prazosin and urapidil
prazosin has been researched along with urapidil in 50 studies
Research
Studies (50)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 22 (44.00) | 18.7374 |
1990's | 13 (26.00) | 18.2507 |
2000's | 7 (14.00) | 29.6817 |
2010's | 8 (16.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors
Authors | Studies |
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Topliss, JG; Yoshida, F | 1 |
Lombardo, F; Obach, RS; Waters, NJ | 1 |
Campillo, NE; Guerra, A; Páez, JA | 1 |
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV | 1 |
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ | 1 |
Kondo, S; Morita, T | 1 |
Fingerle, J; Fotev, Z; Sanders, KH | 1 |
Gagało, I; Szreder, Z | 1 |
Lewczuk, J; Wrabec, K | 1 |
Ramage, AG | 2 |
Beller, KD; Boer, R; Sanders, KH; Walter, B | 1 |
Betteridge, DJ; Prichard, BN; Smith, CC | 1 |
Kirsten, R; Ochs, JG; Storck, J | 1 |
Anastasi, N; Browne, RK; Dias Souza, J; Dretchen, KL; Gillis, RA; Hill, K; Namath, I; Quest, JA | 1 |
Aoki, K; Asano, M; Matsuda, T | 1 |
Friedman, E; Gillis, RA; Hamosh, P; Kellar, KJ; Mandal, AK; Pineo, SV | 1 |
Cichini, G; Kraupp, O; Singer, EA; Valenta, B | 1 |
Gross, G; Hanft, G | 1 |
Shebuski, RJ; Zimmerman, BG | 1 |
Goering, J; Zimmerman, BG | 1 |
Zeigler, DW; Zimmerman, BG | 1 |
Dollery, CT; Warren, JB | 1 |
Magometschnigg, D; Schütz, W | 1 |
Kaneko, Y | 1 |
Bacher, S; Beck, A; Kraupp, O; Raberger, G; Skoda, H | 1 |
Becker, H; Ganten, D; Lang, RE; Luft, FC; Unger, T; Veelken, R | 1 |
Jurna, I; Sanders, KH | 1 |
Beckeringh, JJ; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B | 1 |
Bonham, AC; Brody, MJ; Mangiapane, ML; Porter, JP; Trapani, AJ; Webb, RL | 1 |
Buller, A; Conforti, A; Dias Souza, J; Gillis, RA; Kellar, KJ; Quest, JA; Spera, AC | 1 |
Kaplan, HR; Smith, RD | 1 |
Timmermans, PB; van Zwieten, PA | 1 |
Timmermans, PB; Van Brummelen, P; Van Zwieten, PA | 1 |
Frohlich, ED; Gallo, AJ; Kobrin, I; Natsume, T; Pegram, BL | 1 |
Grassi, G; Mancia, G; Seravalle, G; Zanchetti, A | 1 |
Compagnon, P; Fresel, J; Joannidès, R; Moore, N; Thuillez, C | 1 |
Asano, M; Honda, K; Inagaki, O; Kawabe, K; Kimura, R; Mori, R; Suzuki, M; Takenaka, T; Tanaka, C; Yamada, S | 1 |
Ebihara, A; Fujimura, A; Harada, K; Kumagai, Y; Ohashi, K | 1 |
Heintz, B; Kirsten, D; Kirsten, R; Nelson, K | 1 |
Grassi, G; Mancia, G; Seravalle, G; Stella, ML; Turri, C; Zanchetti, A | 1 |
Eckert, RE; Karsten, AJ; Utz, J; Ziegler, M | 1 |
Edwards, LP; George, OK; Gonzalez, RR | 1 |
Miyata, K; Ohtake, A; Saitoh, C; Sasamata, M; Sato, S; Yuyama, H | 1 |
Miyata, K; Ohtake, A; Sasamata, M; Sato, S | 1 |
Jiang, W; Ma, Y; Wang, L; Zhang, Y; Zhou, G | 1 |
Hatanaka, T; Noguchi, Y; Ohtake, A; Sasamata, M; Sato, S; Suzuki, M; Ueshima, K; Yanai-Inamura, H | 1 |
Araki, M; Araki, T; Monden, K | 1 |
Reviews
5 review(s) available for prazosin and urapidil
Article | Year |
---|---|
[Value of vasodilator agents in the treatment of diseases with pulmonary hypertension caused by chronic obstructive lung diseases].
