Page last updated: 2024-08-16

prazosin and bmy 7378

prazosin has been researched along with bmy 7378 in 90 studies

Research

Studies (90)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's32 (35.56)18.2507
2000's49 (54.44)29.6817
2010's7 (7.78)24.3611
2020's2 (2.22)2.80

Authors

AuthorsStudies
Audinot, V; Bervoets, K; Brocco, M; Canton, H; Gobert, A; Le Marouille-Girardon, S; Millan, MJ; Peglion, JL1
Bock, MG; Broten, TP; Chang, RS; DiSalvo, J; Forray, C; Patane, MA; Ransom, RW; Scott, AL1
Bolognesi, ML; Budriesi, R; Chiarini, A; Leonardi, A; Melchiorre, C; Poggesi, E1
Pedretti, A; Testa, B; Villa, L; Vistoli, G1
Araújo, CV; Barreiro, EJ; Castro, HC; da Silva Ferreira, M; da Silva, LL; Fraga, CA; Miranda, AL; Nascimento, JB; Noël, F; Romeiro, LA; Silva, CL; Tibiriçá, E1
Ballard, S; Blagg, J; Fox, D; Kenny, B1
Budriesi, R; Chiarini, A; Leonardi, A; Melchiorre, C; Minarini, A1
Barrett, JE; Gleeson, S1
Moser, PC1
Bengtsson, HJ; Hjorth, S; Lundberg, JF; Milano, S; Sharp, T1
Chalmers, DH; Kenny, BA; Naylor, AM; Philpott, PC1
Chemtob, S; Deng, XF; Varma, DR1
Hasegawa, Y; Mizuchi, A; Ono, H; Otsu, T; Wada, T1
Deng, XF; Varma, DR1
DeMey, JG; Janssen, GM; Stassen, FR; Willemsen, MJ1
Macmillan, JB; McGrath, JC; Smith, KM1
Hussain, MB; Marshall, I2
Daniel, EE; Gaspar, V; Kwan, CY; Low, AM; Lu-Chao, H1
Endoh, M; Yang, HT1
Hasegawa, Y; Ono, H; Wada, T1
Kadavil, EA; Oriowo, MA; Yousif, M1
Brown, RD; Daniel, EE; Kwan, CY; Low, AM; Lu-Chao, H; Wang, YF1
Foster, HE; Latifpour, J; Nishi, K; Saito, M; Weiss, RM; Yoshida, M1
Dang, H; Gruber, DD; Scofield, MA; Shimozono, M; Wangemann, P1
Du, XJ; Han, C; Yan, M; Zhang, Y1
Hiraoka, Y; Kato, H; Morikawa, K; Muramatsu, I; Nagata, O; Ohmura, T; Oshita, M; Taniguchi, T; Watanabe, Y1
Errasti, AE; Rothlin, RP; Sardi, SP; Torres, RM; Velo, MP1
Saxena, PR; Stam, WB; Van der Graaf, PH1
Enomoto, K; Koike, K; Satoh, M; Takayanagi, I1
Han, QD; Zhang, YY; Zhu, WZ1
Avellar, MC; Megale, A; Porto, CS; Silva, MA1
Berkowitz, DE; Booth, JV; Cozart, KL; D'Amico, EB; El-Moalem, H; Funk, BL; Marucci, L; Page, SO; Richardson, CD; Rudner, XL; Schwinn, DA; Winters, B1
Arias-Montaño, JA; Berger, VA; Soria-Jasso, LE; Young, JM1
García-Sáinz, JA; Gottfried-Blackmore, A; Romero-Avila, MT; Vázquez-Prado, J1
Sasa, M; Tanimitsu, N; Tsuru, H; Yajin, K1
Daly, CJ; Heeley, RP; MacKenzie, JF; McGrath, JC; Pediani, JD1
D'Ocon, P; Gisbert, R; Ivorra, MD; Noguera, MA1
Saxena, PR; Valdivia, LF; Villalón, CM; Willems, EW1
Gaivin, RJ; Gonzalez-Cabrera, P; Perez, DM; Ross, SA; Waugh, DJ; Yun, J; Zuscik, MJ1
De Vries, P; Heiligers, JP; Kapoor, K; Saxena, PR; Tom, B; Villalón, CM; Willems, EW1
Coats, P; Hillier, C; Jarajapu, YP; MacDonald, A; McGrath, JC1
Hillier, C; Jarajapu, YP; MacDonald, A1
Gaitanaki, C; Lazou, A; Seraskeris, S1
Koike, K; Yamamoto, Y2
García-Sáinz, JA; González-Espinosa, C; González-Espinosa, D; Mora-Rodríguez, DM; Romero-Avila, MT1
Chiba, S; Taguchi, Y; Yang, XP1
Anselmi, E; D'Ocon, P; Gisbert, R; Ivorra, MD; Miquel, R; Noguera, MA; Ziani, K1
D'Ocon, P; Gisbert, R; Ivorra, MD; Noguera, MA; Ziani, K1
Katus, HA; Kemken, D; Kurz, T; Mier, K; Richardt, G1
Brodde, OE; Dhein, S; Giessler, C; Silber, RE; Wangemann, T1
Dyer, DC; Ioudina, MV1
Horinouchi, T; Koike, K; Shibano, M; Tanaka, Y; Yamamoto, Y1
Cleary, L; Docherty, JR; Vandeputte, C1
Koss, MC; Yu, Y1
Campos, M; Morais, Pde L; Pupo, AS1
Guarneri, L; Leonardi, A; Testa, R; Velasco, C1
Capello, SA; Chou, EC; Levin, RM; Longhurst, PA1
Hillier, C; MacDonald, A; Zacharia, J2
Eltze, M; Jähnichen, S; Pertz, HH1
Hiraizumi-Hiraoka, Y; Israilova, M; Kunitomo, M; Muramatsu, I; Shinozuka, K; Suzuki, F; Taki, N; Tanaka, T; Taniguchi, T; Zhang, L1
Hieble, JP1
Colston, JF; Deighan, C; McGrath, JC; Woollhead, AM1
Chen, K; Chen, M; Han, C; Lu, Z; Song, Y; Yan, J; Zhang, Y1
Alewood, D; Chen, Z; Kamikihara, SY; Lewis, RJ; Lima, V; Minneman, KP; Mueller, A; Pupo, AS; Raymundi, V1
Ding, X; McCune, DF; Murray, PA; Perez, DM; Sohn, JT1
Cotecchia, S; Hiroyama, M; Hosoda, C; Kitamura, T; Koike, K; Koshimizu, TA; Shibano, M; Tanaka, Y; Tanoue, A; Tsujimoto, G1
Hallberg, M; Lindblom, J; Magnusson, K; Nyberg, F; Petrovska, R; Uhlén, S1
Cunha, FQ; de Andrade, CR; de Godoy, MA; de Oliveira, AM; de Souza, HP; Eberlin, MN; Fukada, SY; Haddad, R; Laurindo, FR; Olivon, VC1
Gallardo-Ortiz, IA; Gómez-Zamudio, JH; Ibarra, M; López-Guerrero, JJ; Parés-Hipólito, J; Santamaría-Ortiz, J; Villalobos-Molina, R1
Doze, VA; Hillman, KL; Porter, JE1
Chartier, D; Ehrlich, JR; Hébert, TE; Nattel, S; Qi, X; Yeh, YH1
Bexis, S; Docherty, JR1
Bustamante, S; García-Sacristán, A; Hernández, M; Martínez, MP; Navarro-Dorado, J; Orensanz, LM; Prieto, D; Recio, P1
Anisuzzaman, AS; Morishima, S; Muramatsu, I; Sathi, ZS; Suzuki, F; Tanaka, T; Yoshiki, H1
Dmitrieva, N; Nagabukuro, H; Zhang, G1
Clair, DK; García-Cazarín, ML; Piascik, MT; Smith, JL1
Hoyano, Y; Itoh, Y; Kobayashi, S; Kohri, K; Kubota, Y; Kusama, H; Tomiyama, Y; Yamazaki, Y1
Chu, CC; Lin, MT; Shieh, JP; Wang, JJ1
Kobayashi, S; Kohri, K; Kojima, Y; Kubota, Y; Sasaki, S; Tomiyama, Y1
Bockman, CS; Dang, HK; Gruber, DD; Scofield, MA; Wangemann, P; Witt, KM1
Docherty, JR2
Fields, AM; Hoover, JM; Ibrahim, IN; Kaye, AD1
Fisher, SA; Mauban, JR; Raina, H; Wier, WG; Zacharia, J1
Chapple, CR; Chess-Williams, R; Davis, BJ; Sellers, DJ; Wiener, M1
Alsufyani, HA; Docherty, JR; McCormick, PA1
Alsufyani, HA; Daly, C; Docherty, JR1

