Page last updated: 2024-08-16

prazosin and urapidil

prazosin has been researched along with urapidil in 50 studies

Research

Studies (50)

TimeframeStudies, this research(%)All Research%
pre-199022 (44.00)18.7374
1990's13 (26.00)18.2507
2000's7 (14.00)29.6817
2010's8 (16.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Lombardo, F; Obach, RS; Waters, NJ1
Campillo, NE; Guerra, A; Páez, JA1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Kondo, S; Morita, T1
Fingerle, J; Fotev, Z; Sanders, KH1
Gagało, I; Szreder, Z1
Lewczuk, J; Wrabec, K1
Ramage, AG2
Beller, KD; Boer, R; Sanders, KH; Walter, B1
Betteridge, DJ; Prichard, BN; Smith, CC1
Kirsten, R; Ochs, JG; Storck, J1
Anastasi, N; Browne, RK; Dias Souza, J; Dretchen, KL; Gillis, RA; Hill, K; Namath, I; Quest, JA1
Aoki, K; Asano, M; Matsuda, T1
Friedman, E; Gillis, RA; Hamosh, P; Kellar, KJ; Mandal, AK; Pineo, SV1
Cichini, G; Kraupp, O; Singer, EA; Valenta, B1
Gross, G; Hanft, G1
Shebuski, RJ; Zimmerman, BG1
Goering, J; Zimmerman, BG1
Zeigler, DW; Zimmerman, BG1
Dollery, CT; Warren, JB1
Magometschnigg, D; Schütz, W1
Kaneko, Y1
Bacher, S; Beck, A; Kraupp, O; Raberger, G; Skoda, H1
Becker, H; Ganten, D; Lang, RE; Luft, FC; Unger, T; Veelken, R1
Jurna, I; Sanders, KH1
Beckeringh, JJ; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Bonham, AC; Brody, MJ; Mangiapane, ML; Porter, JP; Trapani, AJ; Webb, RL1
Buller, A; Conforti, A; Dias Souza, J; Gillis, RA; Kellar, KJ; Quest, JA; Spera, AC1
Kaplan, HR; Smith, RD1
Timmermans, PB; van Zwieten, PA1
Timmermans, PB; Van Brummelen, P; Van Zwieten, PA1
Frohlich, ED; Gallo, AJ; Kobrin, I; Natsume, T; Pegram, BL1
Grassi, G; Mancia, G; Seravalle, G; Zanchetti, A1
Compagnon, P; Fresel, J; Joannidès, R; Moore, N; Thuillez, C1
Asano, M; Honda, K; Inagaki, O; Kawabe, K; Kimura, R; Mori, R; Suzuki, M; Takenaka, T; Tanaka, C; Yamada, S1
Ebihara, A; Fujimura, A; Harada, K; Kumagai, Y; Ohashi, K1
Heintz, B; Kirsten, D; Kirsten, R; Nelson, K1
Grassi, G; Mancia, G; Seravalle, G; Stella, ML; Turri, C; Zanchetti, A1
Eckert, RE; Karsten, AJ; Utz, J; Ziegler, M1
Edwards, LP; George, OK; Gonzalez, RR1
Miyata, K; Ohtake, A; Saitoh, C; Sasamata, M; Sato, S; Yuyama, H1
Miyata, K; Ohtake, A; Sasamata, M; Sato, S1
Jiang, W; Ma, Y; Wang, L; Zhang, Y; Zhou, G1
Hatanaka, T; Noguchi, Y; Ohtake, A; Sasamata, M; Sato, S; Suzuki, M; Ueshima, K; Yanai-Inamura, H1
Araki, M; Araki, T; Monden, K1

Reviews

5 review(s) available for prazosin and urapidil

ArticleYear
[Value of vasodilator agents in the treatment of diseases with pulmonary hypertension caused by chronic obstructive lung diseases].
    Pneumonologia i alergologia polska, 1991, Volume: 59, Issue:3-4

    Topics: Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Blood Pressure; Calcium Channel Blockers; Drug Evaluation; Humans; Hydralazine; Hypertension, Pulmonary; Lung Diseases, Obstructive; Piperazines; Prazosin; Pulmonary Heart Disease; Vasodilator Agents

1991
The usefulness of alpha-adrenoceptor blockade in the treatment of hypertension.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1988, Volume: 6, Issue:2

    Topics: Adrenergic alpha-Antagonists; Antihypertensive Agents; Humans; Hypertension; Indoramin; Labetalol; Piperazines; Prazosin

