Page last updated: 2024-08-18

pyrroles and pk 11195

pyrroles has been researched along with pk 11195 in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's0 (0.00)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Anzini, M; Botta, M; Cagnotto, A; Cappelli, A; Vomero, S1
Bernasconi, P; Campiani, G; Ciani, SM; Fiorini, I; Garofalo, A; Greco, G; Mennini, T; Nacci, V; Novellino, E1
Anderson, LE; Dring, AM; Hamel, LD; Stoner, MA1

Other Studies

3 other study(ies) available for pyrroles and pk 11195

ArticleYear
5-HT and benzodiazepine receptor ligands. III. Synthesis and receptor affinities of 1,2,4-triazolo[4',3':1,6]pyridazino[4,5-b]quinoline and 2,3-dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinoline-1-one derivatives.
    Farmaco (Societa chimica italiana : 1989), 1990, Volume: 45, Issue:11

    Topics: Animals; Binding, Competitive; Brain; Cerebellum; Flumazenil; In Vitro Techniques; Isoquinolines; Ligands; Pyrroles; Quinolones; Rats; Receptors, GABA-A; Receptors, Serotonin

1990
A comparative molecular field analysis model for 6-arylpyrrolo[2,1-d] [1,5]benzothiazepines binding selectively to the mitochondrial benzodiazepine receptor.
    Journal of medicinal chemistry, 1994, Nov-25, Volume: 37, Issue:24

    Topics: Animals; Isoquinolines; Ligands; Male; Mitochondria; Models, Molecular; Molecular Conformation; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Regression Analysis; Structure-Activity Relationship; Thiazepines

1994
Modulation of constitutive androstane receptor (CAR) and pregnane X receptor (PXR) by 6-arylpyrrolo[2,1-d][1,5]benzothiazepine derivatives, ligands of peripheral benzodiazepine receptor (PBR).
    Toxicology letters, 2011, Apr-25, Volume: 202, Issue:2

    Topics: Aryl Hydrocarbon Hydroxylases; Cell Line; Constitutive Androstane Receptor; Cytochrome P-450 CYP2B6; Cytochrome P-450 CYP3A; Hepatocytes; Humans; Indoleacetic Acids; Isoquinolines; Liver; Oxidoreductases, N-Demethylating; Pregnane X Receptor; Pyrroles; Receptors, Cytoplasmic and Nuclear; Receptors, GABA-A; Receptors, Steroid; Reverse Transcriptase Polymerase Chain Reaction; RNA; Thiazepines; Transfection

2011