Reviews

1 review(s) available for prazosin and bmy 7378

ArticleYear
Pharmacological options in the treatment of benign prostatic hyperplasia.
    Journal of medicinal chemistry, 1997, Apr-25, Volume: 40, Issue:9

    Topics: 5-alpha Reductase Inhibitors; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Controlled Clinical Trials as Topic; Endothelins; Enzyme Inhibitors; Humans; Male; Prostate; Prostatic Hyperplasia; Receptors, Adrenergic, alpha; Structure-Activity Relationship

1997

Other Studies

89 other study(ies) available for prazosin and bmy 7378

ArticleYear
Characterization of potent and selective antagonists at postsynaptic 5-HT1A receptors in a series of N4-substituted arylpiperazines.
    Journal of medicinal chemistry, 1995, Sep-29, Volume: 38, Issue:20

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Male; Piperazines; Rats; Rats, Wistar; Serotonin Antagonists; Structure-Activity Relationship

1995
4-Amino-2-[4-[1-(benzyloxycarbonyl)-2(S)- [[(1,1-dimethylethyl)amino]carbonyl]-piperazinyl]-6, 7-dimethoxyquinazoline (L-765,314): a potent and selective alpha1b adrenergic receptor antagonist.
    Journal of medicinal chemistry, 1998, Apr-09, Volume: 41, Issue:8

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Humans; Male; Organ Specificity; Prazosin; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Spinal Cord; Structure-Activity Relationship

1998
Design, synthesis, and biological activity of prazosin-related antagonists. Role of the piperazine and furan units of prazosin on the selectivity for alpha1-adrenoreceptor subtypes.
    Journal of medicinal chemistry, 1998, Nov-19, Volume: 41, Issue:24

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; CHO Cells; Cricetinae; Drug Design; Furans; Humans; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Piperazine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Spleen; Structure-Activity Relationship; Vas Deferens

1998
Range and sensitivity as descriptors of molecular property spaces in dynamic QSAR analyses.
    Journal of medicinal chemistry, 2005, Jul-28, Volume: 48, Issue:15

    Topics: Chemical Phenomena; Chemistry, Physical; Ligands; Models, Molecular; Molecular Conformation; Monte Carlo Method; Quantitative Structure-Activity Relationship; Receptors, Adrenergic, alpha-1; Solvents

2005
Discovery of LASSBio-772, a 1,3-benzodioxole N-phenylpiperazine derivative with potent alpha 1A/D-adrenergic receptor blocking properties.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:7