Topics: Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Blood Pressure; Calcium Channel Blockers; Drug Evaluation; Humans; Hydralazine; Hypertension, Pulmonary; Lung Diseases, Obstructive; Piperazines; Prazosin; Pulmonary Heart Disease; Vasodilator Agents | 1991 |
The usefulness of alpha-adrenoceptor blockade in the treatment of hypertension.
Topics: Adrenergic alpha-Antagonists; Antihypertensive Agents; Humans; Hypertension; Indoramin; Labetalol; Piperazines; Prazosin | 1988 |
Cardiovascular alpha 2-receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Affinity Labels; Animals; Blood Pressure; Brain; Calcium Channel Blockers; Cardiovascular Physiological Phenomena; Guanosine Triphosphate; Heart Rate; Humans; Ketanserin; Kidney; Muscle, Smooth, Vascular; Piperazines; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Synaptic Membranes; Tritium; Vasoconstriction | 1983 |
Role of alpha adrenoceptors in hypertension and in antihypertensive drug treatment.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Azepines; Blood Pressure; Calcium Channel Blockers; Clonidine; Guanfacine; Guanidines; Humans; Hypertension; Ketanserin; Methyldopa; Muscle, Smooth, Vascular; Phenylacetates; Piperazines; Piperidines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha; Vascular Resistance | 1984 |
Clinical pharmacokinetics of vasodilators. Part II.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Alprostadil; Amrinone; Carbazoles; Carvedilol; Enoximone; Female; Humans; Iloprost; Imidazoles; Indoramin; Isosorbide Dinitrate; Labetalol; Milrinone; Molsidomine; Nitroglycerin; Nitroprusside; Oxyfedrine; Pentaerythritol Tetranitrate; Phosphodiesterase Inhibitors; Piperazines; Prazosin; Pregnancy; Propanolamines; Pyridones; Theophylline; Trapidil; Vasodilator Agents | 1998 |
Trials
5 trial(s) available for prazosin and urapidil
Article | Year |
---|---|
Double-blind comparison of urapidil and prazosin in the treatment of patients with essential hypertension.
Topics: Adult; Aged; Antihypertensive Agents; Clinical Trials as Topic; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hypertension; Male; Middle Aged; Piperazines; Prazosin; Random Allocation | 1988 |
A comparison of the hemodynamic effects of urapidil, prazosin, and clonidine in healthy volunteers.
Topics: Adult; Antihypertensive Agents; Blood Pressure; Clonidine; Drug Administration Schedule; Heart Rate; Humans; Male; Norepinephrine; Piperazines; Prazosin; Vascular Resistance | 1994 |
Effect of alpha 1-adrenoceptor antagonists, prazosin and urapidil, on a finger skin vasoconstrictor response to cold stimulation.
Topics: Administration, Oral; Adrenergic alpha-Antagonists; Adult; Analysis of Variance; Cold Temperature; Humans; Laser-Doppler Flowmetry; Male; Piperazines; Prazosin; Regional Blood Flow; Skin; Vasoconstriction | 1996 |
Sympathoexcitatory responses to the acute blood pressure fall induced by central or peripheral antihypertensive drugs.
Topics: Adult; Antihypertensive Agents; Blood Pressure; Cross-Over Studies; Double-Blind Method; Heart Rate; Humans; Hypertension; Male; Muscle, Skeletal; Norepinephrine; Piperazines; Prazosin; Sympathetic Nervous System; Sympatholytics | 2000 |
Comparison of 7 α(1)-adrenoceptor antagonists in patients with lower urinary tract symptoms associated with benign prostatic hyperplasia:a short-term crossover study.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adult; Aged; Aged, 80 and over; Cross-Over Studies; Doxazosin; Humans; Indoles; Lower Urinary Tract Symptoms; Male; Middle Aged; Naphthalenes; Piperazines; Prazosin; Prostatic Hyperplasia; Sulfonamides; Tamsulosin; Treatment Outcome | 2013 |
Other Studies
40 other study(ies) available for prazosin and urapidil
Article | Year |
---|---|
QSAR model for drug human oral bioavailability.
Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship | 2000 |
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical | 2010 |
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations | 2010 |
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics | 2010 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests | 2013 |
[Comparison of selective alpha-1 blockades for alpha-receptors in human hypertrophied prostatic adenomas].
Topics: Adenoma; Adrenergic alpha-Antagonists; Aged; Humans; Male; Piperazines; Prazosin; Prostatic Hyperplasia; Prostatic Neoplasms; Quinazolines; Radioligand Assay; Receptors, Adrenergic, alpha | 1992 |
Alpha 1-receptor antagonists urapidil and prazosin inhibit neointima formation in rat carotid artery induced by balloon catheter injury.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Carotid Arteries; Carotid Artery Injuries; Cell Division; DNA; Heart Rate; Male; Muscle, Smooth, Vascular; Piperazines; Prazosin; Rats; Rats, Inbred Strains | 1991 |
The effect of doxazosin, urapidil and indoramin pretreatment on fever produced by E. coli lipopolysaccharide in rabbits.
Topics: Adrenergic alpha-Antagonists; Animals; Anti-Inflammatory Agents, Non-Steroidal; Body Temperature Regulation; Doxazosin; Escherichia coli; Female; Fever; Indoramin; Lipopolysaccharides; Male; Piperazines; Prazosin; Rabbits | 1991 |
The mechanism of the sympathoinhibitory action of urapidil: role of 5-HT1A receptors.
Topics: Anesthesia; Animals; Blood Pressure; Cats; Clonidine; Heart; Heart Rate; Kidney; Male; Piperazines; Prazosin; Receptors, Serotonin; Regional Blood Flow; Spiperone; Splanchnic Nerves; Sympatholytics | 1991 |
Is blockade of alpha 1-adrenoceptors favourable in hypotension induced by stimulation of serotonin1A receptors in conscious dogs?
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Heart Rate; Male; Piperazines; Prazosin; Rats; Receptors, Serotonin; Stimulation, Chemical; Swine; Tetrahydronaphthalenes | 1990 |
Platelet in vitro responses to urapidil and prazosin.
Topics: Adult; Antihypertensive Agents; Blood Platelets; Epinephrine; Female; Humans; Male; Norepinephrine; Piperazines; Platelet Aggregation; Prazosin | 1990 |
Effects of urapidil on 5-hydroxytryptamine induced platelet aggregation and on 14C-5-hydroxytryptamine uptake in platelets.
Topics: Administration, Oral; Adult; Blood Platelets; Carbon Radioisotopes; Epinephrine; Humans; Ketanserin; Nafronyl; Piperazines; Platelet Aggregation Inhibitors; Prazosin; Serotonin; Serotonin Antagonists | 1990 |
Hypotensive effect of urapidil: CNS site and relative contribution.
Topics: Animals; Blood Pressure; Brain; Cats; Female; Heart Rate; Male; Piperazines; Prazosin; Respiration; Sympathetic Nervous System | 1987 |
Antagonism of alpha 1-adrenoceptor-mediated vascular contraction by urapidil in isolated arterial strips of spontaneously hypertensive rats.
Topics: Age Factors; Animals; Antihypertensive Agents; Dose-Response Relationship, Drug; Hypertension; In Vitro Techniques; Male; Norepinephrine; Phentolamine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha; Vasoconstriction; Yohimbine | 1988 |
Importance of central nervous system serotonin-1A receptors for mediating the hypotensive effect of urapidil.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antihypertensive Agents; Blood Pressure; Cats; Heart Rate; Medulla Oblongata; Piperazines; Prazosin; Receptors, Serotonin; Respiration; Spiperone; Tetrahydronaphthalenes | 1989 |
Effects of urapidil on catecholamine turnover and release in the central nervous system of the rat.
