinpirole and u-50488

quinpirole has been researched along with u-50488 in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19901 (11.11)18.7374
1990's7 (77.78)18.2507
2000's0 (0.00)29.6817
2010's1 (11.11)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berzetei-Gurske, IP; Guerrieri, E; Schmidhammer, H; Spetea, M1
Bot, G; Brent, PJ1
Heijna, MH; Hogenboom, F; Mulder, AH; Padt, M; Schoffelmeer, AN1
Heijna, MH; Hogenboom, F; Mulder, AH; Padt, M; Portoghese, PS; Schoffelmeer, AN1
Rooney, KF; Sewell, RD1
Bot, G; Chahl, LA1
Shieh, GJ; Walters, DE1
Crawford, CA; Garmsen, GM; McDougall, SA; Meier, TL1
Koch, H; Müller, T; Szabo, B1

Other Studies

9 other study(ies) available for quinpirole and u-50488

ArticleYear
Discovery and pharmacological evaluation of a diphenethylamine derivative (HS665), a highly potent and selective κ opioid receptor agonist.
    Journal of medicinal chemistry, 2012, Nov-26, Volume: 55, Issue:22

    Topics: Acetic Acid; Analgesics; Animals; Drug Discovery; Mice; Nociception; Pain; Phenethylamines; Receptors, Opioid, kappa

2012
Morphine, D-Pen2, D-Pen5 enkephalin and U50,488H differentially affect the locomotor activity and behaviours induced by quinpirole in guinea-pigs.
    Psychopharmacology, 1992, Volume: 107, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Behavior, Animal; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ergolines; Female; Guinea Pigs; Hypnotics and Sedatives; Injections, Intraventricular; Male; Morphine; Motor Activity; Piloerection; Pyrrolidines; Quinpirole

1992
Opioid-receptor-mediated inhibition of [3H]dopamine but not [3H]noradrenaline release from rat mediobasal hypothalamus slices.
    Neuroendocrinology, 1991, Volume: 54, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Dopamine; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ergolines; Hypothalamus, Middle; Male; Naloxone; Narcotic Antagonists; Norepinephrine; Oxymetazoline; Pyrrolidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1991
Opioid receptor-mediated inhibition of dopamine and acetylcholine release from slices of rat nucleus accumbens, olfactory tubercle and frontal cortex.
    European journal of pharmacology, 1990, Jun-08, Volume: 181, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acetylcholine; Animals; Benzomorphans; Cerebral Cortex; Corpus Striatum; Dopamine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ergolines; In Vitro Techniques; Male; Naloxone; Naltrexone; Nucleus Accumbens; Olfactory Bulb; Oxymetazoline; Pyrrolidines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Opioid; Septal Nuclei

1990
Evaluation of selective actions of dopamine D-1 and D-2 receptor agonists and antagonists on opioid antinociception.
    European journal of pharmacology, 1989, Sep-22, Volume: 168, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Dopamine Agents; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ergolines; Fentanyl; Injections, Intraventricular; Male; Mice; Narcotics; Nociceptors; Pyrrolidines; Quinpirole; Reaction Time; Receptors, Dopamine; Sufentanil; Sulpiride

1989
Effects of pertussis toxin on behavioural responses of guinea-pigs to centrally administered substance P, quinpirole, carbachol, U-50,488H, morphine and morphine withdrawal.
    European journal of pharmacology, 1993, Jan-26, Volume: 231, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Behavior, Animal; Carbachol; Dopamine Agents; Ergolines; Female; Guinea Pigs; Injections, Intraventricular; Male; Morphine; Motor Activity; Naloxone; Pertussis Toxin; Pyrrolidines; Quinpirole; Receptors, Opioid, kappa; Substance P; Substance Withdrawal Syndrome; Virulence Factors, Bordetella

1993
Altered neurochemical and behavioral development of 10-day-old rats perinatally exposed to the kappa opioid agonist U-50,488H.
    Neuroscience letters, 1994, Jul-18, Volume: 176, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Ergolines; Feeding Behavior; Female; Litter Size; Male; Motor Activity; Nucleus Accumbens; Pregnancy; Prenatal Exposure Delayed Effects; Pyrrolidines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Opioid, kappa; Weight Gain

1994
Kappa opioid mediated locomotor activity in the preweanling rat: role of pre- and postsynaptic dopamine receptors.
    Psychopharmacology, 1997, Volume: 133, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; alpha-Methyltyrosine; Animals; Animals, Suckling; Corpus Striatum; Dopamine; Dopamine Agonists; Female; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Opioid, kappa

1997
Effects of cannabinoids on dopamine release in the corpus striatum and the nucleus accumbens in vitro.
    Journal of neurochemistry, 1999, Volume: 73, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzoxazines; Cannabinoids; Corpus Striatum; Cyclohexanols; Dopamine; Dopamine Agonists; Electric Stimulation; Electrophysiology; In Vitro Techniques; Male; Membrane Potentials; Morpholines; Naphthalenes; Nucleus Accumbens; Patch-Clamp Techniques; Quinpirole; Rats; Rats, Wistar; Receptor, Cannabinoid, CB2; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid, kappa

1999
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