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Aorta; Benzodioxoles; Cell Membrane; Hepatocytes; Humans; Liver; Male; Phenylephrine; Piperazines; Prazosin; Protein Binding; Protein Isoforms; Rabbits; Rats; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Tissue Culture Techniques; Tritium; Vasoconstriction

2011
Search for alpha 1-adrenoceptor subtypes selective antagonists: design, synthesis and biological activity of cystazosin, an alpha 1D-adrenoceptor antagonist.
    Bioorganic & medicinal chemistry letters, 1998, Jun-02, Volume: 8, Issue:11

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Drug Design; Humans; In Vitro Techniques; Male; Quinazolines; Quinoxalines; Rats; Receptors, Adrenergic, alpha-1; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Spleen; Structure-Activity Relationship; Vas Deferens

1998
Discriminative stimulus effects of 8-OH-DPAT in pigeons: antagonism studies with the putative 5-HT1A receptor antagonists BMY 7378 and NAN-190.
    European journal of pharmacology, 1992, Jul-07, Volume: 217, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Columbidae; Discrimination, Psychological; Dose-Response Relationship, Drug; Indoles; Pindolol; Piperazines; Prazosin; Serotonin Antagonists

1992
The effect of putative 5-HT1A receptor antagonists on 8-OH-DPAT-induced hypothermia in rats and mice.
    European journal of pharmacology, 1991, Feb-07, Volume: 193, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Body Temperature; Dioxanes; Dose-Response Relationship, Drug; Hypothermia, Induced; Male; Mice; Piperazines; Prazosin; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1991
Studies on the role of 5-HT1A autoreceptors and alpha 1-adrenoceptors in the inhibition of 5-HT release--I. BMY7378 and prazosin.
    Neuropharmacology, 1995, Volume: 34, Issue:6

    Topics: Animals; Dose-Response Relationship, Drug; Hippocampus; Male; Microdialysis; Pindolol; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Serotonin; Serotonin; Time Factors

1995
Characterization of an alpha 1D-adrenoceptor mediating the contractile response of rat aorta to noradrenaline.
    British journal of pharmacology, 1995, Volume: 115, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Aorta; Binding, Competitive; Dose-Response Relationship, Drug; Doxazosin; Male; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Vasodilation

1995
Characterization of alpha 1 D-adrenoceptor subtype in rat myocardium, aorta and other tissues.
    British journal of pharmacology, 1996, Volume: 119, Issue:2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Blood Pressure; Cardiotonic Agents; In Vitro Techniques; Liver; Male; Myocardial Contraction; Myocardium; Phenylephrine; Piperazines; Prazosin; Prostate; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Salivary Glands; Spleen; Tritium; Vas Deferens

1996
Characterization of alpha 1-adrenoceptor subtypes in rat spinal cord.
    European journal of pharmacology, 1996, Sep-26, Volume: 312, Issue:2

    Topics: Animals; Male; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spinal Cord

1996
Alpha 1D-adrenoceptors do not contribute to inotropic responses of neonatal rat myocardium.
    Journal of cardiovascular pharmacology, 1997, Volume: 29, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Aorta; Cell Membrane; Cerebral Cortex; Heart Ventricles; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Myocardium; Phenylephrine; Piperazines; Prazosin; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Vasoconstrictor Agents; Ventricular Function

1997
Alpha 1-adrenoceptor subtypes in rat aorta and mesenteric small arteries are preserved during left ventricular dysfunction post-myocardial infarction.
    Cardiovascular research, 1997, Volume: 33, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Calcium Channel Blockers; Dihydropyridines; In Vitro Techniques; Male; Mesenteric Arteries; Myocardial Infarction; Piperazines; Prazosin; Protein Binding; Radioligand Assay; Rats; Rats, Inbred WKY; Rats, Wistar; Receptors, Adrenergic, alpha-1; Ventricular Dysfunction, Left

1997
Investigation of alpha1-adrenoceptor subtypes mediating vasoconstriction in rabbit cutaneous resistance arteries.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Acetonitriles; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Male; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha-1; Skin; Tetrahydronaphthalenes; Vascular Resistance; Vasoconstriction

1997
Characterization of alpha1-adrenoceptor subtypes mediating contractions to phenylephrine in rat thoracic aorta, mesenteric artery and pulmonary artery.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Dioxanes; Dioxins; Dose-Response Relationship, Drug; In Vitro Techniques; Indoles; Indoramin; Isometric Contraction; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Oxathiins; Phenylephrine; Piperazines; Prazosin; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Spiro Compounds; Vasoconstrictor Agents

1997
Characterization of alpha-adrenoceptors in canine mesenteric vein.
    Journal of cardiovascular pharmacology, 1997, Volume: 30, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Dogs; Female; Male; Mesenteric Veins; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Yohimbine

1997
Pharmacological evidence for alpha(1D)-adrenoceptors in the rabbit ventricular myocardium: analysis with BMY 7378.
    British journal of pharmacology, 1997, Volume: 122, Issue:8

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Calcium Channel Blockers; Dihydropyridines; Dioxanes; Dose-Response Relationship, Drug; Heart; Heart Ventricles; Male; Myocardial Contraction; Myocardium; Papillary Muscles; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha-1

1997
Characterization of alpha1-adrenoceptor subtypes in facilitation of rat spinal motoneuron activity.
    European journal of pharmacology, 1997, Dec-04, Volume: 340, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Bridged-Ring Compounds; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Epinephrine; Male; Methoxamine; Motor Neurons; Norepinephrine; Oxazines; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Spinal Cord