Topics: Animals; Blood Pressure; Brain Chemistry; Catecholamines; Chromatography, High Pressure Liquid; Dioxanes; Dopamine; Electric Stimulation; Haloperidol; Idazoxan; In Vitro Techniques; Male; Methoxyhydroxyphenylglycol; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Inbred Strains | 1989 |
Subclassification of alpha 1-adrenoceptor recognition sites by urapidil derivatives and other selective antagonists.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Dioxanes; Heart; In Vitro Techniques; Male; Myocardium; Phenethylamines; Phentolamine; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tetralones; Yohimbine | 1989 |
Suppression of reflex tachycardia by central administration of the alpha-1 adrenoceptor antagonists urapidil and prazosin in anesthetized dogs.
Topics: Adrenergic alpha-Antagonists; Anesthesia; Animals; Antihypertensive Agents; Blood Pressure; Bradykinin; Brain; Dogs; Female; Heart Rate; Indoramin; Male; Phenylephrine; Piperazines; Prazosin; Pressoreceptors; Quinazolines; Reflex; Vascular Resistance | 1985 |
Analysis of adrenoceptor blockade and hypotension elicited by urapidil and prazosin in conscious rat.
Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Antihypertensive Agents; Arginine Vasopressin; Blood Pressure; Enalapril; Enalaprilat; Male; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Renin-Angiotensin System | 1986 |
Effect of alpha 1-adrenoceptor blockade on blood pressure and iliac vascular resistance in normotensive and Goldblatt hypertensive dogs; influence of dietary salt and DOCA-salt.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Captopril; Desoxycorticosterone; Dogs; Female; Hypertension, Renovascular; Iliac Artery; Male; Phenylephrine; Piperazines; Prazosin; Regional Blood Flow; Sodium, Dietary; Vascular Resistance | 1987 |
A clinical approach for the identification of peripheral pre- and post-synaptic alpha-adrenergic receptors.
Topics: Adult; Blood Pressure; Heart Rate; Humans; Male; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Synapses; Yohimbine | 1986 |
A comparison of the effects of doxazosin and alfuzosin with those of urapidil on preganglionic sympathetic nerve activity in anaesthetised cats.
Topics: Action Potentials; Animals; Blood Pressure; Cats; Doxazosin; Male; Piperazines; Prazosin; Quinazolines; Receptors, Adrenergic, alpha; Sympathetic Nervous System; Vascular Resistance | 1986 |
Characterization of vasodilators by comparison of their effects on blood pressure, counterregulation and myocardial oxygen demand in conscious normotensive dogs.
Topics: Animals; Blood Pressure; Dihydralazine; Dogs; Female; Heart Rate; Isosorbide Dinitrate; Labetalol; Male; Molsidomine; Myocardium; Oxygen Consumption; Piperazines; Prazosin; Pyridazines; Renin; Sydnones; Vasodilator Agents | 1985 |
Effect of urapidil, clonidine, and prazosin on sympathetic tone in conscious rats.
Topics: Animals; Blood Pressure; Clonidine; Electrodes; Heart Rate; Piperazines; Prazosin; Pressoreceptors; Rats; Rats, Inbred SHR; Splanchnic Nerves; Sympathetic Nervous System | 1986 |
Effects of urapidil, clonidine, prazosin and propranolol on autonomic nerve activity, blood pressure and heart rate in anaesthetized rats and cats.
Topics: Anesthesia; Animals; Antihypertensive Agents; Autonomic Nervous System; Blood Pressure; Cats; Clonidine; Female; Heart Rate; Hemodynamics; In Vitro Techniques; Male; Neurons; Piperazines; Prazosin; Propranolol; Quinazolines; Rats; Rats, Inbred Strains; Species Specificity; Splanchnic Nerves; Sympathetic Nervous System; Vagus Nerve | 1985 |
Cardiovascular effects and interaction with adrenoceptors of urapidil.