1988
Cardiovascular alpha 2-receptors.
    Journal of molecular and cellular cardiology, 1983, Volume: 15, Issue:11

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Affinity Labels; Animals; Blood Pressure; Brain; Calcium Channel Blockers; Cardiovascular Physiological Phenomena; Guanosine Triphosphate; Heart Rate; Humans; Ketanserin; Kidney; Muscle, Smooth, Vascular; Piperazines; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Synaptic Membranes; Tritium; Vasoconstriction

1983
Role of alpha adrenoceptors in hypertension and in antihypertensive drug treatment.
    The American journal of medicine, 1984, Oct-05, Volume: 77, Issue:4A

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Azepines; Blood Pressure; Calcium Channel Blockers; Clonidine; Guanfacine; Guanidines; Humans; Hypertension; Ketanserin; Methyldopa; Muscle, Smooth, Vascular; Phenylacetates; Piperazines; Piperidines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha; Vascular Resistance

1984
Clinical pharmacokinetics of vasodilators. Part II.
    Clinical pharmacokinetics, 1998, Volume: 35, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Alprostadil; Amrinone; Carbazoles; Carvedilol; Enoximone; Female; Humans; Iloprost; Imidazoles; Indoramin; Isosorbide Dinitrate; Labetalol; Milrinone; Molsidomine; Nitroglycerin; Nitroprusside; Oxyfedrine; Pentaerythritol Tetranitrate; Phosphodiesterase Inhibitors; Piperazines; Prazosin; Pregnancy; Propanolamines; Pyridones; Theophylline; Trapidil; Vasodilator Agents

1998

Trials

5 trial(s) available for prazosin and urapidil

ArticleYear
Double-blind comparison of urapidil and prazosin in the treatment of patients with essential hypertension.
    Drugs, 1988, Volume: 35 Suppl 6

    Topics: Adult; Aged; Antihypertensive Agents; Clinical Trials as Topic; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hypertension; Male; Middle Aged; Piperazines; Prazosin; Random Allocation

1988
A comparison of the hemodynamic effects of urapidil, prazosin, and clonidine in healthy volunteers.
    Blood pressure. Supplement, 1994, Volume: 4

    Topics: Adult; Antihypertensive Agents; Blood Pressure; Clonidine; Drug Administration Schedule; Heart Rate; Humans; Male; Norepinephrine; Piperazines; Prazosin; Vascular Resistance

1994
Effect of alpha 1-adrenoceptor antagonists, prazosin and urapidil, on a finger skin vasoconstrictor response to cold stimulation.
    European journal of clinical pharmacology, 1996, Volume: 49, Issue:5

    Topics: Administration, Oral; Adrenergic alpha-Antagonists; Adult; Analysis of Variance; Cold Temperature; Humans; Laser-Doppler Flowmetry; Male; Piperazines; Prazosin; Regional Blood Flow; Skin; Vasoconstriction

1996
Sympathoexcitatory responses to the acute blood pressure fall induced by central or peripheral antihypertensive drugs.
    American journal of hypertension, 2000, Volume: 13, Issue:1 Pt 1

    Topics: Adult; Antihypertensive Agents; Blood Pressure; Cross-Over Studies; Double-Blind Method; Heart Rate; Humans; Hypertension; Male; Muscle, Skeletal; Norepinephrine; Piperazines; Prazosin; Sympathetic Nervous System; Sympatholytics

2000
Comparison of 7 α(1)-adrenoceptor antagonists in patients with lower urinary tract symptoms associated with benign prostatic hyperplasia:a short-term crossover study.
    Acta medica Okayama, 2013, Volume: 67, Issue:4

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adult; Aged; Aged, 80 and over; Cross-Over Studies; Doxazosin; Humans; Indoles; Lower Urinary Tract Symptoms; Male; Middle Aged; Naphthalenes; Piperazines; Prazosin; Prostatic Hyperplasia; Sulfonamides; Tamsulosin; Treatment Outcome

2013

Other Studies

40 other study(ies) available for prazosin and urapidil

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
[Comparison of selective alpha-1 blockades for alpha-receptors in human hypertrophied prostatic adenomas].
    Nihon Hinyokika Gakkai zasshi. The japanese journal of urology, 1992, Volume: 83, Issue:3

    Topics: Adenoma; Adrenergic alpha-Antagonists; Aged; Humans; Male; Piperazines; Prazosin; Prostatic Hyperplasia; Prostatic Neoplasms; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha

1992
Alpha 1-receptor antagonists urapidil and prazosin inhibit neointima formation in rat carotid artery induced by balloon catheter injury.
    Basic research in cardiology, 1991, Volume: 86 Suppl 1

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Carotid Arteries; Carotid Artery Injuries; Cell Division; DNA; Heart Rate; Male; Muscle, Smooth, Vascular; Piperazines; Prazosin; Rats; Rats, Inbred Strains

1991
The effect of doxazosin, urapidil and indoramin pretreatment on fever produced by E. coli lipopolysaccharide in rabbits.
    General pharmacology, 1991, Volume: 22, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Anti-Inflammatory Agents, Non-Steroidal; Body Temperature Regulation; Doxazosin; Escherichia coli; Female; Fever; Indoramin; Lipopolysaccharides; Male; Piperazines; Prazosin; Rabbits

1991
The mechanism of the sympathoinhibitory action of urapidil: role of 5-HT1A receptors.
    British journal of pharmacology, 1991, Volume: 102, Issue:4

    Topics: Anesthesia; Animals; Blood Pressure; Cats; Clonidine; Heart; Heart Rate; Kidney; Male; Piperazines; Prazosin; Receptors, Serotonin; Regional Blood Flow; Spiperone; Splanchnic Nerves; Sympatholytics

1991
Is blockade of alpha 1-adrenoceptors favourable in hypotension induced by stimulation of serotonin1A receptors in conscious dogs?
    Drugs, 1990, Volume: 40 Suppl 4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Heart Rate; Male; Piperazines; Prazosin; Rats; Receptors, Serotonin; Stimulation, Chemical; Swine; Tetrahydronaphthalenes

1990
Platelet in vitro responses to urapidil and prazosin.
    Drugs, 1990, Volume: 40 Suppl 4

    Topics: Adult; Antihypertensive Agents; Blood Platelets; Epinephrine; Female; Humans; Male; Norepinephrine; Piperazines; Platelet Aggregation; Prazosin

1990
Effects of urapidil on 5-hydroxytryptamine induced platelet aggregation and on 14C-5-hydroxytryptamine uptake in platelets.
    International journal of clinical pharmacology, therapy, and toxicology, 1990, Volume: 28, Issue:7

    Topics: Administration, Oral; Adult; Blood Platelets; Carbon Radioisotopes; Epinephrine; Humans; Ketanserin; Nafronyl; Piperazines; Platelet Aggregation Inhibitors; Prazosin; Serotonin; Serotonin Antagonists

1990
Hypotensive effect of urapidil: CNS site and relative contribution.
    Journal of cardiovascular pharmacology, 1987, Volume: 9, Issue:1

    Topics: Animals; Blood Pressure; Brain; Cats; Female; Heart Rate; Male; Piperazines; Prazosin; Respiration; Sympathetic Nervous System

1987
Antagonism of alpha 1-adrenoceptor-mediated vascular contraction by urapidil in isolated arterial strips of spontaneously hypertensive rats.
    Journal of cardiovascular pharmacology, 1988, Volume: 12, Issue:2

    Topics: Age Factors; Animals; Antihypertensive Agents; Dose-Response Relationship, Drug; Hypertension; In Vitro Techniques; Male; Norepinephrine; Phentolamine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha; Vasoconstriction; Yohimbine

1988
Importance of central nervous system serotonin-1A receptors for mediating the hypotensive effect of urapidil.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antihypertensive Agents; Blood Pressure; Cats; Heart Rate; Medulla Oblongata; Piperazines; Prazosin; Receptors, Serotonin; Respiration; Spiperone; Tetrahydronaphthalenes

1989
Effects of urapidil on catecholamine turnover and release in the central nervous system of the rat.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:3

    Topics: Animals; Blood Pressure; Brain Chemistry; Catecholamines; Chromatography, High Pressure Liquid; Dioxanes; Dopamine; Electric Stimulation; Haloperidol; Idazoxan; In Vitro Techniques; Male; Methoxyhydroxyphenylglycol; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Inbred Strains

1989
Subclassification of alpha 1-adrenoceptor recognition sites by urapidil derivatives and other selective antagonists.
    British journal of pharmacology, 1989, Volume: 97, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Dioxanes; Heart; In Vitro Techniques; Male; Myocardium; Phenethylamines; Phentolamine; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones; Yohimbine

1989
Suppression of reflex tachycardia by central administration of the alpha-1 adrenoceptor antagonists urapidil and prazosin in anesthetized dogs.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 234, Issue:2