1997
Heterogeneity of alpha 1-adrenoceptor subtypes mediating noradrenaline-induced contractions of the rat superior mesenteric artery.
    Pharmacology, 1998, Volume: 56, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dopamine Antagonists; Dose-Response Relationship, Drug; Male; Mesenteric Artery, Superior; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spiperone; Vasoconstriction; Vasoconstrictor Agents

1998
Pharmacological and immunocytochemical characterization of subtypes of alpha-1 adrenoceptors in dog aorta.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 285, Issue:2

    Topics: Animals; Aorta; Clonidine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Immunohistochemistry; Indoles; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Spiro Compounds

1998
Characterization, localization and distribution of alpha1 adrenoceptor subtype in male rabbit urethra.
    The Journal of urology, 1998, Volume: 160, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Autoradiography; Dioxanes; Immunohistochemistry; Male; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha-1; Spiperone; Urethra

1998
Alpha1A-adrenergic receptors mediate vasoconstriction of the isolated spiral modiolar artery in vitro.
    Hearing research, 1998, Volume: 119, Issue:1-2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Arteries; Cochlea; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gerbillinae; Nitric Oxide Synthase; Nitroarginine; Norepinephrine; Piperazines; Polymerase Chain Reaction; Prazosin; Propanolamines; Receptors, Adrenergic, alpha-1; RNA; Vasoconstriction; Yohimbine

1998
Functional assessment of alpha 1-adrenoceptor subtypes in porcine coronary artery.
    Clinical and experimental pharmacology & physiology, 1998, Volume: 25, Issue:9

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Coronary Vessels; Dioxanes; Humans; In Vitro Techniques; Kinetics; Male; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Swine; Vasoconstriction

1998
Binding and functional characterization of alpha1-adrenoceptor subtypes in the rat prostate.
    European journal of pharmacology, 1999, Jan-29, Volume: 366, Issue:1

    Topics: Acetonitriles; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Dioxanes; Dose-Response Relationship, Drug; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Prostate; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Tritium

1999
Characterization of alpha1-adrenoceptor subtypes mediating vasoconstriction in human umbilical vein.
    British journal of pharmacology, 1999, Volume: 126, Issue:2

    Topics: Adrenergic Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Humans; In Vitro Techniques; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Umbilical Veins; Vasoconstriction; Vasoconstrictor Agents

1999
Analysis of alpha 1L-adrenoceptor pharmacology in rat small mesenteric artery.
    British journal of pharmacology, 1999, Volume: 127, Issue:3

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Cresols; Imidazoles; In Vitro Techniques; Indoles; Male; Mesenteric Arteries; Norepinephrine; Piperazines; Potassium; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Tetrahydronaphthalenes

1999
Analysis of alpha1-adrenoceptor subtypes in rabbit aorta and arteries: regional difference and co-existence.
    European journal of pharmacology, 1999, Jun-18, Volume: 374, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Arteries; Dose-Response Relationship, Drug; Drug Interactions; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Piperazines; Prazosin; Protein Binding; Rabbits; Receptors, Adrenergic, alpha-1

1999
Characterization of subtype of alpha 1-adrenoceptor mediating vasoconstriction in perfused rat mesenteric vascular bed.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1999, Volume: 20, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Indoles; Male; Mesenteric Artery, Superior; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vasoconstriction; Yohimbine

1999
Expression and pharmacological characterization of alpha1-adrenoceptors in rat seminal vesicle.
    European journal of pharmacology, 1999, Sep-24, Volume: 381, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium Channel Blockers; Clonidine; Dioxanes; Epinephrine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Phenoxybenzamine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Seminal Vesicles

1999
Subtype specific regulation of human vascular alpha(1)-adrenergic receptors by vessel bed and age.
    Circulation, 1999, Dec-07, Volume: 100, Issue:23

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Aged; Aging; Aorta; Arteries; Celiac Artery; Dopamine Antagonists; Female; Femoral Artery; Gene Expression; Hepatic Artery; Humans; Iliac Artery; In Vitro Techniques; Male; Mammary Arteries; Middle Aged; Phenylephrine; Piperazines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha-1; Renal Artery; RNA, Messenger; Saphenous Vein; Spiperone; Splenic Artery; Vasoconstriction

1999
Characterisation of alpha1B-adrenoceptors linked to inositol phosphate formation and calcium mobilisation in human astrocytoma U373 MG cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 360, Issue:5

    Topics: Adrenergic alpha-Antagonists; Astrocytoma; Calcium; Cell Membrane; Clonidine; Dihydropyridines; Dioxanes; Dose-Response Relationship, Drug; Humans; Inositol Phosphates; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Thymidine; Tumor Cells, Cultured

1999
Protein kinase C-mediated phosphorylation and desensitization of human alpha(1b)-adrenoceptors.
    European journal of pharmacology, 1999, Dec-03, Volume: 385, Issue:2-3

    Topics: Animals; Binding, Competitive; Calcium; Cell Line; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Indoles; Inositol Phosphates; Membranes; Norepinephrine; Phentolamine; Phosphorylation; Piperazines; Prazosin; Precipitin Tests; Protein Kinase C; Radioligand Assay; Receptors, Adrenergic, alpha-1; RNA, Messenger; Sulfur Radioisotopes; Tetradecanoylphorbol Acetate; Tritium

1999
alpha(1)-adrenoceptor subtypes and effect of alpha(1A)-adrenoceptor agonist NS-49 on guinea pig nasal mucosa vasculature.
    European journal of pharmacology, 2000, Jan-03, Volume: 387, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anilides; Animals; Blood Vessels; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Male; Nasal Mucosa; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Spiperone; Vasoconstriction; Yohimbine