Topics: Animals; Antihypertensive Agents; Binding, Competitive; Cats; Clonidine; Decerebrate State; Female; Hemodynamics; Hexobarbital; In Vitro Techniques; Infusions, Parenteral; Male; Membranes; Mice; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Piperazines; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rats, Inbred WKY; Receptors, Adrenergic | 1985 |
Comparative central and peripheral antihypertensive mechanisms of urapidil and prazosin.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Brain; Heart Rate; Injections, Intravenous; Injections, Intraventricular; Male; Piperazines; Prazosin; Pressoreceptors; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Sympathectomy; Vascular Resistance | 1984 |
Comparative effects of urapidil, prazosin, and clonidine on ligand binding to central nervous system receptors, arterial pressure, and heart rate in experimental animals.
Topics: Animals; Antihypertensive Agents; Binding, Competitive; Blood Pressure; Brain; Cats; Clonidine; Dose-Response Relationship, Drug; Female; Heart Rate; Injections, Intravenous; Injections, Intraventricular; Male; Piperazines; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Muscarinic | 1984 |
Antihypertensive drugs: proposed sites and mechanisms of action.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Cats; Clonidine; Denervation; Dogs; Heart Rate; Methysergide; Moxisylyte; Phentolamine; Piperazines; Prazosin; Uracil | 1981 |
Systemic and regional hemodynamic effects of acute and prolonged treatment with urapidil or prazosin in normotensive and spontaneously hypertensive rats.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Cardiac Output; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Hypertension; Male; Piperazines; Prazosin; Pressoreceptors; Quinazolines; Rats; Rats, Inbred SHR; Regional Blood Flow; Time Factors; Vascular Resistance | 1984 |
Hemodynamic and neural effects of urapidil and prazosin in essential hypertensives.
Topics: Administration, Oral; Antihypertensive Agents; Blood Pressure; Heart Rate; Humans; Hypertension; Peroneal Nerve; Piperazines; Prazosin; Sympathetic Fibers, Postganglionic | 1994 |
Comparative study on alpha 1-adrenoceptor antagonist binding in human prostate and aorta.
Topics: Adrenergic alpha-Antagonists; Aged; Aorta; Binding Sites; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Humans; Kinetics; Male; Middle Aged; Naphthalenes; Piperazines; Prazosin; Prostate; Sulfonamides; Tamsulosin | 1994 |
Regulation of renal artery smooth muscle tone by alpha1-adrenoceptors: role of voltage-gated calcium channels and intracellular calcium stores.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cell Membrane; Diltiazem; Dioxanes; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Ischemia; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Phenoxybenzamine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Renal Artery; Renal Circulation; Swine; Thapsigargin; Verapamil | 2000 |
Moxonidine, an antihypertensive agent, is permissive to alpha1-adrenergic receptor pathway in the rat-tail artery.
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Antihypertensive Agents; Drug Interactions; Imidazoles; Male; Muscle, Smooth, Vascular; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Vasoconstriction; Yohimbine | 2004 |
Effects of tamsulosin on hypogastric nerve stimulation-induced intraurethral pressure elevation in male and female dogs under anesthesia.
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Dogs; Female; Hypogastric Plexus; Male; Naphthalenes; Piperazines; Prazosin; Pressure; Sex Factors; Sulfonamides; Tamsulosin; Urethra | 2004 |
Effects of tamsulosin on resting urethral pressure and arterial blood pressure in anaesthetized female dogs.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Female; Piperazines; Prazosin; Pressure; Sulfonamides; Tamsulosin; Urethra | 2006 |
Synthesis of a quinazoline derivative: a new α₁-adrenoceptor ligand for conjugation to quantum dots to study α₁-adrenoceptors in living cells.
Topics: Adrenergic alpha-1 Receptor Antagonists; Biological Assay; Biotin; Drug Design; Drug Evaluation, Preclinical; HEK293 Cells; Humans; Ligands; Molecular Structure; Molecular Weight; Piperazines; Polyethylene Glycols; Prazosin; Protein Binding; Quantum Dots; Quinazolines; Receptors, Adrenergic, alpha-1 | 2011 |
Effects of α1-adrenoceptor antagonists on phenylephrine-induced salivary secretion and intraurethral pressure elevation in anesthetized rats.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Dose-Response Relationship, Drug; Drug Interactions; Indoles; Male; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Saliva; Salivary Glands; Sulfonamides; Tamsulosin; Urethra | 2012 |