    Topics: Adrenergic alpha-Antagonists; Anesthesia; Animals; Antihypertensive Agents; Blood Pressure; Bradykinin; Brain; Dogs; Female; Heart Rate; Indoramin; Male; Phenylephrine; Piperazines; Prazosin; Pressoreceptors; Quinazolines; Reflex; Vascular Resistance

1985
Analysis of adrenoceptor blockade and hypotension elicited by urapidil and prazosin in conscious rat.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Antihypertensive Agents; Arginine Vasopressin; Blood Pressure; Enalapril; Enalaprilat; Male; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Renin-Angiotensin System

1986
Effect of alpha 1-adrenoceptor blockade on blood pressure and iliac vascular resistance in normotensive and Goldblatt hypertensive dogs; influence of dietary salt and DOCA-salt.
    Journal of hypertension, 1987, Volume: 5, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Captopril; Desoxycorticosterone; Dogs; Female; Hypertension, Renovascular; Iliac Artery; Male; Phenylephrine; Piperazines; Prazosin; Regional Blood Flow; Sodium, Dietary; Vascular Resistance

1987
A clinical approach for the identification of peripheral pre- and post-synaptic alpha-adrenergic receptors.
    Journal of hypertension, 1986, Volume: 4, Issue:4

    Topics: Adult; Blood Pressure; Heart Rate; Humans; Male; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Synapses; Yohimbine

1986
A comparison of the effects of doxazosin and alfuzosin with those of urapidil on preganglionic sympathetic nerve activity in anaesthetised cats.
    European journal of pharmacology, 1986, Oct-07, Volume: 129, Issue:3

    Topics: Action Potentials; Animals; Blood Pressure; Cats; Doxazosin; Male; Piperazines; Prazosin; Quinazolines; Receptors, Adrenergic, alpha; Sympathetic Nervous System; Vascular Resistance

1986
Characterization of vasodilators by comparison of their effects on blood pressure, counterregulation and myocardial oxygen demand in conscious normotensive dogs.
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:1A

    Topics: Animals; Blood Pressure; Dihydralazine; Dogs; Female; Heart Rate; Isosorbide Dinitrate; Labetalol; Male; Molsidomine; Myocardium; Oxygen Consumption; Piperazines; Prazosin; Pyridazines; Renin; Sydnones; Vasodilator Agents

1985
Effect of urapidil, clonidine, and prazosin on sympathetic tone in conscious rats.
    Hypertension (Dallas, Tex. : 1979), 1986, Volume: 8, Issue:4

    Topics: Animals; Blood Pressure; Clonidine; Electrodes; Heart Rate; Piperazines; Prazosin; Pressoreceptors; Rats; Rats, Inbred SHR; Splanchnic Nerves; Sympathetic Nervous System

1986
Effects of urapidil, clonidine, prazosin and propranolol on autonomic nerve activity, blood pressure and heart rate in anaesthetized rats and cats.
    European journal of pharmacology, 1985, Apr-02, Volume: 110, Issue:2

    Topics: Anesthesia; Animals; Antihypertensive Agents; Autonomic Nervous System; Blood Pressure; Cats; Clonidine; Female; Heart Rate; Hemodynamics; In Vitro Techniques; Male; Neurons; Piperazines; Prazosin; Propranolol; Quinazolines; Rats; Rats, Inbred Strains; Species Specificity; Splanchnic Nerves; Sympathetic Nervous System; Vagus Nerve

1985
Cardiovascular effects and interaction with adrenoceptors of urapidil.
    Archives internationales de pharmacodynamie et de therapie, 1985, Volume: 276, Issue:2

    Topics: Animals; Antihypertensive Agents; Binding, Competitive; Cats; Clonidine; Decerebrate State; Female; Hemodynamics; Hexobarbital; In Vitro Techniques; Infusions, Parenteral; Male; Membranes; Mice; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Piperazines; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rats, Inbred WKY; Receptors, Adrenergic

1985
Comparative central and peripheral antihypertensive mechanisms of urapidil and prazosin.
    The American journal of medicine, 1984, Oct-05, Volume: 77, Issue:4A

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Brain; Heart Rate; Injections, Intravenous; Injections, Intraventricular; Male; Piperazines; Prazosin; Pressoreceptors; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Sympathectomy; Vascular Resistance

1984
Comparative effects of urapidil, prazosin, and clonidine on ligand binding to central nervous system receptors, arterial pressure, and heart rate in experimental animals.
    The American journal of medicine, 1984, Oct-05, Volume: 77, Issue:4A