2000
Alpha(1)-adrenoceptor subtypes mediating contractions of the rat mesenteric artery.
    European journal of pharmacology, 2000, Apr-21, Volume: 395, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; Endothelium, Vascular; Imidazoles; In Vitro Techniques; Indoles; Indoramin; Male; Mesenteric Arteries; Methoxamine; Oxathiins; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Vasoconstriction; Vasoconstrictor Agents

2000
Single-cell recombinant pharmacology: bovine alpha(1a)-adrenoceptors in rat-1 fibroblasts release intracellular ca(2+), display subtype-characteristic agonism and antagonism, and exhibit an antagonist-reversible inverse concentration-response phase.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Calcium Signaling; Cattle; Dioxanes; Dose-Response Relationship, Drug; Imidazoles; Phenylalanine; Piperazines; Prazosin; Rats; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; Tetrahydronaphthalenes

2000
Functional evidence of a constitutively active population of alpha(1D)-adrenoceptors in rat aorta.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 295, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Arteries; Calcium; Female; In Vitro Techniques; Inositol Phosphates; Muscle Contraction; Muscle Hypertonia; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tail

2000
The role of several alpha(1)- and alpha(2)-adrenoceptor subtypes mediating vasoconstriction in the canine external carotid circulation.
    British journal of pharmacology, 2001, Volume: 132, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Carotid Artery, External; Dogs; Female; Imidazoles; Indoles; Isoindoles; Male; Phenylephrine; Piperazines; Prazosin; Quinolizines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Regional Blood Flow; Vasoconstriction

2001
Phe-308 and Phe-312 in transmembrane domain 7 are major sites of alpha 1-adrenergic receptor antagonist binding. Imidazoline agonists bind like antagonists.
    The Journal of biological chemistry, 2001, Jul-06, Volume: 276, Issue:27

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Cell Membrane; Clonidine; Conserved Sequence; Cricetinae; Dihydropyridines; Dioxanes; Humans; Imidazoles; Models, Molecular; Molecular Sequence Data; Oxymetazoline; Phenylalanine; Piperazines; Prazosin; Protein Structure, Secondary; Rats; Receptors, Adrenergic, alpha-1; Structure-Activity Relationship

2001
Alpha1-adrenoceptor subtypes mediating vasoconstriction in the carotid circulation of anaesthetized pigs: possible avenues for antimigraine drug development.
    Cephalalgia : an international journal of headache, 2001, Volume: 21, Issue:2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Dose-Response Relationship, Drug; Female; Hemodynamics; Infusions, Intra-Arterial; Migraine Disorders; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Swine; Vasoconstriction

2001
Functional characterization of alpha(1)-adrenoceptor subtypes in human skeletal muscle resistance arteries.
    British journal of pharmacology, 2001, Volume: 133, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Arteries; Clonidine; Dose-Response Relationship, Drug; Humans; Imidazoles; In Vitro Techniques; Muscle, Skeletal; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes; Vasoconstriction

2001
The alpha(1A)-adrenoceptor subtype mediates contraction in rat femoral resistance arteries.
    European journal of pharmacology, 2001, Jun-22, Volume: 422, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Femoral Artery; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Naphthyridines; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes; Vascular Resistance; Vasoconstriction

2001
alpha(1D)-Adrenoceptors do not contribute to phosphoinositide hydrolysis in adult rat cardiac myocytes.
    Archives of biochemistry and biophysics, 2001, Aug-01, Volume: 392, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Epinephrine; Heart; Hydrolysis; Kinetics; Male; Models, Cardiovascular; Myocardium; Phosphatidylinositols; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1

2001
Characterization of alpha1-adrenoceptor-mediated contraction in the mouse thoracic aorta.
    European journal of pharmacology, 2001, Jul-20, Volume: 424, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Buspirone; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Epinephrine; In Vitro Techniques; Male; Methoxamine; Mice; Models, Biological; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Serotonin Receptor Agonists; Statistics as Topic; Vasoconstriction

2001
Molecular cloning and functional expression of the guinea pig alpha(1a)-adrenoceptor.
    European journal of pharmacology, 2001, Aug-31, Volume: 426, Issue:3

    Topics: Adrenergic Agonists; Adrenergic Antagonists; Amino Acid Sequence; Animals; Base Sequence; Binding, Competitive; Cloning, Molecular; COS Cells; DNA, Complementary; Dose-Response Relationship, Drug; Epinephrine; Gene Expression; Guinea Pigs; Methoxamine; Molecular Sequence Data; Norepinephrine; Oxathiins; Oxymetazoline; Phentolamine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Sequence Alignment; Sequence Analysis, DNA; Sequence Homology, Amino Acid; Sulfonamides; Tamsulosin; Tritium

2001
Existence of alpha(1A)- and alpha(1B)-adrenoceptor subtypes in canine mandibular alveolar arteries.
    Clinical and experimental pharmacology & physiology, 2001, Volume: 28, Issue:9

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Alveolar Process; Animals; Arteries; Clonidine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Male; Mandible; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Vasoconstriction; Xylazine; Yohimbine

2001
alpha(1)-Adrenoceptor subtypes in the mouse mesenteric artery and abdominal aorta.
    British journal of pharmacology, 2001, Volume: 134, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Abdominal; Dioxanes; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Mesenteric Arteries; Mice; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Vasoconstriction

2001
Pathological role of a constitutively active population of alpha(1D)-adrenoceptors in arteries of spontaneously hypertensive rats.
    British journal of pharmacology, 2002, Volume: 135, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Age Factors; Animals; Antihypertensive Agents; Aorta, Thoracic; Arteries; Captopril; Dose-Response Relationship, Drug; Hemodynamics; Hypertension; Iliac Artery; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Tail; Vasoconstriction; Vasodilation

2002
Modulatory role of a constitutively active population of alpha(1D)-adrenoceptors in conductance arteries.
    American journal of physiology. Heart and circulatory physiology, 2002, Volume: 282, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta; Arteries; Calcium; Clonidine; Dose-Response Relationship, Drug; Female; Iliac Artery; Mesenteric Arteries; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vascular Resistance

2002
Adrenergic activation of cardiac phospholipase D: role of alpha(1)-adrenoceptor subtypes.
    Cardiovascular research, 2002, Volume: 54, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Cardiomegaly; Clonidine; Dioxanes; Male; Myocardium; Norepinephrine; Perfusion; Phospholipase D; Piperazines; Prazosin; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Signal Transduction; Stimulation, Chemical

2002
Noradrenaline-induced contraction of human saphenous vein and human internal mammary artery: involvement of different alpha-adrenoceptor subtypes.
    Naunyn-Schmiedeberg's archives of pharmacology, 2002, Volume: 366, Issue:2

    Topics: Adrenergic alpha-Antagonists; Aged; Clonidine; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Male; Mammary Arteries; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha; Regression Analysis; Saphenous Vein; Yohimbine

2002
Pharmacological characterization of alpha1-adrenoceptor subtypes in the bovine tail artery.
    Journal of veterinary pharmacology and therapeutics, 2002, Volume: 25, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Cattle; Dioxanes; Dose-Response Relationship, Drug; Imidazoles; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Tail; Tetrahydronaphthalenes; Vasoconstriction

2002
Pharmacological characterization of alpha1-adrenoceptor in mouse iliac artery.
    European journal of pharmacology, 2002, Dec-05, Volume: 456, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; Iliac Artery; In Vitro Techniques; Male; Mice; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Vasoconstriction

2002
Investigation of postjunctional alpha1- and alpha2-adrenoceptor subtypes in vas deferens from wild-type and alpha(2A/D)-adrenoceptor knockout mice.
    British journal of pharmacology, 2003, Volume: 138, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Cocaine; Electric Stimulation; Imidazoles; Indoles; Isoindoles; Isometric Contraction; Male; Mice; Mice, Knockout; Nifedipine; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Purinergic; Suramin; Thymine; Vas Deferens; Yohimbine

2003
Functional characterization of alpha-adrenoceptors mediating pupillary dilation in rats.
    European journal of pharmacology, 2003, Jun-20, Volume: 471, Issue:2

    Topics: Adrenergic alpha-Antagonists; Adrenergic Fibers; Animals; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Injections, Intravenous; Male; Mydriasis; Norepinephrine; Phenoxybenzamine; Phentolamine; Piperazines; Prazosin; Pupil; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Yohimbine

2003
Effects of castration and of testosterone replacement on alpha(1)-adrenoceptor subtypes in the rat vas deferens.
    European journal of pharmacology, 2003, Jun-20, Volume: 471, Issue:2

    Topics: Animals; Castration; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Male; Muscle Contraction; Neuronal Plasticity; Norepinephrine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Testosterone; Time Factors; Vas Deferens; Yohimbine

2003
Effects of intravenous and infravesical administration of suramin, terazosin and BMY 7378 on bladder instability in conscious rats with bladder outlet obstruction.
    BJU international, 2003, Volume: 92, Issue:1

    Topics: Administration, Intravesical; Adrenergic alpha-Antagonists; Animals; Female; Infusions, Intravenous; Ligation; Piperazines; Prazosin; Purinergic Antagonists; Rats; Rats, Sprague-Dawley; Suramin; Urethral Obstruction; Urinary Bladder Neck Obstruction; Urination; Urination Disorders; Urodynamics

2003
Excitatory alpha1-adrenergic receptors predominate over inhibitory beta-receptors in rabbit dorsal detrusor.
    The Journal of urology, 2003, Volume: 170, Issue:6 Pt 1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Piperazines; Prazosin; Rabbits; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Urinary Bladder

2003
Alpha1-adrenoceptor subtypes involved in vasoconstrictor responses to exogenous and neurally released noradrenaline in rat femoral resistance arteries.
    British journal of pharmacology, 2004, Volume: 141, Issue:6

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Cocaine; Dose-Response Relationship, Drug; Electric Stimulation; Femoral Artery; In Vitro Techniques; Male; Muscle, Skeletal; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Vascular Resistance; Vasoconstriction; Vasoconstrictor Agents

2004
Evidence that alpha(1B)-adrenoceptors are involved in noradrenaline-induced contractions of rat tail artery.
    European journal of pharmacology, 2004, Mar-19, Volume: 488, Issue:1-3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Algorithms; Animals; Arteries; Clonidine; Dioxins; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Piperazines; Prazosin; Pyrimidinones; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tail

2004
Alpha-1D adrenoceptors are involved in reserpine-induced supersensitivity of rat tail artery.
    British journal of pharmacology, 2004, Volume: 142, Issue:4

    Topics: Animals; Aorta, Thoracic; Arteries; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Hypersensitivity; Gene Expression; Indoles; Japan; Male; Phenylephrine; Piperazines; Potassium Chloride; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Reserpine; RNA, Messenger; Serotonin; Spleen; Tail; Time Factors; Tritium

2004
Alpha1-adrenoceptor subtype substitution in knockout mice.
    British journal of pharmacology, 2004, Volume: 142, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Binding, Competitive; Hepatocytes; Mice; Mice, Knockout; Piperazines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha-1; Thymine; Tritium

2004
Hepatocytes from alpha1B-adrenoceptor knockout mice reveal compensatory adrenoceptor subtype substitution.
    British journal of pharmacology, 2004, Volume: 142, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Binding, Competitive; Boron Compounds; Cell Membrane; Genotype; Hepatocytes; Kinetics; Male; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Microscopy, Confocal; Piperazines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha-1; Thymine; Tritium