    Topics: Animals; Antihypertensive Agents; Binding, Competitive; Blood Pressure; Brain; Cats; Clonidine; Dose-Response Relationship, Drug; Female; Heart Rate; Injections, Intravenous; Injections, Intraventricular; Male; Piperazines; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Muscarinic

1984
Antihypertensive drugs: proposed sites and mechanisms of action.
    Federation proceedings, 1981, Volume: 40, Issue:8

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Cats; Clonidine; Denervation; Dogs; Heart Rate; Methysergide; Moxisylyte; Phentolamine; Piperazines; Prazosin; Uracil

1981
Systemic and regional hemodynamic effects of acute and prolonged treatment with urapidil or prazosin in normotensive and spontaneously hypertensive rats.
    The American journal of medicine, 1984, Oct-05, Volume: 77, Issue:4A

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cardiac Output; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Hypertension; Male; Piperazines; Prazosin; Pressoreceptors; Quinazolines; Rats; Rats, Inbred SHR; Regional Blood Flow; Time Factors; Vascular Resistance

1984
Hemodynamic and neural effects of urapidil and prazosin in essential hypertensives.
    Blood pressure. Supplement, 1994, Volume: 4

    Topics: Administration, Oral; Antihypertensive Agents; Blood Pressure; Heart Rate; Humans; Hypertension; Peroneal Nerve; Piperazines; Prazosin; Sympathetic Fibers, Postganglionic

1994
Comparative study on alpha 1-adrenoceptor antagonist binding in human prostate and aorta.
    Clinical and experimental pharmacology & physiology, 1994, Volume: 21, Issue:5

    Topics: Adrenergic alpha-Antagonists; Aged; Aorta; Binding Sites; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Humans; Kinetics; Male; Middle Aged; Naphthalenes; Piperazines; Prazosin; Prostate; Sulfonamides; Tamsulosin

1994
Regulation of renal artery smooth muscle tone by alpha1-adrenoceptors: role of voltage-gated calcium channels and intracellular calcium stores.
    Urological research, 2000, Volume: 28, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Diltiazem; Dioxanes; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Ischemia; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Phenoxybenzamine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Renal Artery; Renal Circulation; Swine; Thapsigargin; Verapamil

2000
Moxonidine, an antihypertensive agent, is permissive to alpha1-adrenergic receptor pathway in the rat-tail artery.
    Journal of cardiovascular pharmacology, 2004, Volume: 43, Issue:2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Antihypertensive Agents; Drug Interactions; Imidazoles; Male; Muscle, Smooth, Vascular; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Vasoconstriction; Yohimbine

2004
Effects of tamsulosin on hypogastric nerve stimulation-induced intraurethral pressure elevation in male and female dogs under anesthesia.
    European journal of pharmacology, 2004, Aug-30, Volume: 497, Issue:3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Dogs; Female; Hypogastric Plexus; Male; Naphthalenes; Piperazines; Prazosin; Pressure; Sex Factors; Sulfonamides; Tamsulosin; Urethra

2004
Effects of tamsulosin on resting urethral pressure and arterial blood pressure in anaesthetized female dogs.
    The Journal of pharmacy and pharmacology, 2006, Volume: 58, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Female; Piperazines; Prazosin; Pressure; Sulfonamides; Tamsulosin; Urethra

2006
Synthesis of a quinazoline derivative: a new α₁-adrenoceptor ligand for conjugation to quantum dots to study α₁-adrenoceptors in living cells.
    Bioorganic & medicinal chemistry letters, 2011, Oct-01, Volume: 21, Issue:19

    Topics: Adrenergic alpha-1 Receptor Antagonists; Biological Assay; Biotin; Drug Design; Drug Evaluation, Preclinical; HEK293 Cells; Humans; Ligands; Molecular Structure; Molecular Weight; Piperazines; Polyethylene Glycols; Prazosin; Protein Binding; Quantum Dots; Quinazolines; Receptors, Adrenergic, alpha-1

2011
Effects of α1-adrenoceptor antagonists on phenylephrine-induced salivary secretion and intraurethral pressure elevation in anesthetized rats.
    European journal of pharmacology, 2012, Mar-15, Volume: 679, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Dose-Response Relationship, Drug; Drug Interactions; Indoles; Male; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Saliva; Salivary Glands; Sulfonamides; Tamsulosin; Urethra

2012
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