2004
Different roles of alpha1-adrenoceptor subtypes in mediating cardiomyocyte protein synthesis in neonatal rats.
    Clinical and experimental pharmacology & physiology, 2004, Volume: 31, Issue:9

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Cell Enlargement; Cells, Cultured; Dioxanes; Indoles; Leucine; Muscle Proteins; Myocytes, Cardiac; Norepinephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1

2004
Pharmacological characterization of alpha1-adrenoceptors in mouse isolated femoral small arteries.
    European journal of pharmacology, 2004, Oct-25, Volume: 503, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Algorithms; Animals; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Femoral Artery; In Vitro Techniques; Male; Mice; Mice, Inbred DBA; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Vascular Resistance; Vasoconstriction; Vasoconstrictor Agents

2004
Differential antagonism by conotoxin rho-TIA of contractions mediated by distinct alpha1-adrenoceptor subtypes in rat vas deferens, spleen and aorta.
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Cell Line; Cell Membrane; Conotoxins; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Iodine Radioisotopes; Male; Muscle Contraction; Norepinephrine; Piperazines; Potassium Chloride; Prazosin; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spleen; Tetralones; Vas Deferens

2005
Fentanyl attenuates alpha1B-adrenoceptor-mediated pulmonary artery contraction.
    Anesthesiology, 2005, Volume: 103, Issue:2

    Topics: Anesthetics, Intravenous; Animals; Clonidine; Dogs; Dose-Response Relationship, Drug; Fentanyl; Hydrogen-Ion Concentration; In Vitro Techniques; Phenylephrine; Piperazines; Prazosin; Pulmonary Artery; Receptors, Adrenergic, alpha-1; Vasoconstriction

2005
Correlation between vasoconstrictor roles and mRNA expression of alpha1-adrenoceptor subtypes in blood vessels of genetically engineered mice.
    British journal of pharmacology, 2005, Volume: 146, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Gene Expression Regulation; In Vitro Techniques; Indoles; Male; Mesenteric Arteries; Mice; Mice, Knockout; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; RNA, Messenger; Vasoconstriction

2005
Nandrolone treatment decreases the alpha1B-adrenoceptor mRNA level in rat kidney, but not the density of alpha1B-adrenoceptors in cultured MDCK-D1 kidney cells.
    European journal of pharmacology, 2005, Dec-19, Volume: 527, Issue:1-3

    Topics: Adrenergic alpha-Antagonists; Animals; Cell Line; Dogs; Down-Regulation; Gene Expression; Kidney; Male; Methiothepin; Nandrolone; Piperazines; Polymerase Chain Reaction; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Androgen; RNA, Messenger; Species Specificity; Tritium

2005
Alpha1D-adrenoceptor-induced relaxation on rat carotid artery is impaired during the endothelial dysfunction evoked in the early stages of hyperhomocysteinemia.
    European journal of pharmacology, 2006, Aug-14, Volume: 543, Issue:1-3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Carotid Arteries; Disease Models, Animal; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Hyperhomocysteinemia; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Superoxide Dismutase; Superoxides; Vasoconstriction; Vasodilation

2006
Selective agonists reveal alpha(1A)- and alpha(1B)-adrenoceptor subtypes in caudal artery of the young rat.
    Autonomic & autacoid pharmacology, 2006, Volume: 26, Issue:4

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Carbachol; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Indoles; Male; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tail; Tetrahydronaphthalenes; Thymine

2006
Alpha1A-adrenergic receptors are functionally expressed by a subpopulation of cornu ammonis 1 interneurons in rat hippocampus.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:3

    Topics: Action Potentials; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electrophysiology; Hippocampus; In Vitro Techniques; Interneurons; Isoproterenol; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1

2007
Adrenergic control of a constitutively active acetylcholine-regulated potassium current in canine atrial cardiomyocytes.
    Cardiovascular research, 2007, Jun-01, Volume: 74, Issue:3

    Topics: Acetylcholine; Action Potentials; Adrenergic Agents; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Bee Venoms; Clonidine; Cyclic AMP-Dependent Protein Kinases; Dihydropyridines; Dogs; Dose-Response Relationship, Drug; Estrenes; Heart Atria; Imidazoles; Indoles; Isoproterenol; Isoquinolines; Maleimides; Myocytes, Cardiac; Patch-Clamp Techniques; Phenylephrine; Phorbol 12,13-Dibutyrate; Piperazines; Potassium Channels; Prazosin; Propanolamines; Propranolol; Protein Kinase C; Pyrrolidinones; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Sulfonamides; Type C Phospholipases

2007
Role of alpha1-adrenoceptor subtypes in the effects of methylenedioxy methamphetamine (MDMA) on body temperature in the mouse.
    British journal of pharmacology, 2008, Volume: 153, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Body Temperature; Fever; Male; Mice; N-Methyl-3,4-methylenedioxyamphetamine; Piperazines; Prazosin; Quinazolines; Quinoxalines; Receptors, Adrenergic, alpha-1; Thymine

2008
Noradrenergic vasoconstriction of pig prostatic small arteries.
    Naunyn-Schmiedeberg's archives of pharmacology, 2008, Volume: 376, Issue:6

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Arteries; Brimonidine Tartrate; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Signaling; Dose-Response Relationship, Drug; Electric Stimulation; Guanethidine; In Vitro Techniques; Indoles; Male; Norepinephrine; Piperazines; Prazosin; Prostate; Quinoxalines; Swine; Thymine; Vasoconstriction; Yohimbine

2008
Different affinities of native alpha1B-adrenoceptors for ketanserin between intact tissue segments and membrane preparations.
    European journal of pharmacology, 2008, Apr-28, Volume: 584, Issue:2-3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Arteries; Binding, Competitive; Cell Line; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Humans; Indoles; Ketanserin; Male; Piperazines; Prazosin; Protein Binding; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Subcellular Fractions; Tail; Transfection; Vasoconstriction

2008
Increased alpha1D adrenergic receptor activity and protein expression in the urinary bladder of aged rats.
    World journal of urology, 2008, Volume: 26, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Animals; Blotting, Western; Fluorescent Antibody Technique; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Inbred F344; Receptors, Adrenergic, alpha-1; Sympathetic Nervous System; Urinary Bladder

2008
The alpha1D-adrenergic receptor induces vascular smooth muscle apoptosis via a p53-dependent mechanism.
    Molecular pharmacology, 2008, Volume: 74, Issue:4

    Topics: Acetophenones; Adrenergic alpha-1 Receptor Antagonists; Anthracenes; Aorta; Apoptosis; Benzothiazoles; Cells, Cultured; Culture Media, Serum-Free; Dioxanes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Mitochondria; Muscle, Smooth, Vascular; Phenylephrine; Piperazines; Prazosin; Pyridines; Reactive Oxygen Species; Receptors, Adrenergic, alpha-1; Time Factors; Toluene; Tumor Suppressor Protein p53

2008
Gene expressions and mechanical functions of α1-adrenoceptor subtypes in mouse ureter.
    World journal of urology, 2009, Volume: 27, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Epinephrine; Gene Expression; Indoles; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Norepinephrine; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; RNA, Messenger; Ureter

2009
Epinephrine, phenylephrine, and methoxamine induce infiltrative anesthesia via alpha1-adrenoceptors in rats.
    Acta pharmacologica Sinica, 2009, Volume: 30, Issue:9

    Topics: Adrenergic alpha-1 Receptor Antagonists; Anesthesia, Local; Anesthetics, Local; Animals; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Male; Methoxamine; Nifedipine; Nitroglycerin; Pain Measurement; Phentolamine; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1

2009
Characterization of α1-adrenoceptor subtypes mediating contraction in human isolated ureters.
    Urology, 2011, Volume: 77, Issue:3

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adult; Aged; Aged, 80 and over; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Indoles; Male; Middle Aged; Muscle Contraction; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Ureter; Young Adult

2011
Molecular and pharmacological characteristics of the gerbil α(1a)-adrenergic receptor.
    Hearing research, 2012, Volume: 283, Issue:1-2

    Topics: Adrenergic alpha-1 Receptor Antagonists; Amino Acid Sequence; Animals; Arteries; Chlorocebus aethiops; Clonidine; Cloning, Molecular; Cochlea; Conserved Sequence; COS Cells; Dioxanes; Dose-Response Relationship, Drug; Gerbillinae; Humans; Mice; Molecular Sequence Data; Piperazines; Prazosin; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Sequence Analysis, Protein; Transfection; Vasoconstriction

2012
Yohimbine antagonises α1A- and α1D-adrenoceptor mediated components in addition to the α2A-adrenoceptor component to pressor responses in the pithed rat.
    European journal of pharmacology, 2012, Mar-15, Volume: 679, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Dose-Response Relationship, Drug; Drug Interactions; Ethanolamines; Idazoxan; Male; Phenylephrine; Piperazines; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Thymine; Vasoconstriction; Xylazine; Yohimbine

2012
Ma huang and alpha subtype adrenoceptors in the cat pulmonary vascular bed.
    Journal of dietary supplements, 2008, Volume: 5, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cats; Clonidine; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Ephedra sinica; Female; Lung; Male; Phentolamine; Piperazines; Prazosin; Prospective Studies; Pulmonary Circulation; Receptors, Adrenergic; Vasoconstrictor Agents

2008
High vascular tone of mouse femoral arteries in vivo is determined by sympathetic nerve activity via α1A- and α1D-adrenoceptor subtypes.
    PloS one, 2013, Volume: 8, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic Fibers; Animals; Arginine; Calcium; Femoral Artery; Isoquinolines; Mice; Microscopy, Fluorescence; Muscle Tonus; Muscle, Smooth, Vascular; Myography; Myosin-Light-Chain Kinase; Naphthyridines; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Suramin; Thymine

2013
Prazosin has low potency at α1A-adrenoceptors and high potency at α1D -adrenoceptors in rat vas deferens.
    Autonomic & autacoid pharmacology, 2013, Volume: 33, Issue:3-4

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic Uptake Inhibitors; Animals; Cocaine; Dose-Response Relationship, Drug; Drug Interactions; In Vitro Techniques; Male; Muscle Contraction; Norepinephrine; Piperazines; Prazosin; Rats; Receptors, Adrenergic, alpha-1; Thymine; Vas Deferens

2013
Functional and radioligand binding characterization of the α1L-adrenoceptor subtype of the human vas deferens.
    Autonomic & autacoid pharmacology, 2015, Volume: 34, Issue:3-4

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Humans; Imidazoles; Indoles; Male; Phenylephrine; Piperazines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Tetrahydronaphthalenes; Tritium; Vas Deferens

2015
Both α
    Pharmacological reports : PR, 2021, Volume: 73, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Dose-Response Relationship, Drug; Male; Muscle Contraction; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Quinazolines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spleen; Thymine; Yohimbine

2021
Interaction between α
    Basic & clinical pharmacology & toxicology, 2021, Volume: 129, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Female; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle Contraction; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Spleen; Thymine; Yohimbine

2021
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